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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 277 / 349
Propylthiouracil Approved DB00550
small molecule | CAS: 51-52-5

A thiourea antithyroid agent. Propythiouracil inhibits the synthesis of thyroxine and inhibits the peripheral conversion of throxine to tri-iodothyronine. It is used in the treatment of hyperthyroidism. (From Martindale, The Extra Pharmacopeoia, 30th ed, p534)

Kategori:
Agents Causing Muscle ToxicityAntimetabolitesAntithyroid agents +14
Target Protein:
Type I iodothyronine deiodinaseThyroid peroxidase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Propyphenazone DB13524
small molecule | CAS: 479-92-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
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Proquazone DB13649
small molecule | CAS: 22760-18-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +14
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Proscillaridin DB13307
small molecule | CAS: 466-06-8

Proscillaridin is a cardiac glycoside that is derived from plants of the genus Scilla and in Drimia maritima (Scilla maritima). Studies suggest the potential cytotoxic and anticancer property of proscillaridin, based on evidence of the drug potently disruptin…

Kategori:
BufanolidesCarbohydratesCardanolides +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prosetin DB18649
small molecule

Prosetin is an orally administered blocker of MAP4K under investigation for the treatment of amyotrophic lateral sclerosis.[L48360]

Waktu Paruh-
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Prosopis juliflora pollen Approved DB10371
biotech

Prosopis juliflora pollen is the pollen of the Prosopis juliflora plant. Prosopis juliflora pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prosopis velutina seed Approved DB15510
biotech

Prosopis velutina seed allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 13367-85-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 41598-07-6

The principal cyclooxygenase metabolite of arachidonic acid. It is released upon activation of mast cells and is also synthesized by alveolar macrophages. Among its many biological actions, the most important are its bronchoconstrictor, platelet-activating-fa…

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Target Protein:
Prostaglandin D2 receptorProstaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtype +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

A cyclic endoperoxide intermediate produced by the action of CYCLOOXYGENASE on ARACHIDONIC ACID. It is further converted by a series of specific enzymes to the series 2 prostaglandins. [PubChem]

Kategori:
AnionsAutacoidsBiological Factors +14
Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prostalene DB11454
small molecule | CAS: 54120-61-5

Analog of prostaglandin F2 alpha.

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine DB13700
small molecule | CAS: 9012-00-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesCoagulants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine sulfate Approved DB09141
biotech | CAS: 9009-65-8

Since it's earliest discovery in salmon rine sperm heads in the late 1800's to its formal introduction via US FDA approval in 1939, protamine sulfate has occupied an important therapeutic niche as perhaps the only viable option for reversing the anticoagulant…

Kategori:
Amino Acids, Peptides, and ProteinsAntiheparin AgentsHematologic Agents +5
Waktu ParuhThe half-life of pr…
Vol. DistribusiIn a study group of…
KlirensIn a study group of…
Genetik -
Protego-PD DB18279
biotech

Protego-PD is a post-delivery placental extract.

Waktu Paruh-
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Protein C Approved DB11312
biotech

Protein C is an endogenously occurring plasma protein that plays a key role within the coagulation cascade. Protein C is a zymogen, or enzyme precursor, of a vitamin K-dependent anticoagulant glycoprotein (serine protease) that is synthesized in the liver. It…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBiological Factors +15
Target Protein:
Coagulation factor VCoagulation factor VIII
Waktu ParuhInitial half life =…
Vol. DistribusiVolume of distribut…
KlirensCL = 0.0533 dL/kg/h
Genetik -
Protein hydrolysate Approved DB09356
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProtein HydrolysatesProteins
Waktu Paruh-
Vol. Distribusi-
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Protein S human Approved DB13149
biotech

Protein S human is a vitamin K-dependent plasma glycoprotein which has antcoagulant properties [A19561]. It serves as a negative feedback mechanism in the coagulation cascade.

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBiological Factors +8
Target Protein:
Coagulation factor VCoagulation factor XVitamin K-dependent protein C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prothipendyl DB12958
small molecule | CAS: 303-69-5

Prothipendyl has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsNervous System +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prothrombin Approved DB11311
biotech | CAS: 9001-26-7

Prothrombin Complex Concentrate (Human), is indicated for the urgent reversal of acquired coagulation factor deficiency induced by Vitamin K antagonist (VKA, e.g., warfarin) therapy in adult patients with acute major bleeding.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +7
Target Protein:
Fibrinogen alpha chainFibrinogen beta chainCoagulation factor XIII A chain +1
Waktu ParuhApproximately 60h […
Vol. Distribusi-
Klirens-
Genetik -
Protiofate DB13632
small molecule | CAS: 58416-00-5

Deskripsi belum tersedia.

Kategori:
Genito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protionamide Approved DB12667
small molecule | CAS: 14222-60-7

Prothionamide has been used in trials studying the treatment of MDR-TB and HIV Infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +5
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protirelin Approved DB09421
small molecule | CAS: 24305-27-9

Protirelin is the pharmaceutically available synthetic analogue of the endogenous peptide thyrotropin-releasing hormone (TRH). It is a tri-peptide tropic hormone, released by the hypothalamus, that stimulates the release of Thyroid Stimulating Hormone (TSH) a…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +12
Target Protein:
Thyrotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 139-85-5

Also known as protocatechuic aldehyde, protocatechualdehyde is a naturally-occuring phenolic aldehyde that is found in barley, green cavendish bananas, grapevine leaves and root of the herb S. miltiorrhiza [A27224]. Protocatechualdehyde possesses antiprolifer…

Kategori:
AldehydesAnticoagulantsBenzene Derivatives +2
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protokylol Approved DB06814
small molecule | CAS: 136-70-9

Protokylol is a ?-adrenergic receptor agonist used as a bronchodilator in Europe and the United States.

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +15
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protoporphyrin DB02285
small molecule | CAS: 553-12-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsDermatologicalsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Hematopoietic prostaglandin D synthaseFerritin light chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prostaglandin G/H synthase 1Cytochrome c
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protriptyline Approved DB00344
small molecule | CAS: 438-60-8

Protriptyline hydrochloride is a dibenzocycloheptene-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents that produce hypertension +24
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proxalutamide DB16065
small molecule | CAS: 1398046-21-3

Proxalutamide is under investigation in clinical trial NCT03899467 (The Safety and Tolerability of Proxalutamide (GT0918) in Subjects With Metastatic Castrate Resistant Prostate Cancer).

Kategori:
HydantoinsImidazolesImidazolidines
Waktu Paruh-
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Genetik -
Proxazole DB13819
small molecule | CAS: 5696-09-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal DisordersOxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proxibarbal Approved DB13253
small molecule | CAS: 2537-29-3

Proxibarbal is a derivative of barbiturates, which has been used to treat migraines. Proxibarbal was approved in France but was withdrawn from the market due to the risk of inducing immunoallergic thrombocytopenia [L5476].

Kategori:
Barbiturates, PlainCentral Nervous System AgentsCentral Nervous System Depressants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proxyphylline DB13449
small molecule | CAS: 603-00-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRTX-100 DB05947
small molecule

PRTX-100 is a highly-purified form of Staphylococcal Protein A that binds directly to monocytes and a subset of B-cells that are involved in the development and progression of various autoimmune diseases. These binding interactions enable the compound to modu…

Waktu Paruh-
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Genetik -
Prucalopride Approved DB06480
small molecule | CAS: 179474-81-8

Prucalopride is a dihydrobenzofurancarboxamide derivative from the benzofurane family that selectively stimulates 5-HT4 receptors and thus, it presents enterokinetic properties.[A37348] The high selectivity of prucalopride allowed further development as it pr…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsCentral Nervous System Depressants +17
Target Protein:
5-hydroxytryptamine receptor 4
Waktu ParuhThe reported half-l…
Vol. DistribusiThe mean volume of …
KlirensPrucalopride renal …
Genetik -
Prulifloxacin DB11892
small molecule | CAS: 123447-62-1

Prulifloxacin has been investigated for the treatment of Urinary Tract Infection.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 4 subunit ADNA gyrase subunit ADNA gyrase subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Prunus armeniaca seed is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prussian blue Approved DB06783
small molecule | CAS: 14038-43-8

Prussian blue is described as a deep blue pigment that is produced when the oxidation of ferrous ferrocyanide salts occurs. It contains ferric hexacyanoferrate(II) in a cubic lattice crystal structure. It is insoluble in water but also tends to form a colloid…

Kategori:
AnionsAntidotesChelating Activity +11
Waktu Paruh-
Vol. DistribusiHistopathological e…
KlirensThe clearance from …
Genetik -
Pruvanserin DB13094
small molecule | CAS: 443144-26-1

Pruvanserin has been used in trials studying the treatment of Sleep Initiation and Maintenance Disorders.

Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-03140 DB05596
small molecule | CAS: 869493-21-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-07034 DB05993
small molecule | CAS: 903580-39-2

Deskripsi belum tersedia.

Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-08066 DB05607
small molecule

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-ASL DB17679
biotech

PRX-ASL is an intracellular enzyme replacement therapy designed to replace the missing or defective enzyme in patients with argininosuccinate lyase deficiency.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PRX-OTC DB17680
biotech

PRX-OTC is an intracellular enzyme replacement therapy designed to replace missing or defective enzyme in patients with ornithine transcarbamylase deficiency.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PS386113 DB05211
small molecule

PS386113 is a small molecule drug candidate under investigation for the treatment of inflammatory disorders. It is being developed by Schering-Plough and Pharmacopeia. Little information has been released about PS386113.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pseudoephedrine Approved DB00852
small molecule | CAS: 90-82-4

Pseudoephedrine is structurally related to [ephedrine] but exerts a weaker effect on the sympathetic nervous system.[A188820,A188823] Both drugs naturally occur in in ephedra plant which have a history of use in traditional Eastern medicine and were first res…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +30
Target Protein:
Sodium-dependent noradrenaline transporterD(2) dopamine receptorSodium-dependent dopamine transporter +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe apparent volume…
KlirensA 60mg oral dose of…
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 567-19-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pseudotropine DB04026
small molecule | CAS: 135-97-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pseudotsuga menziesii pollen Approved DB10986
biotech

Pseudotsuga menziesii pollen is the pollen of the Pseudotsuga menziesii plant. Pseudotsuga menziesii pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PSI-352938 DB12896
small molecule | CAS: 1199809-32-9

PSI-352938 has been used in trials studying the treatment of Hepatitis C and Hepatitis C, Chronic.

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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