Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 266 / 282
Trimethoprim Approved DB00440
small molecule | CAS: 738-70-5

Trimethoprim is an antifolate antibacterial agent that inhibits bacterial dihydrofolate reductase (DHFR), a critical enzyme that catalyzes the formation of tetrahydrofolic acid (THF) - in doing so, it prevents the synthesis of bacterial DNA and ultimately con…

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAnti-Infective Agents +32
Target Protein:
Dihydrofolate reductaseDihydrofolate reductase
Waktu ParuhTrimethoprim half-l…
Vol. DistribusiTrimethoprim is ext…
KlirensFollowing oral admi…
Genetik -
small molecule | CAS: 2453-03-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethyllysine DB03977
small molecule | CAS: 19253-88-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Calmodulin-2Calmodulin-1Calmodulin-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10182-92-0

Deskripsi belum tersedia.

Kategori:
AminesCompounds used in a research, industrial, or household settingDetergents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetrexate Approved DB01157
small molecule | CAS: 52128-35-5

A nonclassical folic acid inhibitor through its inhibition of the enzyme dihydrofolate reductase. It is being tested for efficacy as an antineoplastic agent and as an antiparasitic agent against pneumocystis pneumonia in AIDS patients. Myelosuppression is its…

Kategori:
Acids, AcyclicAcids, AldehydicAnti-Infective Agents +18
Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh11 to 20 hours
Vol. Distribusi* 20 ± 8 L/m2 * 36…
Klirens* 38 +/- 15 mL/min/…
Genetik -
Trimipramine Approved DB00726
small molecule | CAS: 739-71-9

Tricyclic antidepressant similar to imipramine, but with more antihistaminic and sedative properties.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +44
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +15
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +5
Waktu Paruh11-18 hrs
Vol. Distribusi-
Klirens-
Genetik 8 Varian
Trinitrotoluene DB01676
small molecule | CAS: 118-96-7

Trinitrotoluene is an explosive chemical that can cause skin irritation and other toxic consequences.

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingExplosive Agents
Target Protein:
Pentaerythritol tetranitrate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trioxsalen Approved DB04571
small molecule | CAS: 3902-71-4

Trioxsalen (trimethylpsoralen, trioxysalen or trisoralen) is a furanocoumarin and a psoralen derivative obtained from several plants, mainly Psoralea corylifolia. Like other psoralens it causes photosensitization of the skin. It is administered either topical…

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +11
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tripamide DB15959
small molecule | CAS: 73803-48-2

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingMembrane Transport Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tripelennamine Approved DB00792
small molecule | CAS: 91-81-6

A histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation. It is used to treat asthma; HAY fever; urticaria; and rhinitis; and also in veterinary applications. Tripelennamine is administered by various routes, including topic…

Kategori:
AminesAminopyridinesAnti-Allergic Agents +17
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triphendiol DB06588
small molecule | CAS: 1213777-80-0

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10380-08-2

Used as water softener, peptizing agent, emulsifier & dispersing agent; ingredient of cleansers; meat preservative.

Kategori:
AcidsAcids, NoncarboxylicAnions +5
Target Protein:
Poly(A) polymerase alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Dehydrosqualene synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triprolidine Approved DB00427
small molecule | CAS: 486-12-4

First generation histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria. It is a component of cough and cold medicines. It may cause drowsiness.

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +7
Target Protein:
Histamine H1 receptor
Waktu Paruh4 to 6 hours.
Vol. Distribusi-
Klirens-
Genetik -
biotech

Tripterygium wilfordii whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triptolide DB12025
small molecule | CAS: 38748-32-2

Triptolide has been used in trials studying the treatment of HIV, Crohn's Disease, Intestinal Diseases, Gastrointestinal Diseases, and Digestive System Diseases, among others.

Kategori:
Adrenal Cortex HormonesAlkylating DrugsAntineoplastic Agents +10
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triptorelin Approved DB06825
small molecule | CAS: 57773-63-4

Triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH). Possessing greater potency than endogenous LHRH, triptorelin reversibly represses gonadotropin secretion. After chronic, continuous administration, this age…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +23
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiAfter a single IV d…
KlirensIn healthy male vol…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Chlorocatechol 1,2-dioxygenaseAlpha-lytic protease
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trisaccharide A DB17689
small molecule | CAS: 49777-13-1

Deskripsi belum tersedia.

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trisaccharide B DB17690
small molecule | CAS: 49777-14-2

Deskripsi belum tersedia.

Kategori:
ABO Blood-Group SystemCarbohydratesOligosaccharides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trivanadate DB04219
small molecule

Deskripsi belum tersedia.

Kategori:
Vanadates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRK-001 DB18577
biotech

TRK-001 is an autologous regulatory T-cell therapy. It is being investigated for the prevention of graft rejection following solid organ transplantation.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRK-250 DB18500
biotech

TRK-250 is a small interfering RNA agent that targets human transforming growth factor-beta 1 (TGF-?1) messenger RNA.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRO40303 DB16031
small molecule | CAS: 14291-24-8

TRO40303 is under investigation in clinical trial NCT01374321 (Safety and Efficacy Study of TRO40303 for Reduction of Reperfusion Injury in Patients Undergoing Percutaneous Coronary Intervention for Acute Myocardial Infarction).

Kategori:
AminesFused-Ring CompoundsHydroxylamines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troclosene DB15960
small molecule | CAS: 2782-57-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiviral Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trofinetide Approved DB06045
small molecule | CAS: 853400-76-7

Trofinetide is a novel synthetic analog of [glypromate], also known as glycine–proline–glutamate (GPE), a naturally occurring protein in the brain and the N-terminal tripeptide of insulin-like growth factor 1 (IGF-1).[A258438] Trofinetide was approved by the …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +11
Waktu ParuhThe effective elimi…
Vol. DistribusiFollowing oral admi…
KlirensNo information is a…
Genetik -
Trofosfamide DB12902
small molecule | CAS: 22089-22-1

Trofosfamide has been used in trials studying the treatment of Ependymomas, Medulloblastomas, Sarcoma, Soft Tissue, Supratentorial PNETs, and Recurrent Brain Tumors.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troglitazone Approved DB00197
small molecule | CAS: 97322-87-7

Troglitazone was withdrawn in 2000 due to risk of hepatotoxicity. It was superseded by [pioglitazone] and [rosiglitazone].

Kategori:
Alimentary Tract and MetabolismBenzopyransBlood Glucose Lowering Agents +38
Target Protein:
Peroxisome proliferator-activated receptor gammaEstrogen-related receptor gammaSteroid hormone receptor ERR1 +6
Waktu Paruh16-34 hours
Vol. Distribusi-
Klirens-
Genetik -
Trolamine Approved DB13747
small molecule | CAS: 102-71-6

Trolamine, which is also referred to as triethanolamine (TEA), is a tertiary amine and a triol. It is a bifunctional compound that exhibits both properties of alcohols and amines. Trolamine contains small amounts of diethanolamine and ethanolamine and may als…

Kategori:
AlcoholsAminesAmino Alcohols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trolamine salicylate Approved DB11079
small molecule | CAS: 2174-16-5

Trolamine salicylate is an organic compound or a salt formed between triethanolamine and salicylic acid. Triethanolamine neutralizes the acidity of the salicylic acid. It is a topical analgesic used for temporary relief of minor pain associated with arthritis…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnti-Inflammatory Agents +11
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. DistribusiTopical administrat…
Klirens-
Genetik -
Troleandomycin Approved DB13179
small molecule | CAS: 2751-09-9

A macrolide antibiotic that is similar to erythromycin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +18
Target Protein:
50S ribosomal protein L3250S ribosomal protein L4Nuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tromantadine Approved DB13288
small molecule | CAS: 53783-83-8

Tromantadine is marketed as Viru-Merz in the Czech Republic [L5740]. It is an antiviral used in the treatment of herpes zoster and simplex.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tromethamine Approved DB03754
small molecule | CAS: 77-86-1

An organic amine proton acceptor. It is used in the synthesis of surface-active agents and pharmaceuticals; as an emulsifying agent for cosmetic creams and lotions, mineral oil and paraffin wax emulsions, as a biological buffer, and used as an alkalizer. (Fro…

Kategori:
AlcoholsBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +12
Target Protein:
S-adenosylmethionine decarboxylase proenzymeAmyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropatepine DB13252
small molecule | CAS: 27574-24-9

Tropatepine has been used in France for its antiparkinsons activities [A175024].

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropicamide Approved DB00809
small molecule | CAS: 1508-75-4

Tropicamide is an alkaloid atropine?derived anticholinergic drug and a non?selective antagonist of muscarinic acetylcholine (mACh) receptors.[A230103] Usually available in ophthalmic formulations, tropicamide is used to cause mydriasis and cycloplegia for eye…

Kategori:
Anticholinergic AgentsAutonomic AgentsCholinergic Agents +8
Target Protein:
Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhTropicamide has a p…
Vol. DistribusiNo information can …
KlirensNo information can …
Genetik -
Tropifexor DB16343
small molecule | CAS: 1383816-29-2

Tropifexor is under investigation in clinical trial NCT02516605 (A Multi-part, Double Blind Study to Assess Safety, Tolerability and Efficacy of Tropifexor (LJN452) in PBC Patients).

Kategori:
Heterocyclic Compounds, Fused-RingThiazoles
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropinone DB01874
small molecule | CAS: 532-24-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troriluzole DB15079
small molecule | CAS: 1926203-09-9

Troriluzole is under investigation in clinical trial NCT03701399 (Troriluzole in Adult Subjects With Spinocerebellar Ataxia).

Kategori:
Nervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trospium Approved DB00209
small molecule | CAS: 47608-32-2

Trospium is an antispasmodic agent used to treat the symptoms of overactive bladder, a condition that causes the bladder muscles to contract uncontrollably.[L6208] An overactive bladder leads to an increased urge to urinate, frequent urination, and sometimes,…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +22
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu ParuhThe half-life of tr…
Vol. DistribusiThe volume of distr…
KlirensThe total apparent …
Genetik -
Trotabresib DB17421
small molecule | CAS: 1706738-98-8

Trotabresib is an oral, potent, and reversible inhibitor of the epigenetic target bromodomain and extra-terminal (BET) proteins.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trout Approved DB10626
biotech

Trout allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trovafloxacin Approved DB00685
small molecule | CAS: 147059-72-1

Trovafloxacin is a broad spectrum antibiotic that has been commonly marketed under the brand name Trovan by Pfizer. It exerts its antibacterial activity by inhibiting the uncoiling of supercoiled DNA in various bacteria by blocking the activity of DNA gyrase …

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhFollowing oral admi…
Vol. Distribusi-
Klirens-
Genetik -
Troxerutin DB13124
small molecule | CAS: 7085-55-4

Troxerutin has been used in trials studying the treatment of Chronic Venous Insufficiency.

Kategori:
AnticoagulantsBenzopyransCapillary Stabilizing Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRV-120027 DB12199
small molecule | CAS: 1234510-46-3

TRV120027 has been used in trials studying the treatment of Heart Failure and Kidney Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
AmicyaninMethylamine dehydrogenase heavy chainMethylamine dehydrogenase light chain +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-518 DB17534
biotech | CAS: 1427683-53-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-E-002-1 DB17264
small molecule | CAS: 1803036-93-2

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypan blue free acid Approved DB09158
small molecule | CAS: 2538-83-2

Trypan blue is a diazo dye used in ophthalmic cataract surgery to stain the anterior capsule in the presence of a mature cataract. This is done to aid in visualization before creating the continuous curvilinear capsulorhexis.

Kategori:
ArylsulfonatesArylsulfonic AcidsAzo Compounds +12
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypsin Approved DB11237
small molecule | CAS: 9002-07-7

Trypsin is a serine protease that plays an essential role in protein hydrolysis and absorption in mammals. When converted from its zymogen trypsinogen, trypsin is available as an active peptide hydrolase (EC 3.4.21.4) form to cleave peptide chains, mainly at …

Kategori:
Blood and Blood Forming OrgansDermatologicalsEndopeptidases +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tryptamine DB08653
small molecule | CAS: 61-54-1

Deskripsi belum tersedia.

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Target Protein:
Amine oxidase [flavin-containing] B5-hydroxytryptamine receptor 2AAmine oxidase [flavin-containing] A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13251–13300 dari 14063
Sebelumnya Halaman 266 / 282 Berikutnya