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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 268 / 272
Yellow fever vaccine Approved DB10805
biotech

Yellow fever vaccine prevents against Yellow Fever, a viral hemorrhagic disease caused by the transmission of a _flavivirus_ through the bite of an infected mosquito. Symptoms of Yellow fever can range from asymptomatic, to mild flu-like illness, to more seve…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Yersinia pestis 195/p antigen (formaldehyde inactivated) is under investigation in clinical trial NCT02596308 (Immunogenicity and Safety of Subunit Plague Vaccine).

Kategori:
Actively Acquired ImmunityBacterial VaccinesBiological Products +3
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Yimitasvir DB18768
small molecule | CAS: 1959593-23-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Yinfenidone DB18330
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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YK-4-279 DB17428
small molecule | CAS: 1037184-44-3

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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YKP-1358 DB06109
small molecule

YKP1358 is a novel serotonin (5-HT2A) and dopamine (D2) antagonist that has demonstrated potent activity in animals that relates to both positive and negative symptoms of schizophrenia. In addition, the YKP1358 pharmacological profile suggests a very low pote…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsDopamine Agents +7
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Yohimbine Approved DB01392
small molecule | CAS: 146-48-5

A plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of impotence. It is also alleged to be an aphrodisiac.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +35
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor +9
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
YT-001 DB18564
small molecule | CAS: 1072301-78-0

Deskripsi belum tersedia.

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Yttrium Y-90 Approved DB13076
small molecule | CAS: 10098-91-6

Yttrium 90 has been investigated for the treatment of Colon Cancer and Colorectal Cancer.

Kategori:
Acids, AcyclicAnti-Inflammatory AgentsElements +11
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 943976-23-6

Yttrium Y-90 clivatuzumab tetraxetan is under investigation in clinical trial NCT00603863 (Safety and Efficacy Study of Different Doses of 90Y-hPAM4 Combined With Gemcitabine in Pancreatic Cancer).

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biotech | CAS: 501423-25-2

Deskripsi belum tersedia.

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biotech | CAS: 501423-27-4

Deskripsi belum tersedia.

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Z-160 DB12743
small molecule | CAS: 41332-24-5

Z160 has been used in trials studying the treatment of Postherpetic Neuralgia and Lumbosacral Radiculopathy.

Kategori:
Antiarrhythmic agentsBenzene DerivativesCalcium Channel Blockers +3
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
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Z-Ala Prolinal DB04033
small molecule

Deskripsi belum tersedia.

Target Protein:
Prolyl endopeptidase Pep
Waktu Paruh-
Vol. Distribusi-
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Z-Pro-Prolinal DB03535
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Prolyl endopeptidaseProlyl endopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 161401-82-7

Non-methylated, competitive, and irreversible inhibitor of caspase 1, as well as other caspases,1 which can be used directly with purified enzymes. It does not require an esterase to hydrolyze the O-methyl ester like the cell-permeable form, Z-Val-Ala-Asp(O-M…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCaspase Inhibitors +7
Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zabedosertib DB18767
small molecule | CAS: 1931994-81-8

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Interleukin-1 receptor-associated kinase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zafiride DB18371
biotech

Zafiride is a human tumor necrosis factor coupled to the C terminus of CNGRCG peptide.

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Zafirlukast Approved DB00549
small molecule | CAS: 107753-78-6

Zafirlukast is an oral leukotriene receptor antagonist (LTRA) for the maintenance treatment of asthma, often used in conjunction with an inhaled steroid and/or long-acting bronchodilator. It is available as a tablet and is usually dosed twice daily. Another l…

Kategori:
Acids, AcyclicAgents to Treat Airway DiseaseAmides +37
Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh10 hours
Vol. Distribusi* 70 L
Klirens* apparent oral CL=…
Genetik -
Zagociguat DB18315
small molecule | CAS: 2201048-82-8

Deskripsi belum tersedia.

Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zagotenemab DB16674
biotech | CAS: 2019133-28-7

Zagotenemab is under investigation in clinical trial NCT03518073 (A Study of LY3303560 in Participants With Early Symptomatic Alzheimer's Disease).

Waktu Paruh-
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Zalcitabine Approved DB00943
small molecule | CAS: 7481-89-2

A dideoxynucleoside compound in which the 3'-hydroxyl group on the sugar moiety has been replaced by a hydrogen. This modification prevents the formation of 5' to 3' phosphodiester linkages, which are needed for the elongation of DNA chains, thus resulting in…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh2 hours
Vol. Distribusi* 0.304 to 0.734 L/…
Klirens* 285 mL/min [HIV-i…
Genetik -
Zaleplon Approved DB00962
small molecule | CAS: 151319-34-5

Zaleplon is a sedative/hypnotic, mainly used for insomnia. It is known as a nonbenzodiazepine hypnotic. Zaleplon interacts with the GABA receptor complex and shares some of the pharmacological properties of the benzodiazepines. Zaleplon is a schedule IV drug …

Kategori:
AcetatesAcids, AcyclicAmides +22
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhApproximately 1 hour
Vol. Distribusi* 1.4 L/kg
Klirens* 1 L/h/kg
Genetik -
Zalifrelimab DB15632
biotech | CAS: 2148321-69-9

Zalifrelimab is under investigation in clinical trial NCT03894215 (Phase 2 Study of Anti-pd-1 Independently or in Combination With Anti-ctla-4 in Second-line Cervical Cancer).

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Zaltoprofen DB06737
small molecule | CAS: 74711-43-6

A non-steroidal anti-inflammatory drug approved for use in Japan in 1993.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +19
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Zalunfiban DB18766
small molecule | CAS: 1448313-27-6

Deskripsi belum tersedia.

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Zalutumumab DB12202
biotech | CAS: 667901-13-5

Zalutumumab is a fully human IgG1 monoclonal antibody designed to bind with selectivity to the epidermal growth factor receptor (EGFR). Zalutumumab has been investigated for the treatment of Squamous Cell Cancer and Head and Neck Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zalypsis DB12454
small molecule | CAS: 308359-57-1

Zalypsis has been used in trials studying the treatment of Lymphoma, Solid Tumors, Ewing's Sarcoma, Endometrial Cancer, and Uterine Cervical Cancer, among others.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIsoquinolines
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Zamerovimab DB17766
biotech | CAS: 2419087-87-7

Deskripsi belum tersedia.

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Zamicastat DB12389
small molecule | CAS: 1080028-80-3

Zamicastat has been used in trials studying the treatment of Hypertension and Chronic Heart Failure.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
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Zampilimab DB16381
biotech | CAS: 2098280-42-1

Zampilimab is under investigation in clinical trial NCT04335578 (A Study to Evaluate Safety, Tolerability, Pharmacokinetics, and Efficacy of UCB7858 in Adult Kidney Transplant Recipients With Chronic Allograft Injury).

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Zanamivir Approved DB00558
small molecule | CAS: 139110-80-8

A guanido-neuraminic acid that is used to inhibit neuraminidase.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +15
Target Protein:
NeuraminidaseNeuraminidaseSialidase-2
Waktu Paruh2.5-5.1 hours
Vol. Distribusi-
Klirens* 2.5 - 10.9 L/h [F…
Genetik -
Zandatrigine DB19051
small molecule | CAS: 2154406-04-7

Zandatrigine is under investigation in clinical trial NCT05226780 (Extension Study to Evaluate How Safe and Tolerable NBI-921352 Is as an Adjunctive Therapy for Participants With SCN8A-DEE).

Waktu Paruh-
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Zandelisib DB18245
small molecule | CAS: 1401436-95-0

Deskripsi belum tersedia.

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Zanidatamab Approved DB15471
biotech | CAS: 2169946-15-8

Zanidatamab is a bispecific antibody that binds two non-overlapping sites of HER2 (ERBB2).[A264718] It has been investigated for the treatment of HER2-positive solid tumors, including gastroesophageal, colorectal, and biliary tract cancers.[A264718] In No…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhBased on population…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
biotech | CAS: 2329698-82-8

According to Zymeworks, "ZW49 (zanidatamab zovodotin) is a bispecific anti-HER2 ADC that is based on the same antibody framework as [ZW25] but armed with a cytotoxic payload."[L8234] It is being investigated for several indications characterized by HER2 expre…

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Zanolimumab DB17376
biotech | CAS: 652153-01-0

Zanolimumab is a fully human monoclonal antibody directed against CD4.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zansecimab DB16389
biotech | CAS: 2415205-37-5

Zansecimab is under investigation in clinical trial NCT04342897 (A Study of LY3127804 in Participants With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Zanthoxylum clava-herculis bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Genetik -
biotech

Zanthoxylum clava-herculis whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Zanubrutinib Approved DB15035
small molecule | CAS: 1691249-45-2

Zanubrutinib is a novel Bruton's tyrosine kinase (BTK) inhibitor used for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy.[L10163] Mantle cell lymphoma is an aggressive mature B-cell non-Hodgkin lym…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +19
Target Protein:
Tyrosine-protein kinase BTKEpidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2 +12
Waktu ParuhFollowing administr…
Vol. DistribusiThe geometric mean …
KlirensThe mean (%CV) appa…
Genetik -
Zanzalintinib DB17525
small molecule | CAS: 2367004-54-2

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zapnometinib DB18244
small molecule | CAS: 303175-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminesAminobenzoates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zardaverine DB02918
small molecule | CAS: 101975-10-4

Deskripsi belum tersedia.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +4
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
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Zasocitinib DB19278
small molecule | CAS: 2272904-53-5

Deskripsi belum tersedia.

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Zastumotide DB14926
biotech | CAS: 949885-73-8

Zastumotide is a recombinant MAGE-A3 Antigen-Specific Cancer Immunotherapeutic (MAGE-A3 ASCI) also known as astuprotimut-R. It is under investigation in clinical trial NCT00257738 (0804 GCC: MAGE-A3/HPV 16 Vaccine for Squamous Cell Carcinoma of the Head and N…

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Zatolmilast DB14790
small molecule | CAS: 1606974-33-7

BPN-14770 is under investigation in clinical trial NCT02840279 (A Multiple Ascending Dose Study of BPN14770 in Healthy Young and Elderly Male or Female Subjects).

Kategori:
Acids, AcyclicEnzyme InhibitorsFatty Acids +5
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
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Zavegepant Approved DB15688
small molecule | CAS: 1337918-83-8

Zavegepant (BHV-3500) is a calcitonin gene-related peptide (CGRP) receptor antagonist.[L45505] CGRP is released from sensory nerves and acts as a strong vasodilator, and thanks to these properties, it is involved in pain pathways. CGRP receptors are expressed…

Kategori:
Antimigraine PreparationsCalcitonin Gene-Related Peptide (CGRP) AntagonistsCalcitonin Gene-Related Peptide Receptor Antagonists +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhFollowing a 10 mg d…
Vol. DistribusiIntranasal zavegepa…
KlirensIntranasal zavegepa…
Genetik -
ZB131 DB17164
biotech

ZB131 is a monoclonal antibody with a high affinity and specificity for cancer-specific plectin (CSP), a cell surface protein identified in a wide range of cancers that correlates with poor prognosis and aggressive tumors.[L44081]

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