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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (13591)

Halaman 257 / 272
small molecule | CAS: 2453-03-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethyllysine DB03977
small molecule | CAS: 19253-88-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Calmodulin-2Calmodulin-1Calmodulin-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10182-92-0

Deskripsi belum tersedia.

Kategori:
AminesCompounds used in a research, industrial, or household settingDetergents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetrexate Approved DB01157
small molecule | CAS: 52128-35-5

A nonclassical folic acid inhibitor through its inhibition of the enzyme dihydrofolate reductase. It is being tested for efficacy as an antineoplastic agent and as an antiparasitic agent against pneumocystis pneumonia in AIDS patients. Myelosuppression is its…

Kategori:
Acids, AcyclicAcids, AldehydicAnti-Infective Agents +18
Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh11 to 20 hours
Vol. Distribusi* 20 ± 8 L/m2 * 36…
Klirens* 38 +/- 15 mL/min/…
Genetik -
Trimipramine Approved DB00726
small molecule | CAS: 739-71-9

Tricyclic antidepressant similar to imipramine, but with more antihistaminic and sedative properties.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +44
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +15
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +5
Waktu Paruh11-18 hrs
Vol. Distribusi-
Klirens-
Genetik 8 Varian
Trinitrotoluene DB01676
small molecule | CAS: 118-96-7

Trinitrotoluene is an explosive chemical that can cause skin irritation and other toxic consequences.

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingExplosive Agents
Target Protein:
Pentaerythritol tetranitrate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trioxsalen Approved DB04571
small molecule | CAS: 3902-71-4

Trioxsalen (trimethylpsoralen, trioxysalen or trisoralen) is a furanocoumarin and a psoralen derivative obtained from several plants, mainly Psoralea corylifolia. Like other psoralens it causes photosensitization of the skin. It is administered either topical…

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +11
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tripamide DB15959
small molecule | CAS: 73803-48-2

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingMembrane Transport Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triphendiol DB06588
small molecule | CAS: 1213777-80-0

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10380-08-2

Used as water softener, peptizing agent, emulsifier & dispersing agent; ingredient of cleansers; meat preservative.

Kategori:
AcidsAcids, NoncarboxylicAnions +5
Target Protein:
Poly(A) polymerase alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triprolidine Approved DB00427
small molecule | CAS: 486-12-4

First generation histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria. It is a component of cough and cold medicines. It may cause drowsiness.

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +7
Target Protein:
Histamine H1 receptor
Waktu Paruh4 to 6 hours.
Vol. Distribusi-
Klirens-
Genetik -
Triptolide DB12025
small molecule | CAS: 38748-32-2

Triptolide has been used in trials studying the treatment of HIV, Crohn's Disease, Intestinal Diseases, Gastrointestinal Diseases, and Digestive System Diseases, among others.

Kategori:
Adrenal Cortex HormonesAlkylating DrugsAntineoplastic Agents +10
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triptorelin Approved DB06825
small molecule | CAS: 57773-63-4

Triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH). Possessing greater potency than endogenous LHRH, triptorelin reversibly represses gonadotropin secretion. After chronic, continuous administration, this age…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +23
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiAfter a single IV d…
KlirensIn healthy male vol…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Chlorocatechol 1,2-dioxygenaseAlpha-lytic protease
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
AzurinThiazole tautomerasePantothenate synthetase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trisaccharide A DB17689
small molecule | CAS: 49777-13-1

Deskripsi belum tersedia.

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trisaccharide B DB17690
small molecule | CAS: 49777-14-2

Deskripsi belum tersedia.

Kategori:
ABO Blood-Group SystemCarbohydratesOligosaccharides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tritoqualine Approved DB13711
small molecule | CAS: 14504-73-5

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UseCholagogues and CholereticsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRK-001 DB18577
biotech

TRK-001 is an autologous regulatory T-cell therapy. It is being investigated for the prevention of graft rejection following solid organ transplantation.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRO40303 DB16031
small molecule | CAS: 14291-24-8

TRO40303 is under investigation in clinical trial NCT01374321 (Safety and Efficacy Study of TRO40303 for Reduction of Reperfusion Injury in Patients Undergoing Percutaneous Coronary Intervention for Acute Myocardial Infarction).

Kategori:
AminesFused-Ring CompoundsHydroxylamines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trodusquemine DB06333
small molecule | CAS: 186139-09-3

Trodusquemine, a spermine metabolite of cholesterol, is a naturally occurring aminosterol that inhibits protein tyrosine phosphatase 1B. It has demonstrated the ability to stimulate regeneration of heart and multiple other tissues in animal models [A176600].

Kategori:
AminesBiogenic AminesBiogenic Polyamines +3
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trofinetide Approved DB06045
small molecule | CAS: 853400-76-7

Trofinetide is a novel synthetic analog of [glypromate], also known as glycine–proline–glutamate (GPE), a naturally occurring protein in the brain and the N-terminal tripeptide of insulin-like growth factor 1 (IGF-1).[A258438] Trofinetide was approved by the …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +11
Waktu ParuhThe effective elimi…
Vol. DistribusiFollowing oral admi…
KlirensNo information is a…
Genetik -
Troglitazone Approved DB00197
small molecule | CAS: 97322-87-7

Troglitazone was withdrawn in 2000 due to risk of hepatotoxicity. It was superseded by [pioglitazone] and [rosiglitazone].

Kategori:
Alimentary Tract and MetabolismBenzopyransBlood Glucose Lowering Agents +38
Target Protein:
Peroxisome proliferator-activated receptor gammaEstrogen-related receptor gammaSteroid hormone receptor ERR1 +6
Waktu Paruh16-34 hours
Vol. Distribusi-
Klirens-
Genetik -
Trolamine Approved DB13747
small molecule | CAS: 102-71-6

Trolamine, which is also referred to as triethanolamine (TEA), is a tertiary amine and a triol. It is a bifunctional compound that exhibits both properties of alcohols and amines. Trolamine contains small amounts of diethanolamine and ethanolamine and may als…

Kategori:
AlcoholsAminesAmino Alcohols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Various ear diseases and infections are treated with eardrops containing triethanolamine polypeptide oleate-condensate, such as Cerumenex in the United States and Canada.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trolamine salicylate Approved DB11079
small molecule | CAS: 2174-16-5

Trolamine salicylate is an organic compound or a salt formed between triethanolamine and salicylic acid. Triethanolamine neutralizes the acidity of the salicylic acid. It is a topical analgesic used for temporary relief of minor pain associated with arthritis…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnti-Inflammatory Agents +11
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. DistribusiTopical administrat…
Klirens-
Genetik -
Troleandomycin Approved DB13179
small molecule | CAS: 2751-09-9

A macrolide antibiotic that is similar to erythromycin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +18
Target Protein:
50S ribosomal protein L3250S ribosomal protein L4Nuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trolnitrate DB13719
small molecule | CAS: 7077-34-1

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tromantadine Approved DB13288
small molecule | CAS: 53783-83-8

Tromantadine is marketed as Viru-Merz in the Czech Republic [L5740]. It is an antiviral used in the treatment of herpes zoster and simplex.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tromethamine Approved DB03754
small molecule | CAS: 77-86-1

An organic amine proton acceptor. It is used in the synthesis of surface-active agents and pharmaceuticals; as an emulsifying agent for cosmetic creams and lotions, mineral oil and paraffin wax emulsions, as a biological buffer, and used as an alkalizer. (Fro…

Kategori:
AlcoholsBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +12
Target Protein:
S-adenosylmethionine decarboxylase proenzymeAmyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropatepine DB13252
small molecule | CAS: 27574-24-9

Tropatepine has been used in France for its antiparkinsons activities [A175024].

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropicamide Approved DB00809
small molecule | CAS: 1508-75-4

Tropicamide is an alkaloid atropine?derived anticholinergic drug and a non?selective antagonist of muscarinic acetylcholine (mACh) receptors.[A230103] Usually available in ophthalmic formulations, tropicamide is used to cause mydriasis and cycloplegia for eye…

Kategori:
Anticholinergic AgentsAutonomic AgentsCholinergic Agents +8
Target Protein:
Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhTropicamide has a p…
Vol. DistribusiNo information can …
KlirensNo information can …
Genetik -
Tropifexor DB16343
small molecule | CAS: 1383816-29-2

Tropifexor is under investigation in clinical trial NCT02516605 (A Multi-part, Double Blind Study to Assess Safety, Tolerability and Efficacy of Tropifexor (LJN452) in PBC Patients).

Kategori:
Heterocyclic Compounds, Fused-RingThiazoles
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropinone DB01874
small molecule | CAS: 532-24-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropisetron Approved DB11699
small molecule | CAS: 89565-68-4

Tropisetron is an indole derivative with antiemetic activity. As a selective serotonin receptor antagonist, tropisetron competitively blocks the action of serotonin at 5HT3 receptors, resulting in suppression of chemotherapy- and radiotherapy-induced nausea a…

Kategori:
Alimentary Tract and MetabolismAntiarrhythmic agentsAntidepressive Agents +14
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh5.7 h.
Vol. Distribusi400-600 L.
Klirens1800 ml/min.
Genetik -
biotech | CAS: 931101-84-7

Troplasminogen alfa is under investigation in clinical trial NCT00144014 (Safety and Efficacy Study in Acute Ischaemic Stroke).

Kategori:
Amino Acids, Peptides, and ProteinsBeta-GlobulinsBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troriluzole DB15079
small molecule | CAS: 1926203-09-9

Troriluzole is under investigation in clinical trial NCT03701399 (Troriluzole in Adult Subjects With Spinocerebellar Ataxia).

Kategori:
Nervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trospium Approved DB00209
small molecule | CAS: 47608-32-2

Trospium is an antispasmodic agent used to treat the symptoms of overactive bladder, a condition that causes the bladder muscles to contract uncontrollably.[L6208] An overactive bladder leads to an increased urge to urinate, frequent urination, and sometimes,…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +22
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu ParuhThe half-life of tr…
Vol. DistribusiThe volume of distr…
KlirensThe total apparent …
Genetik -
Trotabresib DB17421
small molecule | CAS: 1706738-98-8

Trotabresib is an oral, potent, and reversible inhibitor of the epigenetic target bromodomain and extra-terminal (BET) proteins.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troxerutin DB13124
small molecule | CAS: 7085-55-4

Troxerutin has been used in trials studying the treatment of Chronic Venous Insufficiency.

Kategori:
AnticoagulantsBenzopyransCapillary Stabilizing Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troxipide DB13419
small molecule | CAS: 30751-05-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRV-120027 DB12199
small molecule | CAS: 1234510-46-3

TRV120027 has been used in trials studying the treatment of Heart Failure and Kidney Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
AmicyaninMethylamine dehydrogenase heavy chainMethylamine dehydrogenase light chain +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-518 DB17534
biotech | CAS: 1427683-53-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-E-002-1 DB17264
small molecule | CAS: 1803036-93-2

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX1 DB05863
biotech

TRX1 is a humanized antibody that binds to the CD4 receptor found on a subset of T cells. TRX1 is being developed for the potential treatment of autoimmune diseases in collaboration with Genentech, Inc. TolerRx is currently conducting a Phase I clinical study…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypan blue free acid Approved DB09158
small molecule | CAS: 2538-83-2

Trypan blue is a diazo dye used in ophthalmic cataract surgery to stain the anterior capsule in the presence of a mature cataract. This is done to aid in visualization before creating the continuous curvilinear capsulorhexis.

Kategori:
ArylsulfonatesArylsulfonic AcidsAzo Compounds +12
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypanothione DB03470
small molecule

Deskripsi belum tersedia.

Kategori:
AminesAmino Acids, Peptides, and ProteinsBiogenic Amines +5
Target Protein:
Trypanothione reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypsin Approved DB11237
small molecule | CAS: 9002-07-7

Trypsin is a serine protease that plays an essential role in protein hydrolysis and absorption in mammals. When converted from its zymogen trypsinogen, trypsin is available as an active peptide hydrolase (EC 3.4.21.4) form to cleave peptide chains, mainly at …

Kategori:
Blood and Blood Forming OrgansDermatologicalsEndopeptidases +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tryptamine DB08653
small molecule | CAS: 61-54-1

Deskripsi belum tersedia.

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Target Protein:
Amine oxidase [flavin-containing] B5-hydroxytryptamine receptor 2AAmine oxidase [flavin-containing] A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12801–12850 dari 13591
Sebelumnya Halaman 257 / 272 Berikutnya