Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (16004)

Halaman 274 / 321
Scopolamine Approved DB00747
small molecule | CAS: 51-34-3

Scopolamine is a tropane alkaloid isolated from members of the _Solanaceae_ family of plants, similar to [atropine] and [hyoscyamine], all of which structurally mimic the natural neurotransmitter [acetylcholine].[A228423, A228763] Scopolamine was first synthe…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhThe half-life of sc…
Vol. DistribusiThe volume of distr…
KlirensIV infusion of 0.5 …
Genetik -
Scriptaid DB17053
small molecule | CAS: 287383-59-9

Scriptaid is a histone deacetylase (HDAC) inhibitor researched for its anti-tumor properties.[A253127]

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Scutellaria baicalensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Scutellaria lateriflora Approved DB14339
biotech

Scutellaria lateriflora is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SCY-635 DB12451
small molecule | CAS: 210759-10-7

SCY-635 has been investigated for the treatment of Chronic Hepatitis C and Hepatitis C Infection.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic
Target Protein:
Guided entry of tail-anchored proteins factor CAMLG
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
scyllo-inositol DB03106
small molecule | CAS: 488-59-5

An isomer of glucose that has traditionally been considered to be a B vitamin although it has an uncertain status as a vitamin and a deficiency syndrome has not been identified in man. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1379) Inositol phosph…

Kategori:
AlcoholsCarbohydratesStereoisomerism +1
Target Protein:
Lysosomal acid glucosylceramidase1-phosphatidylinositol phosphodiesteraseCDP-diacylglycerol--inositol 3-phosphatidyltransferase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD-0006 DB07943
small molecule | CAS: 271576-80-8

Deskripsi belum tersedia.

Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD118 DB05207
small molecule

SD118 was previously under investigation in Japan for a different indication and now, following re-profiling and evaluation in experimental animal models, has demonstrated its potential as a new oral therapy for neuropathic pain.

Target Protein:
Tumor necrosis factorInterleukin-1 receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD146 DB02729
small molecule | CAS: 183854-21-9

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Selenium Compounds
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEA-BCMA DB18309
biotech | CAS: 2115084-53-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEA-CD70 DB17555
biotech

SEA-CD70 is an investigational humanized, non-fucosylated monoclonal antibody targeting CD70. SEA-CD70 is under investigation in clinical trial NCT04227847 (A Safety Study of SEA-CD70 in Patients With Myeloid Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sebacic acid DB07645
small molecule | CAS: 111-20-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsLipids
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sebelipase alfa Approved DB11563
biotech | CAS: 1276027-63-4

The lysosomal acid lipase (LAL) enzyme is found in lysosomes and is primarily responsible for the metabolism of lipids, and its absence or deficiency results in the accumulation of lipids in various organs. This lipid accumulation can lead to end-organ damage…

Kategori:
Alimentary Tract and MetabolismCarboxylic Ester HydrolasesCholesterol Ester Storage Disease, drug therapy +7
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients 4-11 ye…
KlirensAcross all age grou…
Genetik -
Sebetralstat DB18305
small molecule | CAS: 1933514-13-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secalciferol DB18406
small molecule | CAS: 55721-11-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seclidemstat DB17117
small molecule | CAS: 1423715-37-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysine-specific histone demethylase 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secnidazole Approved DB12834
small molecule | CAS: 3366-95-8

Secnidazole is a second-generation 5-nitroimidazole antimicrobial agent. It is structurally related to other 5-nitroimidazoles, including [DB00916] and [DB00911], but displays improved oral absorption and a longer terminal elimination half-life than other dru…

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +18
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe total body clea…
Genetik -
Secobarbital Approved DB00418
small molecule | CAS: 76-73-3

Secobarbital (marketed by Eli Lilly and Company under the brand names Seconal and Tuinal) is a barbiturate derivative drug with anaesthetic, anticonvulsant, sedative and hypnotic properties. It is commonly known as quinalbarbitone in the United Kingdom.

Kategori:
AdjuvantsAdjuvants, AnesthesiaAnticholinergic Agents +27
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29388-59-8

Secoisolariciresinol has been used in trials studying the prevention of Breast Cancer.

Kategori:
AlcoholsBenzene DerivativesBenzyl Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secretin human Approved DB09532
biotech | CAS: 108153-74-8

Human secretin is a gastrointestinal peptide hormone that regulates secretions in the stomach, pancreas, and liver. The hormone is produced from the enterochromaffin cells in the duodenum in response to the duodenal content with the pH less than 4.5 [L1875]. …

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGastrointestinal Agents +11
Target Protein:
Secretin receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of sy…
Genetik -
Secretin porcine Approved DB09527
biotech | CAS: 17034-35-4

Secretin porcine stimulates pancreatic and gastric secretions to aid in the diagnosis of pancreatic exocrine dysfunction and the diagnosis of gastrinoma.

Kategori:
Gastrointestinal AgentsSecretin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secukinumab Approved DB09029
biotech | CAS: 1229022-83-6

Secukinumab is a fully human monoclonal IgG1/? antibody against interleukin-17A (IL-17A), a proinflammatory cytokine implicated in various chronic immune-mediated inflammatory disorders, such as plaque psoriasis.[L39600] By blocking the actions of IL-17A, sec…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +14
Target Protein:
Interleukin-17A
Waktu ParuhThe half-life range…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
Genetik -
Segesterone DB14584
small molecule | CAS: 7690-08-6

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesProgestins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Segesterone acetate Approved DB14583
small molecule | CAS: 7759-35-5

Segesterone acetate is a steroidal progestin or synthetic progesterone and a 19-norprogesterone derivative with no CH3 group radical in position 6 [A37048]. In animal studies, segesterone acetate was shown to be one of the most potent progestins [A37090]. It …

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +24
Target Protein:
Progesterone receptorAndrogen receptorGlucocorticoid receptor
Waktu ParuhThe mean (SD) half …
Vol. DistribusiThe volume of distr…
KlirensNo pharmacokinetic …
Genetik -
SEL-24 DB18082
small molecule | CAS: 1616359-00-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEL-302 DB18434
biotech

SEL-302 is a recombinant adeno-associated virus vector-based gene therapy expressing the methylmalonyl-CoA mutase (MMUT) transgene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1609522-33-9

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 19Cyclin-dependent kinase 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seladelpar Approved DB12390
small molecule | CAS: 851528-79-5

Seladelpar is a peroxisome proliferator-activated receptor (PPAR)-delta (?) agonist. Seladelpar is a single enantiomer of the R-configuration.[L51149] On August 14, 2024, seladelpar was granted accelerated approval by the FDA for the treatment of primary bili…

Kategori:
Acids, AcyclicAntimetabolitesBCRP/ABCG2 Substrates +13
Target Protein:
Peroxisome proliferator-activated receptor delta
Waktu ParuhFollowing administr…
Vol. DistribusiSeladelpar steady s…
KlirensThe apparent oral c…
Genetik -
Selamectin DB11459
small molecule | CAS: 220119-17-5

Selamectin is a topical parasiticide and antihelminthic used on dogs and cats to treat and prevent infections of heartworms, fleas, ear mites, sarcoptic mange, and certain types of ticks in dogs as well as prevent heartworms, fleas, ear mites, hookworms, and …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selatogrel DB15163
small molecule | CAS: 1159500-34-1

Selatogrel is under investigation in clinical trial NCT03814200 (A Study to Investigate the Effect of Rifampicin on the Uptake and Breakdown of ACT-246475 in Healthy Subjects).

Kategori:
Organophosphorus Compounds
Target Protein:
P2Y purinoceptor 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selegiline Approved DB01037
small molecule | CAS: 14611-51-9

A selective, irreversible inhibitor of Type B monoamine oxidase. It is used in newly diagnosed patients with Parkinson's disease. It may slow progression of the clinical disease and delay the requirement for levodopa therapy. It also may be given with levodop…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +42
Target Protein:
Amine oxidase [flavin-containing] BSubstance-P receptorAmine oxidase [flavin-containing] A
Waktu Paruh1.2-2 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Selenium Compounds
Target Protein:
Inosine-5'-monophosphate dehydrogenase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenic acid Approved DB11068
small molecule | CAS: 7783-08-6

Selenic acid is an organic compound with the chemical formula H2SeO4. It may be found in over-the-counter daily dietary supplements as a source of [DB11135], an essential trace mineral for human health.

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +10
Waktu ParuhFollowing single or…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Selenious acid Approved DB11127
small molecule | CAS: 7783-00-8

Selenious acid is the acid form of sodium selenite, a form of selenium [L1910]. Selenium is an essential trace element and antioxidant. It is a cofactor metabolic enzyme regulation. It also plays an important role in maintaining the general health of tissu…

Kategori:
Alimentary Tract and MetabolismBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +14
Waktu Paruh30 days in beagle d…
Vol. DistribusiFollowing oral inta…
Klirens-
Genetik -
Selenium Approved DB11135
small molecule | CAS: 7782-49-2

Selenium is a trace metal in the human body particularly important as a component of glutathione peroxidase, an important enzyme in the prevention of cellular damage by free radicals and reactive oxygen species [FDA Label]

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +14
Waktu ParuhHalf life was obser…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 63795-61-9

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsSelenium CompoundsVarious Diagnostic Radiopharmaceuticals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenium Sulfide Approved DB00971
small molecule | CAS: 7488-56-4

Selenium Sulfide is an antifungal agent as well as a cytostatic agent, slowing the growth of hyperproliferative cells in seborrhea. Selenium Sulfide is the active ingredient often used in shampoos for the treatment of dandruff, seborrheic dermatitis and tinea…

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenocysteine DB02345
small molecule | CAS: 10236-58-5

A naturally occurring amino acid in both eukaryotic and prokaryotic organisms. It is found in tRNAs and in the catalytic site of some enzymes. The genes for glutathione peroxidase and formate dehydrogenase contain the TGA codon, which codes for this amino aci…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +5
Target Protein:
Cathelicidin antimicrobial peptideNucleoside diphosphate kinase AFormate dehydrogenase H +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenoinosine DB02753
small molecule | CAS: 40093-99-0

Deskripsi belum tersedia.

Kategori:
Selenium Compounds
Target Protein:
Nucleoside 2-deoxyribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenomethionine Approved DB11142
small molecule | CAS: 3211-76-5

Selenomethionine is a naturally occuring amino acid in some plant materials such as cereal grains, soybeans and enriched yeast but it cannot be synthesized from animals or humans. It can be produced from post-structural modifications. *In vivo*, selenomethion…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsOrganoselenium Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenomethionine Se-75 Approved DB09400
small molecule | CAS: 1187-56-0

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsOrganoselenium Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selepressin DB12495
small molecule | CAS: 876296-47-8

Selepressin has been used in trials studying the treatment of Septic Shock.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +11
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seletalisib DB12706
small molecule | CAS: 1362850-20-1

Seletalisib has been used in trials studying the treatment and basic science of Primary Sjogren's Syndrome.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seletracetam DB05885
small molecule | CAS: 357336-74-4

Seletracetam is a pyrrolidone derivative and with a structural similarity to newer generation antiepileptic drug levetiracetam. It binds to the same target as levetiracetam but with higher affinity and has shown potent seizure suppression in models of acquire…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +6
Target Protein:
Synaptic vesicle glycoprotein 2AVoltage-dependent N-type calcium channel subunit alpha-1BGlycine receptor (alpha-1/beta)
Waktu ParuhApproximately 8 hou…
Vol. DistribusiThe volume of distr…
KlirensThe total apparent …
Genetik -
Selexipag Approved DB11362
small molecule | CAS: 475086-01-2

Selexipag was approved by the United States FDA on December 22, 2015 for the treatment of pulmonary arterial hypertension (PAH) to delay disease progression and reduce risk of hospitalization. PAH is a relatively rare disease with usually a poor prognosis req…

Kategori:
AcetatesAcids, AcyclicAmides +19
Target Protein:
Prostacyclin receptor
Waktu ParuhSelexipag's termina…
Vol. Distribusi-
KlirensOn average, 35 L/ho…
Genetik -
Selgantolimod DB16324
small molecule | CAS: 2004677-13-6

Selgantolimod is under investigation in clinical trial NCT03491553 (Safety, Tolerability and Antiviral Activity of Selgantolimod in Virally-suppressed Adults With Chronic Hepatitis B).

Kategori:
AlcoholsFatty AlcoholsLipids
Target Protein:
Toll-like receptor 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seliciclib DB06195
small molecule | CAS: 186692-46-6

R-roscovitine (Seliciclib or CYC202) is a cyclin-dependent kinase (CDK) inhibitor that preferentially inhibits multiple enzyme targets including CDK2, CDK7 and CDK9, which alter the growth phase of treated cells. Developed by Cyclacel, seliciclib is being res…

Kategori:
Anti-Infective AgentsAntineoplastic AgentsEnzyme Inhibitors +3
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 7Cyclin-dependent kinase 1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selicrelumab DB14958
biotech | CAS: 1622140-49-1

Selicrelumab is under investigation in clinical trial NCT01008527 (Phase I Oncovir Poly IC:LC and NY-ESO-1/gp100).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seliforant DB15220
small molecule | CAS: 1164115-89-2

Seliforant is under investigation in clinical trial NCT01260753 (Proof of Activity Study of UR-63325 in Allergic Rhinitis Induced by Nasal Challenge).

Kategori:
Azetines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13651–13700 dari 16004
Sebelumnya Halaman 274 / 321 Berikutnya