Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (16004)

Halaman 270 / 321
RVT-3101 DB18718
biotech

RVT-3101 is a fully human monoclonal antibody targeting vascular endothelial growth inhibitor, also known as TNF-like ligand 1A (TL1A) and TNF superfamily member 15. It is being investigated for ulcerative colitis.

Target Protein:
Tumor necrosis factor ligand superfamily member 15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RWJ-51084 DB03251
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +4
Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RWJ-56423 DB02812
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RWJ-800088 DB18693
biotech | CAS: 257287-15-3

RWJ-800088 is a synthetic PEGylated thrombopoietin (TPO) mimetic (TPOm) peptide with no sequence homology to endogenous TPO.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsPeptides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 40281-79-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase, inducibleNitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseDelta-aminolevulinic acid dehydratase3',5'-cyclic-AMP phosphodiesterase 4B +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ThermonucleaseListeriolysin regulatory protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 26289-39-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHaptensOligopeptides +1
Target Protein:
Glutathione S-transferase Mu 1Glutathione S-transferase Mu 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycylpeptide N-tetradecanoyltransferase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acyl carrier protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acyl carrier protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glutathione S-transferase P
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6803-19-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Glutathione S-transferase P
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Betaine--homocysteine S-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Toll-like receptor 2Capsid scaffolding proteinGag-Pol polyprotein +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Elongation factor-like GTPase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Hydroxyacylglutathione hydrolase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lactoylglutathione lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Arginase-1Arginase-2, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-23 DB07419
small molecule | CAS: 1010396-29-8

An androgen receptor modulator.

Kategori:
AmidesAminesAniline Compounds +2
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-3304 DB12149
small molecule | CAS: 203640-27-1

S-3304 has been used in trials studying the treatment of Lung Cancer, Solid Tumors, Non Small Cell Lung Cancer, Stage IIIB Non Small Cell Lung Cancer, and Stage IIIA Non Small Cell Lung Cancer, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingMatrix Metalloproteinase Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-38093 DB16893
small molecule | CAS: 862896-30-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAza Compounds +2
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-3APG DB17419
small molecule

S-3APG (S-3-[3-amino-phthalimido]-glutarimide) is a derivative of thalidomide with dual activity against B-cell neoplasias.[A255168]

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingIsoindoles +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glutaryl-CoA dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-40503 DB13938
small molecule | CAS: 404920-28-1

S-40503 is an investigational selective androgen receptor modulator (SARM) developed for the treatment of osteoporosis by the Japanese company Kaken Pharmaceuticals.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-49076 DB16821
small molecule | CAS: 1265965-22-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingSulfur Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-55746 DB18365
small molecule | CAS: 1448584-12-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingOxazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-777469 DB16321
small molecule | CAS: 885496-53-7

S-777469 is under investigation in clinical trial NCT00703573 (A Randomized, Double-blind Study to Evaluate the Safety and Efficacy of 2 Doses of S-777469 in Patients With Atopic Dermatitis).

Kategori:
Pyridines
Target Protein:
Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-8510 DB06504
small molecule

S-8510 / SB-737552 is a BZD inverse agonist investigated for the treatment of Alzheimer’s disease and mild to moderate senile dementia. It was being codeveloped by Shionogi and GlaxoSmithKline.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14047-27-9

Deskripsi belum tersedia.

Target Protein:
Thymidine kinase, cytosolicThymidine kinaseAdenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Histone acetyltransferase KAT5Acetyl-CoA acetyltransferase3-oxoacyl-[acyl-carrier-protein] synthase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 76426-40-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Polyamine aminopropyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 979-92-0

5'-S-(3-Amino-3-carboxypropyl)-5'-thioadenosine. Formed from S-adenosylmethionine after transmethylation reactions.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +7
Target Protein:
DNA (cytosine-5)-methyltransferase 3BHistamine N-methyltransferaseCap-specific mRNA (nucleoside-2'-O-)-methyltransferase +34
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Selenium Compounds
Target Protein:
tRNA (cmo5U34)-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-Apomorphine DB16927
small molecule | CAS: 39478-62-1

Deskripsi belum tersedia.

Target Protein:
D(1A) dopamine receptorD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Arsenate reductaseProtein ArsC3-mercaptopyruvate sulfurtransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
S-azabisabolene DB02099
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3054-01-1

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +3
Target Protein:
Methylated-DNA--protein-cysteine methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsLactoylglutathione Lyase, antagonists & inhibitorsOligopeptides +1
Target Protein:
Lactoylglutathione lyaseGlutathione S-transferase A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetyl-CoA acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase 1Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2986-20-1

S-Ethylisothiourea is a nitric oxide synthase inhibitor.

Kategori:
AmidesCardiovascular AgentsCentral Nervous System Agents +7
Target Protein:
Nitric oxide synthase, inducibleNitric oxide synthase 3Nitric oxide synthase oxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 24425-56-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsLactoylglutathione Lyase, antagonists & inhibitors +2
Target Protein:
Hematopoietic prostaglandin D synthaseLactoylglutathione lyaseGlutathione S-transferase Mu 4 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13451–13500 dari 16004
Sebelumnya Halaman 270 / 321 Berikutnya