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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 256 / 282
Tenofovir alafenamide Approved DB09299
small molecule | CAS: 379270-37-8

Tenofovir alafenamide is a novel [tenofovir] prodrug developed in order to improve renal safety when compared to the counterpart [tenofovir disoproxil].[A178060] Both of these prodrugs were first created to cover the polar phosphonic acid group on tenofovir b…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntiinfectives for Systemic Use +25
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyproteinReverse transcriptase +1
Waktu ParuhThe reported half-l…
Vol. DistribusiIn clinical trials,…
KlirensThe reported cleara…
Genetik -
small molecule | CAS: 1571076-26-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tenofovir disoproxil Approved DB00300
small molecule | CAS: 201341-05-1

Tenofovir disoproxil fumarate (a prodrug of tenofovir), marketed by Gilead Sciences under the trade name _Viread_, belongs to a class of antiretroviral drugs known as nucleotide analogue reverse transcriptase inhibitors (nRTIs). This drug is prescribed in co…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +19
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHProtein P
Waktu ParuhWhen a single oral …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of te…
Genetik -
small molecule | CAS: 911208-73-6

Tenofovir exalidex is under investigation in clinical trial NCT01080820 (A Safety, Tolerability and Pharmacokinetic Study of a Single Dose of CMX157 in Healthy Volunteers).

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1208229-58-6

Deskripsi belum tersedia.

Target Protein:
Nuclear factor NF-kappa-B p105 subunitTranscription factor RelBNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teplizumab Approved DB06606
biotech | CAS: 876387-05-2

Teplizumab (teplizumab-mzwv) is a humanized IgG1 kappa CD3-directed monoclonal antibody used to delay the onset of type 1 diabetes (T1D).[A241480,A241045,A241475,L44091] T1D is an autoimmune condition in which T cell-mediated destruction of pancreatic ? cells…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhIn a 60 kg subject,…
Vol. DistribusiIn a 60 kg subject,…
KlirensIn a 60 kg subject,…
Genetik -
Tepotinib Approved DB15133
small molecule | CAS: 1100598-32-0

Tepotinib is a MET tyrosine kinase inhibitor intended to treat a variety of MET-overexpressing solid tumors.[A228058] It was originally developed in partnership between EMD Serono and the University of Texas M.D. Anderson Cancer Center in 2009 and has since b…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +23
Target Protein:
Hepatocyte growth factor receptorNischarinMelatonin receptor type 1B
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe mean apparent v…
KlirensThe apparent cleara…
Genetik -
Teprasiran DB15064
biotech | CAS: 1231737-88-4

Teprasiran is under investigation in clinical trial NCT03510897 (QPI-1002 Phase 3 for Prevention of Major Adverse Kidney Events (MAKE) in Subjects at High Risk for AKI Following Cardiac Surgery).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teprenone DB15955
small molecule | CAS: 6809-52-5

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsDrugs for Acid Related Disorders +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teprotumumab Approved DB06343
biotech | CAS: 1036734-93-6

Teprotumumab is a fully human IgG1 monoclonal antibody directed against the human insulin-like growth factor-1 receptor.[L11359] Following a clinical trial in which its efficacy in the treatment of thyroid eye disease (TED) was assessed, it received "breakthr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Insulin-like growth factor 1 receptor
Waktu ParuhThe half-life of te…
Vol. DistribusiFollowing the stand…
KlirensThe estimated mean …
Genetik -
Terameprocol DB12226
small molecule | CAS: 24150-24-1

Terameprocol has been investigated for the treatment of Brain and Central Nervous System Tumors.

Kategori:
Benzene DerivativesBenzyl CompoundsCatechols +2
Target Protein:
Transcription factor Sp1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terazosin Approved DB01162
small molecule | CAS: 63590-64-7

Terazosin is a quinazoline derivative alpha-1-selective adrenergic blocking agent indicated for benign prostatic hyperplasia and hypertension[FDA Label][A176831]. Terazosin blocks adrenaline's action on alpha-1 adrenergic receptors, causing relaxation of smoo…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +14
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +4
Waktu ParuhTerazosin has a mea…
Vol. Distribusi25L to 30L[A176831].
KlirensPlasma clearance is…
Genetik -
Terbinafine Approved DB00857
small molecule | CAS: 91161-71-6

Terbinafine hydrochloride (Lamisil) is a synthetic allylamine antifungal.[L9065,L9068] It is highly lipophilic in nature and tends to accumulate in skin, nails, and fatty tissues.[A1279] Like other allylamines, terbinafine inhibits ergosterol synthesis by inh…

Kategori:
Agents Causing Muscle ToxicityAllylamine AntifungalAllylamines +24
Target Protein:
Squalene monooxygenaseSqualene monooxygenase
Waktu ParuhOral terbinafine ha…
Vol. DistribusiA single 250mg oral…
KlirensA single 250mg oral…
Genetik -
Terbogrel DB12204
small molecule | CAS: 149979-74-8

Terbogrel has been used in trials studying the treatment of Hypertension, Pulmonary.

Target Protein:
Thromboxane A2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terbutaline Approved DB00871
small molecule | CAS: 23031-25-6

Terbutaline was first synthesized in 1966[A230333] and described in the literature in the late 1960s and early 1970s.[A230328] It is a selective beta-2 adrenergic agonist used as a bronchodilator in asthmatic patients.[A230333,L32093,L32098] Terbutaline wa…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +26
Target Protein:
Beta-2 adrenergic receptorBeta-3 adrenergic receptorBeta-1 adrenergic receptor
Waktu ParuhAn oral dose of ter…
Vol. DistribusiTerbutaline has a m…
KlirensThe average clearan…
Genetik -
Terbutryn DB08215
small molecule | CAS: 886-50-0

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingHerbicides +2
Target Protein:
Photosynthetic reaction center cytochrome c subunitReaction center protein H chainReaction center protein L chain +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terconazole Approved DB00251
small molecule | CAS: 67915-31-5

Terconazole is an anti-fungal drug that is mainly used to treat vaginal yeast infections (or vaginal candidiasis). It is classified as a _triazole ketal derivative_.[A178096] Terconazole was initially approved by the FDA in 1987.[FDA label] This drug is avail…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungal Agents (Vaginal) +4
Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh6.9 hours (range 4.…
Vol. Distribusi-
Klirens-
Genetik -
Terevalefim DB16397
small molecule | CAS: 1070881-42-3

Terevalefim is under investigation in clinical trial NCT02474667 (Reduce the Severity of DGF in Recipients of a Deceased Donor Kidney).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terfenadine Approved DB00342
small molecule | CAS: 50679-08-8

In the U.S., Terfenadine was superseded by fexofenadine in the 1990s due to the risk of cardiac arrhythmia caused by QT interval prolongation.

Kategori:
Anticholinergic AgentsAntihistamines for Systemic UseBenzene Derivatives +31
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1 +4
Waktu Paruh3.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Teriflunomide Approved DB08880
small molecule | CAS: 163451-81-8

Teriflunomide is the active metabolite of leflunomide, and it acts as an immunomodulatory agent by inhibiting pyrimidine synthesis. It is marketed under the name Aubagio® and is indicated for the treatment of multiple sclerosis, specifically relapsing forms. …

Kategori:
Acids, AcyclicAminesAnalgesics +32
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial3-hydroxy-3-methylglutaryl-coenzyme A reductaseDihydroorotate dehydrogenase (quinone), mitochondrial
Waktu ParuhThe median half-lif…
Vol. DistribusiAfter a single intr…
KlirensAfter a single IV d…
Genetik -
Teriparatide Approved DB06285
biotech | CAS: 52232-67-4

Teriparatide is a recombinant parathyroid hormone (PTH) analog and a potent osteoanabolic agent.[A251395] It is made up of the first amino(N)-terminal 34 amino acids of the human PTH.[A251395] First approved in the United States in November 2002 and in Europe…

Kategori:
Amino Acids, Peptides, and ProteinsBone Anabolic AgentsBone Density Conservation Agents +10
Target Protein:
Parathyroid hormoneParathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe half-life of te…
Vol. DistribusiThe volume of distr…
KlirensSystemic clearance …
Genetik -
Terizidone Approved DB12954
small molecule | CAS: 25683-71-0

Terizidone has been used in trials studying the treatment of Tuberculosis, HIV Infections, Multidrug Resistant Tuberculosis, and Extensively-drug Resistant Tuberculosis.

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsDrugs for Treatment of Tuberculosis +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terlipressin Approved DB02638
biotech | CAS: 14636-12-5

Terlipressin is a synthetic analogue of vasopressin, which is an endogenous neurohormone that acts as a vasoconstrictor.[A2601] It is a prodrug of [lypressin], or lysine vasopressin. Compared to endogenous vasopressin, terlipressin has a longer half life and …

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsHormones +18
Target Protein:
Vasopressin V1a receptorVasopressin V1b receptorVasopressin V2 receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of te…
Genetik -
TERN-101 DB16045
small molecule | CAS: 1103500-20-4

TERN-101 is under investigation in clinical trial NCT04328077 (LIFT Study: A Safety, Tolerability, Efficacy, and Pharmacokinetics Study of TERN-101 in Subjects With Non-cirrhotic Non-alcoholic Steatohepatitis (NASH)).

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terodiline DB13725
small molecule | CAS: 15793-40-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAlkanesAmines +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teropavimab DB18916
biotech | CAS: 2417213-72-8

Teropavimab is under investigation in clinical trial NCT05729568 (A Study of GS-5423 and GS-2872 in Combination With Capsid Inhibitor Lenacapavir in Virologically Suppressed Adults With HIV-1 Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terpin hydrate Approved DB13163
small molecule | CAS: 2451-01-6

Terpin hydrate is an expectorant, commonly used to loosen mucus and ease congestion in patients presenting with acute or chronic bronchitis, and related pulmonary conditions. It is derived from sources such as turpentine, oregano, thyme and eucalyptus. It was…

Kategori:
AlcoholsCyclohexane MonoterpenesCyclohexanes +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terpinen-4-ol DB12816
small molecule | CAS: 562-74-3

Terpinen-4-ol is under investigation in clinical trial NCT01647217 (Demodex Blepharitis Treatment Study).

Kategori:
Cytochrome P-450 CYP2A6 SubstratesCytochrome P-450 Substrates
Target Protein:
AcetylcholinesteraseApoptosis regulator Bcl-2E3 ubiquitin-protein ligase XIAP +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TERT-572 DB17286
biotech | CAS: 255706-49-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCarrier ProteinsDNA Nucleotidyltransferases +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
HTH-type transcriptional regulator EthR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Collagenase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Queuine tRNA-ribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Methionine aminopeptidase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tertomotide DB12747
biotech | CAS: 915019-08-8

Tertomotide is under investigation in clinical trial NCT01223209 (A Study, Combination, Immunologic Study of LTX-315 as adjunct to tertomotide in Patients Following Curative Surgery for Carcinoma). It is a peptide vaccine that activates the immune system so t…

Target Protein:
Telomerase reverse transcriptase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesaglitazar DB06536
small molecule | CAS: 251565-85-2

Tesaglitazar is a dual peroxisome proliferator-activated receptor alpha/gamma agonist which improves apolipoprotein levels in non-diabetic subjects with insulin resistance. Tesaglitazar is a proposed treatment for type 2 diabetes and has completed several pha…

Kategori:
Acids, CarbocyclicAlkanesAlkanesulfonic Acids +4
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesamorelin Approved DB08869
biotech | CAS: 218949-48-5

Tesamorelin is a stabilized synthetic peptide analogue of the hypothalamic peptide, Growth Hormone Releasing Hormone (GHRH) indicated for the reduction of excess abdominal fat in HIV-infected patients with lipodystrophy. Lipodystrophy is a metabolic condition…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone Releasing Factor Analog +17
Target Protein:
Growth hormone-releasing hormone receptor
Waktu Paruh26 and 38 minutes i…
Vol. Distribusi9.4±3.1 L/kg in hea…
Klirens-
Genetik -
Tesetaxel DB12019
small molecule | CAS: 333754-36-2

Tesetaxel has been used in trials studying the treatment of Cancer, Melanoma, Prostate Cancer, Gastric Carcinoma, and Advanced Melanoma, among others.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesevatinib DB11973
small molecule | CAS: 781613-23-8

Tesevatinib has been used in trials studying the treatment of Cancer, Stomach Cancer, Brain Metastases, Esophageal Cancer, and Leptomeningeal Metastases, among others. Tesevatinib is a potent inhibitor of multiple RTKs implicated in driving tumor cell prol…

Kategori:
Antineoplastic AgentsAza CompoundsEnzyme Inhibitors +6
Target Protein:
Ephrin type-B receptor 4Pro-epidermal growth factorReceptor tyrosine-protein kinase erbB-2
Waktu Paruh50-70 hours
Vol. Distribusi-
Klirens-
Genetik -
Tesidolumab DB11926
biotech | CAS: 1531594-08-7

Tesidolumab has been used in trials studying the treatment of Geographic Atrophy, Non-infectious Panuveitis, Exudative Macular Degeneration, Non-infectious Posterior Uveitis, and Age-related Macular Degeneration, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesmilifene DB04905
small molecule | CAS: 98774-23-3

Tesmilifene is a novel potentiator of chemotherapy which, when added to doxorubicin, achieved an unexpected and very large survival advantage over doxorubicin alone in a randomized trial in advanced breast cancer.

Kategori:
Antiplatelet agentsBenzene DerivativesCytochrome P-450 CYP2D6 Substrates +18
Target Protein:
ATP-dependent translocase ABCB1Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesnatilimab DB16377
biotech | CAS: 2242758-08-1

Tesnatilimab is under investigation in clinical trial NCT04655807 (A Study of JNJ-64304500 as Add-on Therapy in Participants With Active Crohn's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Testolactone Approved DB00894
small molecule | CAS: 968-93-4

An antineoplastic agent that is a derivative of progesterone and used to treat advanced breast cancer.

Kategori:
AndrostadienesAndrostanesAndrostenes +7
Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Testosterone Approved DB00624
small molecule | CAS: 58-22-0

Testosterone is a steroid sex hormone indicated to treat primary hypogonadism and hypogonadotropic hypogonadism.[L8983,L8935,L8938,L8986,L8989,L8992,L8995] Testosterone antagonizes the androgen receptor to induce gene expression that causes the growth and dev…

Kategori:
3-Oxoandrosten (4) DerivativesAnabolic SteroidsAndrogens +33
Target Protein:
Androgen receptorEstrogen receptorMineralocorticoid receptor
Waktu ParuhThe half life of te…
Vol. DistribusiThe volume of distr…
KlirensThe mean metabolic …
Genetik -
Testosterone cypionate Approved DB13943
small molecule | CAS: 58-20-8

Testosterone cypionate is a synthetic derivative of testosterone in the form of an oil-soluble 17 (beta)-cyclopentylpropionate ester. Its benefit compared to other testosterone derivatives is the slow rate of release after injection and longer half-life. It w…

Kategori:
Anabolic AgentsAndrogensAndrostanes +33
Target Protein:
Androgen receptorEstrogen receptorMineralocorticoid receptor
Waktu ParuhThe half-life of te…
Vol. DistribusiThe volume of distr…
KlirensTestosterone cypion…
Genetik -
small molecule | CAS: 5721-91-5

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18625-33-7

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12751–12800 dari 14063
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