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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 276 / 321
Sertaconazole Approved DB01153
small molecule | CAS: 99592-32-2

Sertaconazole nitrate is an antifungal medication of the imidazole class. It is available in topical formulations for the treatment of skin infections such as athlete's foot.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +8
Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sertindole Approved DB06144
small molecule | CAS: 106516-24-9

Sertindole, a neuroleptic, is one of the newer antipsychotic medications available. Serdolect is developed by the Danish pharmaceutical company H. Lundbeck. It is a phenylindole derivative used in the treatment of schizophrenia. It was first marketed in 1996 …

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +22
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C +5
Waktu Paruh3 days
Vol. Distribusi-
Klirens-
Genetik -
Sertraline Approved DB01104
small molecule | CAS: 79617-96-2

Sertraline is a popular antidepressant medication commonly known as a selective serotonin reuptake inhibitor (SSRI), and is similar to drugs such as [Citalopram] and [Fluoxetine]. Despite marked structural differences between compounds in this drug class, SSR…

Kategori:
Agents that reduce seizure thresholdAminesAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent dopamine transporterSigma receptor +2
Gen Terkait:
CYP2C19 CYP2C19
Waktu ParuhThe elimination hal…
Vol. DistribusiSertraline is widel…
KlirensIn pharmacokinetic …
Genetik 2 Varian
Sesame oil DB11172
biotech | CAS: 8008-74-0

Sesame oil is a commonly used vegetable oil in Asia and flavoring enhancer in various culinary practices. It is extracted from sesame seeds and contains linoleic acid, oleic acid, palmitic acid, stearic acid and other fatty acids. Sesame oil is reported to po…

Kategori:
Biological ProductsComplex MixturesDiet, Food, and Nutrition +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2379806-98-9

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setanaxib DB16869
small molecule | CAS: 1218942-37-0

Deskripsi belum tersedia.

Kategori:
PyrazolesPyridines
Target Protein:
NADPH oxidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setipiprant DB12562
small molecule | CAS: 866460-33-5

Setipiprant has been investigated for the treatment of Seasonal Allergic Rhinitis, asthma and scalp hair loss (Androgenetic Alopecia).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prostaglandin D2 receptorProstaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setiptiline DB09304
small molecule | CAS: 57262-94-9

Setiptiline is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). In Japan, the company Mochida started its commercialization for the treatment of depression started in 1989.

Kategori:
Antidepressive Agents, TetracyclicDibenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Alpha-2 adrenergic receptorsSerotonin Receptors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setmelanotide Approved DB11700
small molecule | CAS: 920014-72-8

Setmelanotide is the first available treatment for patients with pro-opiomelanocortin, proprotein subilisin/kexin type 1, or leptin deficiencies.[L24474] It is an agonist of the melanocortin 4 receptor.[A224449] Earlier attempts at agonizing MC4R (such as LY2…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Obesity Agents +19
Target Protein:
Melanocortin receptor 4
Waktu ParuhThe elimination had…
Vol. DistribusiThe apparent volume…
KlirensA 3mg subcutaneous …
Genetik -
Setogepram DB15447
small molecule | CAS: 1002101-19-0

Setogepram is under investigation in clinical trial NCT03184584 (Open-Label Rollover Study of PBI 4050 in Subjects With Alström Syndrome).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
G-protein coupled receptor 84Free fatty acid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setrobuvir DB12051
small molecule | CAS: 1071517-39-9

Setrobuvir has been used in trials studying the treatment of Hepatitis C, Chronic.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolinesSulfonamides +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setrusumab DB14778
biotech | CAS: 1847394-95-9

Setrusumab is under investigation in clinical trial NCT01406548 (Safety and Efficacy of Multiple Dosing Regimens of BPS804 in Post Menopausal Women With Low Bone Mineral Density).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevasemten DB18983
small molecule | CAS: 2417395-15-2

Sevasemten is under investigation in clinical trial NCT05291091 (Phase 2 Study of EDG-5506 in Becker Muscular Dystrophy (GRAND CANYON)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevelamer Approved DB00658
small molecule | CAS: 52757-95-6

Sevelamer is a phosphate binding drug used to prevent hyperphosphataemia in patients with chronic renal failure. It is marketed by Genzyme under the trade name Renagel.

Kategori:
AminesBile Acid SequestrantsChelating Agents +9
Target Protein:
Phosphate
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seviprotimut-L DB16328
biotech

Seviprotimut-L is under investigation in clinical trial NCT01546571 (Study of a Melanoma Vaccine in Stage Iib, Iic, and III Melanoma Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevirumab DB17771
biotech | CAS: 138660-96-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seviteronel DB12275
small molecule | CAS: 1610537-15-9

Seviteronel has been used in trials studying the treatment of CRPC, Prostate Cancer, and Castration-resistant Prostate Cancer.

Kategori:
Antineoplastic AgentsCytochrome P-450 Enzyme InhibitorsEnzyme Inhibitors
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevoflurane Approved DB01236
small molecule | CAS: 28523-86-6

Sevoflurane is an ether inhalation anesthetic agent used to induce and maintain general anesthesia.[L42340] It is a volatile, non-flammable compound with a low solubility profile and blood/gas partition coefficient.[L42340] Sevoflurane was patented in 1972, w…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +17
Target Protein:
GABA(A) ReceptorGlycine receptor subunit alpha-1Glutamate receptor 1 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiPatients given low-…
KlirensIn patients given l…
Genetik -
Sevuparin DB15007
small molecule

Sevuparin is under investigation in clinical trial NCT03853421 (Placebo-controlled Study to Determine the Safety and Tolerability of Subcutaneous Doses of Sevuparin).

Kategori:
CarbohydratesGlycosaminoglycansPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SF1126 DB05210
small molecule

SF1126 is an integrin-targeted PI3 kinase inhibitor.

Kategori:
Amino Acids, Peptides, and ProteinsBenzopyransHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Phosphatidylinositol 3-kinase regulatory subunit alphaPhosphatidylinositol 3-kinase regulatory subunit betaPhosphatidylinositol 3-kinase regulatory subunit gamma +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGI-1776 DB12494
small molecule | CAS: 1025065-69-3

SGI-1776 has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGN-1 DB18135
biotech

SGN-1 is a genetically modified strain of _Salmonella enterica_ comprising methioninase.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGN-15 DB05818
biotech

SGN-15 is studied in the treatment of cancer. It combines a monoclonal antibody with the anticancer drug doxorubicin. Monoclonal antibodies are substances that are made in the laboratory and that can locate and bind to cancer cells. Doxorubicin is a type of a…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGN-30 DB05471
biotech

SGN-30 is an engineered monoclonal antibody (mAb) that reacts with significant affinity to the CD30 antigen, which is highly expressed on a variety of hematologic malignancies as compared to on normal cells. SGN-30 has been shown to induce direct anti-cancer…

Target Protein:
Nuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGN-B6A DB18377
biotech | CAS: 2764774-91-4

Sigvotatug vedotin (SGN-B6A) is a humanized immunoglobulin G1 anti-integrin beta-6 monoclonal antibody conjugated to monomethyl auristatin E.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGS-742 DB05010
small molecule | CAS: 123690-78-8

SGS-742 has been used in trials studying the treatment of Seizures and Metabolic Disease.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingGABA Agents +4
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
SGX-523 DB06314
small molecule | CAS: 1022150-57-7

A MET receptor tyrosine kinase inhibitor.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Shark liver oil DB11088
biotech | CAS: 68990-63-6

Shark oil is extracted from the livers of sharks, which can account for up to 25% of their total body weight. The 3 main targeted species are the deep sea shark (Centrophorus squamosus), the dogfish (Sqaulus acanthias), and the basking shark (Cetorhinus maxim…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Shea butter DB14311
biotech | CAS: 194043-92-0

Shea butter is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanecarboxylic AcidsCyclohexanes +3
Target Protein:
3-phosphoshikimate 1-carboxyvinyltransferase3-phosphoshikimate 1-carboxyvinyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SHR-A1904 DB18702
biotech

SHR-A1904 is under investigation in clinical trial NCT04877717 (A Study of SHR-A1904 in Patients With Advanced Solid Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siagoside DB12351
small molecule | CAS: 100345-64-0

Siagoside (Sygen, AGF 2) has been investigated for the treatment of Parkinson Disease. It is a naturally occurring substance in the nerve cell’s membrane that is thought to play a role in cell growth, development, and repair. Siagoside completed phase 2 trial…

Kategori:
Acidic GlycosphingolipidsCarbohydratesGangliosides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sibeprenlimab DB18919
biotech | CAS: 2382896-07-1

Sibeprenlimab is under investigation in clinical trial NCT05248659 (Phase 2/3 Open-label Trial of Sibeprenlimab in the Treatment of Immunoglobulin a Nephropathy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sibofimloc DB16400
small molecule | CAS: 1616113-45-1

Sibofimloc is under investigation in clinical trial NCT03943446 (TAK-018 for Prevention of the Recurrence of Postoperative Crohn's Disease (CD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sibutramine Approved DB01105
small molecule | CAS: 106650-56-0

Sibutramine (trade name Meridia in the USA, Reductil in Europe and other countries), usually as sibutramide hydrochloride monohydrate, is an orally administered agent for the treatment of obesity. It is a centrally acting stimulant chemically related to amphe…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +23
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Gen Terkait:
GNB3
Waktu Paruh1.1 hours
Vol. Distribusi-
Klirens* Oral cl=1750 L/h …
Genetik 1 Varian
Sifalimumab DB12773
biotech | CAS: 1006877-41-3

Sifalimumab is a fully human monoclonal antibody targeting interferon-alpha. The levels of interferon-alpha are elevated in many patients with active systemic lupus erythematosus (SLE, or lupus) and other autoimmune disorders, and may be associated with disea…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Interferon alpha-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIG-001 DB17826
biotech

SIG-001 is a cultured human retinal pigment epithelial cell line (ARPE-19) genetically modified with a non-viral vector to express B domain deleted human factor VIII protein, encapsulated within two-layer modified alginate spheres.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIG-007 DB17710
biotech

SIG-007 is a gene therapy that consists of cells that are genetically modified with a non-viral vector to express human alpha-galactosidase A. Developed by Sigilon Therapeutics, t is being investigated for the treatment of Fabry Disease.[L46153]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIG-205 DB18548
biotech

SIG-205 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express human native alpha-L-iduronidase enzyme (hIDUA), encapsulated within two-layer modified alginate spheres

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIG-207 DB18547
biotech

SIG-207 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express Human alpha-galactosidase A (alpha-Gal A), encapsulated within two-layer modified alginate spheres

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silanol Approved DB11343
small molecule | CAS: 70131-67-8

Silanol is an FDA-approved food contact substance that is commonly used in organosilicon chemistry and silicate mineralogy.

Kategori:
Silicon Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silatecan DB12384
small molecule | CAS: 220913-32-6

Silatecan has been used in trials studying the treatment of GBM, Tumors, Gliosarcoma, Solid Malignancies, and Glioblastoma Multiforme, among others.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sildenafil Approved DB00203
small molecule | CAS: 139755-83-2

In eliciting its mechanism of action, sildenafil ultimately prevents or minimizes the breakdown of cyclic guanosine monophosphate (cGMP) by inhibiting cGMP specific phosphodiesterase type 5 (PDE5) [F3850, F3853, F3856, F3859, F3883, F3886, L5611, L5614]. The …

Kategori:
Agents Causing Muscle ToxicityAmidesCardiovascular Agents +33
Target Protein:
Plasma protease C1 inhibitorcGMP-specific 3',5'-cyclic phosphodiesteraseRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma +3
Gen Terkait:
ACE GNB3
Waktu ParuhThe terminal phase …
Vol. DistribusiThe mean steady-sta…
KlirensThe total body clea…
Genetik 2 Varian
Silibinin DB09298
small molecule | CAS: 22888-70-6

Silibinin is the major active constituent of silymarin, a standardized extract of the milk thistle seeds, containing a mixture of flavonolignans consisting of silibinin, isosilibinin, silicristin, silidianin and others. Silibinin is presented as a mixture of …

Kategori:
Alimentary Tract and MetabolismAntineoplastic AgentsAntineoplastic Agents, Phytogenic +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 68611-44-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silicic acid DB14138
small molecule | CAS: 1343-98-2

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicSilicon Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silicon Approved DB12982
small molecule | CAS: 7440-21-3

Silicon is under investigation in clinical trial NCT00103246 (Photodynamic Therapy Using Silicon Phthalocyanine 4 in Treating Patients With Actinic Keratosis, Bowen's Disease, Skin Cancer, or Stage I or Stage II Mycosis Fungoides).

Kategori:
Diet, Food, and NutritionElementsFood +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silicon dioxide Approved DB11132
small molecule | CAS: 7631-86-9

Silicon dioxide, or silica, is an oxide of silicon with the chemical formula SiO2. It is found in nature as agate, amethyst, chalcedony, cristobalite, flint, sand, QUARTZ, and tridymite as transparent and tasteless crystals. Inhalation of fine crystals is tox…

Kategori:
ColloidsComplex MixturesCompounds used in a research, industrial, or household setting +6
Target Protein:
Macrophage receptor MARCO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silk sericin DB15531
biotech | CAS: 1190590-38-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsArthropod ProteinsBiopolymers +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silmitasertib DB15408
small molecule | CAS: 1009820-21-6

Silmitasertib is under investigation in clinical trial NCT03904862 (Testing the Safety and Tolerability of CX-4945 in Patients With Recurrent Medulloblastoma Who May or May Not Have Surgery).

Kategori:
Casein Kinase II, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Casein kinase II subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13751–13800 dari 16004
Sebelumnya Halaman 276 / 321 Berikutnya