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6694

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4518 (67.5%)
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3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 27 / 134
Basifungin DB14058
small molecule | CAS: 127785-64-2

Basifungin, also known as _aureuobacidin A_, is a phosphorylceramide synthase inhibitor [L2960], [A33381].

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +3
Target Protein:
Inositol phosphorylceramide synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Basiliximab Approved DB00074
biotech | CAS: 179045-86-4

A recombinant chimeric (murine/human) monoclonal antibody (IgG1k) that functions as an immunosuppressive agent, specifically binding to and blocking the interleukin-2 receptor a-chain (IL-2R alpha, also known as CD25 antigen) on the surface of activated T-lym…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu Paruh7.2 +/- 3.2 days (a…
Vol. Distribusi* 7.8 ± 5.1 L [Pedi…
Klirens* 41 +/- 19 mL/h [A…
Genetik -
Basmisanil DB11877
small molecule | CAS: 1159600-41-5

Basmisanil has been used in trials studying the treatment and basic science of Down Syndrome.

Kategori:
Oxazines
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batabulin DB16103
small molecule | CAS: 195533-53-0

Batabulin is under investigation in clinical trial NCT00057382 (T138067 Versus Doxorubicin in Chemotherapy-naive, Unresectable, Hepatocellular Carcinoma Patients).

Kategori:
AmidesBenzene DerivativesHydrocarbons, Fluorinated +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Batroxobin DB09005
biotech | CAS: 9039-61-6

Batroxobin is a defibrinogenating hemostatic agent derived from the venom of a pit viper, Bothrops atrox moojeni. In addition to batroxobin, the venom of Bothrops atrox has a composition of 10.2% neutral carbohydrate. Batroxobin is a serine protease, which cl…

Kategori:
Biological FactorsBlood and Blood Forming OrgansCardiovascular Agents +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bavisant DB12299
small molecule | CAS: 929622-08-2

Bavisant has been used in trials studying the basic science and treatment of Alcoholism, Pharmacokinetics, Drug Interactions, Attention Deficit Hyperactivity Disorder, and Attention Deficit Disorders With Hyperactivity.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BAX 335 DB17845
biotech

BAX 335 is an adeno-associated virus vector 8 (AAV8)–based FIX gene therapy being investigated for the treatment of hemophilia B.[A259791]

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Baxdrostat DB19090
small molecule | CAS: 1428652-17-8

Baxdrostat is under investigation in clinical trial NCT06344104 (A Phase III Study to Investigate the Efficacy and Safety of Baxdrostat in Asian Participants With Uncontrolled Hypertension on Two or More Medications Including Participants With Resistant Hyper…

Target Protein:
Cytochrome P450 11B2, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bazedoxifene Approved DB06401
small molecule | CAS: 198481-32-2

Bazedoxifene is a third generation selective estrogen receptor modulator (SERM), developed by Pfizer following the completion of their takeover of Wyeth Pharmaceuticals. In late 2013, Pfizer received approval for bazedoxifene as part of the combination drug D…

Kategori:
Bone Density Conservation AgentsEstrogen Agonist/AntagonistEstrogen Receptor Modulators +8
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh~30 hours.
Vol. DistribusiFollowing intraveno…
KlirensThe apparent oral c…
Genetik -
BBIBP-CorV DB15807
biotech

BBIBP-CorV vaccine contains a SARS-CoV-2 strain inactivated inside Vero Cells. Investigation shows this vaccine induces neutralizing antibodies in several mammalian species while also showing protective efficacy with SARS-CoV-2 challenge in rhesus macaques[A2…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBM-H803 DB17700
biotech

BBM-H803 is a recombinant adeno-associated virus (AAV) based gene therapy drug for hemophilia A developed and manufactured by Belief BioMed. It consists of an adeno-associated virus vector containing an expression cassette of the human Factor VIII transgene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBM-H901 DB17704
biotech

BBM-H901 is a liver-tropic adeno-associated viral (AAV) vector carrying cassette coding hyperactive Padua factor IX (FIX) protein. It is being investigated for the treatment of hemophilia B.[A259048]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBV152 DB15847
biotech

BBV152 is a vaccine candidate created by the Indian Council of Medical Research (ICMR). The candidate, a whole virion inactivated SARS-CoV-2 vaccine, was developed from a well-known SARS-CoV-2 strain and a vero cell platform (CCL-81) with adjuncts of either a…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCc1 DB16504
small molecule

BCc1 is a nanomedicine that demonstrated potent anticancer effects in both in vitro and in vivo studies.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCG vaccine Approved DB12768
biotech

BCG vaccine has been investigated for the treatment of Neoplasms, Bladder Cancer, Neoplasms by Site, Urologic Diseases, and Urologic Neoplasms, among others.

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBacterial Vaccines +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCX9250 DB18069
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BDB-001 DB16480
biotech

BDB-001, was under investigation in multiple clinical trials to evaluate its safety, tolerability, and efficacy across various conditions. In NCT05075304 and NCT04449588, BDB-001 was studied in mild to severe COVID-19 patients. It was also explored for solid …

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bebtelovimab DB16755
biotech | CAS: 2578319-11-4

Bebtelovimab (LY-COV1404, LY-3853113) is a human monoclonal antibody approved for emergency use in the treatment of COVID-19. It binds to a portion of the SARS-CoV-2 spike (S) protein's receptor-binding domain, thereby preventing spike protein interaction wit…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesApproved Treatments for COVID-19 +6
Target Protein:
Spike glycoprotein
Waktu ParuhFollowing a single …
Vol. DistribusiAt steady-state, th…
KlirensFollowing a single …
Genetik -
Becatecarin DB06362
small molecule | CAS: 119673-08-4

Becatecarin is a derivative of [rebeccamycin].

Kategori:
CarbohydratesGlycosidesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
DNA topoisomerase 1DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beclomethasone dipropionate Approved DB00394
small molecule | CAS: 5534-09-8

Beclomethasone dipropionate is a second-generation[A179842] synthetic corticosteroid and diester of beclomethasone, which is structurally similar to [dexamethasone].[L6871] It is a prodrug of an active metabolite beclomethasone 17-monopropionate (17-BMP)[A179…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +40
Target Protein:
Glucocorticoid receptor
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Becocalcidiol DB04891
small molecule | CAS: 524067-21-8

Becocalcidiol is a vitamin D(3) analogue which has not caused hypercalcaemia or significant irritation in preclinical trials.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Mediator of RNA polymerase II transcription subunit 1Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Becotatug DB19069
biotech | CAS: 2648260-93-7

Becotatug is under investigation in clinical trial NCT06380348 (JMT101 in Combination With Osimertinib, Versus Cisplatin-pemetrexed in Participants With Locally Advanced or Metastatic Non-small Cell Lung Cancer (NSCLC) Characterized by Epithermal Growth Facto…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bedaquiline Approved DB08903
small molecule | CAS: 843663-66-1

Bedaquiline is a bactericidal antimycobacterial drug belonging to the class of diarylquinoline. The quinolinic central heterocyclic nucleus with alcohol and amine side chains is responsible for bedaquiline-mediated antimycobacterial activity.[A261866] Althoug…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +10
Target Protein:
ATP synthase subunit c
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe volume of distr…
KlirensBedaquiline has a l…
Genetik -
Beeswax Approved DB11600
biotech | CAS: 8012-89-3

The wax obtained from the honeycomb of the bee. It consists primarily of myricyl palmitate, cerotic acid esters and some high-carbon paraffins. Beeswax is used as a stiffening agent in ointments and creams, and enables water to be incorporated to produce wate…

Kategori:
BeesLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Befovacimab DB16188
biotech | CAS: 2156634-62-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Begacestat DB12263
small molecule | CAS: 769169-27-9

Begacestat has been used in trials studying the treatment and basic science of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein SecretasesEnzyme Inhibitors +3
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bekanamycin DB13673
small molecule | CAS: 4696-76-8

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belatacept Approved DB06681
biotech | CAS: 706808-37-9

Belatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1). Structurally, abatacept is a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents, Immunological +15
Target Protein:
T-lymphocyte activation antigen CD86T-lymphocyte activation antigen CD80
Waktu ParuhMean terminal elimi…
Vol. DistribusiVd, steady state, t…
KlirensIncreased body weig…
Genetik -
Belimumab Approved DB08879
biotech | CAS: 356547-88-1

Belimumab is a fully human recombinant IgG1? monoclonal antibody that inhibits soluble human B lymphocyte stimulator protein (BLyS, also referred to as BAFF and TNFSF13B), a B cell survival factor.[L42630] BLyS levels are often elevated in immunodeficient and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Tumor necrosis factor ligand superfamily member 13B
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Belinostat Approved DB05015
small molecule | CAS: 866323-14-0

Belinostat is a novel agent that inhibits the enzyme histone deacetylase (HDAC) with a sulfonamide-hydroxamide structure. It was developed as an orphan drug to target hematological malignancies and solid tumors by TopoTarget. The safety and efficacy of belino…

Kategori:
AmidesAminesAntineoplastic Agents +31
Target Protein:
Histone deacetylase
Gen Terkait:
UGT1A1 UGT1A1
Waktu ParuhDisplays a three-co…
Vol. DistribusiThe volume of distr…
Klirens1240 mL/min
Genetik 2 Varian
Belladonna Approved DB13913
biotech

Belladonna, also known as atropa belladonna or deadly nightshade, is a perennial herbaceous plant in the nightshade family _Solanaceae_. Its roots, leaves and fruits contain [DB00424], [DB00747], and mostly, [DB00572]. These alkaloids are naturally-occurring …

Kategori:
Anticholinergic AgentsAntimuscarinics AntispasmodicsMuscarinic Antagonists
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Belrestotug DB19066
biotech | CAS: 2574438-65-4

Belrestotug is under investigation in clinical trial NCT05565378 (A Platform Study of Novel Immunotherapy Combinations in Participants With Previously Untreated, Advanced/metastatic Non-small-cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Beludavimab DB18952
biotech | CAS: 2423016-74-2

Beludavimab is under investigation in clinical trial NCT04746183 (AGILE (Early Phase Platform Trial for COVID-19)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belumosudil Approved DB16703
small molecule | CAS: 911417-87-3

Belumosudil is used in the treatment of chronic graft-versus-host disease (GVHD) and has been investigated for the treatment of pulmonary arterial hypertension.[A236634] It is an inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK), with …

Kategori:
AcetatesAcids, AcyclicAmides +25
Target Protein:
Rho-associated protein kinase 2Rho-associated protein kinase 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing a single …
KlirensThe mean clearance …
Genetik -
Belzutifan Approved DB15463
small molecule | CAS: 1672668-24-4

Belzutifan is an inhibitor of hypoxia-inducible factor 2? (HIF-2?) used in the treatment of von Hippel-Lindau (VHL) disease-associated cancers.[L35995] The HIF-2? protein was first identified in the 1990s by researchers at UT Southwestern Medical Center as a …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Endothelial PAS domain-containing protein 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Bemiparin Approved DB09258
small molecule | CAS: 91449-79-5

Bemiparin is an antithrombotic and belongs to the group of drugs known as the low molecular weight heparins (LMWH). Like semuloparin, bemiparin is classified as an ultra-LMH because of its low mean molecular mass of 3600 daltons, which is a unique property of…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +6
Target Protein:
Coagulation factor XAntithrombin-IIIHeparin cofactor 2
Waktu ParuhBemiparin, when adm…
Vol. Distribusi5.1 L [A32018].
KlirensElimination occurs …
Genetik -
Bemotrizinol Approved DB11206
small molecule | CAS: 187393-00-6

Bemotrizinol, or bis-ethylhexyloxyphenol methoxyphenyl triazine, is an organic UV filter found in over-the-counter sunscreen products. It primarily absorbs UV-A rays. Compared to older broad-spectrum chemical agents, bemotrizinol is more more fat soluble (oil…

Kategori:
Benzene DerivativesSunscreen Agents
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Bempedoic acid Approved DB11936
small molecule | CAS: 738606-46-7

High levels of LDL cholesterol (LDL-C) are a major risk factor for cardiovascular events. Caused by genetic mutations or lifestyle factors, hypercholesterolemia can significantly reduce quality of life and increase the risk of mortality from cardiovascular di…

Kategori:
Acids, AcyclicAdenosine Triphosphate-Citrate Lyase InhibitorAdenosine Triphosphate-Citrate Lyase Inhibitors +11
Target Protein:
ATP-citrate synthase
Waktu ParuhThe half-life of be…
Vol. DistribusiThe apparent volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1939126-74-5

Bempegaldesleukin is under investigation in clinical trial NCT03729245 (A Study of NKTR-214 in Combination With Nivolumab Compared With the Investigator's Choice of a Tyrosine Kinase Inhibitor (TKI) Therapy (Either Sunitinib or Cabozantinib Monotherapy) for A…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benactyzine DB09023
small molecule | CAS: 302-40-9

Benactyzine is an anticholinergic drug used as an antidepressant in the treatment of depression and associated anxiety. Benactyzine is no longer widely used in medicine, although it is still a useful drug for scientific research. It does not possess any an…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAnticholinergic Agents +14
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benazeprilat DB14125
small molecule | CAS: 86541-78-8

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bencyclane DB13488
small molecule | CAS: 2179-37-5

A vasodilator agent found to be effective in a variety of peripheral circulation disorders. It has various other potentially useful pharmacological effects. Its mechanism may involve block of calcium channels.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bendazac Approved DB13501
small molecule | CAS: 20187-55-7

Bendazac is an oxyacetic acid [A39863, A39869]. Despite possessing anti-inflammatory, anti-necrotic, choleretic, and anti-lipidemic characteristics, most research has revolved around studying and demonstrating the agent's principal action in inhibiting the de…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Target Protein:
Free radicalsProstaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Benfluorex DB09022
small molecule | CAS: 23602-78-0

Benfluorex is an anorectic and hypolipidemic agent that is structurally related to fenfluramine. It was patented and manufactured by a French pharmaceutical company Servier. The European Medicines Agency (EMA) recommended withdrawing all benfluorex containing…

Kategori:
Alimentary Tract and MetabolismAminesAnti-Obesity Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benidipine DB09231
small molecule | CAS: 105979-17-7

Benidipine has the formula 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridine-dicarboxylic acid methyl 1-(phenylmethyl)-3-piperidinyl ester hydrochloride. It is a synthetic dihydropyridine derivative that has anti-hypertensive and anti-anginal actions.[A…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +19
Target Protein:
Voltage-dependent L-type calcium channelVoltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent T-type calcium channel
Waktu ParuhThe elimination hal…
Vol. DistribusiBenidipine is highl…
Klirens-
Genetik -
Benoxaprofen Approved DB04812
small molecule | CAS: 51234-28-7

The use of benoxaprofen, formerly marketed as Oraflex tablets, was associated with fatal cholestatic jaundice among other serious adverse reactions. The holder of the approved application voluntarily withdrew Oraflex tablets from the market on August 5, 1982.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Acetyl-CoA acetyltransferase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benralizumab Approved DB12023
biotech | CAS: 1044511-01-4

Benralizumab is a humanized recombinant monoclonal antibody of the isotype IgG1k immunoglobulin that specifically binds to the alpha chain of the interleukin 5 receptor (IL-5R) expressed on eosinophils and basophils.[A31294] It inhibits the binding of IL-5 as…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +13
Target Protein:
Interleukin-5 receptor subunit alphaLow affinity immunoglobulin gamma Fc region receptor III-A
Waktu ParuhThe half-life of Be…
Vol. DistribusiPharmacokinetic rep…
KlirensFor a subject weigh…
Genetik -
Benserazide Approved DB12783
small molecule | CAS: 322-35-0

When levodopa is used by itself as a therapy for treating Parkinson's disease, its ubiquitous metabolism into dopamine is responsible for a resultant increase in the levels of circulating dopamine in the blood and to various extracerebral tissues. This can re…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsAromatic L-amino Acid Decarboxylase Inhibitors +6
Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu ParuhThe half-life of be…
Vol. DistribusiReadily accessible …
KlirensReadily accessible …
Genetik -
Bentracimab DB16659
biotech | CAS: 2260568-31-6

Bentracimab is under investigation in clinical trial NCT04286438 (Bentracimab (PB2452) in Ticagrelor-treated Patients With Uncontrolled Major or Life-threatening Bleeding or Requiring Urgent Surgery or Invasive Procedure).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Neutralizing +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1301–1350 dari 6694
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