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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 260 / 272
Unoprostone Approved DB06826
small molecule | CAS: 120373-36-6

Unoprostone isopropyl is a prostaglandin analogue. Ophthalmic Solution 0.15% is a synthetic docosanoid. Unoprostone isopropyl has the chemical name isopropyl (+)-(Z)-7-[(1R,2R,3R,5S)-3,5 dihydroxy-2-(3-oxodecyl)cyclopentyl]-5-heptenoate. The main indication …

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +12
Waktu ParuhHalf-life of Unopr…
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Upadacitinib Approved DB15091
small molecule | CAS: 1310726-60-3

Upadacitinib is an oral Janus kinase (JAK)1-selective inhibitor and a disease-modifying antirheumatic drug (DMARD) used in the treatment of rheumatoid arthritis to slow down disease progression. Rheumatoid arthritis is a chronic autoimmune inflammatory diseas…

Kategori:
Antineoplastic and Immunomodulating AgentsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +16
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe volume of distr…
KlirensThe apparent oral c…
Genetik -
Upamostat DB13052
small molecule | CAS: 1191101-18-4

Upamostat has been used in trials studying the treatment of Pancreatic Cancer.

Kategori:
AmidesAminesHydroxylamines +3
Target Protein:
Urokinase-type plasminogen activator
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Upanovimab DB16505
biotech | CAS: 2500633-46-3

Upanovimab (SCTA01) was under investigation in clinical trials (NCT04683328, NCT04644185, NCT04709328 and NCT05156645) to evaluate its safety and efficacy in patients with severe COVID-19

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Genetik -
biotech | CAS: 2254119-00-9

Upinitatug rilsodotin is under investigation in clinical trial NCT05329545 (Upifitamab Rilsodotin Maintenance in Platinum-sensitive Recurrent Ovarian Cancer (UP-NEXT)).

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Uprifosbuvir DB15206
small molecule | CAS: 1496551-77-9

Uprifosbuvir is under investigation in clinical trial NCT02332707 (Efficacy and Safety of Grazoprevir (MK-5172) and Uprifosbuvir (MK-3682) With Elbasvir (MK-8742) or Ruzasvir (MK-8408) for Chronic Hepatitis C Genotype (GT)1 and GT2 Infection (MK-3682-011)).

Kategori:
Anti-Infective AgentsAntiviral AgentsNucleic Acids, Nucleotides, and Nucleosides +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Uproleselan DB14829
small molecule | CAS: 1983970-12-2

Uproleselan is a novel, specific E-Selectin antagonist under investigation in clinical trial NCT02306291 (Study to Determine Safety, Pharmacokinetics and Efficacy of GMI-1271 in Combination With Chemotherapy in AML).

Kategori:
CarbohydratesE-Selectin, antagonists & inhibitorsGlycoconjugates +1
Target Protein:
E-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uprosertib DB11969
small molecule | CAS: 1047634-65-0

Uprosertib has been used in trials studying the treatment of Cancer, Melanoma, Solid Tumours, Cervical Cancer, and HER2/Neu Negative, among others.

Kategori:
AminesPolyamines
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Urabrelimab DB17209
biotech | CAS: 2249722-58-3

Deskripsi belum tersedia.

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Genetik -
Uracil DB03419
small molecule | CAS: 66-22-8

Deskripsi belum tersedia.

Kategori:
Fluorouracil and prodrugsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Uridine-cytidine kinase-like 1Uracil-DNA glycosylase +4
Waktu Paruh-
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Genetik -
Uracil C-13 DB16345
small molecule | CAS: 35803-45-3

Uracil C-13 is under investigation in clinical trial NCT01677338 (Phase 2 Study to Evaluate the Preliminary Performance of the C13-URA Breath Test Kit in Dyspeptic Subjects).

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Uracil mustard Approved DB00791
small molecule | CAS: 66-75-1

Nitrogen mustard derivative of uracil. It is a alkylating antineoplastic agent that is used in lymphatic malignancies, and causes mainly gastrointestinal and bone marrow damage.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +10
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Urapidil DB12661
small molecule | CAS: 34661-75-1

Urapidil has been investigated for the treatment of Hypertension During Pre-Eclampsia.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +12
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Urea Approved DB03904
small molecule | CAS: 57-13-6

A compound formed in the liver from ammonia produced by the deamination of amino acids. It is the principal end product of protein catabolism and constitutes about one half of the total urinary solids.

Kategori:
AmidesBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +7
Target Protein:
Dihydrofolate reductaseArginase-1Carbonic anhydrase 2 +2
Waktu Paruh-
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Urea C-13 Approved DB09510
small molecule | CAS: 58069-82-2

Urea 13C is a urea molecule radiolabelled with the non-radioactive element carbon-13. It is currently used for the Urea Breath Test (UBT) and is available as a rapid diagnostic test (marketed as Pranactin-Citric) for the detection of Helicobacter pylori infec…

Kategori:
Diagnostic AgentsHelicobacter pylori Diagnostic
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Urea C-14 Approved DB09513
small molecule | CAS: 594-05-8

Urea 14C is a urea molecule radiolabelled with a radioactive carbon-14. It is currently used for the Urea Breath Test (UBT) and is available as a rapid diagnostic test (marketed as PyTest) for the detection of Helicobacter pylori infections. H pylori is a com…

Kategori:
Radioactive Diagnostic Agent
Waktu Paruh14C-urea that is no…
Vol. Distribusi-
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Urelumab DB12077
biotech | CAS: 934823-49-1

Urelumab has been used in trials studying the treatment of Leukemia, Multiple Myeloma, Malignant Tumors, and Cancer - Solid Tumors and B-Cell Non-Hodgkin's Lymphoma. Urelumab is a fully human antibody that targets CD137. The antibody product was developed usi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Tumor necrosis factor receptor superfamily member 9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Urethane Approved DB04827
small molecule | CAS: 51-79-6

Urethane, formerly marketed as an inactive ingredient in Profenil injection, was determined to be carcinogenic and was removed from the Canadian, US, and UK markets in 1963.

Kategori:
Acids, AcyclicAnestheticsAnesthetics, General +8
Waktu Paruh-
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Uric acid DB08844
small molecule | CAS: 69-93-2

Uric acid is the last product of purine metabolism in humans. The formation of uric acid is through the enzyme xanthine oxidase, which oxidizes oxypurines. Normally a small amount of uric acid is present in the body, but when there is an excess amount in the …

Kategori:
AlkaloidsAntioxidantsBiological Factors +6
Target Protein:
Glycogen phosphorylase, liver form
Waktu Paruh-
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Genetik -
small molecule | CAS: 63-39-8

Uridine 5'-(tetrahydrogen triphosphate). A uracil nucleotide containing three phosphate groups esterified to the sugar moiety.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Target Protein:
P2Y purinoceptor 2P2Y purinoceptor 6P2Y purinoceptor 4 +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 133-89-1

A key intermediate in carbohydrate metabolism. Serves as a precursor of glycogen, can be metabolized into UDPgalactose and UDPglucuronic acid which can then be incorporated into polysaccharides as galactose and glucuronic acid. Also serves as a precursor of s…

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides +8
Target Protein:
Galactose-1-phosphate uridylyltransferaseUDP-glucose 4-epimeraseAlpha,alpha-trehalose-phosphate synthase [UDP-forming] +7
Waktu Paruh-
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Genetik -
small molecule | CAS: 58-97-9

5'-Uridylic acid. A uracil nucleotide containing one phosphate group esterified to the sugar moiety in the 2', 3' or 5' position.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Target Protein:
Thymidylate synthaseUridine-cytidine kinase-like 1Galactose-1-phosphate uridylyltransferase +11
Waktu Paruh-
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Uridine triacetate Approved DB09144
small molecule | CAS: 4105-38-8

Uridine triacetate, formerly known as vistonuridine, is an orally active prodrug of the naturally occurring nucleoside uridine. It is used for the treatment of hereditary orotic aciduria (Xuriden), or for the emergency treatment of fluorouracil or capecitabin…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismFatty Acids +9
Waktu Paruh2 to 2.5 hours
Vol. DistribusiCirculating uridine…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Vanadates
Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 58-98-0

A uracil nucleotide containing a pyrophosphate group esterified to C5 of the sugar moiety. [PubChem]

Target Protein:
UDP-N-acetylglucosamine 2-epimeraseHisto-blood group ABO system transferaseGalactose-1-phosphate uridylyltransferase +13
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Alpha,alpha-trehalose-phosphate synthase [UDP-forming]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-N-acetylmuramoylalanine--D-glutamate ligaseUDP-N-acetylmuramate--L-alanine ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligaseUDP-N-acetylmuramoylalanine--D-glutamate ligase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-N-acetylglucosamine 1-carboxyvinyltransferaseUDP-N-acetylhexosamine pyrophosphorylaseUDP-N-acetylglucosamine 1-carboxyvinyltransferase +6
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
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Urocortin-2 DB13033
biotech | CAS: 351999-18-3

Urocortin 2 has been investigated for the basic science of Heart Failure and Cardiovascular Disease.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +3
Target Protein:
Corticotropin-releasing factor receptor 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Urofollitropin Approved DB00094
biotech | CAS: 97048-13-0

Urofollitropin is a urinary-derived follicle-stimulating hormone (FSH) that is extracted and purified from human urine samples. It consists of two non-covalently linked, non-identical glycoproteins designated as the alpha- and beta- subunits. The alpha- and b…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesGonadotropins +9
Target Protein:
Follicle-stimulating hormone receptor
Waktu ParuhCirculation half li…
Vol. DistribusiTime to peak in pla…
Klirens-
Genetik -
Urokinase Approved DB00013
biotech | CAS: 9039-53-6

Urokinase is an endogenous peptide that is cleaved in the presence of plasmin between lysine 158 and isoleucine 159 to yield active urokinase.[A191943] Urokinase remains connected between these 2 chains by a sulfhydryl bond.[A191943] Urokinase was granted …

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +15
Target Protein:
PlasminogenUrokinase plasminogen activator surface receptorPlasminogen activator inhibitor 1 +5
Waktu ParuhUrokinase has a hal…
Vol. DistribusiThe volume of distr…
KlirensData regarding the …
Genetik -
Urolithin A DB15464
small molecule | CAS: 1143-70-0

Urolithin A is a metabolite of ellagic acid. It has been demonstrated to stimulate mitophagy and improve muscle health in old animals and in preclinical models of aging.[A179494]

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
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Genetik -
Ursadiol DB14555
small molecule | CAS: 37384-13-7

Deskripsi belum tersedia.

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Ursodeoxycholic acid Approved DB01586
small molecule | CAS: 128-13-2

Ursodeoxycholic acid (UDCA), also known as ursodiol, is a naturally-occurring bile acid that constitutes a minor fraction of the human bile acid pool.[A256272,A256277] UDCA has been used to treat liver disease for decades: its first use in traditional medicin…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +15
Target Protein:
Aldo-keto reductase family 1 member C2Biliverdin reductase ASolute carrier family 23 member 2 +1
Waktu ParuhThe estimated half-…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Urtica dioica pollen Approved DB10763
biotech

Urtica dioica pollen is the pollen of the Urtica dioica plant. Urtica dioica pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
Usistapide DB12414
small molecule | CAS: 403989-79-7

Usistapide has been used in trials studying the treatment of Obesity, Overweight, Metabolic Diseases, Nutrition Disorders, and Nutritional and Metabolic Diseases.

Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
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USL-311 DB15265
small molecule | CAS: 1373268-67-7

USL-311 is under investigation in clinical trial NCT02765165 (Phase 1/2 Study of USL311 Alone and in Combination With Lomustine in Subjects With Advanced Solid Tumors and Relapsed/Recurrent Glioblastoma Multiforme (GBM)).

Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Usnea barbata Approved DB14351
biotech

Usnea barbata is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Ustekinumab Approved DB05679
biotech | CAS: 815610-63-0

Ustekinumab is a human immunoglobulin (Ig) G1 kappa monoclonal antibody directed against interleukin(IL)-12 and IL-23, which are cytokines that are involved in immune and inflammatory responses.[A187349] It was generated via recombinant human IL-12 immunizati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Interleukin-23Interleukin-12 subunit beta
Waktu ParuhFollowing administr…
Vol. DistribusiThe total volume of…
KlirensThe median apparent…
Genetik -
Ustilago cynodontis Approved DB10834
biotech

Ustilago cynodontis is a fungus which can provoke allergic reactions. Ustilago cynodontis extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
Ustilago maydis Approved DB10443
biotech

Ustilago maydis is a fungus which can provoke allergic reactions. Ustilago maydis extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Ustilago nuda hordei Approved DB10835
biotech

Ustilago nuda hordei is a fungus which can provoke allergic reactions. Ustilago nuda hordei extract is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +5
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Genetik -
Uteroglobin DB14880
biotech

Uteroglobin is under investigation in clinical trial NCT01473264 (Safety, Pk and Anti-inflammatory Effects of CC10 Protein in Premature Infants With Respiratory Distress Syndrome (RDS)).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsSecretoglobins
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Utomilumab DB15113
biotech | CAS: 1417318-27-4

Utomilumab is under investigation in clinical trial NCT03318900 (T Cell Immunotherapy for Advanced Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Utreloxastat DB18154
small molecule | CAS: 1213269-96-5

Deskripsi belum tersedia.

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Genetik -
Uttroside B DB18633
small molecule | CAS: 88048-09-3

Deskripsi belum tersedia.

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Genetik -
UX053 DB18558
biotech

UX053 is an mRNA encoding the human glycogen debranching enzyme.

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UX701 DB18317
biotech

Deskripsi belum tersedia.

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Menampilkan 12951–13000 dari 13591
Sebelumnya Halaman 260 / 272 Berikutnya