Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 270 / 282
Ursolic acid DB15588
small molecule | CAS: 77-52-1

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +13
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Phospholipase A2DNA polymerase catalytic subunit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urtoxazumab DB17806
biotech | CAS: 502496-16-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Usistapide DB12414
small molecule | CAS: 403989-79-7

Usistapide has been used in trials studying the treatment of Obesity, Overweight, Metabolic Diseases, Nutrition Disorders, and Nutritional and Metabolic Diseases.

Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
USL-311 DB15265
small molecule | CAS: 1373268-67-7

USL-311 is under investigation in clinical trial NCT02765165 (Phase 1/2 Study of USL311 Alone and in Combination With Lomustine in Subjects With Advanced Solid Tumors and Relapsed/Recurrent Glioblastoma Multiforme (GBM)).

Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ustekinumab Approved DB05679
biotech | CAS: 815610-63-0

Ustekinumab is a human immunoglobulin (Ig) G1 kappa monoclonal antibody directed against interleukin(IL)-12 and IL-23, which are cytokines that are involved in immune and inflammatory responses.[A187349] It was generated via recombinant human IL-12 immunizati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Interleukin-23Interleukin-12 subunit beta
Waktu ParuhFollowing administr…
Vol. DistribusiThe total volume of…
KlirensThe median apparent…
Genetik -
Uteroglobin DB14880
biotech

Uteroglobin is under investigation in clinical trial NCT01473264 (Safety, Pk and Anti-inflammatory Effects of CC10 Protein in Premature Infants With Respiratory Distress Syndrome (RDS)).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsSecretoglobins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Utidelone DB17575
small molecule

Utidelone (UTD1), a novel microtubule stabilizing agent, is an epothilone B analogue produced by genetic engineering.[A257544,A257549] It is under investigation in clinical trials for various cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Utomilumab DB15113
biotech | CAS: 1417318-27-4

Utomilumab is under investigation in clinical trial NCT03318900 (T Cell Immunotherapy for Advanced Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Utreloxastat DB18154
small molecule | CAS: 1213269-96-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uttroside B DB18633
small molecule | CAS: 88048-09-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
UV1 DB18470
biotech

UV1 is a cancer vaccine consisting of p719-20, p728, and p725 synthetic peptides representing fragments of the hTERT subunit

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uzansertib DB17571
small molecule | CAS: 2088852-47-3

Uzansertib is under investigation in clinical trial NCT02587598 (Study of INCB053914 in Subjects With Advanced Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V-SARS DB15812
biotech

[COVID-19 convalescent plasma] is currently being acquired from recovered COVID-19 patients and used as prophylaxis for the virus. This therapeutic concept was applied to the development of V-SARS, which heat inactivates the plasma, and packages it into a onc…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V24343 DB05201
small molecule

The anti-obesity drug, V24343, acts by targeting the CB1 receptor in the brain and suppressing a person's appetite.

Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V590 DB16437
biotech

The V590 vaccine was developed on Merck’s recombinant vesicular stomatitis virus (rVSV) platform that was previously used to develop its Ebola Zaire virus vaccine, ERVEBO®[A226818, L30573, L30578]. By teaming up with IAVI, Merk developed a vaccine that does n…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V591 DB16438
biotech

The V591 vaccine, part of Merck’s COVID-19 vaccine programming, was developed using a modified measles vaccine virus as a vector for COVID-19 antigen delivery[L30593]. Through Merck’s acquisition of Thermis in May 2020, they were able to leverage Thermis’ pla…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VA-MENGOC-BC® DB15800
biotech

VA-MENGOC-BC is a meningococcal B and C vaccine and an outer membrane vesicle (OMV)-based vaccine. The OMVs contain over 100 proteins, and are derived from meningococcal group B and capsular polysaccharide of meningococcal group C. As there already exists a p…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vabicaserin DB12071
small molecule | CAS: 887258-95-9

Vabicaserin has been used in trials studying the health services research and treatment of Schizophrenia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vaborbactam Approved DB12107
small molecule | CAS: 1360457-46-0

Vaborbactam is a ?-lactamase inhibitor based on a cyclic boronic acid pharmacophore.[A32053] It has been used in trials investigating the treatment of bacterial infections in subjects with varying degrees of renal insufficiency. In August 2017, a combination …

Kategori:
AcidsAcids, NoncarboxylicAnti-Infective Agents +6
Target Protein:
Beta-lactamaseBeta-lactamaseCarbapenem-hydrolyzing beta-lactamase KPC +7
Waktu ParuhThe half life of va…
Vol. DistribusiThe steady-state vo…
KlirensThe mean renal clea…
Genetik -
VAC-52150 DB17781
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vactosertib DB15310
small molecule | CAS: 1352608-82-2

Vactosertib is under investigation in clinical trial NCT03724851 (Vactosertib in Combination With Pembrolizumab in Metastatic Colorectal or Gastric Cancer).

Kategori:
AminesEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
TGF-beta receptor type-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VAD-044 DB17697
small molecule

VAD-044 is an allosteric AKT inhibitor developed by Vaderis Therapeutics AG. It is being investigated for the treatment of Hereditary Hemorrhagic Telangiectasia.[L46098]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vadadustat Approved DB12255
small molecule | CAS: 1000025-07-9

One of the most common symptoms of advanced renal disease is anemia, caused primarily by the inability of the kidney to respond to anemic conditions with a corresponding increase in [erythropoietin] (EPO) production.[A244165] The treatment of anemia associate…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntianemic Preparations +20
Target Protein:
Egl nine homolog 1Prolyl hydroxylase EGLN2Prolyl hydroxylase EGLN3 +2
Waktu ParuhIn patients with di…
Vol. DistribusiThe apparent volume…
KlirensIn healthy subjects…
Genetik -
Vadimezan DB06235
small molecule | CAS: 117570-53-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +4
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vafidemstat DB16446
small molecule | CAS: 1357362-02-7

Vafidemstat is under investigation in clinical trial NCT03867253 (Testing the Safety and Preliminary Efficacy of the New Drug ORY-2001 in Mild to Moderate Alzheimer's Disease).

Kategori:
Oxazoles
Target Protein:
Lysine-specific histone demethylase 1AAmine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valaciclovir Approved DB00577
small molecule | CAS: 124832-26-4

Valaciclovir (valacyclovir), also known as _Valtrex_, is an antiviral drug that has been used to manage and treat various herpes infections for more than 2 decades. It was initially approved by the FDA in 1995 [FDA label] and marketed by GlaxoSmithKline [L56…

Kategori:
Acyclovir and prodrugAmino AcidsAmino Acids, Branched-Chain +19
Target Protein:
Thymidine kinaseDNA polymerase catalytic subunit
Waktu ParuhThe plasma eliminat…
Vol. DistribusiCerebrospinal fluid…
KlirensRenal clearance of …
Genetik -
Valanafusp alfa DB15336
biotech | CAS: 1815583-32-4

Valanafusp alfa is under investigation in clinical trial NCT03071341 (Extension Study Evaluating Long Term Safety and Activity of AGT-181 in Children With MPS I).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valbenazine Approved DB11915
small molecule | CAS: 1025504-45-3

Valbenazine is a modified metabolite of [tetrabenazine], and it is currently being approved for the treatment of various movement disorders, particularly tardive dyskinesia and chorea associated with Huntington's disease.[L47885,A261135] Tardive dyskinesia ha…

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +11
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhBoth Valbenazine an…
Vol. DistribusiThe mean steady-sta…
KlirensValbenazine has a m…
Genetik -
Valdecoxib Approved DB00580
small molecule | CAS: 181695-72-7

Valdecoxib was removed from the Canadian, U.S., and E.U. markets in 2005 due to concerns about a possible increased risk of heart attack and stroke.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +29
Target Protein:
Prostaglandin G/H synthase 2Carbonic anhydrase 2Carbonic anhydrase 3
Waktu Paruh8-11 hours
Vol. Distribusi* 86 L
Klirens* oral cl=6 L/h * …
Genetik -
Valemetostat DB18314
small molecule | CAS: 1809336-39-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valethamate DB13497
small molecule | CAS: 16376-74-2

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAminesAmmonium Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 238401-16-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1034190-08-3

Valiltramiprosate is under investigation in clinical trial NCT06304883 (Long-term Extension of Phase 3 Study of ALZ- 801 in APOE4/4 Early AD Subjects).

Kategori:
AlkanesAlkanesulfonic AcidsAmino Acids +7
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valine Approved DB00161
small molecule | CAS: 72-18-4

Valine is a branched-chain essential amino acid that has stimulant activity. It promotes muscle growth and tissue repair. It is a precursor in the penicillin biosynthetic pathway.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Propionyl-CoA carboxylase beta chain, mitochondrialBranched-chain-amino-acid aminotransferase, cytosolicValine--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 897937-73-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valinomycin DB14057
small molecule | CAS: 2001-95-8

A cyclododecadepsipeptide ionophore antibiotic produced by Streptomyces fulvissimus and related to the enniatins. It is composed of 3 moles each of L-valine, D-alpha-hydroxyisovaleric acid, D-valine, and L-lactic acid linked alternately to form a 36-membered …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valoctocogene roxaparvovec Approved DB15561
biotech | CAS: 1819334-78-5

Valoctocogene roxaparvovec is an adeno-associated virus serotype 5 (AAV5) based gene therapy vector that expresses the B-domain deleted SQ form of human coagulation factor VIII (hFVIII-SQ).[L43282] The expression of hFVIII-SQ is driven by a liver-specific pro…

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsBiological Factors +9
Target Protein:
Coagulation factor VIII (F8)
Waktu Paruh-
Vol. Distribusi-
KlirensThe maximum time to…
Genetik -
small molecule | CAS: 195156-77-5

Valomaciclovir stearate is under investigation in clinical trial NCT00831103 (A Phase 2b Trial of EPB-348 for the Treatment of Herpes Zoster).

Kategori:
Antiviral AgentsHerpes ZosterHeterocyclic Compounds, Fused-Ring +4
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valopicitabine DB13920
small molecule | CAS: 640281-90-9

The 3-O-valine ester prodrug of the nucleoside analog 2'-C-methylcytidine with anti-hepatitis C virus (HCV) activity. Upon administration, valopicitabine is converted into 2'-C-methylcytidine; upon phosphorylation into its 5-triphosphate form, this metabolite…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidines
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valproate bismuth Approved DB13910
small molecule | CAS: 60364-28-5

Valproate bismuth is available in Canada in the over-the-counter medication Neo-Laryngobis.

Kategori:
Bismuth containing drugsEENT Drugs, MiscellaneousNeurotoxic agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valproic acid Approved DB00313
small molecule | CAS: 99-66-1

Valproic acid, or valproate, is an fatty acid derivative and anticonvulsant originally synthesized in 1881 by Beverly S. Burton.[A178051] It enjoyed use as a popular organic solvent in industry and pharmaceutical manufacturing for nearly a century. In 1963, a…

Kategori:
Acids, AcyclicAnti-epileptic AgentAnticonvulsants +68
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialGlycogen synthase kinase-3 alphaHistone deacetylase 9 +13
Gen Terkait:
POLG POLG
Waktu Paruh13-19 hours.[label]…
Vol. Distribusi11 L/1.73m<sup>2</s…
Klirens0.56 L/hr/m<sup>2</…
Genetik 2 Varian
Valrocemide DB06657
small molecule | CAS: 92262-58-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valrubicin Approved DB00385
small molecule | CAS: 56124-62-0

Valrubicin (N-trifluoroacetyladriamycin-14-valerate) is a chemotherapy drug commonly marketed under the trade name VALSTAR. It is a semisynthetic analog of the [doxorubicin], which is an anthracycline drug. Used in the treatment of the bladder cancer, valrub…

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +9
Target Protein:
DNADNA topoisomerase 2-betaDNA topoisomerase 2-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valsartan Approved DB00177
small molecule | CAS: 137862-53-4

Valsartan belongs to the angiotensin II receptor blocker (ARB) family of drugs, which also includes [telmisartan], [candesartan], [losartan], [olmesartan], and [irbesartan]. ARBs selectively bind to angiotensin receptor 1 (AT1) and prevent the protein angiote…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +22
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhAfter intravenous (…
Vol. DistribusiThe steady-state vo…
KlirensFollowing intraveno…
Genetik -
Valspodar DB11869
small molecule | CAS: 121584-18-7

Valspodar has been used in trials studying the treatment of Cancer, Sarcoma, Leukemia, Lymphoma, and Breast Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsATP Binding Cassette Transporter, Subfamily B, Member 1Drug Resistance, Multiple +6
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valziflocept DB17728
biotech | CAS: 1804910-11-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vamifeport DB17692
small molecule | CAS: 2095668-10-1

Vamifeport is being investigated for the treatment of beta-thalassemia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vamikibart DB18896
biotech | CAS: 2744320-12-3

Vamikibart is under investigation in clinical trial NCT05642312 (A Study to Investigate Vamikibart in Participants With Uveitic Macular Edema).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vamorolone Approved DB15114
small molecule | CAS: 13209-41-1

Vamorolone is a novel and fully synthetic glucocorticoid developed by Santhera Pharmaceuticals. It is used to manage inflammation and immune dysregulation in patients with Duchenne muscular dystrophy (DMD), a neuromuscular disorder characterized by the insidi…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +20
Target Protein:
Glucocorticoid receptorMineralocorticoid receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
Menampilkan 13451–13500 dari 14063
Sebelumnya Halaman 270 / 282 Berikutnya