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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 277 / 321
Silodosin Approved DB06207
small molecule | CAS: 160970-54-7

Silodosin is a selective antagonist of alpha(?)-1 adrenergic receptors that binds to the ?<sub>1A</sub> subtype with the highest affinity. ?1-adrenergic receptors regulate smooth muscle tone in the bladder neck, prostate, and prostatic urethra: the ?<sub>1A</…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +15
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu ParuhThe elimination hal…
Vol. DistribusiSilodosin has an ap…
KlirensAfter intravenous a…
Genetik -
Silodrate Approved DB14116
small molecule | CAS: 12408-47-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siltuximab Approved DB09036
biotech | CAS: 541502-14-1

Siltuximab is a chimeric (human-mouse) monoclonal immunoglobulin G1-kappa antibody produced in a Chinese hamster ovary (CHO) cell line by recombinant DNA technology. Siltuximab prevents the binding of IL-6 to soluble and membrane-bound IL-6 receptors by formi…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Interleukin-6
Waktu ParuhThe mean terminal h…
Vol. DistribusiBased on population…
KlirensBody weight was ide…
Genetik -
Silver Approved DB12965
small molecule | CAS: 7440-22-4

Silver (Ag) is a chemical element that belongs in the family of transition metals in the periodic table. It has a high electrical conductivity, thermal conductivity, and reflectivity. Silver exists as a pure elemental form, alloy with other metals, and minera…

Kategori:
Antiseptics and DisinfectantsDermatologicalsElements +4
Target Protein:
MetallothioneinCeruloplasminAlbumin +1
Waktu ParuhThe biological half…
Vol. DistribusiFollowing exposure …
Klirens-
Genetik -
Silver cation DB14521
small molecule | CAS: 14701-21-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver citrate DB11233
small molecule | CAS: 126-45-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver nitrate Approved DB11080
small molecule | CAS: 7761-88-8

Silver nitrate is an inorganic compound with the chemical formula AgNO3. In its solid form, silver nitrate is coordinated in a trigonal planar arrangement. It is often used as a precursor to other silver-containing compounds. It is used in making photographic…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver oxide DB15668
small molecule | CAS: 20667-12-3

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Infective AgentsElectrolytes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 9015-51-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Infective Agents, Local +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver sulfadiazine Approved DB05245
small molecule | CAS: 22199-08-2

Silver sulfadiazine is a sulfa derivative topical antibacterial used primarily on second- and third-degree burns.

Kategori:
AmidesAminesAniline Compounds +14
Target Protein:
DNADihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simendan DB12286
small molecule | CAS: 131741-08-7

Simendan is under investigation in clinical trial NCT00527059 (Renal Effects of Levosimendan in Patients Admitted With Acute Decompensated Heart Failure).

Kategori:
Antiarrhythmic agentsCardiotonic AgentsCardiovascular Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 910562-13-9

Simenepag isopropyl has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simeprevir Approved DB06290
small molecule | CAS: 923604-59-5

Simeprevir is a hepatitis C virus (HCV) NS3/4A protease inhibitor indicated in patient's with HCV genotype 1 for the treatment of chronic hepatitis C virus (HCV) infection. HCV is a single-stranded RNA virus that is categorized into nine distinct genotypes, w…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +37
Target Protein:
Genome polyproteinNS3 proteaseGenome polyprotein
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of si…
Genetik -
Simethicone Approved DB09512
small molecule | CAS: 8050-81-5

Simethicone is a silicon based surfactant that decreases the surface tension of gastrointestinal gas bubbles to facilitate their elimination.[A228308] It has a favourable safety profile as it is not systemically absorbed.[A228308] Simethicone has been in u…

Kategori:
Antifoaming AgentsCompounds used in a research, industrial, or household settingDermatologicals +9
Waktu ParuhSimethicone is not …
Vol. DistribusiSimethicone is not …
KlirensSimethicone is not …
Genetik -
Simfibrate DB13433
small molecule | CAS: 14929-11-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1776942-10-9

RO6874281 is under investigation in clinical trial NCT03193190 (A Study of Multiple Immunotherapy-based Treatment Combinations in Participants With Metastatic Pancreatic Ductal Adenocarcinoma (Morpheus-pancreatic Cancer)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Simmondsia chinensis seed is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simoctocog alfa Approved DB09108
biotech | CAS: 1219013-68-9

Simoctocog alfa is a recombinant B-domain deleted (BDD) rFVIII produced in genetically modified human embryonic kidney (HEK) 293F cells. The harvested product is concentrated and purified by a series of chromatography steps. It is an antihemorrhagic agent use…

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +1
Target Protein:
von Willebrand factor
Waktu ParuhAt initial assessme…
Vol. DistribusiIt is observed that…
KlirensAt initial assessme…
Genetik -
Simotaxel DB15384
small molecule | CAS: 791635-59-1

Simotaxel is under investigation in clinical trial NCT00088647 (Study Evaluating MST-997 in Advanced Malignant Solid Tumors).

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simpinicline DB17065
small molecule | CAS: 753015-44-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simtuzumab DB12152
biotech | CAS: 1318075-13-6

Simtuzumab has been used in trials studying the treatment and basic science of Myelofibrosis, Pancreatic Cancer, Colorectal Cancer, and Idiopathic Pulmonary Fibrosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simufilam DB18817
small molecule | CAS: 1224591-33-6

Deskripsi belum tersedia.

Target Protein:
Filamin-A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simurosertib DB16330
small molecule | CAS: 1330782-76-7

Simurosertib is under investigation in clinical trial NCT03261947 (A Study to Evaluate the Safety, Tolerability, and Activity of TAK-931 in Participants With Metastatic Pancreatic Cancer, Metastatic Colorectal Cancer, and Other Advanced Solid Tumors).

Kategori:
Pyrazoles
Target Protein:
Cell division cycle 7-related protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simvastatin Approved DB00641
small molecule | CAS: 79902-63-9

Simvastatin, also known as the brand name product Zocor, is a lipid-lowering drug derived synthetically from a fermentation product of _Aspergillus terreus_. It belongs to the statin class of medications, which are used to lower the risk of cardiovascular dis…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +37
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-LHistone deacetylase 2
Gen Terkait:
KIF6 HMGCR SLCO1B1
Waktu Paruh4.85 hours[A181571]
Vol. DistribusiRat studies indicat…
Klirens-
Genetik 3 Varian
Sinapic acid DB08587
small molecule | CAS: 7362-37-0

Sinapic acid is a matrix for matrix-assisted laser desorption technique for protein MW determination. It is also a constituent of propolis.

Kategori:
Acids, CarbocyclicCinnamatesCompounds used in a research, industrial, or household setting +2
Target Protein:
Endo-1,4-beta-xylanase Y
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinapultide Approved DB11332
small molecule | CAS: 138531-07-4

Sinapultide (also known as KL4 peptide) is a synthetic protein used to mimic human lung surfactant protein B.[L2502] This protein has a weight of 2469.40.[L2502] Sinapultide is a 21-residue peptide made up of lysine (K) and leucine (L) residues with the se…

Kategori:
Amino Acids, Peptides, and ProteinsPulmonary Surfactants
Target Protein:
Lung epithelial cells
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinbaglustat DB17619
small molecule | CAS: 441061-33-2

Deskripsi belum tersedia.

Kategori:
CarbohydratesImines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sincalide Approved DB09142
biotech | CAS: 25126-32-3

Sincalide is a medication given by injection to assist in the diagnosis of gallbladder and pancreas disorders. It is identified as the 8-amino acid C-terminal segment of cholecystokinin and is also known as _CCK-8_. Naturally occurring cholecystokinin is a ga…

Kategori:
Amino Acids, Peptides, and ProteinsCholecystokinin AnalogDiagnostic Agents +7
Target Protein:
Cholecystokinin receptor type AGastrin/cholecystokinin type B receptor
Waktu ParuhLimited information…
Vol. DistribusiLimited information…
Klirens-
Genetik -
Sinecatechins Approved DB01266
small molecule | CAS: 188265-33-0

Sinecatechins is a botanical drug product for topical use. It is a partially purified fraction of the water extract of green tea leaves from Camellia sinensis, and is a mixture of catechins and other green tea components. Catechins constitute 85 to 95% (by we…

Kategori:
Antiviral AgentsBenzopyransChromans +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinefungin DB01910
small molecule | CAS: 58944-73-3

Sinefungin is a solid. This compound belongs to the purine nucleosides and analogues. These are compounds comprising a purine base attached to a sugar. The proteins that adenosyl-ornithine target include RdmB, modification methylase TaqI, rRNA (adenine-N6-)-m…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiparasitic Agents +7
Target Protein:
Modification methylase RsrIAclacinomycin 10-hydroxylase RdmBrRNA adenine N-6-methyltransferase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinomenine DB16892
small molecule | CAS: 115-53-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntirheumatic AgentsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sintilimab DB15765
biotech | CAS: 2072873-06-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siplizumab DB06371
biotech | CAS: 288392-69-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
T-cell surface antigen CD2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sipoglitazar DB19312
small molecule | CAS: 342026-92-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +4
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siponimod Approved DB12371
small molecule | CAS: 1230487-00-9

Siponimod, also known as _Mayzent_, by Novartis, is a new drug formulated for the management of Multiple Sclerosis (MS). It was approved by the FDA on March 26, 2019 [L5792] and by Health Canada on February 20, 2020.[L12171] This drug is considered a _sphingo…

Kategori:
Agents that produce hypertensionAntineoplastic and Immunomodulating AgentsAzetines +18
Target Protein:
Sphingosine 1-phosphate receptor 1Sphingosine 1-phosphate receptor 5
Waktu ParuhThe apparent elimin…
Vol. DistribusiSiponimod distribut…
KlirensApparent systemic c…
Genetik -
Sipuleucel-T Approved DB06688
biotech | CAS: 917381-47-6

Sipuleucel-T is a personalized, autologous, cellular immunotherapy. Sipuleucel-T is a therapeutic cancer vaccine for prostate cancer. Sipuleucel-T selectively targets the prostate-specific antigen (PSA) known as prostatic acid phosphatase (PAP) that is expres…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsAutologous Cellular Immunotherapy +6
Target Protein:
Prostatic acid phosphatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siramesine DB06555
small molecule | CAS: 147817-50-3

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siremadlin DB16331
small molecule | CAS: 1448867-41-1

Deskripsi belum tersedia.

Target Protein:
E3 ubiquitin-protein ligase Mdm2Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sirexatamab DB17515
biotech | CAS: 2414962-49-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sirna-027 DB05896
small molecule

Sirna-027 is a chemically modified short interfering RNA(siRNA) targeting Vascular Endothelial Growth Factor Receptor-1(VEGFR-1). VEGFR-1 is a key component of the clinically validated vascular endothelial growth factor (VEGF) pathway. Sirna-027 is developed …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siroheme DB02832
small molecule | CAS: 52553-42-1

Deskripsi belum tersedia.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingMetalloporphyrins +2
Target Protein:
Sulfite reductase [NADPH] hemoprotein beta-component
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sirolimus Approved DB00877
small molecule | CAS: 53123-88-9

Sirolimus, also known as rapamycin, is a macrocyclic lactone antibiotic produced by bacteria _Streptomyces hygroscopicus_, which was isolated from the soil of the Vai Atari region of Rapa Nui (Easter Island).[A242412] It was first isolated and identified as a…

Kategori:
Agents causing angioedemaAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu ParuhThe mean ± SD termi…
Vol. DistribusiThe mean (± SD) blo…
KlirensIn adult renal tran…
Genetik -
Sirpiglenastat DB17536
small molecule | CAS: 2079939-05-0

Sirpiglenastat, also known as DRP-104, is a prodrug of [6-diazo-5-oxo-L-norleucine] (DON), which is a broad-acting glutamine antagonist. It is under investigation in clinical trial NCT04471415 (Study to Investigate DRP-104 in Adults With Advanced Solid Tumors…

Kategori:
AcetatesAcids, AcyclicAmides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sirukumab DB11803
biotech | CAS: 1194585-53-9

Sirukumab has been used in trials studying the treatment and basic science of Giant Cell Arteritis and Arthritis, Rheumatoid.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIS-101-ADO DB18085
biotech

SIS-101-ADO is a siRNA therapeutic under investigation for the treatment of Autosomal Dominant Osteopetrosis Type 2 (ADO2).[L48091]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sisomicin DB12604
small molecule | CAS: 32385-11-8

Sisomicin has been used in trials studying the treatment of Pyoderma.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sisunatovir DB15674
small molecule | CAS: 1903763-82-5

Sisunatovir is under investigation in clinical trial NCT04267822 (Study of RV521 in the Treatment of Adult Subjects Who Have Undergone HCT With an URTI With RSV).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fusion glycoprotein F0
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sitafloxacin DB13261
small molecule | CAS: 163253-35-8

Deskripsi belum tersedia.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sitagliptin Approved DB01261
small molecule | CAS: 486460-32-6

Sitagliptin is an oral dipeptidyl peptidase-4 (DPP-4) inhibitor used in conjunction with diet and exercise to improve glycemic control in patients with type 2 diabetes mellitus[FDA label,A2260,A2255,A2256]. The effect of this medication leads to glucose depen…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +17
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhApproximately 12.4 …
Vol. Distribusi198L[FDA label,A226…
Klirens350mL/min[FDA label…
Genetik -
Sitamaquine DB04909
small molecule | CAS: 57695-04-2

Sitamaquine (WR-6026) is an orally active 8-aminoquinoline analog in development by the Walter Reed Army Institute, in collaboration with GlaxoSmithKline (formerly SmithKline Beecham), for the potential treatment of visceral leishmaniasis.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13801–13850 dari 16004
Sebelumnya Halaman 277 / 321 Berikutnya