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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 268 / 349
biotech

PIKA rabies vaccine is a novel vaccine developed by YS Biopharma.

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Pilaralisib DB11772
small molecule | CAS: 934526-89-3

Pilaralisib is an orally available small molecule that selectively inhibits the activity of phosphoinositide-3 kinase (PI3K). Pilaralisib has been used in trials studying the treatment of Cancer, Lymphoma, Solid Tumors, Glioblastoma, and Breast Cancer, among …

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
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Pilocarpine Approved DB01085
small molecule | CAS: 92-13-7

A naturally occurring alkaloid derived from the _Pilocarpus_ plants, pilocarpine is a muscarinic acetylcholine agonist.[A262016, A262036] Pilocarpine is associated with parasympathomimetic effects by selectively working on muscarinic receptors.[A262036] Piloc…

Kategori:
AlkaloidsAntiglaucoma Preparations and MioticsAutonomic Agents +20
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThere is no informa…
KlirensThere is no informa…
Genetik -
Pilsicainide DB12712
small molecule | CAS: 88069-67-4

Pilsicainide has been investigated for the treatment of Paroxysmal Atrial Fibrillation.

Kategori:
AcetanilidesAmidesAmines +9
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Pimagedine DB05383
small molecule | CAS: 79-17-4

Pimagedine has been developed by Synvista Therapeutics, Inc for the treatment of diabetic kidney disease. It is an advanced glycation end product inhibitor which manages diabetic nephropathy, either alone or in combination with other therapies. It is benefici…

Kategori:
AmidinesEnzyme InhibitorsNitric Oxide Synthase, antagonists & inhibitors +1
Target Protein:
Nitric oxide synthase, inducibleC-C chemokine receptor type 2Diamine oxidase [copper-containing] +2
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Pimasertib DB14904
small molecule | CAS: 1236699-92-5

Pimasertib is under investigation in clinical trial NCT01378377 (Combination Trial of Pimasertib (MSC1936369B) With Temsirolimus).

Kategori:
Nicotinic AcidsProtein Kinase InhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase kinase (MAPKK)
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Pimavanserin Approved DB05316
small molecule | CAS: 706779-91-1

Pimavanserin is an atypical antipsychotic indicated for the treatment of psychiatric disorders.[L48236] Although the exact mechanism of action is unknown, it is thought that pimavanserin interacts with the serotonin receptors, particularly the 5-HT<sub>2A</su…

Kategori:
AmidesAntidepressive AgentsCentral Nervous System Agents +14
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CSigma non-opioid intracellular receptor 1
Waktu ParuhThe average plasma …
Vol. DistribusiFollowing administr…
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Pimecrolimus Approved DB00337
small molecule | CAS: 137071-32-0

Pimecrolimus is an immunomodulating agent that was first marketed by Novartis under the trade name Elidel. It is now promoted in Canada by Galderma since early 2007. It is currently available as a topic cream used in the treatment of atopic dermatitis (eczema…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAnalgesicsAnalgesics, Non-Narcotic +15
Target Protein:
Protein phosphatase 3 catalytic subunit alphaSerine/threonine-protein kinase mTORPeptidyl-prolyl cis-trans isomerase FKBP1A
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Pimelic Acid DB01856
small molecule | CAS: 111-16-0

A group of compounds that are derivatives of heptanedioic acid with the general formula R-C7H11O4. [PubChem]

Kategori:
Acids, AcyclicDicarboxylic Acids
Target Protein:
2,3,4,5-tetrahydropyridine-2,6-dicarboxylate N-succinyltransferase
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Pimethixene Approved DB13292
small molecule | CAS: 314-03-4

Pimethixene is approved for use in Brazil and is marketed under the trade name Muricalm. It is an anticholinergic used in the treatment of bronchitis.

Kategori:
Antihistamines for Systemic UseHeterocyclic Compounds, Fused-RingSulfur Compounds +1
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Pimicotinib DB18972
small molecule

Pimicotinib is under investigation in clinical trial NCT05804045 (Study of Pimicotinib (ABSK021) for Tenosynovial Giant Cell Tumor (MANEUVER)).

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Pimivalimab DB16667
biotech | CAS: 2293951-22-9

Pimivalimab is under investigation in clinical trial NCT04549025 (Study of PD-1 Inhibitor JTX-4014 Alone and in Combination With Vopratelimab in Biomarker-selected Subjects With Metastatic NSCLC After One Prior Platinum-containing Regimen).

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Pimobendan DB11450
small molecule | CAS: 74150-27-9

Deskripsi belum tersedia.

Kategori:
Cardiotonic AgentsCardiovascular AgentsCompounds used in a research, industrial, or household setting +6
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Pimodivir DB14974
small molecule | CAS: 1629869-44-8

Pimodivir is under investigation in clinical trial NCT02658825 (A Study to Evaluate the Effect of JNJ-63623872 on Cardiac Repolarization Interval in Healthy Participants).

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Pimonidazole DB12485
small molecule | CAS: 70132-50-2

Pimonidazole is under investigation for the diagnostic of Prostate Cancer and Head and Neck Cancer.

Kategori:
ImidazolesNitro CompoundsRadiation-Sensitizing Agents
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Pimozide Approved DB01100
small molecule | CAS: 2062-78-4

A diphenylbutylpiperidine that is effective as an antipsychotic agent and as an alternative to haloperidol for the suppression of vocal and motor tics in patients with Tourette syndrome. Although the precise mechanism of action is unknown, blockade of postsyn…

Kategori:
Agents that reduce seizure thresholdAnti-Dyskinesia AgentsAntipsychotic Agents +38
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorVoltage-gated inwardly rectifying potassium channel KCNH2 +1
Waktu Paruh29 &plusmn; 10 hour…
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Pinacidil Approved DB06762
small molecule | CAS: 60560-33-0

Pinacidil is a cyanoguanidine drug that acts by opening ATP-sensitive potassium channels, leading to peripheral vasodilatation of arterioles and decreasing peripheral vascular resistance. The above processes result in reduced blood pressure. This drug has bee…

Kategori:
AmidinesAntihypertensive AgentsArteriolar Smooth Muscle, Agents Acting On +9
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biotech | CAS: 1313706-14-7

Pinatuzumab vedotin is under investigation in clinical trial NCT01691898 (A Study of Pinatuzumab Vedotin (DCDT2980S) Combined With Rituximab or Polatuzumab Vedotin (DCDS4501A) Combined With Rituximab or Obinutuzumab in Participants With Relapsed or Refractory…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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Pinaverium Approved DB09090
small molecule | CAS: 59995-65-2

Pinaverium is a spasmolytic agent used for functional gastrointestinal disorders. It is a quaternary ammonium compound that acts as an atypical calcium antagonist to restore normal bowel function. It is shown to relieve GI spasm and pain, transit disturbances…

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismAntiarrhythmic agents +17
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1S
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIt is selectively d…
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Pinazepam DB13335
small molecule | CAS: 52463-83-9

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +7
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
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Pindolol Approved DB00960
small molecule | CAS: 13523-86-9

Pindolol is a first generation non-selective beta blocker used in the treatment of hypertension.[L32353] Early research into the use of pindolol found it had chronotropic effects, and so further investigation focused on the treatment of arrhythmia.[A231059] R…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu ParuhThe half life of pi…
Vol. DistribusiThe volume of distr…
KlirensIn otherwise health…
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biotech | CAS: 8000-26-8

Pine needle oil is obtained from the needles of *Pinus mugo* tree via steam distillation. Major components of pine needle oil (pinus mugo) include ?-Pinene, ?-pinene, ?-3-carene, limonene, ?-phellandrene, (E)-caryophyllene, and germacrene D. It is present in …

Kategori:
Herbs and Natural Products
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Pine tar Approved DB15840
biotech | CAS: 8011-48-1

Deskripsi belum tersedia.

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Pineapple Approved DB10558
biotech

Pineapple allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Pinometostat DB12920
small molecule | CAS: 1380288-87-8

Pinometostat has been used in trials studying the treatment of Leukemia, Acute Leukemias, Acute Myeloid Leukemia, Myelodysplastic Syndrome, and Acute Lymphocytic Leukemia, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Histone-lysine N-methyltransferase, H3 lysine-79 specific
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Pinus banksiana pollen Approved DB10922
biotech

Pinus banksiana pollen is the pollen of the Pinus banksiana plant. Pinus banksiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus contorta pollen Approved DB10894
biotech

Pinus contorta pollen is the pollen of the Pinus contorta plant. Pinus contorta pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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biotech

Deskripsi belum tersedia.

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Pinus echinata pollen Approved DB10487
biotech

Pinus echinata pollen is the pollen of the Pinus echinata plant. Pinus echinata pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus elliottii pollen Approved DB10747
biotech

Pinus elliottii pollen is the pollen of the Pinus elliottii plant. Pinus elliottii pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus monticola pollen Approved DB10749
biotech

Pinus monticola pollen is the pollen of the Pinus monticola plant. Pinus monticola pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus nigra pollen Approved DB10924
biotech

Pinus nigra pollen is the pollen of the Pinus nigra plant. Pinus nigra pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus palustris pollen Approved DB10745
biotech

Pinus palustris pollen is the pollen of the Pinus palustris plant. Pinus palustris pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus ponderosa pollen Approved DB10746
biotech

Pinus ponderosa pollen is the pollen of the Pinus ponderosa plant. Pinus ponderosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus resinosa pollen Approved DB10923
biotech

Pinus resinosa pollen is the pollen of the Pinus resinosa plant. Pinus resinosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus rigida pollen Approved DB10896
biotech

Pinus rigida pollen is the pollen of the Pinus rigida plant. Pinus rigida pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus strobus pollen Approved DB10486
biotech

Pinus strobus pollen is the pollen of the Pinus strobus plant. Pinus strobus pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus sylvestris pollen Approved DB10895
biotech

Pinus sylvestris pollen is the pollen of the Pinus sylvestris plant. Pinus sylvestris pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus taeda pollen Approved DB10744
biotech

Pinus taeda pollen is the pollen of the Pinus taeda plant. Pinus taeda pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus thunbergii pollen Approved DB10925
biotech

Pinus thunbergii pollen is the pollen of the Pinus thunbergii plant. Pinus thunbergii pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pinus virginiana pollen Approved DB10748
biotech

Pinus virginiana pollen is the pollen of the Pinus virginiana plant. Pinus virginiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Pioglitazone Approved DB01132
small molecule | CAS: 111025-46-8

Pioglitazone is an antihyperglycemic used as an adjunct to diet, exercise, and other antidiabetic medications to manage type 2 diabetes mellitus.[L11416,L11419,L11422,L11425] It is administered as a racemic mixture, though there is no pharmacologic difference…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP2C8 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor gammaAmine oxidase [flavin-containing] B
Waktu ParuhThe mean serum half…
Vol. DistribusiThe average apparen…
KlirensThe apparent cleara…
Genetik -
Pipamperone DB09286
small molecule | CAS: 1893-33-0

Pipamperone is a typical antipsychotic of the _butyrophenone_ family used in the treatment of schizophrenia. It was developed by Janssen Pharmaceutica in 1961 and started its first round of clinical trials in 1963 [L1514, L1518]. In an effort to improve [h…

Kategori:
Antidepressive AgentsAntipsychotic AgentsButyrophenone Derivatives +15
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AAlpha-1 adrenergic receptors +5
Waktu Paruh17-26h [L1522]
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Pipazethate DB08796
small molecule | CAS: 2167-85-3

A non-narcotic oral antitussive agent.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +4
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Pipecuronium Approved DB01338
small molecule | CAS: 68399-58-6

Pipecuronium is a piperazinyl androstane derivative which is a non-depolarizing neuromuscular blocking agent.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCentral Nervous System Depressants +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhPipecuronium has an…
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Pipemidic acid DB13823
small molecule | CAS: 51940-44-4

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Urinary +11
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Pipendoxifene DB05414
small molecule | CAS: 198480-55-6

ER modulator, ERA-923(Pipendoxifene) is a estrogen receptor modulator being evaluated for the treatment of breast cancer. Pipendoxifene is a new 2-phenyl indole selective estrogen receptor modulators (SERM )that exhibits an excellent preclinical pharmacologic…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Estrogen receptorEstrogen receptor betaIntegrase, catalytic core
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Pipenzolate DB13844
small molecule | CAS: 13473-38-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
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Pipequaline DB13991
small molecule | CAS: 77472-98-1

Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It presents a unique chemical structure that does not follow the structural properties of other drugs of its class. Pipequaline has a simil…

Kategori:
Central Nervous System AgentsHeterocyclic Compounds, Fused-Ring
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Piperacetazine Approved DB06808
small molecule | CAS: 3819-00-9

Piperacetazine was an antipsychotic.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
D(2) dopamine receptor
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