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13591

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10177 (74.9%)
Target
7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 264 / 272
VidPrevtyn Beta Approved DB16427
biotech

VidPrevtyn Beta is an adjuvanted, recombinant COVID-19 vaccine developed collaboratively by GlaxoSmithKline (GSK) and Sanofi Pasteur.[L49691] It comprises a recombinant SARS-CoV-2 spike protein (B.1.351 strain) - produced by recombinant DNA technology using a…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vidupiprant DB12272
small molecule | CAS: 1169483-24-2

Vidupiprant has been used in trials studying the treatment and basic science of Asthma.

Kategori:
Acids, CarbocyclicAmidesSulfones +1
Target Protein:
Prostaglandin D2 receptor 2Prostaglandin D2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vidutolimod DB17500
biotech | CAS: 147063-80-7

Vidutolimod is a Toll-like receptor 9 (TLR9) agonist. It is an investigational cancer vaccine.

Waktu Paruh-
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Genetik -
Vigabatrin Approved DB01080
small molecule | CAS: 68506-86-5

Vigabatrin is an analog of gamma-aminobutyric acid ([GABA]), the main inhibitory neurotransmitter in the central nervous system, used in the treatment of refractory seizures and infantile spasms.[L13616] It irreversibly inhibits the enzyme responsible for GAB…

Kategori:
Acids, AcyclicAminobutyratesAnti-epileptic Agent +15
Target Protein:
4-aminobutyrate aminotransferase, mitochondrial
Waktu ParuhThe terminal half-l…
Vol. DistribusiVigabatrin is widel…
KlirensThe oral clearance …
Genetik -
Vilamakitug DB18978
biotech | CAS: 2458202-06-5

Vilamakitug is under investigation in clinical trial NCT05201352 (Evaluation of Efficacy of Trifluridine/tipiracil Plus an Anti-il-1? True Human Antibody Versus Trifluridine/tipiracil Plus Placebo in Metastatic Colorectal Cancer Patients After Failure of Oxal…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vilanterol Approved DB09082
small molecule | CAS: 503068-34-6

Vilanterol is a selective long-acting ?2-adrenergic agonist (LABA) with inherent 24-hour activity for the once-daily treatment of COPD and asthma.[A7737] This is in response to the need for longer-acting ?2-adrenergic agonists to overcome poor patient complia…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +19
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhThe effective half-…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Vilastobart DB19327
biotech | CAS: 2760549-50-4

Vilastobart is under investigation in clinical trial NCT04896697 (Vilastobart (XTX101) Monotherapy and Vilastobart and Atezolizumab Combination Therapy in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Vildagliptin Approved DB04876
small molecule | CAS: 274901-16-5

Vildagliptin (LAF237) is an orally active antihyperglycemic agent that selectively inhibits the dipeptidyl peptidase-4 (DPP-4) enzyme. It is used to manage type II diabetes mellitus, where GLP-1 secretion and insulinotropic effects are impaired.[A232488] By i…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +11
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensAfter intravenous a…
Genetik -
Vilobelimab DB16416
biotech | CAS: 2250440-41-4

Vilobelimab is a chimeric monoclonal immunoglobulin G4 (IgG4) antibody that binds to the soluble form of human C5a with high affinity. It consists of mouse anti-human complement factor 5a (C5a) monoclonal binding sites (variable regions of heavy and light cha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Complement C5
Waktu ParuhThe elimination hal…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Viltolarsen Approved DB15005
biotech | CAS: 2055732-84-6

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albeit a less seve…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD gene (exon 53 viltolarsen target site)
Waktu ParuhViltolarsen has a r…
Vol. DistribusiViltolarsen has a s…
KlirensViltolarsen has a r…
Genetik -
Viminol DB13353
small molecule | CAS: 21363-18-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vimseltinib DB17520
small molecule | CAS: 1628606-05-2

Deskripsi belum tersedia.

Target Protein:
Macrophage colony-stimulating factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinbarbital DB13377
small molecule | CAS: 125-42-8

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61936-68-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsVinca Alkaloids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinburnine DB13793
small molecule | CAS: 4880-88-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +7
Target Protein:
Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vincamine DB13374
small molecule | CAS: 1617-90-9

Vincamine is a monoterpenoid indole alkaloid obtained from the leaves of *Vinca minor* with a vasodilatory property. Studies indicate that vincamine increases the regional cerebral blood flow.

Kategori:
AlkaloidsAntihypertensive AgentsAntineoplastic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vindesine Approved DB00309
small molecule | CAS: 53643-48-4

Vinblastine derivative with antineoplastic activity against cancer. Major side effects are myelosuppression and neurotoxicity. Vindesine is used extensively in chemotherapy protocols (antineoplastic combined chemotherapy protocols).

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +19
Target Protein:
Tubulin beta-1 chain
Waktu Paruh24 hours.
Vol. Distribusi-
Klirens-
Genetik -
Vinflunine Approved DB11641
small molecule | CAS: 162652-95-1

Vinflunine is a third-generation member of the vinca alkaloid family with anti-tumour actions. It was first described in 1998 at the Pierre Fabre research center in France. Like other vinca agents, vinflunine is an anti-mitotic agent that induces a cell cycle…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Tubulin beta chain
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe terminal volume…
KlirensThe total blood cle…
Genetik -
Vinorelbine Approved DB00361
small molecule | CAS: 71486-22-1

Vinorelbine is an anti-mitotic chemotherapy drug that is used in the treatment of several types of malignancies, including breast cancer and non-small cell lung cancer (NSCLC) [L1998]. It was initially approved in the USA in 1990's for the treatment of NSCLC…

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +23
Target Protein:
Tubulin beta chain
Waktu ParuhThe terminal phase …
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Vinpocetine DB12131
small molecule | CAS: 42971-09-5

Vinpocetine has been investigated for the treatment of Epilepsy.

Kategori:
Agents causing hyperkalemiaAlkaloidsAntiarrhythmic agents +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vintafolide DB05168
small molecule | CAS: 742092-03-1

Vintafolide is a folate-targeted chemotherapeutic conjugate (folate vitamin + vinca alkaloid) in clinical stage development as a treatment for folate-receptor positive cancers.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
Folate receptor alphaFolate receptor betaFolate receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinyl ether DB13690
small molecule | CAS: 109-93-3

Deskripsi belum tersedia.

Kategori:
AlkenesAnestheticsAnesthetics, General +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinylbital DB13770
small molecule | CAS: 2430-49-1

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinylglycine DB03214
small molecule | CAS: 70982-53-5

Vinylglycine is an irreversible inhibitor of aspartate aminotransferase.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
L-amino-acid oxidase1-aminocyclopropane-1-carboxylate synthase-like protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1184-84-5

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAlkenes +4
Target Protein:
Phosphonoacetaldehyde hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Violaxanthin DB03460
small molecule | CAS: 126-29-4

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Viomycin Approved DB06827
small molecule | CAS: 32988-50-4

Viomycin is a tuberactinomycin antibiotic that was used to treat Mycobacterium tuberculosis until it was replaced by the less toxic capreomycin. These drugs bind RNA in bacterial ribosomes and inhibit protein synthesis. Viomycin was derived from the actinomyc…

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAnti-Bacterial Agents +8
Target Protein:
16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vipadenant DB06625
small molecule | CAS: 442908-10-3

Deskripsi belum tersedia.

Kategori:
Adenosine A2 Receptor AntagonistsNeurotransmitter AgentsPurinergic Agents +2
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vipoglanstat DB18126
small molecule | CAS: 1360622-01-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Virginiamycin DB11476
small molecule | CAS: 11006-76-1

Virginiamycin is a streptogramin antibiotic similar to pristinamycin and quinupristin/dalfopristin. It is a combination of pristinamycin IIA and virginiamycin S1. Virginiamycin is used in the fuel ethanol industry to prevent microbial contamination and in liv…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 21411-53-0

Pristinamycin IIA is a macrolide antibiotic, a member of the streptogramin A group of antibiotics, and one component of pristinamycin. It is produced by Streptomyces graminofaciens and other bacteria.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
Streptogramin A acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 23152-29-6

One of the components of virginiamycin, a cyclic polypeptide antibiotic complex from streptomyces virginiae, s. Loidensis, s. Mitakaensis, s. Pristina-spiralis, s. Ostreogriseus, and others. It is used to treat infections with gram-positive organisms and as a…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic +1
Target Protein:
Large ribosomal subunit protein eL37
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Virulizin DB17098
biotech | CAS: 216586-46-8

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicBodily SecretionsComplex Mixtures +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Virus Specific T-Cells (VSTs) are a target therapy that are generated for specific viral antigens. These products are generated from virus-naive or virus-experienced autologous or allogenic sources. Antigens identified as an immune target are presented by ant…

Waktu Paruh-
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VIS-410 DB19067
biotech | CAS: 2043950-09-8

VIS-410 is under investigation in clinical trial NCT03040141 (Study of Efficacy and Safety of IV VIS410 Plus Oseltamivir Versus Oseltamivir in Hospitalized Adults With Influenza A).

Waktu Paruh-
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Visilizumab DB12053
biotech | CAS: 219716-33-3

Visilizumab has been investigated for the treatment of Ulcerative Colitis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vismodegib Approved DB08828
small molecule | CAS: 879085-55-9

Vismodegib is an orally active small molecule that inhibits the hedgehog signaling pathway by binding to and inhibiting the transmembrane protein smoothened homologue (SMO).[A258613,A258618,L45803] It was discovered by high-throughput screening of a library o…

Kategori:
AmidesAminesAniline Compounds +18
Target Protein:
Protein smoothened
Waktu ParuhThe half-life of vi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Visnadine DB13355
small molecule | CAS: 477-32-7

Deskripsi belum tersedia.

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingPeripheral Vasodilators +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 934960-96-0

Deskripsi belum tersedia.

Kategori:
AminesBenzoquinonesBenzylammonium Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Visugromab DB18894
biotech | CAS: 2556646-63-8

Visugromab is under investigation in clinical trial NCT06059547 (Neoadjuvant Immunotherapy in Combination With the Anti-gdf-15 Antibody Visugromab (CTL-002) for Treatment of Muscle Invasive Bladder Cancer).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vitamin A Approved DB00162
small molecule | CAS: 68-26-8

Retinol and derivatives of retinol that play an essential role in metabolic functioning of the retina, the growth of and differentiation of epithelial tissue, the growth of bone, reproduction, and the immune response. Dietary vitamin A is derived from a varie…

Kategori:
Adjuvants, ImmunologicAlimentary Tract and MetabolismAlkenes +33
Target Protein:
Retinoic acid receptor RXR-gammaApolipoprotein DProstaglandin-H2 D-isomerase +13
Waktu Paruh1.9 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15713-12-9

Deskripsi belum tersedia.

Target Protein:
5-methyltetrahydrofolate--homocysteine S-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitamin D Approved DB11094
small molecule | CAS: 1406-16-2

Vitamin D ultimately comprises a group of lipid-soluble secosteroids responsible for a variety of biological effects, some of which include increasing the intestinal absorption of calcium, magnesium, and phosphate. With reference to human use, there are 2 mai…

Kategori:
Bone Density Conservation AgentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Vitamin D3 receptorVitamin D-binding protein
Waktu ParuhAlthough certain st…
Vol. Distribusi-
KlirensSome studies propos…
Genetik -
Vitamin E Approved DB00163
small molecule | CAS: 59-02-9

In 1922, vitamin E was demonstrated to be an essential nutrient[A32448]. Vitamin E is a term used to describe 8 different fat soluble tocopherols and tocotrienols, alpha-tocopherol being the most biologically active[A176104]. Vitamin E acts as an antioxidant,…

Kategori:
AntioxidantsBasic Ointments and ProtectantsBenzopyrans +23
Target Protein:
SEC14-like protein 4SEC14-like protein 3SEC14-like protein 2 +7
Waktu Paruh44 hours in prematu…
Vol. Distribusi0.41L/kg in prematu…
Klirens6.5mL/hr/kg in prem…
Genetik -
Vitamin K7 DB15664
small molecule | CAS: 83-69-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Vitex agnus-castus fruit extract is obtained from dry fruits of Vitex agnus-castus. The fruits contain mixture of iridoids, flavonoids and compounds in leaves and flowers that structurally resemble sex hormones. Clinical studies demonstrates effectiveness of …

Kategori:
AngiospermsBiological ProductsComplex Mixtures +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitexin DB16836
small molecule | CAS: 3681-93-4

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vixarelimab DB16350
biotech | CAS: 2243320-83-2

Vixarelimab is under investigation in clinical trial NCT03816891 (A Study to Assess the Efficacy, Safety, and Tolerability of KPL-716 in Reducing Pruritus in Prurigo Nodularis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13151–13200 dari 13591
Sebelumnya Halaman 264 / 272 Berikutnya