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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (17430)

Halaman 275 / 1743
Acebilustat DB15385
small molecule | CAS: 943764-99-6

Acebilustat is under investigation in clinical trial NCT01748838 (Phase 1 Study Assessing the Safety and Tolerability of CTX-4430).

Kategori:
Acids, CarbocyclicAza CompoundsBenzene Derivatives
Target Protein:
Leukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Acebutolol Approved DB01193
small molecule | CAS: 37517-30-9

A cardioselective beta-adrenergic antagonist with little effect on the bronchial receptors. The drug has stabilizing and quinidine-like effects on cardiac rhythm as well as weak inherent sympathomimetic action.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu ParuhThe plasma eliminat…
Vol. Distribusi-
Klirens-
Genetik -
Acecainide DB17602
small molecule | CAS: 32795-44-1

Acecainide is an investigational anti-arrhythmia drug.

Kategori:
Acids, CarbocyclicAminobenzoatesAntiarrhythmic agents +5
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aceclidine Approved DB13262
small molecule | CAS: 827-61-2

Aceclidine has been marketed in Europe but has not been used clinically in the United States. It is used in the treatment of open-angle glaucoma and is a parasympathomimetic agent.

Kategori:
Antiglaucoma Preparations and MioticsAutonomic AgentsMiotics +4
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aceclofenac Approved DB06736
small molecule | CAS: 89796-99-6

Aceclofenac is an oral non-steroidal anti-inflammatory drug (NSAID) with marked anti-inflammatory and analgesic properties used to treat osteoarthritis, rheumatoid arthritis and ankylosing spondylitis. It is reported to have a higher anti-inflammatory action …

Kategori:
Acetic Acid Derivatives and Related SubstancesAcids, CarbocyclicAgents causing hyperkalemia +20
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Acediasulfone DB08926
small molecule | CAS: 80-03-5

Acediasulfone (INN) is an antimicrobial and antimalarial long-acting prodrug of dapsone.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Acedoben DB04500
small molecule | CAS: 556-08-1

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Acefylline DB13573
small molecule | CAS: 652-37-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aceglutamide DB04167
small molecule | CAS: 2490-97-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +2
Target Protein:
o-succinylbenzoate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Acemannan DB19224
small molecule | CAS: 110042-95-0

Acemannan is under investigation in clinical trial NCT03250923 (Celagace™ Orarinse Solution for Treatment of Candidiasis).

Kategori:
Adjuvants, ImmunologicAnti-Infective AgentsAntineoplastic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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