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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 266 / 272
Voxtalisib DB12400
small molecule | CAS: 934493-76-2

Voxtalisib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Breast Cancer, among others.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase mTOR
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VP-14637 DB12195
small molecule | CAS: 235106-62-4

MDT-637 has been investigated for the treatment of Drug Safety.

Kategori:
Benzene DerivativesHydrazines
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VP025 DB05133
small molecule

VP025, a novel drug formulation based on phospholipid microparticles incorporating phosphatidylglycerol, can inhibit neuroinflammation. VP025 may inhibit immune system activation and protect motoneurons from injury. It also shows the ability to reduce inflamm…

Target Protein:
Interleukin-1 beta
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VPO-227 DB18004
small molecule | CAS: 1314873-02-3

Deskripsi belum tersedia.

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VS-4718 DB15273
small molecule | CAS: 1061353-68-1

VS-4718 is under investigation in clinical trial NCT02215629 (Dose Escalation Study in Acute Myeloid or B-Cell Acute Lymphoblastic Leukemia).

Kategori:
AminesFocal Adhesion Protein-Tyrosine Kinases, antagonists & inhibitorsPyridines
Target Protein:
Focal adhesion kinase 1
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VS-5584 DB12986
small molecule | CAS: 1246560-33-7

VS-5584 has been used in trials studying the treatment of Lymphoma, Metastatic Cancer, and Non Hematologic Cancers.

Kategori:
Heterocyclic Compounds, Fused-RingOxazines
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
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VSF-173 DB05753
small molecule

VSF-173 is an oral small molecule. It is an oral compound that has demonstrated effects on animal sleep/wake patterns and gene expression patterns suggestive of a stimulant effect. It is developed for the treatment of excessive sleepiness. Study shows that VS…

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VT-1598 DB17757
small molecule | CAS: 2089320-99-8

Deskripsi belum tersedia.

Target Protein:
Lanosterol 14-alpha demethylase
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VTP-194204 DB11806
small molecule | CAS: 220619-73-8

Nrx194204 has been used in trials studying the treatment of Parkinson's Disease and Non-small Cell Lung Cancer.

Kategori:
Fatty AcidsLigandsLipids +1
Target Protein:
Retinoic acid receptor RXR-gamma
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VTX-803 DB18271
biotech

Deskripsi belum tersedia.

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Vudalimab DB18833
biotech | CAS: 2329669-72-7

Vudalimab is under investigation in clinical trial NCT05005728 (Xmab®20717 (Vudalimab) Alone or in Combination With Chemotherapy or Targeted Therapy in Patients With Metastatic Castration-resistant Prostate Cancer).

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Vunakizumab DB15154
biotech | CAS: 1792181-33-9

Vunakizumab is under investigation in clinical trial NCT03463187 (Multi-Dose Study of SHR-1314 in Subjects With Moderate-to-severe Plaque Psoriasis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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Vurolenatide DB18440
biotech | CAS: 2434640-83-0

Vurolenatide is a recombinant fusion protein comprising exenatide and XTEN.

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Vutrisiran Approved DB16699
biotech | CAS: 1867157-35-4

Vutrisiran is a double-stranded small interfering ribonucleic acid (siRNA) that targets wild-type and mutant transthyretin (TTR) messenger RNA (mRNA).[L42065] This siRNA therapeutic is indicated for the treatment of neuropathies associated with hereditary tra…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Transthyretin mRNA
Waktu ParuhThe median half-lif…
Vol. DistribusiBased on a populati…
KlirensThe apparent cleara…
Genetik -
VX-148 DB06103
small molecule

VX-148 is a second-generation, orally administered inhibitor of inosine monophosphate dehydrogenase (IMPDH). The IMPDH enzyme plays a key role in regulating immune response and proliferation of specific cell types, including lymphocytes. VX-148 is a developed…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Inosine-5'-monophosphate dehydrogenase 2
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VX-702 DB05470
small molecule | CAS: 745833-23-2

VX-702 is a small molecule investigational oral anti-cytokine therapy for treatment of inflammatory diseases, specifically rheumatoid arthritis (RA). It acts as a p38 MAP kinase inhibitor. In the future, VX-702 may be investigated for combination with methotr…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
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VX-765 DB05507
small molecule

VX-765 is the orally available prodrug of a potent and selective competitive inhibitor of ICE/caspase-1 (VRT-043198). VX-765 is currently under clinical development for the treatment of inflammatory and autoimmune conditions, as it blocks the hypersensitive r…

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAminobenzoates +4
Target Protein:
Caspase-1Interleukin-1 beta
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VXA-CoV2-1 DB16433
biotech

VXA-CoV2-1 is a non-replicating adenoviral vector-based oral tableted vaccine candidate that expresses a SARS-CoV-2 antigen and dsRNA adjuvant[L30493]. This oral vaccine aims to induce immunogenicity through induction of potent serum neutralizing antibodies t…

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Warfarin Approved DB00682
small molecule | CAS: 81-81-2

Warfarin is an anticoagulant drug normally used to prevent blood clot formation as well as migration. Although originally marketed as a pesticide (d-Con, Rodex, among others), Warfarin has since become the most frequently prescribed oral anticoagulant in Nort…

Kategori:
4-HydroxycoumarinsAgrochemicalsAnticoagulants +38
Target Protein:
Vitamin K epoxide reductase complex subunit 1Nuclear receptor subfamily 1 group I member 2
Gen Terkait:
CYP2C9 VKORC1 CYP4F2 +2
Waktu ParuhR-warfarin is clear…
Vol. DistribusiVd of 0.14 L/kg.[la…
KlirensClearance of warfar…
Genetik 5 Varian
Water Approved DB09145
small molecule | CAS: 7732-18-5

Water (chemical formula: H2O) is a transparent fluid which forms the world's streams, lakes, oceans and rain, and is the major constituent of the fluids of organisms. As a chemical compound, a water molecule contains one oxygen and two hydrogen atoms that are…

Kategori:
DiluentsEENT Drugs, MiscellaneousIrrigating Solutions +2
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WAY-151693 DB02071
small molecule

Deskripsi belum tersedia.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
Collagenase 3
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Wheat germ oil DB16570
biotech | CAS: 313258-61-6

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesLipids +4
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Willardiine DB04129
small molecule | CAS: 21416-43-3

Willardiine is a compound isolated from seeds of _Acacia willariana_.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsPyrimidines +1
Target Protein:
Glutamate receptor 1Glutamate receptor 2
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WIN 55212-2 DB13950
small molecule | CAS: 131543-22-1

WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure. It is a potent cannabinoid receptor agonist th…

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAnalgesics +21
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2
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WIN-54954 DB08723
small molecule | CAS: 107355-45-3

WIN-54954 is a broad-spectrum antipicornavirus drug.

Target Protein:
Genome polyproteinGenome polyprotein
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Wine grape Approved DB10634
biotech

Wine grape allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
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WL-1002 DB05346
small molecule

WL-1002 is developed by Winston Laboratories which is a topical cream formulation of 075% zucapaicin (also known as civamide), for the treatment of pain due to osteoarthritis.

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WNT-974 DB12561
small molecule | CAS: 1243244-14-5

WNT974 has been used in trials studying the treatment of Metastatic Colorectal Cancer and Squamous Cell Carcinoma, Head And Neck.

Kategori:
Enzyme Inhibitors
Target Protein:
Protein-serine O-palmitoleoyltransferase porcupine
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Wood creosote DB13271
small molecule | CAS: 8021-39-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCough and Cold PreparationsCresols +2
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Wortmannin DB08059
small molecule | CAS: 19545-26-7

Wortmannin is a steroid metabolite of _Penicillium funiculosum_ and _Talaromyces wortmannii_ fungi. This drug acts as a nonspecific, covalent inhibitor of phosphoinositide 3-kinase enzymes (PI3Ks).

Kategori:
AndrostadienesAndrostanesAndrostenes +16
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase PLK1 +2
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WP-1066 DB12679
small molecule | CAS: 857064-38-1

WP1066 has been used in trials studying the treatment of Melanoma, Brain Cancer, Solid Tumors, and Central Nervous System Neoplasms.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Signal transducer and activator of transcription 3
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WP-1122 DB17192
small molecule

WP-1122 is a prodrug of 2-deoxy-D-glucose (2-DG). It was granted FDA orphan designation for the treatment of glioblastoma multiforme.[L47361]

Kategori:
CarbohydratesDeoxy Sugars
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WP-1301 DB17702
biotech | CAS: 1609460-62-9

WP1301 is a synthetic peptide derived from hFVIII. It binds to an MHC class II molecule and is recognized by a Factor VIII-specific T cell.[L46138]

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WRR-112 DB03691
small molecule

Deskripsi belum tersedia.

Target Protein:
CruzipainCathepsin F
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WRR-204 DB04502
small molecule

Deskripsi belum tersedia.

Target Protein:
Cruzipain
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WRR-99 DB03573
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin FCruzipain
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WSD-0922 DB17170
small molecule | CAS: 2226552-64-1

Deskripsi belum tersedia.

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WT-1 122 long DB17353
biotech | CAS: 952720-86-4

Deskripsi belum tersedia.

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WT-1 331 long DB17355
biotech | CAS: 935395-34-9

Deskripsi belum tersedia.

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WT-1 427 long DB17354
biotech | CAS: 935395-33-8

Deskripsi belum tersedia.

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WT-1 A1 DB17352
small molecule | CAS: 852243-39-1

Deskripsi belum tersedia.

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WTx-Bortezomib DB17389
biotech

Deskripsi belum tersedia.

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WU-CART-007 DB18617
biotech

WU-CART-007 consists of allogeneic, fratricide-resistant genetically modified T cells transduced with a 2nd generation 4-1BB-CD3z chimeric antigen receptor targeting human CD7.

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WU-NK-101 DB18350
biotech

WU-NK-101 is an allogeneic CD3-depleted, CD56-enriched activated natural killer-cell product

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WVE-003 DB17870
biotech

WVE-003 is an allele-selective antisense oligonucleotide that works to selectively reduce the toxic mutant huntingtin (mHTT) protein.[L46787]

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WVE-N531 DB17848
biotech

Deskripsi belum tersedia.

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WX-UK1 DB05476
small molecule | CAS: 255374-84-6

WX-UK1 is a 3-amidinophenylalanine-based non-cytotoxic small molecule that belongs to a new class of drugs. In animal models, WX-UK1 blocks tumor cell invasion, metastasis and primary tumor growth by inhibiting serine proteases and the urokinase Plasminogen A…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Urokinase plasminogen activator surface receptor
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WZB-117 DB16764
small molecule | CAS: 1223397-11-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +3
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X-165 DB18053
small molecule | CAS: 1815589-34-4

Deskripsi belum tersedia.

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X-396 DB13104
small molecule | CAS: 1365267-27-1

X-396 has been used in trials studying the treatment of Advanced Solid Tumors and Non-small Cell Lung Cancer.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
ALK tyrosine kinase receptor
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Menampilkan 13251–13300 dari 13591
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