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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 265 / 321
RGG0853 DB18669
biotech

RGG0853 is an E1A lipid complex, a repressor gene complexed with a cationic lipid vector.

Waktu Paruh-
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rGLP-1 DB05433
small molecule

rGLP-1 is a continuous infusion of glucagon-like peptide 1, or GLP-1, targeted for the treatment of congestive heart failure (CHF) in patients ineligible for transplant. GLP-1 is a naturally occurring hormone produced in the intestines in response to food int…

Kategori:
Gastrointestinal HormonesGlucagon-Like PeptidesHormones +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
RGLS-8429 DB18127
biotech

RGLS-8429 is an investigational anti-miR-17 oligonucleotide.

Waktu Paruh-
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RGX-111 DB17632
biotech

RGX-111 is an adeno-associated virus vector AAV9 designed to deliver the ?-L-iduronidase (IDUA) gene. Developed by REGENXBIO Inc., it was investigated for the treatment of mucopolysaccharidosis Type I (MPS I).[L46666]

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RGX-121 DB17681
biotech

RGX-121 is designed to use the NAV AAV9 vector to deliver the human iduronate-2-sulfatase gene to the central nervous system.

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RGX-181 DB17942
biotech

RGX-181 consists of an adeno-associated virus serotype 9 (AAV9) vector designed to deliver the soluble lysosomal enzyme tripeptidyl peptidase I (TPP1) gene. Developed by REGENXBIO, it is being investigated for the treatment of late-infantile neuronal ceroid l…

Waktu Paruh-
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RGX-202 DB18397
biotech

RGX-202 is a recombinant AAV8 that contains a vector genome encoding a miniaturized dystrophin protein (microdystrophin).

Waktu Paruh-
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RGX-501 DB17639
biotech

RGX-501 is an adeno-associated virus vector 8 (AAV8)-mediated gene therapy that delivers a functional copy of the human low-density lipoprotein receptor (LDLR) gene to liver cells. It is being investigated for the treatment of homozygous familial hypercholest…

Waktu Paruh-
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RH-1 DB04090
small molecule | CAS: 221635-42-3

RH-1 has been used in trials studying the treatment of Advanced Solid Tumors and Non-Hodgkin's Lymphoma.

Target Protein:
NAD(P)H dehydrogenase [quinone] 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rhamnetin DB16772
small molecule | CAS: 90-19-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhamnose DB02961
small molecule | CAS: 3615-41-6

A methylpentose whose L- isomer is found naturally in many plant glycosides and some gram-negative bacterial lipopolysaccharides. [PubChem]

Kategori:
CarbohydratesDeoxy Sugars
Target Protein:
L-rhamnose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhein DB13174
small molecule | CAS: 478-43-3

Rhein is an anthraquinone metabolite of rheinanthrone and senna glycoside is present in many medicinal plants including Rheum palmatum, Cassia tora, Polygonum multiflorum, and Aloe barbadensis [A19247]. It is known to have hepatoprotective, nephroprotective, …

Kategori:
AnthracenesCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +10
Target Protein:
Heat shock protein HSP 90-alphaOxysterols receptor LXR-alphaOxysterols receptor LXR-beta +2
Waktu Paruh4-10h [A19300].
Vol. Distribusi15-60L [A19300].
KlirensTotal CL is 1.5 L/h…
Genetik -
Rheinanthrone DB13175
small molecule | CAS: 480-09-1

Rheinanthrone is the active metabolite of senna glycoside [DB11365] known for its laxative effect [A19235]. It is commonly produced by plants of the Rheum species [L772].

Kategori:
Anthracenes
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 644961-22-8

Deskripsi belum tersedia.

Waktu Paruh-
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Rhenium re-186 DB19266
small molecule | CAS: 14998-63-1

Rhenium re-186 is under investigation in clinical trial NCT01906385 (Maximum Tolerated Dose, Safety, and Efficacy of Rhenium Nanoliposomes in Recurrent Glioma (Respect)).

Kategori:
ElementsIsotopesMetals +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsTherapeutic Radiopharmaceuticals
Waktu Paruh-
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Rhenium re-188 DB19267
small molecule | CAS: 14378-26-8

Rhenium re-188 is under investigation in clinical trial NCT03458559 (Rhenium-188-hedp vs. Radium-223-chloride in Patients With Advanced Prostate Cancer Refractory to Hormonal Therapy).

Kategori:
ElementsIsotopesMetals +2
Waktu Paruh-
Vol. Distribusi-
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rhIGFBP-3 DB05897
biotech

rhIGFBP-3 (recombinant human insulin-like growth factor binding protein-3) is Insmed’s proprietary anti-cancer compound that has demonstrated significant decreases in cancerous growth in several models of human. It is developed by Insmed and is currently unde…

Target Protein:
Insulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rhMBL DB05237
biotech

rhMBL is a protein therapeutic being developed by Enzon for the prevention and treatment of severe infections in individuals with low levels of Mannose-Binding Lectin (MBL). Over 10 percent of the general population is estimated to be MBL-deficient. Natural M…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 104114-27-4

Deskripsi belum tersedia.

Waktu Paruh-
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Rhodamine 6G DB03825
small molecule | CAS: 989-38-8

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsColoring AgentsCompounds used in a research, industrial, or household setting +7
Target Protein:
HTH-type transcriptional regulator QacRMultidrug efflux pump subunit AcrB
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhodamine B DB16853
small molecule | CAS: 81-88-9

Deskripsi belum tersedia.

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingCosmetics +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rhThrombin Approved DB04923
biotech | CAS: 1270043-60-1

rhThrombin (recombinant human thrombin) is being developed by ZymoGenetics, Inc. as a general aid to achieving hemostasis during surgery. ZymoGenetics is developing rhThrombin, a recombinant form of human thrombin that is not derived from animal or human bloo…

Waktu ParuhApproximately 15 ho…
Vol. Distribusi-
Klirens-
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Rhubarb Approved DB10651
biotech | CAS: 8016-55-5

Rhubarb allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ribavirin Approved DB00811
small molecule | CAS: 36791-04-5

Producing a broad-spectrum activity against several RNA and DNA viruses, Ribavirin is a synthetic guanosine nucleoside and antiviral agent that interferes with the synthesis of viral mRNA. It is primarily indicated for use in treating hepatitis C and viral he…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +13
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1RNA-directed RNA polymerase LGenome polyprotein +2
Gen Terkait:
IFNL3
Waktu ParuhThe terminal half-l…
Vol. DistribusiRibavirin displays …
KlirensThe total apparent …
Genetik 1 Varian
small molecule | CAS: 1352921-29-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 40925-28-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsCarbohydrates +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ribaxamase DB16311
biotech | CAS: 1792207-66-9

Ribaxamase is under investigation in clinical trial NCT02563106 (A Study of SYN-004 for the Prevention of c.diff in Patients With a LRTI).

Kategori:
AmidohydrolasesAmino Acids, Peptides, and ProteinsEnzymes +3
Waktu Paruh-
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Ribitol DB14704
small molecule | CAS: 488-81-3

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesSugar Alcohols
Waktu Paruh-
Vol. Distribusi-
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Ribociclib Approved DB11730
small molecule | CAS: 1211441-98-3

Ribociclib is a selective cyclin-dependent kinase inhibitor, a class of drugs that help slow the progression of cancer by inhibiting two proteins called cyclin-dependent kinase 4 and 6 (CDK4/6). These proteins, when over-activated, can enable cancer cells to …

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhAt steady-state in …
Vol. DistribusiAt steady-state, th…
KlirensAt steady-state in …
Genetik -
Riboflavin Approved DB00140
small molecule | CAS: 83-88-5

Nutritional factor found in milk, eggs, malted barley, liver, kidney, heart, and leafy vegetables. The richest natural source is yeast. It occurs in the free form only in the retina of the eye, in whey, and in urine; its principal forms in tissues and cells a…

Kategori:
Alimentary Tract and MetabolismBiological FactorsCoenzymes +14
Target Protein:
Riboflavin kinaseRiboflavin synthaseFlavin reductase (NADPH)
Waktu Paruh66-84 minutes
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 752-56-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Riboprine DB11933
small molecule | CAS: 7724-76-7

Ipa has been used in trials studying the treatment of Nausea and Surgical Site Infection.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ribose DB15073
small molecule | CAS: 50-69-1

Ribose is under investigation in clinical trial NCT01727479 (Ribose and Sport Performance).

Kategori:
CarbohydratesMonosaccharidesPentoses
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylaseUridine phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4151-19-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesPentosephosphatesSugar Phosphates
Target Protein:
Ribose-5-phosphate isomerase A2-dehydro-3-deoxyphosphooctonate aldolaseADP-ribose pyrophosphatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ribostamycin Approved DB03615
small molecule | CAS: 25546-65-0

Ribostamycin is an aminoglycoside antibiotic[A187166] isolated from _Streptomyces ribosidificus_[A187178] listed as one of the World Health Organization's critically important antimicrobials.[L9071]

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Target Protein:
30S ribosomal protein S12Protein disulfide-isomeraseAminoglycoside N(6')-acetyltransferase type 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
3-keto-L-gulonate-6-phosphate decarboxylase UlaD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rice bran Approved DB14361
biotech

Rice bran is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Rice bran oil Approved DB11293
biotech

Rice bran oil is extracted from the hard outer brown layer of rice after chaff (rice husk) used for high-temperature cooking methods such as deep frying and stir frying. It contains monosaturated fatty acids, polyunsaturated fatty acids, and saturated fatty a…

Kategori:
Biological ProductsComplex MixturesDietary Fats +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ricinoleic acid DB02955
small molecule | CAS: 141-22-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsFatsFats, Unsaturated +6
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ricolinostat DB12376
small molecule | CAS: 1316214-52-4

Ricolinostat is under investigation for the treatment of Breast Carcinoma and Metastatic Breast Cancer.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ridaforolimus DB06233
small molecule | CAS: 572924-54-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +8
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ridinilazole DB15308
small molecule | CAS: 308362-25-6

Ridinilazole is under investigation in clinical trial NCT02092935 (A Study of SMT19969 Compared With Vancomycin for the Treatment of Clostridium Difficile-Associated Diarrhoea (CDAD)).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ridogrel DB01207
small molecule | CAS: 110140-89-1

Ridogrel is a dual action drug useful for the prevention of systemic thrombo-embolism and as an adjunctive agent to thrombolytic therapy in acute myocardial infarction. However, there currently are no clinical indications for preferential use of ridogrel over…

Kategori:
Acids, AcyclicAntiplatelet agentsEnzyme Inhibitors +7
Target Protein:
Thromboxane-A synthaseThromboxane A2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifabutin Approved DB00615
small molecule | CAS: 72559-06-9

A broad-spectrum antibiotic that is being used as prophylaxis against disseminated Mycobacterium avium complex infection in HIV-positive patients.

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +27
Target Protein:
DNA-directed RNA polymerase subunit alphaDNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta' +2
Waktu Paruh45 (± 17) ho…
Vol. Distribusi-
Klirens* 0.69 +/- 0.32 L/h…
Genetik -
Rifalazil DB04934
small molecule | CAS: 129791-92-0

Rifalazil is a derivative of the antibiotic rifamycin. It is being investigated by ActivBiotics for the treatment of various bacterial infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +7
Target Protein:
DNA-directed RNA polymerase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifampin Approved DB01045
small molecule | CAS: 13292-46-1

Rifampin, also known as rifampicin, is a broad-spectrum antimicrobial [A263748] that was first discovered in 1965 [A263753] and clinically used in 1968.[A263768] Rifampin is used to treat tuberculosis and works by inhibiting the microbial DNA-dependent RNA po…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +55
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhIn healthy adults, …
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Rifamycin Approved DB11753
small molecule | CAS: 6998-60-3

Rifamycin is the prime member of the rifamycin family which are represented by drugs that are a product of fermentation from the gram-positive bacterium _Amycolatopsis mediterranei_, also known as _Streptomyces mediterranei_. The parent compound of rifamycin …

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +49
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'DNA-directed RNA polymerase subunit beta +2
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Rifapentine Approved DB01201
small molecule | CAS: 61379-65-5

Rifapentine is an antibiotic drug used in the treatment of tuberculosis. It inhibits DNA-dependent RNA polymerase activity in susceptible cells. Specifically, it interacts with bacterial RNA polymerase but does not inhibit the mammalian enzyme.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +24
Target Protein:
DNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi* 70.2 ± 9.1 L
Klirens* Apparent Oral cl=…
Genetik -
Menampilkan 13201–13250 dari 16004
Sebelumnya Halaman 265 / 321 Berikutnya