Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (16004)

Halaman 260 / 321
Quisinostat DB12985
small molecule | CAS: 875320-29-9

Quisinostat has been used in trials studying the treatment of Lymphoma, Neoplasms, Myelodysplastic Syndromes, and Advanced or Refractory Leukemia.

Kategori:
AminesHydroxy AcidsHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quisovalimab DB16482
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quisqualic acid DB02999
small molecule | CAS: 52809-07-1

Quisqualic acid is an agonist at two subsets of excitatory amino acid receptors, ionotropic receptors that directly control membrane channels and metabotropic receptors that indirectly mediate calcium mobilization from intracellular stores. The compound is ob…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsExcitatory Amino Acid Agents +4
Target Protein:
Metabotropic glutamate receptor 1Glutamate receptor ionotropic, kainate 1Metabotropic glutamate receptor 2 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quizartinib Approved DB12874
small molecule | CAS: 950769-58-1

Quizartinib is an oral and potent fms-like tyrosine kinase 3 (FLT3) inhibitor and it is the first drug developed specifically targeting FLT3, as other agents with FLT3 inhibition activities were investigated with other targets in mind.[A260641] Additionally, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean (SD) effec…
Vol. DistribusiVolume of distribut…
KlirensTotal body clearanc…
Genetik -
QXL138AM DB18552
biotech

QXL138AM is a masked immunocytokine (MIC) comprised of an anti-CD138 immunoglobulin G1 antibody fused to interferon alpha 2a. It binds the CD138 protein on the surface of the tumour cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 37571-78-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-1487 DB06518
small molecule | CAS: 449811-92-1

Deskripsi belum tersedia.

Kategori:
Mitogen-Activated Protein Kinase 14, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Stromelysin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-30490 DB09179
small molecule | CAS: 60618-49-7

R-30490 is an opioid related to carfentanil used as an animal tranquilizer. It was first synthesized by Janssen Pharmaceutica as part of a structure-activity relationship study of fentanly and its derivatives. R-30490 was found to be the most selective agonis…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-306465 DB12382
small molecule | CAS: 604769-01-9

R306465 has been used in trials studying the treatment of Neoplasms.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-348 DB06321
small molecule | CAS: 916742-11-5

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase JAK3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-82913 DB08598
small molecule | CAS: 126347-69-1

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +7
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-851 DB05747
small molecule

R-851 is part of the family of immune response modifier (IRM) and it acts in a novel way to stimulate the human body's immnune system to attack virus-infected cells and tumor cells. It is expected to be topical treatment for cervical displasia and cervical hi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14047-28-0

Deskripsi belum tersedia.

Target Protein:
Thymidine kinase, cytosolicThymidine kinaseThymidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-95845 DB07327
small molecule | CAS: 163435-77-6

R-95845 is an inhibitor of HIV-1 reverse transcriptase.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-azabisabolene DB03985
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R048-8071 DB02016
small molecule | CAS: 161582-11-2

Deskripsi belum tersedia.

Target Protein:
Lanosterol synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R107474 DB06553
small molecule | CAS: 214548-46-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R112 DB06252
small molecule | CAS: 575474-82-7

R112 is an investigational compound developed to treat Allergic Rhinitis. It's mechanism of action is to inhibit SYK kinase.

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1204 DB05118
small molecule

R1204 is G-protein-coupled receptor modulator. It is developed for the treatment of depression.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R343 DB06316
small molecule | CAS: 575484-78-5

R343, was investigated in clinical trial NCT01591044 to evaluate its safety and efficacy in patients with mild to moderate asthma.

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R3R01 DB18078
small molecule

R3R01 is an investigational lipid-modifying drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R411 DB05468
small molecule

R411 is a non-steroid oral medicine for the treatment of asthma. It is not immunosuppressive, but blocks the activation and recruitment of cells involved in respiratory inflammation. It is a dual-acting competitive integrin antagonist (as compared to previous…

Target Protein:
Integrin alpha-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R450 DB05469
small molecule

R450 is an alpha 1 antagonist that acts to tighten the muscle tone in the bladder. It is being considered for treatment of stress-related urinary incontinence. Phase IIa data for the drug show it reduced the number of incontinent episodes compared to placebo …

Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R673 DB05466
small molecule

R673 is a novel NK1 antagonist that penetrates the blood-brain barrier, has excellent safety and tolerability and shows low P450-based drug interaction potential. The phase II program for treatment of depression and anxiety is ongoing in the US and EU.It is n…

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R906289 DB19126
small molecule | CAS: 2602614-45-7

R906289 is under investigation in clinical trial NCT05308264 (Study of R289 in Participants With Lower-risk Myelodysplastic Syndromes (LR MDS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV1-CB-hAAT DB18724
biotech

rAAV1-CB-hAAT is a recombinant adeno-associated virus alpha 1-antitrypsin vector.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV9-hNAGLU DB18415
biotech

rAAV9-hNAGLU consists of a recombinant AAV9 expressing human alpha-N-acetylglucosaminidase.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV9-rsATP7A DB17664
biotech

A recombinant adeno-associated viral vector gene therapy under investigation for the treatment of Menkes disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rabacfosadine DB12762
small molecule | CAS: 859209-74-8

Rabacfosadine has been used in trials studying the treatment of Multiple Myeloma, Non-Hodgkin's Lymphoma, and Chronic Lymphocytic Leukemia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rabeprazole Approved DB01129
small molecule | CAS: 117976-89-3

Rabeprazole is an antiulcer drug in the class of proton pump inhibitors. It is a prodrug - in the acid environment of the parietal cells it turns into active sulphenamide form. Rabeprazole inhibits the H+, K+ATPase of the coating gastric cells and dose-depend…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcetatesAcid Reducers +47
Target Protein:
Potassium-transporting ATPase alpha chain 1
Waktu Paruh1-2 hours (in plasm…
Vol. Distribusi-
Klirens-
Genetik -
Rabeximod DB05772
small molecule | CAS: 872178-65-9

Rabeximod is an orally administered compound for treatment of moderate or severe active rheumatoid arthritis that is currently undergoing phase II clinical testing in eight European countries.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

IMOGAM Rabies Pasteurized is indicated for post-exposure prophylaxis in persons suspected of exposure to rabies, who have not previously received a complete immunization regimen with a cell culture produced rabies vaccine. Persons previously vaccinated wit…

Kategori:
Human Rabies Immune GlobulinsSerumVaccines
Target Protein:
Rabies Virus Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Rabies virus inactivated antigen, A is an inactivated virus vacine for the intramuscular injection. It is an active immunization against rabies that can be administered pre- or post-exposure to the rabies virus.

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Inactivated rabies virus antigen B is a component of rabies vaccines used for pre- and post-exposure prophylaxis against rabies.[L12795]

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseImmune Sera +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rabusertib DB11662
small molecule | CAS: 911222-45-2

Rabusertib has been used in trials studying the treatment of Cancer, Solid Tumors, Advanced Cancer, Pancreatic Neoplasms, and Non Small Cell Lung Cancer.

Kategori:
AmidesAntineoplastic AgentsBenzene Derivatives +1
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raceanisodamine DB16896
small molecule | CAS: 85760-60-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Racecadotril DB11696
small molecule | CAS: 81110-73-8

Racecadotril has been investigated for the basic science and treatment of Diarrhea, Acute Diarrhea, and Acute Gastroenteritis.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Peptides, and Proteins +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Racemethionine Approved DB13972
small molecule | CAS: 59-51-8

A preparation of methionine that includes a mixture of D-methionine and L-methionine isomers.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Racemetyrosine DB16306
small molecule | CAS: 658-48-0

Racemetyrosine is under investigation in clinical trial NCT03512756 (A Randomized Phase 2/3 Multi-center Study of SM-88 in Patients With Metastatic Pancreatic Cancer).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Racephedrine Approved DB14752
small molecule | CAS: 90-81-3

Deskripsi belum tersedia.

Kategori:
Adrenergic AgonistsAdrenergic alpha-AgonistsAdrenergic beta-Agonists +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Racepinephrine Approved DB11124
small molecule | CAS: 329-65-7

Racepinephrine is a racemic mixture consisting of d-[DB00668] and l-[DB00668] enantiomers. Epinephrine is a non-selective ?- and ?-adrenergic receptor agonist. It is a bronchodilator used in the temporary relief of mild symptoms of intermittent asthma includi…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +30
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-2A adrenergic receptor +6
Waktu ParuhTo refer to the pha…
Vol. DistribusiTo refer to the pha…
KlirensTo refer to the pha…
Genetik -
Racivir DB12753
small molecule | CAS: 143491-54-7

Racivir, also known as RCV, is an oxothiolane nucleoside reverse transcriptase inhibitor similar to emtricitabine and lamivudine. Racivir is a 50:50 mixture of [emtricitabine] and its positive enantiomer. Racivir has been used in trials studying the preventio…

Kategori:
Anti-Infective AgentsAntiviral AgentsDeoxycytidine +5
Target Protein:
Reverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raclopride DB12518
small molecule | CAS: 84225-95-6

Raclopride has been used in trials studying Parkinson Disease.

Kategori:
Acids, CarbocyclicAmidesAntipsychotic Agents +13
Target Protein:
Insulin receptorD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Racotumomab DB13045
biotech | CAS: 946832-34-4

Racotumomab has been used in trials studying the treatment of Glioma, Wilm's Tumor, Neuroblastoma, Retinoblastoma, and Ewing's Sarcoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RAD 502 DB17328
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RAD-140 DB13939
small molecule | CAS: 1182367-47-0

RAD140 is an investigational selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and breast cancer.

Kategori:
Oxazoles
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Radafaxine DB11790
small molecule | CAS: 192374-14-4

Radafaxine has been used in trials studying the treatment of Depressive Disorder, Major.

Kategori:
KetonesPropiophenones
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Radalbuvir DB12065
small molecule | CAS: 1314795-11-3

Radalbuvir has been used in trials studying the treatment of Chronic Hepatitis C, Chronic HCV Infection, and Chronic Hepatitis C Infection.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Radavirsen DB15332
biotech | CAS: 1228284-45-4

Radavirsen is under investigation in clinical trial NCT01375985 (Safety Study of Single Administration Intravenous Treatment for Influenza).

Kategori:
Anti-Infective AgentsAntiviral AgentsMorpholines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12951–13000 dari 16004
Sebelumnya Halaman 260 / 321 Berikutnya