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1977

Total database: 17430
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1074 (54.3%)
Target
1046 (52.9%)
Genomik
39 (2.0%)
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1977 (100.0%)

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Hasil Pencarian (1977)

Halaman 26 / 40
Nurulimab DB18946
biotech | CAS: 2168561-20-2

Nurulimab is under investigation in clinical trial NCT05732805 (A Clinical Study of BCD-217 (Nurulimab + Prolgolimab) Followed by Anti-pd-1 Compared to Anti-pd-1 Monotherapy as First-line Treatment in Subjects With Unresectable/metastatic Melanoma).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nusinersen Approved DB13161
small molecule | CAS: 1258984-36-9

An antisense oligonucleotide that induces survival motor neuron (SMN) protein expression, it was approved by the U.S. FDA in December, 2016 as Spinraza for the treatment of children and adults with spinal muscular atrophy (SMA). It is adminstrated as direct i…

Kategori:
Antisense OligonucleotidesIncreased Protein SynthesisMusculo-Skeletal System +4
Target Protein:
Survival motor neuron protein
Waktu ParuhThe mean terminal e…
Vol. DistribusiCSF: 0.4 L Plasma…
KlirensSlow clearance is o…
Genetik -
Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-5138 DB19180
small molecule | CAS: 2095886-80-7

NV-5138 is under investigation in clinical trial NCT06235905 (Open-label of SPN-820 in Adults With Major Depressive Disorder).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nylidrin Approved DB06152
small molecule | CAS: 447-41-6

Nylidrin, also known as _buphenine_ belongs to the category of drugs called _vasodilators_, which relax blood vessels and increase blood flow. Nylidrin is a peripheral vasodilator. Some studies show the evidence of improving cognitive impairment in selected i…

Kategori:
2-Amino-1-Phenylethanol DerivativesAdrenergic AgentsAdrenergic Agonists +29
Target Protein:
Interferon alpha/beta receptor 2Voltage-dependent T-type calcium channel subunit alpha-1I
Waktu ParuhDuration of action …
Vol. Distribusi-
Klirens-
Genetik -
NYX-2925 DB19149
small molecule | CAS: 2012536-16-0

NYX-2925 is under investigation in clinical trial NCT04146896 (Efficacy and Safety of NYX-2925 in Subjects With Neuropathic Pain Associated With Diabetic Peripheral Neuropathy (DPN)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obeticholic acid Approved DB05990
small molecule | CAS: 459789-99-2

Primary biliary cirrhosis, or PBC, is a progressive and chronic condition that leads to hepatic injury often resulting in end-stage liver failure that requires liver transplantation.[A192786] Obeticholic acid is a farnesoid-X receptor (FXR) agonist used to…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +14
Target Protein:
Bile acid receptor
Waktu ParuhThe biological half…
Vol. DistribusiThe volume of distr…
KlirensClearance informati…
Genetik -
OBI-999 DB17356
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obicetrapib DB14890
small molecule | CAS: 866399-87-3

Obicetrapib is under investigation in clinical trial NCT02241772 (A Study on the Effects of TA-8995 on Lp(a) in Subjects With Elevated Lp(a)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Cholesteryl ester transfer protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ocrelizumab Approved DB11988
biotech | CAS: 637334-45-3

Ocrelizumab is a CD20-directed cytolytic antibody indicated for the treatment of patients with primary progressive or relapsing forms of multiple sclerosis (MS).[L42895] It is a second-generation recombinant humanized monoclonal IgG1 antibody that selectively…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe terminal elimin…
Vol. DistribusiIn a population pha…
KlirensThe constant cleara…
Genetik -
Octocrylene Approved DB09535
small molecule | CAS: 6197-30-4

Octocrylene is a compound often used as an additive in sun screen, and is thought to have skin moisturizing effects because of its emollient properties. What makes this chemical such a popular additive to sun block, is its ability to neutralize UV radiation d…

Kategori:
Acids, AcyclicSunscreen Agents
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Octovalent O-polysaccharide-toxin A conjugate vaccine is currently being investigated to treat Pseudomonas Aeruginosa infection in patients with cystic fibrosis.[A259462]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Octreotide Approved DB00104
biotech | CAS: 83150-76-9

Acromegaly is a disorder caused by excess growth hormone (GH), increasing the growth of body tissues and causing metabolic dysfunction.[L14501] In most cases, it results from an anterior pituitary growth hormone-releasing tumor. Typically, the feet, hands, an…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Hormonal +19
Target Protein:
Somatostatin receptor type 2Somatostatin receptor
Waktu ParuhAfter a subcutaneou…
Vol. DistribusiIn a pharmacokineti…
KlirensThe total body clea…
Genetik -
Odevixibat Approved DB16261
small molecule | CAS: 501692-44-0

Odevixibat, or A4250, is an ileal sodium/bile acid cotransporter inhibitor indicated for the treatment of pruritus in patients older than 3 months, with progressive familial intrahepatic cholestasis (PFIC).[A236808,L34793] Odevixibat is the first approved non…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBenzazepines +9
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu ParuhA 7.2 mg oral dose …
Vol. DistribusiThe majority of adu…
KlirensThe majority of adu…
Genetik -
Ofatumumab Approved DB06650
biotech | CAS: 679818-59-8

Ofatumumab is a novel anti-CD20 monoclonal antibody that targets B-cells. It is an IgG1? human monoclonal antibody produced from a recombinant murine cell line (NS0) via transgenic mouse and hybridoma technology.[L12612] Ofatumumab works by recognizing antige…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhIn patients with CL…
Vol. DistribusiIn patients with CL…
KlirensIn patients with CL…
Genetik -
biotech | CAS: 1476737-24-2

Ofranergene obadenovec is under investigation in clinical trial NCT01229865 (Safety and Efficacy of VB-111 in Subjects With Advanced Differentiated Thyroid Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olacaftor DB16262
small molecule | CAS: 1897384-89-2

Olacaftor is under investigation in clinical trial NCT02951182 (A Study Evaluating the Safety and Efficacy of VX-440 Combination Therapy in Subjects With Cystic Fibrosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olendalizumab DB14834
biotech | CAS: 1337966-73-0

Olendalizumab is under investigation in clinical trial NCT01883544 (Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of ALXN1007 in Healthy Male and Female Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olipudase alfa Approved DB12835
biotech | CAS: 927883-84-9

Olipudase alfa is recombinant human acid sphingomyelinase.[A251590] It is the first and only enzyme replacement therapy in the world for the treatment of Acid Sphingomyelinase Deficiency (ASMD), also known as Niemann–Pick disease.[L42740] ASMD is a rare lysos…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzyme Replacement Therapy +7
Waktu ParuhAfter administratio…
Vol. DistribusiAfter administratio…
KlirensAfter administratio…
Genetik -
Olopatadine Approved DB00768
small molecule | CAS: 113806-05-6

Olopatadine is a selective histamine H1 antagonist and mast cell stabilizer that works by attenuating inflammatory and allergic reactions. It is a structural analog of [doxepin], which has a minimal anti-allergic activity.[L6790] Olopatadine works by blocking…

Kategori:
Anti-Allergic AgentsAnti-Inflammatory AgentsAntiallergic Agents, Excl. Corticosteroids +23
Target Protein:
Histamine H1 receptorHistamine H2 receptorHistamine H3 receptor +5
Waktu ParuhFollowing ocular ad…
Vol. DistribusiIn an open-label st…
KlirensIn an open-label st…
Genetik -
Olorinab DB14998
small molecule | CAS: 1268881-20-4

Olorinab is under investigation in clinical trial NCT03155945 (Tolerability, Pharmacokinetics, and Efficacy of APD371 in Subjects With Crohn's Disease Experiencing Abdominal Pain).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olorofim DB15245
small molecule | CAS: 1928707-56-5

Olorofim is under investigation in clinical trial NCT03340597 (Assessment of Varying Oral Dosing Regimens for F901318 in Healthy Subjects).

Kategori:
AcetatesAcids, AcyclicAmides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olsalazine Approved DB01250
small molecule | CAS: 15722-48-2

Olsalazine is an aminosalicylate and a prodrug of [mesalamine] (5-aminosalicylic acid, 5-ASA).[A257063] It was first developed for delivering mesalamine to the colon without the use of [sulfapyridine].[A257078] Olsalazine comprises two mesalamine molecules jo…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Human CyclooxygenasesThiopurine S-methyltransferaseXanthine dehydrogenase/oxidase
Waktu ParuhOlsalazine has a ve…
Vol. DistribusiThe steady-state vo…
Klirens-
Genetik -
Ombitasvir Approved DB09296
small molecule | CAS: 1258226-87-7

Ombitasvir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
AmidesAminesAmino Acids +18
Target Protein:
Nonstructural protein 5AGenome polyprotein
Waktu ParuhOmbitasvir has a ha…
Vol. DistribusiOmbitasvir has a vo…
KlirensClearance of Ombita…
Genetik -
small molecule

Omega-6 fatty acids are polyunsaturated fatty acids with a final carbon-carbon double bond in the n-6 position, that is, the sixth bond, counting from the methyl end. They are a family of fatty acid molecules that act as precursors to potent lipid mediator si…

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omidenepag isopropyl Approved DB15071
small molecule | CAS: 1187451-19-9

Omidenepag isopropyl is a topical ocular hypotensive agent used to reduce intraocular pressure (IOP) in patients with glaucoma and ocular hypertension.[L43503] Omidenepag isopropyl is quickly metabolized to its active metabolite, omidenepag, a molecule with h…

Kategori:
Antiglaucoma AgentsHypotensive AgentsOphthalmic Solutions +6
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype
Waktu ParuhThe half-life of om…
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
OMS-103HP DB05303
small molecule

OMS103HP is the first drug being developed to improve joint function following arthroscopic surgery, one of the most common procedures performed today by orthopedic surgeons.

Kategori:
Acids, CarbocyclicBenzocycloheptenesDibenzocycloheptenes +3
Target Protein:
Tumor necrosis factorInterleukin-1 receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ondansetron Approved DB00904
small molecule | CAS: 99614-02-5

A competitive serotonin type 3 receptor antagonist. It is effective in the treatment of nausea and vomiting caused by cytotoxic chemotherapy drugs, including cisplatin, and has reported anxiolytic and neuroleptic properties. Having been developed in the 19…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +29
Target Protein:
5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 4Mu-type opioid receptor +2
Gen Terkait:
CYP2D6 CYP2D6
Waktu ParuhThe half-life of on…
Vol. DistribusiThe volume of distr…
KlirensThe clearance value…
Genetik 2 Varian
Onfekafusp alfa DB16269
biotech | CAS: 1957239-88-1

Onfekafusp alfa is under investigation in clinical trial NCT02938299 (Neoadjuvant L19IL2/L19TNF- Pivotal Study).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ongericimab DB18949
biotech | CAS: 2145096-91-7

Ongericimab is under investigation in clinical trial NCT05325203 (A Study to Evaluate the Efficacy and Safety of JS002 in Patients With Heterozygous Familial Hypercholesterolemia (Hefh).).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONO-2952 DB14802
small molecule | CAS: 895169-20-7

ONO-2952 is under investigation in clinical trial NCT01887002 (Study to Evaluate the Effects of ONO-2952 on Pain Perception Produced by Rectal Distention in Female Subjects With Diarrhea-Predominant Irritable Bowel Syndrome (IBS-D)).

Kategori:
CycloparaffinsHeterocyclic Compounds, Fused-Ring
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1620643-19-7

Onvitrelin ucalontide is under investigation in clinical trial NCT01485848 (EP-100 Plus Paclitaxel Versus Paclitaxel Alone in Patients With Ovarian Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OPC1 DB17944
biotech

OPC1 is an oligodendrocyte progenitor cell therapy being investigated for the treatment of acute spinal cord injury.[L47082]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opicapone Approved DB11632
small molecule | CAS: 923287-50-7

Opicapone is a potent, reversible, and peripherally-acting third-generation inhibitor of catechol-o-methyltransferase (COMT), an enzyme involved in the breakdown of various catecholamines including dopamine.[A36938, A203048] Many patients with Parkinson’s dis…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBCRP/ABCG2 Substrates +25
Target Protein:
Catechol O-methyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing oral admi…
KlirensFollowing oral admi…
Genetik -
Opicinumab DB14959
biotech | CAS: 1422268-07-2

Opicinumab is under investigation in clinical trial NCT02641041 (Safety, Tolerability, and Pharmacokinetics of Single and Multiple Doses of BIIB033 in Healthy Japanese Participants).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opiranserin DB16271
small molecule | CAS: 1441000-45-8

Opiranserin is under investigation in clinical trial NCT03997838 (Evaluate the Efficacy and Safety of VVZ-149 Injections for the Treatment of Post-operative Pain Following Abdominoplasty).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orilanolimab DB15312
biotech | CAS: 2066544-85-0

Orilanolimab is under investigation in clinical trial NCT03075878 (A Safety Study of SYNT001 in Subjects With Chronic, Stable Warm Autoimmune Hemolytic Anemia (WAIHA)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orthosiphon aristatus leaf Approved DB15838
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orticumab DB16653
biotech | CAS: 1314241-10-5

Orticumab is under investigation in clinical trial NCT04776629 (A Proof-of-activity Study With Orticumab in Subjects With Psoriasis and Cardiometabolic Risk Factors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Vol. Distribusi-
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Genetik -
Orvepitant DB12427
small molecule | CAS: 579475-18-6

Orvepitant has been used in trials studying the treatment of Depressive Disorder, Depressive Disorder, Major, Post-Traumatic Stress Disorder, and Posttraumatic Stress Disorder (PTSD).

Kategori:
Antidepressive AgentsCentral Nervous System Depressants
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-7904L DB05457
small molecule

OSI-7904L is a liposome encapsulated thymidylate synthase inhibitor, which is indicated for use in advanced gastric and/or gastroesophageal adenocarcinoma (A-G/GEJA). Current treatments also inhibit thymidylate synthase but the innovative lipid coating of OSI…

Kategori:
Acids, AcyclicDicarboxylic AcidsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osilodrostat Approved DB11837
small molecule | CAS: 928134-65-0

Osilodrostat is an inhibitor of 11?-hydroxylase (also referred to as CYP11B1), the enzyme that catalyzes the final step in the biosynthesis of endogenous cortisol.[L12123] It is used to lower circulating cortisol levels in the treatment of Cushing's disease, …

Kategori:
Antiadrenal PreparationsAnticorticosteroidsCortisol Synthesis Inhibitors +32
Target Protein:
Cytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial
Waktu ParuhThe elimination hal…
Vol. DistribusiThe median apparent…
KlirensData regarding the …
Genetik -
Oteracil Approved DB03209
small molecule | CAS: 937-13-3

Oteracil is an adjunct to antineoplastic therapy, used to reduce the toxic side effects associated with chemotherapy. Approved by the European Medicines Agency (EMA) in March 2011, Oteracil is available in combination with [DB09257] and [DB09256] within the c…

Kategori:
Triazines
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Oxaliplatin Approved DB00526
small molecule | CAS: 61825-94-3

Oxaliplatin is a platinum-based chemotherapy drug in the same family as cisplatin and carboplatin. Compared to cisplatin the two amine groups are replaced by diamino cyclohexane (DACH) group to provide a greater antitumor effect.[A797] However, this leads to …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +9
Target Protein:
DNA
Waktu ParuhThe decline of ultr…
Vol. DistribusiAfter a single 2-ho…
KlirensPlatinum was cleare…
Genetik -
Oxaprozin Approved DB00991
small molecule | CAS: 21256-18-8

Oxaprozin is a non-narcotic, non-steroidal anti-inflammatory drug (NSAID), used to relieve the inflammation, swelling, stiffness, and joint pain associated with osteoarthritis and rheumatoid arthritis.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +22
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh54.9 hours
Vol. Distribusi* 11 to 17 L/70 kg
Klirens-
Genetik -
Oxcarbazepine Approved DB00776
small molecule | CAS: 28721-07-5

Oxcarbazepine is an anti-epileptic medication used in the treatment of partial onset seizures that was first approved for use in the United States in 2000.[L8627,L8630,L8633] It is a structural derivative of [carbamazepine][A186101] and exerts a majority of i…

Kategori:
Anti-epileptic AgentAnticonvulsantsCarboxamide Derivatives +29
Target Protein:
Sodium channel protein type 11 subunit alphaSodium channel protein
Gen Terkait:
HLA-B
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensPlasma clearance of…
Genetik 1 Varian
Oxiconazole Approved DB00239
small molecule | CAS: 64211-45-6

Oxiconazole is an antifungal agent that is commonly found in topical formulations. It is marketed under the brand names Oxistat and Oxistat, and is used in the treatment of various skin infections such as athlete's foot, jock itch and ringworm.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +13
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol synthaseNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxitriptan Approved DB02959
small molecule | CAS: 4350-09-8

5-Hydroxytryptophan (5-HTP), also known as oxitriptan (INN), is a naturally occurring amino acid and metabolic intermediate in the synthesis of serotonin and melatonin. 5-HTP is sold over-the-counter in the United Kingdom, United States and Canada as a dietar…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +8
Target Protein:
Tryptophan--tRNA ligase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1251–1300 dari 1977
Sebelumnya Halaman 26 / 40 Berikutnya