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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 271 / 282
Vamotinib DB15396
small molecule | CAS: 1416241-23-0

Vamotinib (PF-114) is under investigation in clinical trial NCT02885766 (Study to Evaluate Tolerability, Safety, Pharmacokinetics and Preliminary Efficacy of PF-114 for Oral Administration in Adults With Ph+ Chronic Myeloid Leukemia, Which is Resistant to the…

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Vanadium Approved DB13971
small molecule | CAS: 7440-62-2

Deskripsi belum tersedia.

Kategori:
Diet, Food, and NutritionElementsFood +6
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Vancomycin Approved DB00512
small molecule | CAS: 1404-90-6

Antibacterial obtained from Streptomyces orientalis. It is a glycopeptide related to ristocetin that inhibits bacterial cell wall assembly and is toxic to kidneys and the inner ear. As of January 29 2018, CutisPharma's Firvanq is the only FDA approved vanc…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +17
Target Protein:
D-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycan
Waktu ParuhHalf-life in normal…
Vol. DistribusiThe volume of distr…
KlirensThe mean plasma cle…
Genetik -
Vandetanib Approved DB05294
small molecule | CAS: 443913-73-3

Vandetanib is an oral once-daily kinase inhibitor of tumour angiogenesis and tumour cell proliferation with the potential for use in a broad range of tumour types. On April 6 2011, vandetanib was approved by the FDA to treat nonresectable, locally advanced…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Vascular endothelial growth factor receptor 2Proto-oncogene tyrosine-protein kinase receptor RetEpidermal growth factor receptor +3
Waktu ParuhMedian half life of…
Vol. DistribusiVd of about 7450 L.
Klirens-
Genetik -
biotech | CAS: 2382896-00-4

Deskripsi belum tersedia.

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Vanillic acid DB02130
small molecule | CAS: 121-34-6

A flavoring agent. It is the intermediate product in the two-step bioconversion of ferulic acid to vanillin. (J Biotechnol 1996;50(2-3):107-13).

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +5
Target Protein:
Chorismate pyruvate-lyase
Waktu Paruh-
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small molecule | CAS: 498-00-0

Vanillyl alcohol has been used in trials studying the treatment of Smoking.

Kategori:
AlcoholsBenzene DerivativesBenzyl Compounds
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Vanillyl butyl ether Approved DB11299
small molecule | CAS: 82654-98-6

Vanillyl butyl ether is an ether of monohydroxybenzoic acid. It is added to food products as a flavoring agent. It is also present in cosmetics and personal care products as a fragrance ingredient, oral care agent, hair conditioning agent, and warming or cool…

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Vaniprevir DB11929
small molecule | CAS: 923590-37-8

Vaniprevir has been used in trials studying the treatment and diagnostic of Hepatitis C, Chronic Hepatitis C, Hepatitis C, Chronic, Chronic Hepatitis C Infection, and Chronic Genotype 1 Hepatitis C Virus Infection.

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +9
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Vanoxerine DB03701
small molecule | CAS: 67469-69-6

Vanoxerine is a highly selective dopamine transporter antagonist. It was synthesized in the late 1970s and developed as a potential treatment for depression.[A19824] Vanoxerine was later evaluated as a potential treatment for cocaine addiction due to its abil…

Kategori:
Antiarrhythmic agentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +6
Target Protein:
Sodium-dependent dopamine transporterHERG human cardiac K+ channel
Waktu ParuhThe mean eliminatio…
Vol. DistribusiVanoxerine is capab…
KlirensAt 25, 75 and 125 m…
Genetik -
Vantictumab DB12956
biotech | CAS: 1345009-45-1

Vantictumab has been used in trials studying the treatment of Solid Tumors, Pancreatic Cancer, and Stage IV Pancreatic Cancer.

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Vanucizumab DB12317
biotech | CAS: 1448221-05-3

Vanucizumab has been used in trials studying the treatment of ColoRectal Cancer and Advanced/Metastatic Solid Tumors.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Angiopoietin-2Vascular endothelial growth factor A, long form
Waktu Paruh-
Vol. Distribusi-
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biotech | CAS: 886584-10-7

Vanutide cridificar has been investigated for the treatment of Alzheimer Disease.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
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Vanzacaftor DB18373
small molecule | CAS: 2374124-49-7

Deskripsi belum tersedia.

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Vapreotide DB04894
biotech | CAS: 103222-11-3

Vapreotide is a synthetic octapeptide somatostatin analog. It was being studied for the treatment of cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntineoplastic Agents +20
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5Substance-P receptor
Waktu Paruh30 minutes
Vol. Distribusi-
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Vardenafil Approved DB00862
small molecule | CAS: 224785-90-4

Vardenafil is a selective inhibitor of cyclic guanosine monophosphate (cGMP)-specific phosphodiesterase type 5 (PDE5) and an oral therapy for the treatment of erectile dysfunction.[L45563,L45568] During sexual stimulation, nitric oxide (NO) is released from n…

Kategori:
Cardiovascular AgentsCytochrome P-450 CYP2C19 InhibitorsCytochrome P-450 CYP2C19 Inhibitors (weak) +30
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gammaRetinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma
Waktu ParuhVardenafil and its …
Vol. DistribusiVardenafil has a st…
KlirensVardenafil has a to…
Genetik -
Varenicline Approved DB01273
small molecule | CAS: 249296-44-4

Varenicline is a prescription medication used to treat smoking addiction. This medication is the first approved nicotinic receptor partial agonist. Specifically, varenicline is a partial agonist of the alpha4/beta2 subtype of the nicotinic acetylcholine recep…

Kategori:
BenzazepinesCholinergic AgentsCholinergic Agonists +17
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-3 +2
Waktu ParuhThe elimination hal…
Vol. Distribusi-
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Varespladib DB11909
small molecule | CAS: 172732-68-2

Varespladib has been investigated for the treatment and prevention of Sickle Cell Disease, Vaso-occlusive Crisis, and Acute Coronary Syndrome.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +4
Target Protein:
Phospholipase A2
Waktu Paruh-
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small molecule | CAS: 172733-08-3

Varespladib methyl has been investigated for the treatment of Acute Coronary Syndrome. Studies showed that Varespladib methyl treatment resulted in significant positive changes on lipoproteins and inflammation.

Kategori:
Acids, AcyclicEnzyme InhibitorsFatty Acids +4
Target Protein:
Phospholipase A2, membrane associatedGroup 10 secretory phospholipase A2
Waktu Paruh-
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Genetik -
biotech

Live attenuated zoster vaccine is available as two products: Zostavax for the prevention of shingles in immunocompetent people over the age of 50, and Varivax for the prevention of chickenpox in individuals 12 months of age and older. While the two vaccines c…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +8
Waktu Paruh-
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biotech

Recombinant zoster vaccine, manufactured as the product Shingrix by GlaxoSmithKline, is an adjuvanted non-live recombinant vaccine indicated for prevention of shingles. First approved in October 2017 by the Food and Drug Administration, Shingrix is the prefer…

Kategori:
VaccinesVaricella Zoster Vaccines
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Varlilumab DB11930
biotech | CAS: 1393344-72-3

Varlilumab has been used in trials studying the treatment of MELANOMA, Skin Ulcer, Burkett's Lymphoma, Mantle cell lymphoma, and Any T-cell Malignancy, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Varlitinib DB05944
small molecule | CAS: 845272-21-1

Varlitinib is an oral, selective, reversible, small molecule tyrosine kinase inhibitor of both ErbB-2 (Her-2/neu) and EGFR. Over-expression of ErbB-2 and EGFR receptors in tumors is predictive of poor prognosis in cancer patients. Varlitinib has shown signifi…

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
Waktu Paruh-
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Varoglutamstat DB18785
small molecule | CAS: 1276021-65-8

Deskripsi belum tersedia.

Target Protein:
Glutaminyl-peptide cyclotransferase
Waktu Paruh-
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small molecule | CAS: 37221-79-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsCentral Nervous System Agents +13
Target Protein:
Vasoactive intestinal polypeptide receptor 1
Waktu Paruh-
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Vasopressin Approved DB00067
biotech | CAS: 11000-17-2

Vasopressin (arginine-vasopressin or antidiuretic hormone) is a nonapeptide primarily produced in the hypothalamus that exhibits diverse physiological functions related to diuresis, hemodynamic modulation, and behaviour.[A110, A111, A112, A113, A228008] Vasop…

Kategori:
Amino Acids, Peptides, and ProteinsAntidiuretic AgentsArginine Vasopressin +22
Target Protein:
Vasopressin V2 receptorVasopressin V1a receptorVasopressin V1b receptor +1
Waktu ParuhVasopressin adminis…
Vol. Distribusi-
KlirensVasopressin has a c…
Genetik -
Vatalanib DB04879
small molecule | CAS: 212141-54-3

Vatalanib (PTK787/ZK-222584) is a new oral antiangiogenic molecule that inhibits all known vascular endothelial growth factor receptors. Vatalanib is under investigation for the treatment of solid tumors.

Kategori:
Enzyme InhibitorsProtein Kinase InhibitorsPyridazines +1
Target Protein:
Epidermal growth factor receptorVascular endothelial growth factor receptor 3Vascular endothelial growth factor receptor 2 +1
Waktu ParuhApproximately 6 hou…
Vol. Distribusi-
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Vatelizumab DB12346
biotech | CAS: 1238217-55-4

Vatelizumab has been used in trials studying the treatment of Ulcerative Colitis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
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Vatiquinone DB11917
small molecule | CAS: 1213269-98-7

Vatiquinone has been investigated for the treatment and prevention of Retinopathy, Rett Syndrome, Genetic Disease, Noise-induced Hearing Loss, and Methylmalonic Aciduria and Homocystinuria,Cblc Type.

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Waktu Paruh-
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biotech | CAS: 897936-89-9

Vatreptacog Alfa (Activated) has been used in trials studying the treatment of Haemophilia B, Haemophilia A, Congenital Bleeding Disorder, Haemophilia A With Inhibitors, and Haemophilia B With Inhibitors.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
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VaxSyn DB17827
biotech

VaxSyn HIV-1 is a recombinant form of the HIV envelope protein gp 160 developed by MicroGeneSys and the National Institute of Allergy and Infectious Diseases (NIAID).

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Vayarin Approved DB09328
biotech

Vayarin is a prescription medical food for the clinical dietary management of certain lipid imbalances blamed to be associated with attention deficit hyperactivity disorder (ADHD) in children. Vayarin contains _Lipirinen_, a proprietary composition containing…

Kategori:
Cytochrome P-450 CYP2E1 InhibitorsCytochrome P-450 CYP2E1 Inhibitors (strength unknown)Cytochrome P-450 Enzyme Inhibitors
Waktu ParuhAbout 2h [L1507]
Vol. Distribusi-
KlirensMainly in the feces…
Genetik -
VB-201 DB15259
small molecule | CAS: 630112-41-3

VB-201 is under investigation in clinical trial NCT01001468 (Study to Assess VB-201 in Patients With Psoriasis).

Kategori:
AlcoholsCarbohydratesGlycerophosphates +10
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VB-309 DB18539
small molecule | CAS: 2699021-75-3

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-310 DB18537
small molecule | CAS: 2699021-76-4

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-311 DB18540
small molecule | CAS: 2699021-77-5

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-312 DB18542
small molecule | CAS: 2699021-78-6

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-313 DB18541
small molecule | CAS: 2699021-79-7

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB10.16 DB17512
biotech

VB10.16 is a novel therapeutic antigen-presenting cell-targeting DNA vaccine developed to treat HPV16-positive cancers. It is composed of three parts, one encodes the E6/E7 fusion protein of human papillomavirus (HPV) type 16 (HPV16), a dimerization entity, a…

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VB2-011 DB05411
biotech

VB2-011 is an antibody developed as an anti-cancer treatment. According to some preclinical studies, it has a potential to inhibit tumour growth in various cancers including lymphoma and melanoma. This drug includes the parent IgM (H11 IgM) and a recombinant …

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VCA-894A DB18609
biotech

VCA-894A is a synthetic 2'-O-methoxyethyl phosphorothioate oligoribonucleotide sodium salt consisting of 19 nucleotide residues with the sequence 5'-MeCMeUGMeUGGAAGMeUGAGGGMeCMeCAG-3'

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VCN-01 DB18193
biotech

VCN-01 is an investigational, genetically modified human adenovirus encoding human PH20.

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vCP2292 DB19292
biotech

vCP2292 is under investigation in clinical trial NCT01982487 (Vaccine Therapy and IDO1 Inhibitor INCB024360 in Treating Patients With Epithelial Ovarian, Fallopian Tube, or Primary Peritoneal Cancer Who Are in Remission).

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Veal Approved DB10612
biotech

Veal allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Vebicorvir DB18784
small molecule | CAS: 2090064-66-5

Deskripsi belum tersedia.

Waktu Paruh-
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Vebreltinib DB16823
small molecule | CAS: 1440964-89-5

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
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Vecabrutinib DB16657
small molecule | CAS: 1510829-06-7

Vecabrutinib is under investigation in clinical trial NCT03037645 (Safety, PK, PD, and Antitumor Activity of Vecabrutinib (SNS-062) in B Lymphoid Cancers).

Kategori:
Amines
Target Protein:
Tyrosine-protein kinase BTK
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Vecuronium Approved DB01339
small molecule | CAS: 86029-43-8

Monoquaternary homolog of pancuronium. A non-depolarizing neuromuscular blocking agent with shorter duration of action than pancuronium. Its lack of significant cardiovascular effects and lack of dependence on good kidney function for elimination as well as i…

Kategori:
AndrostanesAndrostanolsAnticholinergic Agents +15
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2
Waktu Paruh51–80 minutes
Vol. Distribusi-
Klirens-
Genetik -
Vedolizumab Approved DB09033
biotech | CAS: 943609-66-3

Vedolizumab is a recombinant humanized IgG1 monoclonal antibody directed against the human lymphocyte ?4?7 integrin, a key mediator of gastrointestinal inflammation implicated in diseases like ulcerative colitis or Crohn's disease.[L48216] ?4?7 integrin facil…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-4Integrin beta-7
Waktu ParuhVedolizumab has a l…
Vol. DistribusiSerum apparent volu…
KlirensVedolizumab clearan…
Genetik -
Vedroprevir DB12037
small molecule | CAS: 1098189-15-1

Vedroprevir has been investigated for the treatment of Hepatitis C, Chronic.

Kategori:
Antiviral AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
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