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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 260 / 282
Tidutamab DB18839
biotech | CAS: 2148354-90-7

Tidutamab is under investigation in clinical trial NCT04590781 (Safety and Efficacy of Xmab18087 ± Pembrolizumab in Advanced Merkel Cell Carcinoma or Extensive-stage Small Cell Lung Cancer).

Waktu Paruh-
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small molecule | CAS: 144-12-7

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +4
Waktu Paruh-
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Tienilic acid DB04831
small molecule | CAS: 40180-04-9

Tienilic acid, or ticrynafen, is a diuretic drug with uric acid-lowering action which was marketed for the treatment of hypertension. It was withdrawn in 1982 after case reports in the United States suggested a link between ticrynafen and hepatitis. (Manier e…

Kategori:
AcetatesAcids, AcyclicAntigout Preparations +16
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Tifcemalimab DB18914
biotech | CAS: 2236068-83-8

Tifcemalimab is under investigation in clinical trial NCT06095583 (Phase 3 Study of Toripalimab Alone or in Combination With Tifcemalimab as Consolidation Therapy in Patients With Limited-stage Small Cell Lung Cancer (LS-SCLC)).

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Tifuvirtide DB05413
biotech | CAS: 251562-00-2

Tifuvirtide is the first members of a new class of anti-HIV drugs which is also called fusion inhibitors. It has received fast-track designation from the FDA and is in Phase I/II clinical testing.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Viral +14
Target Protein:
Plasma serine protease inhibitor
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Tigatuzumab DB15101
biotech | CAS: 918127-53-4

Tigatuzumab is under investigation in clinical trial NCT00991796 (CS-1008 With Carboplatin/Paclitaxel in Chemotherapy naïve Subjects With Metastatic or Unresectable Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Tigecycline Approved DB00560
small molecule | CAS: 220620-09-7

Tigecycline is a glycylcycline antibiotic developed and marketed by Wyeth under the brand name Tygacil. It was developed in response to the growing prevalence of antibiotic resistance in bacteria such as Staphylococcus aureus. It was granted fast-track approv…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
16S ribosomal RNA30S ribosomal protein S930S ribosomal protein S12 +3
Waktu Paruh27-43 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 943001-56-7

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
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Tigozertinib DB19239
small molecule | CAS: 2660250-10-0

Tigozertinib (BLU-945) is currently under investigation in clinical trial NCT04862780 (Phase 1/?2 Study Targeting EGFR Resistance Mechanisms in NSCLC) for the treatment of NSCLC.

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Tigulixostat DB18799
small molecule | CAS: 1287766-55-5

Deskripsi belum tersedia.

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TIK-301 DB16909
small molecule | CAS: 118702-11-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Melatonin receptor type 1A
Waktu Paruh-
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Tilactase Approved DB13761
biotech | CAS: 9031-11-2

Tilactase is a beta-D-galactosidase obtained from _Aspergillus oryzae_. It is produced as a chewable tablet that has to be taken before the consumption of a lactose-containing meal.[A27172] The beta-D-galactosidase us a large monomeric multi-domain enzyme of …

Kategori:
Alimentary Tract and MetabolismAntifoaming Agentsbeta-Galactosidase +8
Target Protein:
Lactose
Waktu ParuhTilactase half-life…
Vol. DistribusiTilactase is not ab…
KlirensTilactase is not ab…
Genetik -
Tilarginine Approved DB11815
small molecule | CAS: 17035-90-4

Tilarginine has been investigated for the basic science, treatment, and diagnostic of Obesity, Type 2 Diabetes, Ocular Physiology, and Regional Blood Flow.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +4
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
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Tilavonemab DB17014
biotech | CAS: 2096513-89-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
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Tilbroquinol Approved DB13222
small molecule | CAS: 7175-09-9

Tilbroquinol was approved in France, Morocco, and Saudi Arabia but it has been withdrawn in France and Saudi Arabia markets mainly due to its hepatotoxicity risk outweighing the drug benefit [L5467]. In Morocco, the drug has been limited to use in the treatme…

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
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Tildacerfont DB18545
small molecule | CAS: 1014983-00-6

Tildacerfont is a corticotropin-releasing factor receptor-1 antagonist containing an unfused thiazole ring

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Tildipirosin DB11470
small molecule | CAS: 328898-40-4

Tildipirosin is a veterinary antibiotic.

Kategori:
Anti-Bacterial AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +4
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Tildrakizumab Approved DB14004
biotech | CAS: 1326244-10-3

Tildrakizumab is a high-affinity, humanized, IgG1 ? antibody targeting interleukin 23 p19 that shows promise in the evolution of treatment strategy in chronic plaque psoriasis [A32255]. The Food and Drug Administration (FDA) approved ILUMYA (tildrakizumab-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-23
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe geometric mean …
KlirensThe mean (CV%) syst…
Genetik -
Tilia americana pollen Approved DB10732
biotech

Tilia americana pollen is the pollen of the Tilia americana plant. Tilia americana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Tilmanocept Approved DB15373
small molecule | CAS: 1185986-76-8

Tilmanocept is under investigation in clinical trial NCT03241446 (Pharmacokinetics and Dosimetry of Tc 99m Tilmanocept Following a Single Intravenous Dose Administration in Male and Female Subjects Diagnosed With Rheumatoid Arthritis (RA)).

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Tilorone DB17965
small molecule | CAS: 27591-97-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Inflammatory AgentsAntiinfectives for Systemic Use +7
Waktu Paruh-
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Tilpisertib DB18798
small molecule | CAS: 2065153-41-3

Deskripsi belum tersedia.

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small molecule | CAS: 2567459-64-5

Deskripsi belum tersedia.

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Tilsotolimod DB16341
biotech | CAS: 1948266-37-2

Tilsotolimod is under investigation in clinical trial NCT03865082 (Study of Tilsotolimod in Combination With Nivolumab and Ipilimumab for the Treatment of Solid Tumors (ILLUMINATE-206)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Toll-like receptor 9
Waktu Paruh-
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TILT-123 DB17519
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Tiludronic acid Approved DB01133
small molecule | CAS: 89987-06-4

Tiludronate, or (4-chlorophenyl)thio-methylene-1,1-bisphosphonate, is a first generation bisphosphonate similar to [etidronic acid] and [clodronic acid].[A1923,A203111] These drugs were developed to mimic the action of pyrophosphate, a regulator of calcificat…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +6
Target Protein:
HydroxylapatiteAdenosine triphosphate (ATP)Tyrosine-protein phosphatase non-receptor type 12 +3
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe volume of distr…
KlirensTiludronic acid has…
Genetik -
Timbetasin DB19119
biotech | CAS: 77591-33-4

Timbetasin is under investigation in clinical trial NCT05555589 (Assessment of the Safety and Efficacy of 0.1% RGN-259 Ophthalmic Solution for the Treatment of NK: SEER-2).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +5
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Timcodar DB12761
small molecule | CAS: 179033-51-3

Timcodar has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

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Timdarpacept DB17544
biotech | CAS: 2749520-17-8

IMM01 is a recombinant human signal regulatory protein ? (SIRP?) IgG 1 fusion protein.[A257261] IMM01 is under investigation in clinical trial NCT05140811 (A Study of IMM01 Combined With Azacitidine in Patients With Acute Myeloid Leukemia and Myelodysplastic …

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Timepidium DB13850
small molecule | CAS: 97094-64-9

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Timolol Approved DB00373
small molecule | CAS: 26839-75-8

Timolol is a nonselective beta-adrenergic antagonist given in an eye drop solution to reduce intraocular pressure, or pressure in the eyes.[L6724] It is also used in tablet form as a drug to treat hypertension.[L6727] Timolol was first approved by the FDA in …

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +28
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorEndolysin
Waktu ParuhTimolol half-life w…
Vol. Distribusi1.3 - 1.7 L/kg [L6]…
KlirensOne pharmacokinetic…
Genetik -
Timonacic DB12856
small molecule | CAS: 444-27-9

Timonacic has been used in trials studying the treatment of HIV Infections.

Waktu Paruh-
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biotech | CAS: 1905415-02-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Genetik -
small molecule | CAS: 14325-05-4

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesEnzyme Inhibitors +5
Waktu Paruh-
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Tinengotinib DB17384
small molecule | CAS: 2230490-29-4

Deskripsi belum tersedia.

Waktu Paruh-
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Tinidazole Approved DB00911
small molecule | CAS: 19387-91-8

A nitroimidazole antitrichomonal agent effective against _Trichomonas vaginalis_, _Entamoeba histolytica_, and _Giardia lamblia_ infections.

Kategori:
Alimentary Tract and MetabolismAlkylating DrugsAnti-Bacterial Agents +24
Target Protein:
DNA
Waktu ParuhThe elimination hal…
Vol. Distribusi* 50 L
Klirens-
Genetik -
Tinlarebant DB17832
small molecule | CAS: 1821327-95-0

Deskripsi belum tersedia.

Target Protein:
Retinol-binding protein 4
Waktu Paruh-
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Tinlorafenib DB17082
small molecule | CAS: 2573781-75-4

Tinlorafenib (PF-07284890) is a potent, selective, highly brain-penetrant, small-molecule inhibitor of BRAF V600 mutations.[A253992]

Kategori:
Heterocyclic Compounds, Fused-RingSulfonamides
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Tinodasertib DB18796
small molecule | CAS: 1464151-33-4

Deskripsi belum tersedia.

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Tinoridine DB13001
small molecule | CAS: 24237-54-5

Tinoridine is under investigation in clinical trial NCT01224756 (Efficacy of Tinoridine in Treating Pain and Inflammation in Adults).

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
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Tinostamustine DB15147
small molecule | CAS: 1236199-60-2

Tinostamustine is under investigation in clinical trial NCT03452930 (Tinostamustine With or Without Radiation Therapy in Treating Patients With Newly Diagnosed MGMT-Unmethylated Glioblastoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Tinzaparin Approved DB06822
small molecule | CAS: 9041-08-1

Tinzaparin is a low molecular weight heparin (LMWH), produced by enzymatic depolymerization of unfractionated heparin from porcine intestinal mucosa. It is a heterogeneous mixture of with an average molecular weight between 5500 and 7500 daltons. Tinzaparin i…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIIntegrin alpha-4Stromal cell-derived factor 1
Waktu ParuhAnti-Xa activity is…
Vol. DistribusiAnti-Xa activity is…
KlirensClearance is dose-d…
Genetik -
Tioclomarol DB13451
small molecule | CAS: 22619-35-8

Deskripsi belum tersedia.

Kategori:
AnticoagulantsBenzopyransBlood and Blood Forming Organs +3
Waktu Paruh-
Vol. Distribusi-
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Tioconazole Approved DB01007
small molecule | CAS: 65899-73-2

Tioconazole is an imidazole antifungal used to treat fungal and yeast infections. Topical formulations are used for ringworm, jock itch, athlete's foot, and tinea versicolor or "sun fungus". Tioconazole interacts with 14-alpha demethylase, a cytochrome P-450 …

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +21
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tioguanine Approved DB00352
small molecule | CAS: 154-42-7

An antineoplastic compound which also has antimetabolite action. The drug is used in the therapy of acute leukemia.

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
DNA
Gen Terkait:
TPMT TPMT TPMT +1
Waktu ParuhWhen the compound w…
Vol. Distribusi-
Klirens-
Genetik 4 Varian
Tiopronin Approved DB06823
small molecule | CAS: 1953-02-2

Tiopronin is a prescription thiol drug used primarily in the treatment of severe homozygous cystinuria. Patients with cystinuria excrete high levels of cystine in their urine and are at risk for kidney stone formation. Tiopronin is used as a second-line thera…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +7
Waktu ParuhTiopronin has a lon…
Vol. DistribusiThe volume of distr…
KlirensTotal renal clearan…
Genetik -
Tiotropium Approved DB01409
small molecule | CAS: 186691-13-4

Tiotropium is a long-acting, antimuscarinic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD) and asthma.[A180163,L7084,L7087,L7090,L7093] Tiotropium acts mainly on M3 muscarinic receptors located in the airways to produce …

Kategori:
Adrenergics, InhalantsAgents producing tachycardiaAgents to Treat Airway Disease +22
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe terminal half l…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
Tioxidazole DB11472
small molecule | CAS: 61570-90-9

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Waktu Paruh-
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Genetik -
biotech | CAS: 1052105-48-2

Deskripsi belum tersedia.

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Tipelukast DB12435
small molecule | CAS: 125961-82-2

Tipelukast is under investigation for the treatment of IPF and Idiopathic pulmonary fibrosis.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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