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16004

Total database: 17430
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12010 (75.0%)
Target
9041 (56.5%)
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112 (0.7%)
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16004 (100.0%)

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Halaman 269 / 321
Rozanolixizumab Approved DB14919
biotech | CAS: 1584645-37-3

Rozanolixizumab is a humanized high-affinity anti-human neonatal Fc receptor (FcRn) monoclonal antibody (IgG4P) targeting the immunoglobulin G (IgG). Rozonolixizumab itself is an IgG4P, an inactive isotype, to reduce the likelihood of unwanted chain exchange.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
IgG receptor FcRn large subunit p51
Waktu Paruh-
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Rozibafusp Alfa DB19233
biotech | CAS: 2143449-47-0

Rozibafusp Alfa is under investigation in clinical trial NCT04058028 (Efficacy and Safety of AMG 570 in Subjects With Active Systemic Lupus Erythematosus (SLE)).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
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Rozrolimupab DB05209
biotech | CAS: 909402-77-3

Rozrolimupab is a recombinant polyclonal antibody consisting of 25 different anti-Rhesus D (RhD) antibodies to replace existing anti-RhD hyperimmune immunoglobulins for the treatment of Idiopathic Thrombocytopenic Purpura (ITP) and the prevention of Hemolytic…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Target Protein:
Rhesus blood group D antigen
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RP-67580 DB16742
small molecule | CAS: 135911-02-3

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNeurokinin-1 Receptor AntagonistsNeurotransmitter Agents
Target Protein:
Substance-P receptor
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RP-72 DB17156
biotech

Deskripsi belum tersedia.

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RP-A501 DB17647
biotech

RP-A501 is a gene therapy product consisting of a recombinant adeno-associated virus serotype 9 (rAAV9) capsid containing the human LAMP2B transgene (AAV9:LAMP2B), which encodes lysosome-associated membrane protein 2 (LAMP-2). It is being investigated for Dan…

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RP-A601 DB18339
biotech

RP-A601 is an adeno-associated virus serotype rhesus 10 vector expressing the human galactocerebrosidase (GALC) gene

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RP-L201 DB17595
biotech

Deskripsi belum tersedia.

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RP-L301 DB17661
biotech

RP-L301 is a lentiviral vector containing the human liver and erythroid pyruvate kinase gene.

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RP01 DB05751
small molecule

RP01 is a novel anti-IgE immunotherapy for allergic individuals. It is designed to induce the immune system to produce antibodies that block Immunoglobulin E (IgE), the key mediator of an allergic response. It could offer benefit to millions of asthma and all…

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RPI-78M DB05740
small molecule

RPI-78M is being developed for the treatment of multiple sclerosis (MS). Other neurological disorders that may be served by RPI-78M include myasthenia gravis (MG), muscular dystrophy (MD) and amyotrophic lateral sclerosis (ALS).

Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit beta-2Neuronal acetylcholine receptor subunit alpha-7 +3
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RPI-MN DB17957
biotech

RPI-MN is a detoxified or chemically modified alpha-cobratoxin with antiviral properties.[A260132] Being developed by Nutra Pharma under the trade name PEPTERON, it is being investigated for the treatment of neurological and immune disorders.[L47107]

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rPSGL-Ig DB06256
biotech

Recombinant P-selectin glycoprotein ligand IgG fusion protein (rPSGL-Ig) is a fusion protein of human P-selectin ligand and IgG1-Fc.

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RR001 DB17369
biotech

RR001 is an investigational gene therapy consisting of autologous human adipose perivascular stromal cells genetically modified to secrete soluble tumour necrosis factor-related apoptosis-inducing ligand (AD-PC sTRAIL).[L44276]

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RRx-001 DB12060
small molecule | CAS: 925206-65-1

RRx-001 has been used in trials studying the treatment of Lymphomas, Brain Metastases, Cholangiocarcinoma, Colorectal Neoplasms, and Malignant Solid Tumor, among others.

Kategori:
AzetinesCarbon Radioisotopes
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RS-39604 DB17050
small molecule | CAS: 161362-65-8

RS-39604 is a selective 5-HT4 receptor antagonist.[A253112]

Kategori:
AlkanesHydrocarbons, Acyclic
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rsATP7A cDNA DB17854
biotech

Deskripsi belum tersedia.

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rsPSMA Vaccine Approved DB06361
biotech

Prostate-specific membrane antigen (PSMA) is an ?100 kDa transmembrane glycoprotein that is abundantly and preferentially expressed in prostate cancer, including recurrent and hormone-refractory cases. rsPSMA Vaccine is a subunit vaccine based on a novel rsPS…

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RST-001 DB17843
biotech

RST-001 is a non-replicating recombinant adeno-associated virus vector containing a fragment of the gene encoding channel rhodopsin-2 protein.

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RSV-604 DB15197
small molecule | CAS: 676128-63-5

RSV-604 is under investigation in clinical trial NCT00416442 (Safety, Tolerability and Pharmacokinetic Study of Single and Multiple Intravenous Doses of RSV604 in Healthy Subjects.).

Kategori:
AmidesBenzazepinesBenzene Derivatives +1
Waktu Paruh-
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RTA 744 DB05920
small molecule

RTA 744 is a novel anthracycline derivative that crosses the blood-brain barrier and shows significant potential for the treatment of primary and metastatic brain cancers. Anthracyclines are one of the most broadly used and effective classes of cancer therapi…

Target Protein:
DNA topoisomerase 2-alpha
Waktu Paruh-
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RTL-1000 DB17946
biotech | CAS: 1391875-03-8

RTL-1000 is a recombinant T-Cell receptor ligand being investigated for the treatment of multiple sclerosis.

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RTP-801i DB06048
biotech

RTP-801i is an siRNA drug candidate designed to inhibit the expression of the hypoxia-inducible gene RTP801. The proposed primary indication for RTP-801i is the treatment of patients with neovascular (wet) Age-related Macular Degeneration (AMD or ARMD).

Kategori:
Antisense Elements (Genetics)Nucleic AcidsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
DNA damage-inducible transcript 4 protein
Waktu Paruh-
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RU82197 DB03268
small molecule

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
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RU84687 DB01678
small molecule

RU84687 is a subnanomolar and Src SH2 selective binder.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
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RU85053 DB03712
small molecule

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
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Rubella virus vaccine Approved DB10317
biotech

Rubella virus vaccine is a live attenuated virus vaccine for active immunization against rubella (German measles) that is subcutaneously administered. It is prepared from RA 27/3 strain of live attenuated rubella virus. Rubella is a common childhood disease, …

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseLive Attenuated Rubella Virus Vaccine +5
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Rubidium Approved DB11346
small molecule | CAS: 7440-17-7

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Alkali +1
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Rubidium Rb-82 Approved DB09479
small molecule

Rubidium chloride Rb-82 injection is a sterile nonpyrogenic solutions of rubidium Rb 82 chloride. It is indicated for Positron Emission Tomography (PET) imaging of the myocardium under rest or pharmacologic stress conditions to evaluate regional myocardial p…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh1.27 minutes
Vol. Distribusi-
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Rubitecan DB06159
small molecule | CAS: 91421-42-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
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Ruboxistaurin DB11829
small molecule | CAS: 169939-94-0

Ruboxistaurin has been investigated for the basic science of Type 2 Diabetes Mellitus and Type 1 Diabetes Mellitus.

Kategori:
Acids, AcyclicDicarboxylic AcidsEnzyme Inhibitors +4
Target Protein:
Peptide deformylase, mitochondrialProtein kinase C beta type
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Rucaparib Approved DB12332
small molecule | CAS: 283173-50-2

Rucaparib is an anticancer drug and poly (ADP-ribose) polymerase (PARP) inhibitor. PARP is an enzyme that plays an essential role in DNA repair.[A18745] Rucaparib is proposed to work in several PARP-dependent and PARP-independent mechanisms of action; however…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +47
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2Protein mono-ADP-ribosyltransferase PARP3
Waktu ParuhThe mean (coefficie…
Vol. DistribusiThe mean (coefficie…
KlirensThe mean (coefficie…
Genetik -
Rufinamide Approved DB06201
small molecule | CAS: 106308-44-5

Rufinamide is a triazole derivative and an anticonvulsant medication to treat seizure disorders like Lennox-Gastuat syndrome, a form of childhood epilepsy. Clinical trials suggest its efficacy in the treatment of partial seizures.

Kategori:
AnticonvulsantsCarboxamide DerivativesCardiovascular Agents +14
Target Protein:
Sodium channel protein type 9 subunit alphaMetabotropic glutamate receptor 5
Waktu ParuhElimination half-li…
Vol. DistribusiRufinamide was even…
Klirens-
Genetik -
Rufloxacin DB13772
small molecule | CAS: 101363-10-4

Rufloxacin is a quinolone antibiotic. [A31894]

Kategori:
4-QuinolonesAnti-Bacterial AgentsAntibacterials for Systemic Use +13
Waktu Paruh-
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Rugonersen DB18662
biotech | CAS: 2591587-57-2

Rugonersen is a locked nucleic acid antisense oligonucleotide under investigation for the treatment of Angelman Syndrome.

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Rulonilimab DB18922
biotech | CAS: 2417124-95-7

Rulonilimab is under investigation in clinical trial NCT05408221 (The Efficacy and Safety of Rulonilimab in Combination With Lenvatinib in Hepatocellular Carcinoma).

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Rumex crispus whole Approved DB14267
biotech

Rumex crispus whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Runcaciguat DB16700
small molecule | CAS: 1402936-61-1

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCycloparaffins
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1
Waktu Paruh-
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Rupatadine Approved DB11614
small molecule | CAS: 158876-82-5

Rupatadine is a dual histamine H1 receptor and platelet activating factor receptor antagonist that is used for symptomatic relief in seasonal and perennial rhinitis as well as chronic spontaneous urticaria. It was approved for marketing in Canada under the tr…

Kategori:
Antihistamines for Systemic UseBenzocycloheptenesCytochrome P-450 CYP2C19 Substrates +13
Target Protein:
Platelet-activating factor receptorHistamine H1 receptor
Waktu ParuhThe half life of el…
Vol. DistribusiThe apparent volume…
KlirensSystemic clearance …
Genetik -
Rupintrivir DB05102
small molecule | CAS: 223537-30-2

Rupintrivir is a rhinovirus 3C protease inhibitor in development for use against human rhinoviral (HRV) infections. Rupintrivir was active against all 48 HRV serotypes tested in a cell protection assay in H1-HeLa cells. It is designed to combat colds caused b…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Branched-Chain +8
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ruplizumab DB06475
biotech | CAS: 220651-94-5

Ruplizumab is a humanized monoclonal antibody used as an immunosuppressive drug and is a component of Antova.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Target Protein:
CD40 ligand
Waktu Paruh-
Vol. Distribusi-
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Rurioctocog alfa pegol Approved DB16007
biotech | CAS: 1417412-83-9

Rurioctocog alfa pegol is a pegylated recombinant human coagulation factor VIII or antihemophilic factor. Factor VIII is an essential protein involved in normal blood clotting; thus, a deficient level of functional factor VIII is associated with an elevated r…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
Target Protein:
von Willebrand factorCoagulation factor VIII
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
biotech | CAS: 875455-82-6

Chrysalin has been used in trials studying the treatment of Radius Fracture.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +11
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Ruscogenin DB15830
small molecule | CAS: 472-11-7

Deskripsi belum tersedia.

Kategori:
CholestanesFused-Ring CompoundsSapogenins +1
Waktu Paruh-
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Rusfertide DB17724
biotech | CAS: 1628323-80-7

Rusfertide is a hepcidin mimetic currently being developed by Protagonist Therapeutics for the treatment of polycythemia vera and beta-thalassemia.

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Rutin Approved DB01698
small molecule | CAS: 153-18-4

A flavonol glycoside found in many plants, including buckwheat; tobacco; forsythia; hydrangea; viola, etc. It has been used therapeutically to decrease capillary fragility.

Kategori:
BenzopyransCapillary Stabilizing AgentsChromones +12
Target Protein:
Aldo-keto reductase family 1 member C3Carbonyl reductase [NADPH] 1
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RUTI® Vaccine DB15853
biotech

The RUTI® Vaccine contains fragmented, purified and liposomed heat-inactivated Mycobacterium tuberculosis bacilli. The vaccine has demonstrated a reasonable safety profile and potent stimulation of the immune response against tuberculosis. Much like the BCG v…

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Ruxolitinib Approved DB08877
small molecule | CAS: 941678-49-5

Ruxolitinib, formerly known as INCB018424 or INC424, is an anticancer drug and a Janus kinase (JAK) inhibitor. It is a potent and selective inhibitor of JAK1 and JAK2,[A229698] which are tyrosine kinases involved in cytokine signalling and hematopoiesis.[A745…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Urokinase plasminogen activator surface receptorTyrosine-protein kinase JAK2Tyrosine-protein kinase JAK1 +2
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensRuxolitinib clearan…
Genetik -
Ruzasvir DB11713
small molecule | CAS: 1613081-64-3

Ruzasvir has been used in trials studying the treatment of Hepatitis C, Hepatitis C, Chronic, and Hepatitis C Infection.

Kategori:
Anti-Infective AgentsAntiviral AgentsHeterocyclic Compounds, Fused-Ring +1
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Ruzinurad DB19209
small molecule | CAS: 1638327-48-6

Ruzinurad is under investigation in clinical trial NCT04956432 (A Multicentre, Randomized, Double-blind, Allopurinol Controlled Study to Evaluate the Efficacy and Safety of SHR4640 in Subjects With Gout).

Kategori:
CycloparaffinsHeterocyclic Compounds, Fused-Ring
Target Protein:
Solute carrier family 22 member 12
Waktu Paruh-
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