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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 277 / 282
XP21279 DB06319
small molecule

XP21279 is a prodrug of [Levodopa], a dopamine precursor used in the management of Parkinson's disease. XP21279 was under investigation in clinical trial NCT00914602 (An Exploratory Study of XP21279 (With Lodosyn®) and Sinemet® in Parkinson's Disease Subjects…

Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XPro1595 DB16454
biotech | CAS: 2489785-77-3

XPro1595 is an investigational dominant-negative protein that neutralizes soluble TNF.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +10
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XR5944 DB06364
small molecule | CAS: 343247-32-5

XR5944 is a DNA bis-intercalating anticancer drug. It has both intercalating and antineoplastic activities.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
XTL-6865 DB06058
small molecule

XTL-6865 is a combination of two fully human monoclonal antibodies (Ab68 and Ab65) against the hepatitis C virus E2 envelope protein. It is being developed to prevent HCV re-infection following a liver transplant and for the treatment of chronic HCV disease.

Target Protein:
Genome polyprotein
Waktu Paruh-
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Genetik -
XV638 DB02702
small molecule | CAS: 183854-11-7

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
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Xylazine DB11477
small molecule | CAS: 7361-61-7

Xylazine is a clonidine analog used as a non-opioid tranquilizer in veterinary medicine and as an emetic, especially in cats.[A9095,L42675,A251420] It acts as an agonist at ?2 adrenoceptors; however, its affinity is lower than the one reported for other ?2 ad…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +15
Target Protein:
Alpha-2B adrenergic receptorAlpha-2C adrenergic receptorAlpha-2 adrenergic receptors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xylitol DB11195
small molecule | CAS: 87-99-0

Xylitol is a naturally occurring five-carbon sugar alcohol found in most plant material, including many fruits and vegetables. Xylitol-rich plant materials include birch and beechwood [A22081]. It is widely used as a sugar substitute and in "sugar-free" food …

Kategori:
AlcoholsCarbohydratesCompounds used in a research, industrial, or household setting +8
Target Protein:
Xylose isomeraseXylose isomeraseXylose isomerase +2
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Xylometazoline Approved DB06694
small molecule | CAS: 526-36-3

Xylometazoline is an imidazoline derivative [A228523] with sympathomimetic and nasal decongestant activity. Xylometazoline works by binding to alpha (?)-adrenergic receptors to cause vasoconstriction of nasal blood vessels.[A228508] Xylometazoline is avail…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +17
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-1A adrenergic receptor +3
Waktu ParuhNo information is a…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Exoglucanase/xylanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Exoglucanase/xylanase
Waktu Paruh-
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Klirens-
Genetik -
Y-27632 DB08756
small molecule | CAS: 146986-50-7

Y-27632 is an inhibitor of Rho-associated protein kinase. It inhibits calcium sensitization to affect smooth muscle relaxation.

Kategori:
Antihypertensive AgentsCardiovascular AgentsCentral Nervous System Agents +6
Target Protein:
ProthrombincAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alpha +2
Waktu Paruh-
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Genetik -
YA-101 DB18121
small molecule | CAS: 151602-49-2

Deskripsi belum tersedia.

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small molecule | CAS: 9041-22-9

Yeast beta-D-glucan is under investigation in clinical trial NCT00632008 (Soluble Beta-glucan (SBG) as Treatment for Diabetic Foot Ulcers).

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Yellow fever vaccine Approved DB10805
biotech

Yellow fever vaccine prevents against Yellow Fever, a viral hemorrhagic disease caused by the transmission of a _flavivirus_ through the bite of an infected mosquito. Symptoms of Yellow fever can range from asymptomatic, to mild flu-like illness, to more seve…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
Waktu Paruh-
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Genetik -
biotech

Yersinia pestis 195/p antigen (formaldehyde inactivated) is under investigation in clinical trial NCT02596308 (Immunogenicity and Safety of Subunit Plague Vaccine).

Kategori:
Actively Acquired ImmunityBacterial VaccinesBiological Products +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Yimitasvir DB18768
small molecule | CAS: 1959593-23-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral Agents
Waktu Paruh-
Vol. Distribusi-
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YK-4-279 DB17428
small molecule | CAS: 1037184-44-3

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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YKP-1358 DB06109
small molecule

YKP1358 is a novel serotonin (5-HT2A) and dopamine (D2) antagonist that has demonstrated potent activity in animals that relates to both positive and negative symptoms of schizophrenia. In addition, the YKP1358 pharmacological profile suggests a very low pote…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsDopamine Agents +7
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Yohimbine Approved DB01392
small molecule | CAS: 146-48-5

A plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of impotence. It is also alleged to be an aphrodisiac.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +35
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor +9
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
YS-ON-001 DB17291
biotech

YS-ON-001 is a combination of an inactivated purified rabies virus (IPRV) and the PIKA adjuvant (Poly I:C, kanamycin and calcium).

Waktu Paruh-
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YT-001 DB18564
small molecule | CAS: 1072301-78-0

Deskripsi belum tersedia.

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biotech | CAS: 943976-23-6

Yttrium Y-90 clivatuzumab tetraxetan is under investigation in clinical trial NCT00603863 (Safety and Efficacy Study of Different Doses of 90Y-hPAM4 Combined With Gemcitabine in Pancreatic Cancer).

Waktu Paruh-
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Genetik -
biotech | CAS: 501423-25-2

Deskripsi belum tersedia.

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Genetik -
biotech | CAS: 501423-27-4

Deskripsi belum tersedia.

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Z-160 DB12743
small molecule | CAS: 41332-24-5

Z160 has been used in trials studying the treatment of Postherpetic Neuralgia and Lumbosacral Radiculopathy.

Kategori:
Antiarrhythmic agentsBenzene DerivativesCalcium Channel Blockers +3
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
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Genetik -
small molecule | CAS: 161401-82-7

Non-methylated, competitive, and irreversible inhibitor of caspase 1, as well as other caspases,1 which can be used directly with purified enzymes. It does not require an esterase to hydrolyze the O-methyl ester like the cell-permeable form, Z-Val-Ala-Asp(O-M…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCaspase Inhibitors +7
Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zabedosertib DB18767
small molecule | CAS: 1931994-81-8

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Interleukin-1 receptor-associated kinase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zabofloxacin DB12479
small molecule | CAS: 219680-11-2

Zabofloxacin has been used in trials studying the treatment of Community Acquired Pneumonia and Chronic Obstructive Pulmonary Disease.

Kategori:
4-QuinolonesHeterocyclic Compounds, Fused-RingQuinolines +1
Waktu Paruh-
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Klirens-
Genetik -
Zafirlukast Approved DB00549
small molecule | CAS: 107753-78-6

Zafirlukast is an oral leukotriene receptor antagonist (LTRA) for the maintenance treatment of asthma, often used in conjunction with an inhaled steroid and/or long-acting bronchodilator. It is available as a tablet and is usually dosed twice daily. Another l…

Kategori:
Acids, AcyclicAgents to Treat Airway DiseaseAmides +37
Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh10 hours
Vol. Distribusi* 70 L
Klirens* apparent oral CL=…
Genetik -
biotech | CAS: 2567881-78-9

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Zagociguat DB18315
small molecule | CAS: 2201048-82-8

Deskripsi belum tersedia.

Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Zagotenemab DB16674
biotech | CAS: 2019133-28-7

Zagotenemab is under investigation in clinical trial NCT03518073 (A Study of LY3303560 in Participants With Early Symptomatic Alzheimer's Disease).

Waktu Paruh-
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Zalcitabine Approved DB00943
small molecule | CAS: 7481-89-2

A dideoxynucleoside compound in which the 3'-hydroxyl group on the sugar moiety has been replaced by a hydrogen. This modification prevents the formation of 5' to 3' phosphodiester linkages, which are needed for the elongation of DNA chains, thus resulting in…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh2 hours
Vol. Distribusi* 0.304 to 0.734 L/…
Klirens* 285 mL/min [HIV-i…
Genetik -
Zaleplon Approved DB00962
small molecule | CAS: 151319-34-5

Zaleplon is a sedative/hypnotic, mainly used for insomnia. It is known as a nonbenzodiazepine hypnotic. Zaleplon interacts with the GABA receptor complex and shares some of the pharmacological properties of the benzodiazepines. Zaleplon is a schedule IV drug …

Kategori:
AcetatesAcids, AcyclicAmides +22
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhApproximately 1 hour
Vol. Distribusi* 1.4 L/kg
Klirens* 1 L/h/kg
Genetik -
Zalifrelimab DB15632
biotech | CAS: 2148321-69-9

Zalifrelimab is under investigation in clinical trial NCT03894215 (Phase 2 Study of Anti-pd-1 Independently or in Combination With Anti-ctla-4 in Second-line Cervical Cancer).

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Zalunfiban DB18766
small molecule | CAS: 1448313-27-6

Deskripsi belum tersedia.

Waktu Paruh-
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Zalutumumab DB12202
biotech | CAS: 667901-13-5

Zalutumumab is a fully human IgG1 monoclonal antibody designed to bind with selectivity to the epidermal growth factor receptor (EGFR). Zalutumumab has been investigated for the treatment of Squamous Cell Cancer and Head and Neck Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zalypsis DB12454
small molecule | CAS: 308359-57-1

Zalypsis has been used in trials studying the treatment of Lymphoma, Solid Tumors, Ewing's Sarcoma, Endometrial Cancer, and Uterine Cervical Cancer, among others.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIsoquinolines
Waktu Paruh-
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Zamaporvint DB18765
small molecule | CAS: 1900754-56-4

Deskripsi belum tersedia.

Waktu Paruh-
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Zamerovimab DB17766
biotech | CAS: 2419087-87-7

Deskripsi belum tersedia.

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Zamicastat DB12389
small molecule | CAS: 1080028-80-3

Zamicastat has been used in trials studying the treatment of Hypertension and Chronic Heart Failure.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zampilimab DB16381
biotech | CAS: 2098280-42-1

Zampilimab is under investigation in clinical trial NCT04335578 (A Study to Evaluate Safety, Tolerability, Pharmacokinetics, and Efficacy of UCB7858 in Adult Kidney Transplant Recipients With Chronic Allograft Injury).

Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Zanamivir Approved DB00558
small molecule | CAS: 139110-80-8

A guanido-neuraminic acid that is used to inhibit neuraminidase.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +15
Target Protein:
NeuraminidaseNeuraminidaseSialidase-2
Waktu Paruh2.5-5.1 hours
Vol. Distribusi-
Klirens* 2.5 - 10.9 L/h [F…
Genetik -
Zanapezil DB04859
small molecule | CAS: 142852-50-4

Zanapezil (TAK-147) is a selective acetylcholine (ACh) esterase inhibitor under investigation as a drug for Alzheimer's disease (AD) treatment.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zandatrigine DB19051
small molecule | CAS: 2154406-04-7

Zandatrigine is under investigation in clinical trial NCT05226780 (Extension Study to Evaluate How Safe and Tolerable NBI-921352 Is as an Adjunctive Therapy for Participants With SCN8A-DEE).

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Zandelisib DB18245
small molecule | CAS: 1401436-95-0

Deskripsi belum tersedia.

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Zanidatamab Approved DB15471
biotech | CAS: 2169946-15-8

Zanidatamab is a bispecific antibody that binds two non-overlapping sites of HER2 (ERBB2).[A264718] It has been investigated for the treatment of HER2-positive solid tumors, including gastroesophageal, colorectal, and biliary tract cancers.[A264718] In No…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhBased on population…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
biotech | CAS: 2329698-82-8

According to Zymeworks, "ZW49 (zanidatamab zovodotin) is a bispecific anti-HER2 ADC that is based on the same antibody framework as [ZW25] but armed with a cytotoxic payload."[L8234] It is being investigated for several indications characterized by HER2 expre…

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