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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 263 / 272
Velusetrag DB12702
small molecule | CAS: 866933-46-2

Velusetrag has been used in trials studying the treatment of Gastroparesis and Alzheimer's Disease. It is a highly selective serotonin receptor agonist effective in patients with chronic constipation. It is being developed by Theravance. Velusetrag was discov…

Kategori:
Aza Compounds
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
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Genetik -
Vemircopan DB18012
small molecule | CAS: 2086178-00-7

Deskripsi belum tersedia.

Target Protein:
Complement factor D
Waktu Paruh-
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Vemurafenib Approved DB08881
small molecule | CAS: 918504-65-1

Vemurafenib is a competitive kinase inhibitor with activity against BRAF kinase with mutations like V600E.[A31269] It exerts its function by binding to the ATP-binding domain of the mutant BRAF.[A31270] Vemurafenib was co-developed by Roche and Plexxikon and …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimation of t…
KlirensThe total body clea…
Genetik -
Venadaparib DB17105
small molecule | CAS: 1681017-83-3

Deskripsi belum tersedia.

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Venanprubart DB18891
biotech | CAS: 2635407-50-8

Venanprubart is under investigation in clinical trial NCT05781451 (Anti-btla Agonist Therapy in Subjects With Primary Sjogren's Syndrome).

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Venetoclax Approved DB11581
small molecule | CAS: 1257044-40-8

Venetoclax is a BCL-2 inhibitor that was initially approved by the FDA in April 2016 [FDA label]. Proteins in the B cell CLL/lymphoma 2 (BCL-2) family are important regulators of the apoptotic (programmed cell death) process [A18565], [A18566]. Venetoclax is…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe half-life of ve…
Vol. DistribusiThe population esti…
KlirensMainly hepatic [FDA…
Genetik -
Venglustat DB14966
small molecule | CAS: 1401090-53-6

Venglustat is under investigation in clinical trial NCT01674036 (Safety, Tolerability and Pharmacokinetics of Genz-682452 in Healthy Men).

Kategori:
Acids, AcyclicEnzyme Inhibitors
Target Protein:
Ceramide glucosyltransferase
Waktu Paruh-
Vol. Distribusi-
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Venlafaxine Approved DB00285
small molecule | CAS: 93413-69-5

Venlafaxine is an antidepressant and a serotonin and norepinephrine reuptake inhibitor (SNRI). Its active metabolite, [desvenlafaxine], works by blocking the reuptake of serotonin and norepinephrine, which are key neurotransmitters in mood regulation. Venlafa…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAmines +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +2
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe apparent volume…
KlirensMean ± SD plasma ap…
Genetik 5 Varian
Vepdegestrant DB19006
small molecule | CAS: 2229711-68-4

Vepdegestrant is under investigation in clinical trial NCT05909397 (A Study of ARV-471 (PF-07850327) Plus Palbociclib Versus Letrozole Plus Palbociclib in Participants With Estrogen Receptor Positive, Human Epidermal Growth Factor Negative Advanced Breast Can…

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Vepsitamab DB18211
biotech | CAS: 2413453-53-7

Deskripsi belum tersedia.

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Veralipride DB13523
small molecule | CAS: 66644-81-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntipsychotic Agents +12
Waktu Paruh-
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Verapamil Approved DB00661
small molecule | CAS: 52-53-9

Verapamil is a phenylalkylamine calcium channel blocker used in the treatment of high blood pressure, heart arrhythmias, and angina,[L8791] and was the first calcium channel antagonist to be introduced into therapy in the early 1960s.[A188514] It is a member …

Kategori:
ACE Inhibitors and Calcium Channel BlockersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +50
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent P/Q-type calcium channel subunit alpha-1A +10
Gen Terkait:
ADRB1
Waktu ParuhSingle-dose studies…
Vol. DistribusiVerapamil has a ste…
KlirensSystemic clearance …
Genetik 1 Varian
biotech | CAS: 2364604-87-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Vercirnon DB15250
small molecule | CAS: 698394-73-9

Vercirnon is a novel, orally active anti-inflammatory agent that targets a chemokine receptor protein implicated in both Crohn's disease and ulcerative colitis, the two principal forms of IBD. It is under investigation in clinical trial NCT01611805 (Japanese …

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
C-C chemokine receptor type 9
Waktu Paruh-
Vol. Distribusi-
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Verdinexor DB12207
small molecule | CAS: 1392136-43-4

Kpt 335 is under investigation in clinical trial NCT02431364 (Trial of Safety and Tolerability of Oral Verdinexor (Verdinexor) in Healthy Adults).

Kategori:
Acids, AcyclicAcrylatesAmides
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Verdoheme DB04803
small molecule

Deskripsi belum tersedia.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingMetalloporphyrins +2
Target Protein:
Heme oxygenase 1
Waktu Paruh-
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Verekitug DB19096
biotech | CAS: 2768386-15-6

Verekitug is under investigation in clinical trial NCT06164704 (A Study to Investigate the Efficacy and Safety of Verekitug (UPB-101) in Participants With Chronic Rhinosinusitis With Nasal Polyps).

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Vericiguat Approved DB15456
small molecule | CAS: 1350653-20-1

Vericiguat is a direct stimulator of soluble guanylate cyclase (sGC) used in the management of systolic heart failure to reduce mortality and hospitalizations.[L31153] A key component of the NO-sGC-cGMP signaling pathway that helps to regulate the cardiovascu…

Kategori:
BCRP/ABCG2 SubstratesCardiac TherapyGuanylate Cyclase Stimulators +8
Target Protein:
Retinal guanylyl cyclase 1Guanylate cyclase soluble subunit beta-1
Waktu ParuhIn patients with he…
Vol. DistribusiIn healthy subjects…
KlirensVericiguat is a low…
Genetik -
Verinurad DB11873
small molecule | CAS: 1352792-74-5

Verinurad has been used in trials studying the basic science and treatment of Gout, Gout and Hyperuricemia, and Gout and Asymptomatic Hyperuricemia.

Kategori:
Acids, AcyclicAntigout PreparationsAntirheumatic Agents +3
Target Protein:
Solute carrier family 22 member 12
Waktu Paruh-
Vol. Distribusi-
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Vernakalant Approved DB06217
small molecule | CAS: 794466-70-9

Vernakalant was developed by Cardiome Pharma as as an antiarrhythmic drug intended for rapid conversion of atrial fibrillation to sinus rhythm. It acts as an atypical class III antiarrhythmic drug that potentiates its effect in higher heart rates. Intravenous…

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IIIBenzene Derivatives +12
Target Protein:
Sodium channel protein type 5 subunit alphaPotassium voltage-gated channel subfamily A member 5A-type voltage-gated potassium channel KCND3 +1
Waktu ParuhElimination half li…
Vol. DistribusiApproximately 2L/kg.
KlirensThe typical total b…
Genetik -
Verpacamide A DB04433
small molecule

Deskripsi belum tersedia.

Target Protein:
Chitinase B
Waktu Paruh-
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biotech | CAS: 295371-00-5

Verpasep caltespen is a recombinant chimeric protein composed of the heat shock protein 65 (Hsp65) from _Mycobacterium bovis_, and the human papilloma viral (HPV) protein E7. Hsp65, similar to other members of its family of proteins, elicits a strong immune r…

Target Protein:
Keratin, type II cytoskeletal 7E3 ubiquitin-protein ligase UBR4
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Verteporfin Approved DB00460
small molecule | CAS: 129497-78-5

Verteporfin, marketed as Visudyne, is a benzoporphyrin derivative comprising a 50:50 mixture of two isomers: [CL-315555] and [CL-315585]. It is used as a photosensitizer in photodynamic therapy to eliminate abnormal blood vessels in wet form macular degenerat…

Kategori:
Antineovascularisation AgentsDermatologicalsEENT Drugs, Miscellaneous +10
Waktu ParuhFollowing intraveno…
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Veru-111 DB16462
small molecule | CAS: 1332881-26-1

VERU-111, an investigational drug intended for various therapeutic uses, was under investigation in clinical trials NCT04842747, NCT03752099, NCT04388826, NCT04844749, NCT05008510, and NCT05079360. These trials aimed to evaluate its efficacy, safety, and tole…

Kategori:
Experimental Unapproved Treatments for COVID-19Heterocyclic Compounds, Fused-Ring
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Verubecestat DB12285
small molecule | CAS: 1286770-55-5

Verubecestat is under investigation for the treatment of Alzheimer's Disease, Prodromal Alzheimer's disease, and Amnestic Mild Cognitive Impairment. Verubecestat is Merck’s investigational oral ?-site amyloid precursor protein cleaving enzyme (BACE1 or ? …

Kategori:
Sulfur CompoundsThiazines
Target Protein:
Beta-secretase 1
Waktu Paruh-
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Verubulin DB05585
small molecule | CAS: 827031-83-4

Antineoplastic; a small-molecule inhibitor of microtubule formation that is not a substrate for multidrug resistance pumps.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Verzistobart DB18895
biotech | CAS: 2649466-18-0

Verzistobart is under investigation in clinical trial NCT06056895 (Triple Immune Checkpoint Inhibition for Advanced or Metastatic PD-(L)1 Refractory Merkel Cell Carcinoma).

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Vesatolimod DB12687
small molecule | CAS: 1228585-88-3

Vesatolimod has been used in trials studying the treatment of Hepatitis B and Chronic Hepatitis B.

Kategori:
Anti-Infective AgentsAntiviral AgentsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Toll-like receptor 7
Waktu Paruh-
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Vesencumab DB15428
biotech | CAS: 1205533-60-3

Vesencumab is under investigation in clinical trial NCT00747734 (A Study of MNRP1685A in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
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Vesleteplirsen DB16993
biotech

Deskripsi belum tersedia.

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biotech

Vespula germanica venom protein is an extract of Vespula germanica venom. Vespula germanica venom protein is used in allergenic testing.

Kategori:
Bee and Wasp VenomCell-mediated ImmunityIncreased Histamine Release +2
Waktu Paruh-
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Genetik -
biotech

Vespula pensylvanica venom protein is an extract of Vespula pensylvanica venom. Vespula pensylvanica venom protein is used in allergenic testing.

Kategori:
Bee and Wasp VenomCell-mediated ImmunityIncreased Histamine Release +2
Waktu Paruh-
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Klirens-
Genetik -
biotech

Vespula squamosa venom protein is an extract of Vespula squamosa venom. Vespula squamosa venom protein is used in allergenic testing.

Kategori:
Bee and Wasp VenomCell-mediated ImmunityIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Vespula vulgaris venom protein is an extract of Vespula vulgaris venom. Vespula vulgaris venom protein is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
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Vestipitant DB11949
small molecule | CAS: 334476-46-9

Vestipitant has been investigated for the treatment of Tinnitus.

Kategori:
Benzene DerivativesHydrocarbons, FluorinatedHydrocarbons, Halogenated +2
Target Protein:
Substance-P receptor
Waktu Paruh-
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Vestronidase alfa Approved DB12366
biotech | CAS: 1638194-78-1

Vestronidase alfa, or vestronidase alfa-vjbk, is a recombinant human lysosomal beta glucuronidase that is a purified enzyme produced by recombinant DNA technology in a Chinese hamster ovary cell line. The enzyme is a homotetramer consisted of 4 monomers with …

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +3
Waktu ParuhAfter repeated dosi…
Vol. DistribusiAfter repeated dosi…
KlirensAfter repeated dosi…
Genetik -
Veverimer DB18977
small molecule | CAS: 2099678-27-8

Veverimer is under investigation in clinical trial NCT03390842 (Long-term Safety Extension to Study TRCA-301).

Kategori:
Macromolecular Substances
Waktu Paruh-
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VGA039 DB18385
biotech

VGA039 is an IgG4 monoclonal antibody directed against protein S.

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VGV-1 DB05328
small molecule

VGV-1 is a potential salvage therapy for treatment of HIV infected people who have failed anti-retroviral therapy.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Genetik -
biotech

Viagenpumatucel-L is under investigation in clinical trial NCT02117024 (A Phase 2 Study of Viagenpumatucel-l (HS-110) in Patients With Non-small Cell Lung Cancer).

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Vibecotamab DB18872
biotech | CAS: 2138442-13-2

Vibecotamab is under investigation in clinical trial NCT05285813 (A Phase II Study of Vibecotamab (Xmab14045) for MRD- Positive AML and MDS After Hypomethylating Agent Failure).

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Vibegron Approved DB14895
small molecule | CAS: 1190389-15-1

Vibegron is a potent, selective beta-3 adrenergic receptor (?3) agonist that relaxes the detrusor smooth muscle of the bladder, thereby increasing bladder capacity.[L28305] Vibegron was first approved in Japan in September 2018 for the treatment of overactive…

Kategori:
Adrenergic AgonistsAdrenergic beta-3 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-3 adrenergic receptor
Waktu ParuhThe terminal plasma…
Vol. DistribusiThe mean apparent v…
KlirensThere is limited in…
Genetik -
Vibostolimab DB16420
biotech | CAS: 2231305-30-7

Vibostolimab is under investigation in clinical trial NCT04303169 (Substudy 02C: Safety and Efficacy of Pembrolizumab in Combination With Investigational Agents or Pembrolizumab Alone in Participants With Stage III Melanoma Who Are Candidates for Neoadjuvant …

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biotech | CAS: 1704499-30-8

_Vibrio cholerae_ CVD 103-HgR strain live antigen is a component of Vaxchora, an oral vaccine for immunization against _Vibrio cholerae_ serogroup O1.[L12801] Cholera is an acute bacterial disease of the small intestine caused by _Vibrio cholerae_, which is g…

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +3
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiPharmacokinetic inf…
KlirensPharmacokinetic inf…
Genetik -
biotech

Deskripsi belum tersedia.

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Vibriolysin DB05135
small molecule | CAS: 69598-88-5

Vibriolysin is a proteolytic enzyme secreted by the marine microorganism Vibrio proteolyticus. It is a new agent for enzymatic debridement, shown to rapidly and thoroughly hydrolyze burn wound eschar within full-thickness wounds.

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Vicagrel DB16349
small molecule | CAS: 1314081-53-2

Vicagrel is under investigation in clinical trial NCT03599284 (The Efficacy, Safety and Pharmacokinetic of Antiplatelet Therapy for Vicagrel).

Kategori:
Acids, CarbocyclicAntiplatelet agentsCytochrome P-450 CYP2C19 Substrates +2
Target Protein:
P2Y purinoceptor 12
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vicriviroc DB06652
small molecule | CAS: 306296-47-9

Vicriviroc, also known as SCH 417690 and SCH-D, is currently in clinical trials for the management of HIV-1. This pyrimidine based drug inhibits the interaction of HIV-1 with CCR5, preventing viral entry into cells. This drug was developed by Schering-Plough.

Kategori:
Cytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +2
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
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Vidarabine Approved DB00194
small molecule | CAS: 24356-66-9

A nucleoside antibiotic isolated from Streptomyces antibioticus. It has some antineoplastic properties and has broad spectrum activity against DNA viruses in cell cultures and significant antiviral activity against infections caused by a variety of viruses su…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +17
Target Protein:
Adenosine receptor A2bDNA polymerase catalytic subunitThymidine kinase +1
Waktu Paruh-
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Vidofludimus DB15446
small molecule | CAS: 717824-30-1

Vidofludimus is under investigation in clinical trial NCT03722576 (Vidofludimus Calcium for Primary Sclerosing Cholangitis).

Kategori:
Acids, AcyclicBenzene Derivatives
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
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Genetik -
Menampilkan 13101–13150 dari 13591
Sebelumnya Halaman 263 / 272 Berikutnya