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2279

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866 (38.0%)
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1100 (48.3%)
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Halaman 27 / 46
Mannitol busulfan Approved DB12097
small molecule | CAS: 1187-00-4

Mm has been used in trials studying the treatment of Cocaine Dependence and Diabetes Mellitus, Type 2.

Kategori:
Agents causing hyperkalemia
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Mannose DB12907
small molecule | CAS: 3458-28-4

Mannose is under investigation for the basic science of IUGR and Pregnancy.

Kategori:
CarbohydratesHexosesMonosaccharides
Waktu Paruh-
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small molecule | CAS: 3672-15-9

Mannose 6-phosphate has been used in trials studying the treatment of Wound, Cicatrix, Wound-healing, and Re-epithelialisation.

Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu Paruh-
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Mannosulfan DB13334
small molecule | CAS: 7518-35-6

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +7
Waktu Paruh-
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Genetik -
Mant-Adp DB03126
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAdenine NucleotidesAminobenzoates +8
Target Protein:
Myosin-14
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mapatumumab DB18945
biotech | CAS: 658052-09-6

Mapatumumab is under investigation in clinical trial NCT00094848 (Study of TRM-1 (TRAIL-R1 Monoclonal Antibody) in Subjects With Relapsed or Refractory Non-hodgkin's Lymphoma (NHL)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Maplirpacept DB18441
biotech

Maplirpacept is a recombinant fusion protein consisting of the CD47-binding domain of human signal regulatory protein alpha (SIRPa) linked to the IgG4 Fc region of human IgG.

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Maralixibat Approved DB16226
small molecule | CAS: 716313-53-0

Maralixibat (also known as SHP625, LUM001, and lopixibat) is an ileal bile acid transporter inhibitor, like [odevixibat].[A236823,A239249,L38834] Maralixibat is indicated for the treatment of cholestatic pruritus in patients with Alagille syndrome.[L38834] …

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyBile Therapy +9
Target Protein:
Ileal sodium/bile acid cotransporterHepatic sodium/bile acid cotransporter
Waktu ParuhThe mean half life …
Vol. Distribusi-
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Margetuximab Approved DB14967
biotech | CAS: 1350624-75-7

The HER2 oncoprotein, the product of the human _ERBB2_/mouse _neu_ genes, is a member of the HER family of receptor tyrosine kinases that includes the epidermal growth factor receptor (EGFR). Of the various subtypes of breast cancer, HER2-positive breast canc…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhMargetuximab has a …
Vol. DistribusiMargetuximab has a …
KlirensMargetuximab has a …
Genetik -
biotech | CAS: 2760218-55-9

Maridebart Cafraglutide is under investigation in clinical trial NCT05669599 (Dose-ranging Study to Evaluate the Efficacy, Safety, and Tolerability of AMG 133 in Adult Subjects With Overweight or Obesity, With or Without Type 2 Diabetes Mellitus).

Waktu Paruh-
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Marstacimab Approved DB17725
biotech | CAS: 1985638-39-8

Marstacimab is a human monoclonal immunoglobulin G Type 1 (IgG1) antibody produced by Chinese hamster ovary (CHO) cells by recombinant DNA technology.[L51803] It is a tissue factor pathway inhibitor (TFPI) antagonist, which is an endogenous anticoagulant.[A26…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Tissue factor pathway inhibitor
Waktu ParuhIn a study consisti…
Vol. DistribusiIn patients with he…
KlirensIn a study consisti…
Genetik -
Matuzumab DB05101
biotech | CAS: 339186-68-4

Matuzumab (formerly known as the experimental drug, EMD 72000) is a humanized monoclonal antibody used in cancer treatment. It has a high affinity for EGFR (epithelial growth factor receptor), frequently associated with the growth of blood vessels in malignan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epidermal growth factor receptor
Waktu Paruh196 hours
Vol. Distribusi-
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Mavacamten Approved DB14921
small molecule | CAS: 1642288-47-8

Mavacamten is a myosin inhibitor indicated for the treatment of adults with symptomatic New York Heart Association (NYHA) class II-III obstructive hypertrophic cardiomyopathy (HCM). It received initial US FDA approval in 2022, and it is one of the first myosi…

Kategori:
AminesBenzene DerivativesBenzyl Compounds +21
Target Protein:
Myosin-7
Waktu ParuhMavacamten has a va…
Vol. DistribusiThrough the use of …
KlirensMavacamten demonstr…
Genetik -
Mavorixafor Approved DB05501
small molecule | CAS: 558447-26-0

Mavorixafor is a CXC chemokine receptor 4 (CXCR4) antagonist.[L50642] It was first approved by the FDA on April 30, 2024, for the treatment of warts, hypogammaglobulinemia, infections, and myelokathexis (WHIM) syndrome, a genetic immunodeficiency disorder cha…

Kategori:
AlkanesAminesButanes +38
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiMavorixafor volume …
KlirensThe mean (CV%) appa…
Genetik -
MaxAdFVIII DB17713
biotech

MaxAdFVIII is an adenoviral vector that expresses the full-length human Factor VIII (hFVIII) cDNA. First developed by GenStar, it is being investigated for the treatment of hemophilia.

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Maxy-G34 DB05718
biotech

MAXY-G34 is a pegylated variant of human granulocyte-colony stimulating factor (G-CSF). This variant contains multiple non-naturally occurring lysines that have been introduced into alpha helixes of wild type human G-CSF as PEGylation sites, and from which mu…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +15
Waktu Paruh-
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Klirens-
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Mazdutide DB19099
biotech | CAS: 2259884-03-0

Mazdutide is under investigation in clinical trial NCT06143956 (A Chronic Weight Management Master Protocol Study (LY900038) of Multiple Intervention-specific-appendices (Isas) in Adult Participants With Obesity or Overweight).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
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Mazorelvimab DB17767
biotech | CAS: 2419087-89-9

Deskripsi belum tersedia.

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biotech

MB-102 are autologous T cells genetically modified to express CD123-specific, hinge-optimized CD28-costimulatory chimeric receptor and a truncated human epidermal growth factor receptor.

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MBP134 DB18686
biotech

MBP134 is a pan-ebolavirus cocktail comprising two broadly neutralizing human antibodies. It is under investigation for the treatment of Sudan ebolavirus (SUDV).

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MCC DB05282
small molecule

Mycobacterial Cell Wall-DNA Complex (MCC) is formulated from Mycobacterium phlei, a non-pathogenic strain of mycobacteria. MCC has been shown to have immune stimulatory and apoptosis (programmed cell death) activity against cancer cells. The product is a ster…

Target Protein:
Apoptosis-inducing factor 1, mitochondrial
Waktu Paruh-
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MD05 DB06375
small molecule

MD05 is a beta-tricalcium phosphate (beta-TCP) coated with recombinant human growth/differentiation factor-5 (rhGDF-5).

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MDX-018 DB05484
small molecule

MDX-018, also known as HuMax-Inflam, is a fully human antibody that is directed to IL-8 (interleukin-8) and may have potential application in oncology and inflammation. Trials will initially focus on studies to treat glioblastoma, a cancer of the central nerv…

Target Protein:
Interleukin-8
Waktu Paruh-
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MDX-1303 DB05945
biotech | CAS: 915947-57-8

MDX-1303 is a fully human antibody against the inhalation anthrax, the most lethal form of illness in humans caused by the Bacillus anthracis bacterium, and targets a protein component of these lethal toxins known as the anthrax protective antigen.

Target Protein:
Anthrax toxin receptor 2Anthrax toxin receptor 1
Waktu Paruh-
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MDX-214 DB06110
small molecule

MDX-214 consists of recombinant human epidermal growth factor (EGF) genetically linked to a fully human antibody fragment that is designed to activate cytotoxic killing of cancer cells by immune effector cells. It is developed for the treatment of EGF-R overe…

Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
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Genetik -
biotech | CAS: 1570067-55-8

Mecapegfilgrastim is under investigation in clinical trial NCT05463601 (Mecapegfilgrastim for the Prevention of Dalpiciclib -Induced Neutropenia in Advanced Breast Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +13
Waktu Paruh-
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Mecasermin Approved DB01277
biotech | CAS: 68562-41-4

Mecasermin contains recombinant-DNA-engineered human insulin-like growth factor-1 (rhIGF-1)[FDA Label]. IGF-1 consists of 70 amino acids in a single chain with three intramolecular disulfide bridges and a molecular weight of 7649 daltons. The amino acid seque…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesBiological Factors +15
Target Protein:
Insulin-like growth factor 1 receptorInsulin-like growth factor-binding protein 3Insulin receptor +1
Waktu ParuhMean half life of 5…
Vol. Distribusi* 0.257 ± 0.073 L/k…
KlirensClearance of Mecase…
Genetik -
Mecasermin rinfabate Approved DB14751
biotech | CAS: 478166-15-3

Mecasermin rinfabate is approved for severe primary insulin-like growth factor (IGF) deficiency or in patients with GH gene deletion who have developed antibodies to growth hormone (GH)[A176020]. Mecasermin rinfabate is similar to [DB01277] in that both drugs…

Kategori:
Anterior Pituitary Lobe Hormones and AnaloguesPituitary and Hypothalamic Hormones and AnaloguesSomatropin and Somatropin Agonists +1
Target Protein:
Insulin-like growth factor 1 receptorInsulin receptorCation-independent mannose-6-phosphate receptor
Waktu ParuhHalf life ranges fr…
Vol. DistribusiApproximately 1000m…
KlirensClearance ranges fr…
Genetik -
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

Waktu Paruh-
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MEDI-491 DB17859
biotech

MEDI-491 is a recombinant human parvovirus B19 vaccine composed of the VP1 and VP2 capsid proteins.

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MEDI3506 DB16473
biotech | CAS: 2376858-66-9

Tozorakimab (MEDI3506), developed by AstraZeneca, was investigated in multiple clinical trials to evaluate its safety, tolerability, efficacy, and pharmacokinetics across various conditions. These trials include NCT03096795 (completed; healthy participants, C…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Interleukin-33
Waktu Paruh-
Vol. Distribusi-
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MEDI6012 DB14833
biotech

Recombinant human lecithin:cholesterol acyltransferase is under investigation in clinical trial NCT03578809 (A Study to Evaluate the Safety and Efficacy of MEDI6012 in Acute ST Elevation Myocardial Infarction).

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Genetik -
biotech

The use of the plant species _Cannabis sativa_ and _Cannabis indica_, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical conditions as a wave of legalization in North America has changed public …

Kategori:
Agents producing tachycardiaBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +51
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +38
Waktu ParuhThe half life of TH…
Vol. DistribusiAs a very lipophili…
KlirensOne study reported …
Genetik -
Medroxyprogesterone acetate Approved DB00603
small molecule | CAS: 71-58-9

Medroxyprogesterone acetate (MPA) is a [progesterone] derivative that is more resistant to metabolism for improved pharmacokinetic properties.[A14848] MPA can be use to treat secondary amenorrhea, endometrial hyperplasia, abnormal uterine bleeding, osteoporos…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +46
Target Protein:
Progesterone receptorEstrogen receptorATP-dependent translocase ABCB1 +1
Waktu ParuhOral medroxyprogest…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Mefloquine Approved DB00358
small molecule | CAS: 53230-10-7

Malaria is a protozoan disease that places an enormous burden on human health in endemic areas around the world. The 2020 World Health Organization malaria report indicates a 60% decrease in the global malaria fatality rate between 2000 to 2019.[L30618] Despi…

Kategori:
Agents Causing Muscle ToxicityAgents that reduce seizure thresholdAminoquinolines +20
Target Protein:
Fe(II)-protoporphyrin IX80S ribosomal subunitAdenosine receptor A2a
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe systemic cleara…
Genetik -
Melarsoprol DB12864
small molecule | CAS: 494-79-1

Melarsoprol is under investigation in clinical trial NCT00330148 (Randomized Clinical Trial of Three Drug Combinations for Late-Stage Gambiense Human African Trypanosomiasis).

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Memantine Approved DB01043
small molecule | CAS: 19982-08-2

Initially approved by the FDA in 2013, memantine is an N-methyl-D-aspartate (NMDA) receptor antagonist used in the management of Alzheimer's Disease (AD). It is different from many other Alzheimer's Disease medications, as it works by a different mechanism t…

Kategori:
Anti-Dementia DrugsAnti-Dyskinesia AgentsAnti-Parkinson Drugs +20
Target Protein:
Glutamate (NMDA) receptor5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThis drug is cleare…
Genetik -
Menotropins Approved DB00032
biotech | CAS: 9002-68-0

Menotropins contains follicle stimulating hormone (FSH) and luteinizing hormone (LH) purified from the urine of postmenopausal women. It is used as a fertility medication that is injected either subcutaneously or intramuscularly. It is composed of LH with 2 …

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +14
Target Protein:
Follicle-stimulating hormone receptorLutropin-choriogonadotropic hormone receptor
Waktu Paruh-
Vol. Distribusi-
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Meplazumab DB16465
biotech

Meplazumab is a humanized anti-CD147 antibody being investigated as an add-on therapy in patients with COVID-19 pneumonia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepolizumab Approved DB06612
biotech | CAS: 196078-29-2

Eosinophils are involved in inflammatory immune responses, and prolonged hypereosinophilia (typically defined as absolute eosinophil levels of 1500/mm<sup>3</sup> or more) is associated with a spectrum of diseases, including severe asthma, eosinophilic granul…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interleukin-5
Waktu ParuhMepolizumab has a m…
Vol. DistribusiMepolizumab has a p…
KlirensMepolizumab has an …
Genetik -
Meprobamate Approved DB00371
small molecule | CAS: 57-53-4

A carbamate with hypnotic, sedative, and some muscle relaxant properties, although in therapeutic doses reduction of anxiety rather than a direct effect may be responsible for muscle relaxation. Meprobamate has been reported to have anticonvulsant actions aga…

Kategori:
Acids, AcyclicAnti-Anxiety AgentsCarbamates +10
Target Protein:
Peptide deformylase, mitochondrialProtein kinase C epsilon typeGABA(A) Receptor +6
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Mequinol Approved DB09516
small molecule | CAS: 150-76-5

Mequinol is a phenol used in various applications. It is used as an inhibitor for acrylic monomers and acrylonitirles, as a stabilizer for chlorinated hydrocarbons and ethyl cellulose, as an ultraviolet inhibitor, as a chemical intermediate in the manufacture…

Kategori:
AntioxidantsBenzene DerivativesBiological Factors +11
Waktu ParuhMequinol demonstrat…
Vol. DistribusiThe volume of distr…
KlirensReadily accessible …
Genetik -
Merbromin DB13392
small molecule | CAS: 129-16-8

Mercurochrome is a trade name of merbromin commonly used as a topical first-aid antiseptic agent. It is an organomercuric disodium salt compound and a fluorescein that is available in many countries, except Switzerland, France, Germany, and the United States …

Kategori:
Antiseptics and DisinfectantsDermatologicalsFluoresceins +6
Waktu Paruh-
Vol. Distribusi-
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Merimepodib DB04862
small molecule | CAS: 198821-22-6

Merimepodib (VX-497) is a novel noncompetitive inhibitor of IMPDH. Merimepodib is orally bioavailable and inhibits the proliferation of primary human, mouse, rat, and dog lymphocytes at concentrations of approximately 100 nM.

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesoheme DB02577
small molecule

The color-furnishing portion of hemoglobin. It is found free in tissues and as the prosthetic group in many hemeproteins.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mestranol Approved DB01357
small molecule | CAS: 72-33-3

The 3-methyl ether of ethinyl estradiol. It must be demethylated to be biologically active. It is used as the estrogen component of many combination ORAL contraceptives.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +25
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metandienone DB13586
small molecule | CAS: 72-63-9

Metandienone is an orally active anabolic androgenic steroid. It was introduced to the market in the 1960s but later discontinued and withdrawn from the market. Although it is prohibited in and outside competition by the World Anti-Doping Agency, metandienone…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metelimumab DB18695
biotech | CAS: 272780-74-2

Metelimumab (CAT-192) is a monoclonal antibody targeted against transforming growth factor (TGF) beta-1.

Waktu Paruh-
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Genetik -
Metformin Approved DB00331
small molecule | CAS: 657-24-9

Metformin is a biguanide antihyperglycemic agent and first-line pharmacotherapy used in the management of type II diabetes.[L12207,A176173] Metformin is considered an antihyperglycemic drug because it lowers blood glucose concentrations in type II diabete…

Kategori:
Alimentary Tract and MetabolismAmidinesBiguanides +11
Target Protein:
Multidrug and toxin extrusion protein 1Acetyl-CoA carboxylase 2Electron transfer flavoprotein-ubiquinone oxidoreductase, mitochondrial +2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensRenal clearance is …
Genetik -
Methadone Approved DB00333
small molecule | CAS: 76-99-3

Methadone is a potent synthetic analgesic that works as a full µ-opioid receptor (MOR) agonist and N-methyl-d-aspartate (NMDA) receptor antagonist. As a full MOR agonist, methadone mimics the natural effects of the body's opioids, endorphins, and enkephalins …

Kategori:
AnalgesicsAnticholinergic AgentsAntidepressive Agents +50
Target Protein:
Mu-type opioid receptorNMDA receptorDelta-type opioid receptor +5
Waktu ParuhDue to interindivid…
Vol. DistribusiDue to interindivid…
KlirensDue to interindivid…
Genetik -
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