Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 258 / 282
TG01 vaccine DB17123
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG100-115 DB05552
small molecule | CAS: 677297-51-7

An NSAID that inhibits PI-3K gamma and delta.

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG1024 DB06180
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG4010 DB06584
biotech | CAS: 350485-85-7

A bivalent cancer vaccine comprised of a modified vaccinia virus Ankara (MVA) strain encoding human mucin 1 (MUC1) and interleukin-2 (IL-2) with potential immunostimulating and antineoplastic activities. Originally developed for the eradication of smallpox, M…

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsCarbohydrates +6
Target Protein:
Mucin-1Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG4023 DB06108
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TGAAC09 DB06363
biotech

tgAAC09 is an investigational vaccine that utilizes an AAV vector to deliver genes that encode HIV proteins. It was under investigation in clinical trials NCT00482027 and NCT00888446 for the treatment of HIV Infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TGAAC94 DB06175
small molecule

tgAAC94 is a recombinant adeno-associated virus serotype 2 (AAV2) vector containing the cDNA for a human tumor necrosis factor receptor (TNFR)-immunoglobulin (IgG1) Fc fusion (TNFR:Fc) gene. It was under investigation in clinical trials to treat Inflammatory …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
tgAAG-76 DB18421
biotech

tgAAG-76 consists of a recombinant adeno-associated virus (serotype 2) (rAAV2) gene transfer agent expressing RPE65.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
tgAAVCF DB17849
biotech

tgAAVCF is an adeno-associated virus (AAV) vector encoding the human cystic fibrosis transmembrane conductance regulator protein (CFTR) cDNA. It is being investigated for the treatment of cystic fibrosis.[A259821, A259826]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1373958-68-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingXanthenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TH0318 DB05145
biotech

TH0318 is a stabilized analogue of human GLP-1 (glucagon-like peptide-1) under investigation for the treatment of type 2 diabetes.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thalidomide Approved DB01041
small molecule | CAS: 50-35-1

A piperidinyl isoindole originally introduced as a non-barbiturate hypnotic, thalidomide was withdrawn from the market due to teratogenic effects. It has been reintroduced and used for a number of inflammatory disorders and cancers. Thalidomide displays immun…

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +38
Target Protein:
Tumor necrosis factorProtein cereblonDNA +1
Waktu ParuhThe half-life of th…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Thallium Tl-201 DB15361
small molecule | CAS: 15064-65-0

Thallium Tl-201 is under investigation in clinical trial NCT02697760 (The CZT Dynamic Myocardial Perfusion Imaging).

Kategori:
IsotopesRadioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thallous chloride Approved DB09316
small molecule | CAS: 7791-12-0

Thallous chloride (also known as Thallium(I) chloride) is a colourless solid intermediate in the isolation of thallium from its ores. It is created from the treatment of thallium(I) sulfate with hydrochloric acid. This solid crystallizes in the caesium chlori…

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh91% of the blood ra…
Vol. Distribusi3–10 L/kg
KlirensApproximately 4-8% …
Genetik -
Thallous chloride Tl-201 Approved DB16624
small molecule | CAS: 55172-29-7

Deskripsi belum tersedia.

Kategori:
Diagnostic Radiopharmaceuticals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theanine DB12444
small molecule | CAS: 3081-61-6

Theanine, a precursor of ethylamine, is found in green tea. It is under investigation in clinical trial NCT00291070 (Effects of L-Theanine in Boys With ADHD).

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thenalidine Approved DB04826
small molecule | CAS: 86-12-4

Withdrawn from the Canadian, US, and UK markets in 1963 due to concerns involving neutropenia.

Kategori:
Antihistamines for Systemic UseAntihistamines for Topical UseAntipruritics, Incl. Antihistamines, Anesthetics, Etc. +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 326-91-0

Thenoyltrifluoroacetone is a chelating agent and inhibitor of cellular respiration.

Kategori:
ButanonesChelating AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
Liver carboxylesterase 1Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thenyldiamine Approved DB16022
small molecule | CAS: 91-79-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theobromine DB01412
small molecule | CAS: 83-67-0

Theobromine (3,7-dimethylxanthine) is the principle alkaloid in Theobroma cacao (the cacao bean) and other plants. A xanthine alkaloid that is used as a bronchodilator and as a vasodilator. It has a weaker diuretic activity than theophylline and is also a les…

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +15
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theodrenaline DB12927
small molecule | CAS: 13460-98-5

Theodrenaline is under investigation in clinical trial NCT01311414 (Effect of Cafedrine/Theodrenaline and Urapidil on Cerebral Oxygenation).

Kategori:
Adrenergic and Dopaminergic AgentsAgents that produce hypertensionAlcohols +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theophylline Approved DB00277
small molecule | CAS: 58-55-9

A methylxanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant activities. Mechanistically, theophylline acts as a phosphodiesterase inhibitor, adenosine receptor blocker, and histo…

Kategori:
Agents that reduce seizure thresholdAlkaloidsAnti-Asthmatic Agents +32
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +12
Gen Terkait:
CYP1A2
Waktu Paruh8 hours
Vol. Distribusi* 0.3 to 0.7 L/kg
Klirens* 0.29 mL/kg/min [P…
Genetik 1 Varian
Theralizumab DB15717
biotech | CAS: 906068-56-2

Theralizumab is a humanized anti-CD28 monoclonal antibody designed for treating autoimmune diseases and cancer. After the first human trial, it was withdrawn due to severe toxicity (likely due to lymphopenia and human cytokine release).[A216527,A216532]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiabendazole Approved DB00730
small molecule | CAS: 148-79-8

2-Substituted benzimidazole first introduced in 1962. It is active against a variety of nematodes and is the drug of choice for strongyloidiasis. It has CNS side effects and hepatototoxic potential. (From Smith and Reynard, Textbook of Pharmacology, 1992, p91…

Kategori:
AnthelminticsAnti-Infective AgentsAntifungals for Dermatological Use +18
Target Protein:
Fumarate reductase flavoprotein subunit
Waktu ParuhThe half-life for t…
Vol. Distribusi-
Klirens-
Genetik -
Thiacloprid DB08620
small molecule | CAS: 111988-49-9

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +3
Target Protein:
CHRNA7-FAM7A fusion protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamine Approved DB00152
small molecule | CAS: 70-16-6

Thiamine or thiamin, also known as vitamin B1, is a colorless compound with the chemical formula C12H17N4OS. It is soluble in water and insoluble in alcohol. Thiamine decomposes if heated. Thiamine was first discovered by Umetaro Suzuki in Japan when research…

Kategori:
Alimentary Tract and MetabolismDiet, Food, and NutritionFood +10
Target Protein:
Thiamine pyrophosphokinase 1Pyruvate dehydrogenase E1 component
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10023-48-0

Deskripsi belum tersedia.

Target Protein:
Thiamine-phosphate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamphenicol DB08621
small molecule | CAS: 15318-45-3

Deskripsi belum tersedia.

Kategori:
AlcoholsAmphenicolsAnti-Bacterial Agents +8
Target Protein:
Dr hemagglutinin structural subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamylal Approved DB01154
small molecule | CAS: 77-27-0

A barbiturate that is administered intravenously for the production of complete anesthesia of short duration, for the induction of general anesthesia, or for inducing a hypnotic state. (From Martindale, The Extra Pharmacopoeia, 30th ed, p919)

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +22
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3ATP-sensitive inward rectifier potassium channel 8ATP-sensitive inward rectifier potassium channel 11 +1
Waktu ParuhAlthough no studies…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Arsenate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiazinam DB13420
small molecule | CAS: 2338-21-8

Deskripsi belum tersedia.

Kategori:
AminesAntihistamines for Systemic UseAntipsychotic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activatorSerine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thienylfentanyl DB09180
small molecule | CAS: 1165-22-6

Thienylfentanyl is a fentanyl analog analgesic that was sold on the black market in the 1980s until the Federal Analog Act scheduled drugs based on structural similarity rather than scheduling drugs individually. Thienylfentanyl has a similar synthesis pathwa…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiethylperazine Approved DB00372
small molecule | CAS: 1420-55-9

A dopamine antagonist that is particularly useful in treating the nausea and vomiting associated with anesthesia, mildly emetic cancer chemotherapy agents, radiation therapy, and toxins. This piperazine phenothiazine does not prevent vertigo or motion sicknes…

Kategori:
AntiemeticsAntihistamines for Systemic UseAntipsychotic Agents +16
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thimerosal Approved DB11590
small molecule | CAS: 54-64-8

Thiomersal (INN), commonly known in the U.S. as thimerosal, is an organomercury compound. This compound is a well-established and widely used antiseptic and antifungal agent. Developed in 1927, thimerosal has been and is still being used as a preservative…

Kategori:
Alkylmercury CompoundsAntiseptics and DisinfectantsCell-mediated Immunity +11
Target Protein:
Methionine synthaseCystine/glutamate transporterSodium/potassium-transporting ATPase subunit gamma
Waktu ParuhA study was done to…
Vol. Distribusi266 L in one study …
KlirensThe high concentrat…
Genetik -
Thiocamphor DB02851
small molecule | CAS: 7519-74-6

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBornanesBridged-Ring Compounds +4
Target Protein:
Camphor 5-monooxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiocellobiose DB03263
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 602-41-5

Thiocolchicoside is a semi-synthetic derivative of the colchicine, a natural anti-inflammatory glycoside which originates from the flower seeds of _Superba gloriosa_. It is a muscle relaxant with anti-inflammatory and analgesic effects. It has potent convul…

Kategori:
AlkaloidsCentral Nervous System DepressantsMuscle Relaxants +2
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Glycine receptor subunit alpha-2 +6
Waktu ParuhApproximately 7.7h …
Vol. DistribusiThe apparent volume…
KlirensPrimarily extrarena…
Genetik -
Thiocoumarin DB02462
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thioctamide DB15963
small molecule | CAS: 940-69-2

Deskripsi belum tersedia.

Kategori:
CoenzymesEnzymes and CoenzymesFatty Acids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 137314-40-0

A salt of alpha-lipoic acid and tromethamine; may be useful in treating vascular stress in patients with diabetes.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 68-11-1

Thioglycolic acid is under investigation in clinical trial NCT03238105 (Treatment of Periorbicular Hyperchromia Comparing 10% Thioglycolic Acid Peeling Versus Pulsed Intense Light).

Kategori:
AcetatesAcids, AcyclicSulfhydryl Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiohexam Approved DB14200
small molecule | CAS: 95-33-0

Thiohexam is a rubber cure accelerator. It is also a known allergen and dermatological sensitizer. Sensitivity to Thiohexam may be identified with a clinical patch test.

Kategori:
Cell-mediated ImmunityHeterocyclic Compounds, Fused-RingIncreased Histamine Release +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiopental Approved DB00599
small molecule | CAS: 76-75-5

A barbiturate that is administered intravenously for the induction of general anesthesia or for the production of complete anesthesia of short duration. It is also used for hypnosis and for the control of convulsive states. It has been used in neurosurgical p…

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +27
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +9
Waktu Paruh3-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thioproperazine DB01622
small molecule | CAS: 316-81-4

Thioproperazine is a potent neuroleptic with antipsychotic properties. Thioproperazine has a marked cataleptic and antiapomorphine activity associated with relatively slight sedative, hypothermic and spasmolytic effects. It is virtually without antiserotonin …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +18
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12851–12900 dari 14063
Sebelumnya Halaman 258 / 282 Berikutnya