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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 26 / 66
Fluoride ion Approved DB11257
small molecule | CAS: 16984-48-8

Having a chemical formula of F?, fluoride ion is the simplest inorganic, monatomic anion of fluorine with basic properties. It is considered a trace element. Fluoride ions are found in various minerals but are only present in trace amounts in water. Its vario…

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Fluorodopa (18F) Approved DB13848
small molecule | CAS: 92812-82-3

Fluorodopa F 18 is a fluorinated analog of [levodopa] used as a diagnostic agent for positron emission tomography (PET) in the evaluation of Parkinsonian syndromes.[L12849] Fluorodopa F 18 PET is used adjunctly with other diagnostic investigations and serves …

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +8
Waktu ParuhThe plasma half-lif…
Vol. Distribusi-
KlirensThe agent is cleare…
Genetik -
Fluoroestradiol F-18 Approved DB15690
small molecule | CAS: 94153-53-4

Fluoroestradiol F-18 is an imaging agent used with positron emission tomography (PET) to detect estrogen receptor-positive breast cancer lesions.[L14096] The ability to image ER-positive tumors _in vivo_ is advantageous in that, while helping to visualize tum…

Kategori:
Estradiol CongenersEstranesEstrogens +10
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. DistribusiAs fluoroestradiol …
KlirensFluoroestradiol F-1…
Genetik -
small molecule | CAS: 1255-35-2

Fluprednidene acetate is a corticosteroid. It has anti-inflammatory and anti-allergic properties.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Inducers +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flurbiprofen Approved DB00712
small molecule | CAS: 5104-49-4

Flurbiprofen, a propionic acid derivative, is a nonsteroidal anti-inflammatory agent (NSAIA) with antipyretic and analgesic activity. Oral formulations of flurbiprofen may be used for the symptomatic treatment of rheumatoid arthritis, osteoarthritis and ankly…

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +37
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhR-flurbiprofen, 4.7…
Vol. Distribusi* 14 L [Normal Heal…
Klirens-
Genetik -
small molecule | CAS: 1211333-21-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 1274863-98-7

Flutriciclamide F-18 is under investigation in clinical trial NCT02350426 (A Study to Assess Inflammation in Rheumatoid Arthritis Using Molecular Imaging Techniques).

Waktu Paruh-
Vol. Distribusi-
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Fomepizole Approved DB01213
small molecule | CAS: 7554-65-6

Fomepizole is used as an antidote in confirmed or suspected methanol or ethylene glycol poisoning. Fomepizole is a competitive inhibitor of alcohol dehydrogenase, the enzyme that catalyzes the initial steps in the metabolism of ethylene glycol and methanol to…

Kategori:
AntidotesCompounds used in a research, industrial, or household settingCytochrome P-450 CYP2A6 Inhibitors +13
Target Protein:
Alcohol dehydrogenase 1AAll-trans-retinol dehydrogenase [NAD(+)] ADH1BAlcohol dehydrogenase 1C +1
Waktu ParuhThe plasma half-lif…
Vol. Distribusi* 0.6 to 1.02 L/kg
Klirens-
Genetik -
Fonadelpar DB16169
small molecule | CAS: 515138-06-4

Fonadelpar is under investigation in clinical trial NCT03527212 (A Study to Assess the Safety and Effectiveness of SJP-0035 for the Treatment of Patients With Dry Eye Disease).

Waktu Paruh-
Vol. Distribusi-
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Foralumab DB16170
biotech | CAS: 946415-64-1

Foralumab is under investigation in clinical trial NCT03291249 (Assessment of the Safety of Foralumab, an Oral Anti-cd3 Antibody, in Patients With NASH and T2DM).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foretinib DB12307
small molecule | CAS: 849217-64-7

Foretinib has been used in trials studying the treatment of Cancer, Breast Cancer, Carcinoma, Renal Cell, Recurrent Breast Cancer, and Neoplasms, Head and Neck, among others. Foretinib is an orally available small molecule compound designed to target multiple…

Kategori:
AmidesAminesAniline Compounds +3
Target Protein:
Hepatocyte growth factor receptorVascular endothelial growth factor receptor 2Hepatocyte growth factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Forigerimod DB12490
biotech | CAS: 497156-60-2

Forigerimod is under investigation for the treatment of Lupus Erythematosus, Systemic.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesRibonucleoprotein, U1 Small Nuclear
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formoterol Approved DB00983
small molecule | CAS: 73573-87-2

Formoterol is an inhaled beta<sub>2</sub>-agonist used in the management of COPD and asthma that was first approved for use in the United States in 2001.[L10986] It acts on bronchial smooth muscle to dilate and relax airways, and is administered as a racemic …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +29
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe average termina…
Vol. Distribusi-
KlirensRenal clearance of …
Genetik -
Formycin DB02281
small molecule | CAS: 6742-12-7

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
S-methyl-5'-thioadenosine phosphorylase5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosbretabulin DB12577
small molecule | CAS: 222030-63-9

Fosbretabulin has been investigated for the treatment of Anaplastic Thyroid Cancer.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosdagrocorat DB12198
small molecule | CAS: 1044535-58-1

Fosdagrocorat has been used in trials studying the treatment and basic science of Rheumatoid Arthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foslinanib DB16172
small molecule | CAS: 1256037-60-1

Foslinanib is under investigation in clinical trial NCT03600233 (Study of CVM-1118 for Patients With Advanced Neuroendocrine Tumors).

Waktu Paruh-
Vol. Distribusi-
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Fosravuconazole DB15204
small molecule | CAS: 351227-64-0

Fosravuconazole is under investigation in clinical trial NCT03378661 (BENDITA BEnznidazole New Doses Improved Treatment and Associations).

Kategori:
Antifungals for Dermatological UseAntifungals for Systemic UseDermatologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Fostamatinib Approved DB12010
small molecule | CAS: 901119-35-5

Fostamatinib has been investigated for the treatment and basic science of Rheumatoid Arthritis and Immune Thrombocytopenic Purpura (ITP). It was approved on April 17, 2018, under the trade name Tavalisse for use in ITP [L2644, FDA Label]. Fostamatinib has als…

Kategori:
AminesBCRP/ABCG2 InhibitorsBlood and Blood Forming Organs +17
Target Protein:
Tyrosine-protein kinase SYKAdenosine receptor A3Synaptic vesicular amine transporter +297
Waktu ParuhR406 has a half-lif…
Vol. DistribusiR406 has an apparen…
KlirensR406 has an apparen…
Genetik -
Fostemsavir Approved DB11796
small molecule | CAS: 864953-29-7

Fostemsavir is the phosphonooxymethyl prodrug of temsavir, a novel HIV-1 attachment inhibitor.[L14867] It binds to and inhibits the activity of gp120, a subunit within the HIV-1 gp160 envelope glycoprotein that facilitates the attachment of HIV-1 to host cell…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +18
Target Protein:
Envelope glycoprotein gp160
Waktu ParuhThe half-life of te…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 2129993-56-0

Deskripsi belum tersedia.

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small molecule | CAS: 141790-23-0

Fozivudine Tidoxil has been used in trials studying the treatment of HIV Infections.

Kategori:
DeoxyribonucleosidesDideoxynucleosidesNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fresolimumab DB12396
biotech | CAS: 948564-73-6

Fresolimumab has been used in trials studying the treatment of Primary Brain Tumors, Metastatic Breast Cancer, Diffuse Systemic Sclerosis, Pleural Malignant Mesothelioma, and Primary Focal Segmental Glomerulosclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
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Froniglutide DB16178
biotech | CAS: 1417579-81-7

Glymera is under investigation in clinical trial NCT01658501 (Phase 2b Multicenter, Randomized, Double-blind, Placebo- and Active-controlled, Parallel-group Study to Assess the PD Response and Safety of Three Dose Levels of (PB1023) Injection Following 20 Wee…

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Fulranumab DB12102
biotech | CAS: 902141-80-4

Fulranumab has been used in trials studying the treatment of Pain, Cystitis, Neuralgia, Joint Pain, and Arthralgia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fulvestrant Approved DB00947
small molecule | CAS: 129453-61-8

Fulvestrant is a drug treatment of hormone receptor (HR)-positive metastatic breast cancer in post-menopausal women with disease progression following anti-estrogen therapy. It is an estrogen receptor antagonist with no agonist effects, which works both by do…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +20
Target Protein:
Estrogen receptor
Waktu Paruh40 days
Vol. Distribusi* 3 to 5 L/kg
Klirens-
Genetik -
Funapide DB11769
small molecule | CAS: 1259933-16-8

Funapide has been used in trials studying the treatment of Pharmacokinetics, Postherpetic Neuralgia, and Osteoarthritis of the Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Sodium channel protein type 9 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprevir DB12785
small molecule | CAS: 1435923-88-8

Furaprevir is under investigation in clinical trial NCT01523990 (A Study to Evaluate the Safety, Tolerability, and PK in Healthy Volunteers and HCV Genotype 1 Infected Patients).

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazabol DB01514
small molecule | CAS: 1239-29-8

Deskripsi belum tersedia.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Waktu Paruh-
Vol. Distribusi-
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Gabexate DB12831
small molecule | CAS: 39492-01-8

Gabexate is a synthetic serine protease inhibitor which has been used as an anticoagulant. It also known to decrease production of inflammatory cytokines. Gabexate has been investigated for use in cancer, ischemia-reperfusion injury, and pancreatitis.[A19218,…

Kategori:
AmidinesAnticoagulantsEnzyme Inhibitors +4
Target Protein:
Plasma kallikreinProthrombinPlasminogen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gadolinium Approved DB12091
small molecule | CAS: 7440-54-2

Gadolinium is under investigation in Hypertension, ACUTE KIDNEY INJURY, and Chronic Kidney Disease. Gadolinium has been investigated for the basic science of CAD, Multiple Sclerosis, and Coronary Artery Disease.

Kategori:
Anti-Inflammatory AgentsCompounds used in a research, industrial, or household settingContrast Media +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gadoteric acid Approved DB09132
small molecule | CAS: 72573-82-1

Gadoteric acid, commonly used in the salt form gadoterate meglumine, is a macrocyclic, ionic gadolinium-based contrast agent (GBCA).[A263131] It is composed of the organic acid DOTA (1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid) used for its chel…

Kategori:
AlcoholsAmino SugarsCarbohydrates +12
Waktu ParuhFollowing an intrav…
Vol. DistribusiThe volume of distr…
KlirensIn healthy subjects…
Genetik -
Gadoteridol Approved DB00597
small molecule | CAS: 120066-54-8

Gadoteridol is a macrocyclic nonionic gadolinium that provides contrast enhancement of the brain, spine, and surrounding tissues, resulting in improved visualization (compared with unenhanced MRI) of lesions with abnormal vascularity or those thought to disru…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe plasma distribu…
KlirensThe renal and plasm…
Genetik -
Galcanezumab Approved DB14042
biotech | CAS: 1578199-75-3

Galcanezumab is a humanized monoclonal antibody developed by Eli Lilly and Company against human calcitonin gene-related peptide (CGRP).[A33105] Although several small-molecule CGRP receptor antagonists have been developed, humanized monoclonal antibodies lik…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +15
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhBetween 1 and 600 m…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Galeterone DB12415
small molecule | CAS: 851983-85-2

Galeterone has been used in trials studying the treatment of Prostate Cancer.

Kategori:
AndrostanesAndrostenesEnzyme Inhibitors +4
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Galidesivir DB11676
small molecule | CAS: 249503-25-1

Galidesivir is an adenosine analogue that has been investigated for use against Zaire Ebolavirus.[A191451] In animal studies, galidesivir was effective in increasing the survival rates from infections caused by various pathogens, including Ebola, Marburg, Yel…

Kategori:
Anti-Infective AgentsAntiviral AgentsCarbohydrates +9
Target Protein:
RNA-directed RNA polymerase L
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gallium chloride Ga-67 Approved DB14550
small molecule

Gallium chloride Ga-67 is the chloride salt of a gallium radioisotope which is typically complexed with [sodium citrate] to generate [gallium citrate Ga 67], which can be used to image certain cancers and inflammatory lesions.[L12705]

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Gallopamil DB12923
small molecule | CAS: 16662-47-8

Gallopamil has been used in trials studying the treatment of Asthma.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +17
Target Protein:
Sarcoplasmic/endoplasmic reticulum calcium ATPase 2Angiotensin-converting enzymeNeprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Galsulfase Approved DB01279
biotech | CAS: 552858-79-4

Galsufase is a variant form of the polymorphic human enzyme N-acetylgalactosamine 4-sulfatase of recombinant DNA origin. Galsulfase is a glycoprotein with a molecular weight of approximately 56 kD. The recombinant protein is comprised of 495 amino acids and c…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsArylsulfatases +9
Target Protein:
Dermatan sulfate
Waktu Paruh9 (6 to 21) minutes…
Vol. DistribusiWeek 1: 56-323 mL/k…
Klirens-
Genetik -
gamma-Aminobutyric acid Approved DB02530
small molecule | CAS: 56-12-2

The most common inhibitory neurotransmitter in the central nervous system.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +4
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-2Sodium- and chloride-dependent GABA transporter 3Integrin alpha-4 +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gamolenic acid Approved DB13854
small molecule | CAS: 506-26-3

Gamolenic acid, or gamma-linolenic acid (?-Linolenic acid) or GLA, is an essential fatty acid (EFA) comprised of 18 carbon atoms with three double bonds [F27] that is most commonly found in human milk and other botanical sources [A32848]. It is an omega-6 pol…

Kategori:
Agents that reduce seizure thresholdDermatologicalsFatty Acids +5
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Ganaplacide DB16173
small molecule | CAS: 1261113-96-5

Ganaplacide is under investigation in clinical trial NCT03167242 (Efficacy and Safety of KAF156 in Combination With LUM-SDF in Adults and Children With Uncomplicated Plasmodium Falciparum Malaria).

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Gandotinib DB13040
small molecule | CAS: 1229236-86-5

Gandotinib has been used in trials studying the treatment of Myelofibrosis, Polycythemia Vera, Primary Myelofibrosis, Thrombocythemia, Essential, and Myeloproliferative Disorders, among others.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganetespib DB12047
small molecule | CAS: 888216-25-9

Ganetespib is under investigation for the treatment of BREAST CANCER, Small Cell Lung Cancer, Acute Myeloid Leukaemia, and Myelodysplastic Syndrome.

Kategori:
HSP90 Heat-Shock Proteins, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganirelix Approved DB06785
small molecule | CAS: 124904-93-4

Ganirelix is a synthetic decapeptide and a competitive gonadotropin-releasing hormone (GnRH) antagonist. Derived from endogenous GnRH, ganirelix has amino acid substitutions. Ganirelix is indicated for controlled ovarian hyperstimulation in assisted reproduct…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Gonadotropin-Releasing HormonesDecreased GnRH Secretion +16
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean (SD) volum…
KlirensClearance following…
Genetik -
Ganitumab DB12205
biotech | CAS: 905703-97-1

Ganitumab has been used in trials studying the treatment of Colon Cancer, Rectal Cancer, Breast Cancer, Breast Tumors, and Breast Neoplasms, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gantenerumab DB12034
biotech | CAS: 1043556-46-2

Alzheimer's disease (AD) is the most common cause of dementia in elderly patients, with classical histopathological hallmarks including extracellular amyloid-beta (A?) plaques and intraneuronal neurofibrillary tangles (NFTs). As the classical view of AD patho…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhGantenerumab admini…
Vol. Distribusi-
Klirens-
Genetik -
Garadacimab DB15629
biotech | CAS: 2162134-62-3

Garadacimab is under investigation in clinical trial NCT04281524 (A Clinical Study to Test the Efficacy and Safety of CSL312 on Catheter-associated Blood Clot Formation in Subjects With Cancer Who Receive Chemotherapy Through a PICC Line).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garetosmab DB16379
biotech | CAS: 2097125-54-5

Fibrodysplasia ossificans progressiva (FOP) is a rare autosomal dominant disorder of episodic, progressive heterotropic ossification. FOP is characterized by episodic inflammatory episodes, which may be precipitated by trauma, including immunizations and mino…

Target Protein:
Inhibin beta A chain
Waktu Paruh-
Vol. DistribusiGaretosmab had a st…
KlirensWhen administered a…
Genetik -
Gastric intrinsic factor Approved DB09349
biotech

Intrinsic factor (IF), also known as gastric intrinsic factor (GIF), is a glycoprotein produced by the parietal cells of the stomach that is necessary for the absorption of vitamin B12 (cobalamin) later on in the small intestine. When vitamin B12 is provided …

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1251–1300 dari 3253
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