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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 252 / 349
Opium Approved DB11130
small molecule | CAS: 8008-60-4

Opium is the first substance of the diverse group of the opiates. It has been known for a long time, and the first evidence of a poppy culture dates from 5 thousand years by the Sumerians. During the years, opium was used as a sedative and hypnotic, but it wa…

Kategori:
Alimentary Tract and MetabolismAnalgesicsAntidiarrheals +25
Target Protein:
Delta-type opioid receptorKappa-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half-life of op…
Vol. DistribusiOpium presents a la…
Klirens-
Genetik -
biotech | CAS: 945228-48-8

VB4-845 is studied in the treatment of certain types of head and neck cancer. VB4-845 is made by linking a monoclonal antibody fragment to a toxic protein that may kill cancer cells. VB4-845 is a fusion protein containing humanized scFv specific for the epith…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +8
Target Protein:
Epithelial cell adhesion molecule
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oprelvekin Approved DB00038
biotech | CAS: 145941-26-0

Oprelvekin, the active ingredient in Neumega®, is recombinant Interleukin-11 (IL-11), which is produced in Escherichia coli (E. coli) by recombinant DNA technology. With a molecular mass of approximately 19,000 daltons, the non-glycosylated protein is 177 ami…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-11 receptor subunit alpha
Waktu Paruh6.9 +/- 1.7 hrs
Vol. Distribusi-
Klirens-
Genetik -
Oprozomib DB11991
small molecule | CAS: 935888-69-0

Oprozomib has been used in trials studying the treatment of Solid Tumors, Multiple Myeloma, Waldenstrom Macroglobulinemia, Advanced Hepatocellular Carcinoma, and Advanced Non-Central Nervous System (CNS) Malignancies.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OptPA DB18325
biotech

Optimized tPA (OptPA; W253R/R275S-tPA) is an engineered variant of tPA designed to exhibit reduced neurotoxicity.[A261486]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The oral polio vaccine (OPV) is a live attenuated vaccine containing a mixture of one or more strains of poliovirus serotypes. Strains of the virus are selected based on their reduced incidence of spreading to the central nervous system but still having the a…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orange Approved DB10549
biotech

Orange allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orantinib DB12072
small molecule | CAS: 252916-29-3

Orantinib has been used in trials studying the treatment of Lung Cancer, Breast Cancer, Kidney Cancer, Gastric Cancer, and Prostate Cancer, among others.

Kategori:
Acids, AcyclicAlkaloidsEnzyme Inhibitors +9
Target Protein:
Vascular endothelial growth factor receptor 2Aurora kinase AFibroblast growth factor receptor 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orbifloxacin DB11443
small molecule | CAS: 113617-63-3

Orbifloxacin is a fluoroquinolone antibiotic. It is marketed by Schering-Plough Animal Health and approved for certain infections in dogs.

Kategori:
4-QuinolonesAnti-Bacterial AgentsCytochrome P-450 CYP1A2 Inhibitors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORC-13661 DB18903
small molecule | CAS: 1979935-33-5

ORC-13661 is under investigation in clinical trial NCT05730283 (Prevention of Ototoxicity in NTM Patients Treated With IV Amikacin).

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orciprenaline Approved DB00816
small molecule | CAS: 586-06-1

A beta-adrenergic agonist used in the treatment of asthma and bronchospasms. [PubChem]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +26
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh6 hours
Vol. Distribusi-
Klirens-
Genetik -
Ordesekimab DB16649
biotech | CAS: 2394931-19-0

Ordesekimab is under investigation in clinical trial NCT02633020 (Study to Evaluate the Efficacy and Safety of AMG 714 in Adult Patients With Type II Refractory Celiac Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORE-1001 DB12271
small molecule | CAS: 305335-31-3

ORE1001 has been used in trials studying the treatment of Mild to Moderate Ulcerative Colitis. It is an ACE2 inhibitor.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins
Target Protein:
Angiotensin-converting enzyme 2Carboxypeptidase N catalytic chainCarboxypeptidase N subunit 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oregano Approved DB10677
biotech

Oregano allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oregovomab DB04964
biotech | CAS: 213327-37-8

Oregovomab is a murine monoclonal antibody that attaches to the tumor-associated antigen CA125.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Mucin-16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orelabrutinib DB16272
small molecule | CAS: 1655504-04-3

Orelabrutinib is under investigation in clinical trial NCT04305197 (A Study of ICP-022 in Patients With Systemic Lupus Erythematosus (SLE)).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +1
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orellanine DB19263
small molecule | CAS: 37338-80-0

Orellanine is under investigation in clinical trial NCT05287945 (Study of Orellanine in Metastatic Clear-cell or Papillary Renal Cell Carcinoma).

Kategori:
AgaricalesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orforglipron DB18964
small molecule | CAS: 2212020-52-3

Orforglipron is under investigation in clinical trial NCT06010004 (A Long-term Safety Study of Orforglipron (LY3502970) in Participants With Type 2 Diabetes).

Kategori:
Oxazoles
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORG-25435 DB12312
small molecule | CAS: 256456-73-2

Org 25435 has been used in trials studying the treatment of Anaesthesia.

Kategori:
Benzene Derivatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORG-25935 DB12220
small molecule | CAS: 1147011-84-4

Org 25935 has been used in trials studying the treatment of Alcoholism, Schizophrenia, and Panic Disorder.

Kategori:
Naphthalenes
Target Protein:
Sodium- and chloride-dependent glycine transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORG-31710 DB15585
small molecule | CAS: 118968-41-5

ORG-31710 is a progestational hormone antagonist.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORG-34517 DB05423
small molecule | CAS: 189035-07-2

ORG-34517 is currently under investigation by Organon for the treatment of depression. It has potential to treat a number of diseases such as Cushing’s disease, hypertension, diabetes, glaucoma etc, in which the activity of metabolites corticosterone and cor…

Kategori:
DioxolesFused-Ring CompoundsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orgotein DB11444
biotech | CAS: 1569268-91-2

Superoxide is a natural byproduct of oxygen metabolism which, if left unchecked, leads to cell damage. Superoxide dismutase (SOD) is an enzyme that alternately catalyzes the dismutation of the superoxide radical into either the less damaging hydrogen peroxide…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OriCar-017 DB17280
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Oridonin DB19086
small molecule | CAS: 28957-04-2

Oridonin is under investigation in clinical trial NCT05130892 (Effect of Inflammasome Inhibitor on Hscrp in Patients After PCI).

Kategori:
DiterpenesTerpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orilanolimab DB15312
biotech | CAS: 2066544-85-0

Orilanolimab is under investigation in clinical trial NCT03075878 (A Safety Study of SYNT001 in Subjects With Chronic, Stable Warm Autoimmune Hemolytic Anemia (WAIHA)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orismilast DB19042
small molecule | CAS: 1353546-86-7

Orismilast is under investigation in clinical trial NCT05190419 (Study to Assess the Efficacy and Safety of Orismilast in Psoriasis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
Orlistat Approved DB01083
small molecule | CAS: 96829-58-2

The global prevalence of obesity is increasing rapidly. Obesity-related complications lead to significant personal and economic burden by reducing quality of life and increasing the cost of healthcare. In some individuals, diet and exercise are insufficient …

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAntiobesity Preparations, Excl. Diet Products +11
Target Protein:
Pancreatic triacylglycerol lipaseCannabinoid receptor 1Gastric triacylglycerol lipase +1
Waktu ParuhThe half-life of or…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
ORM-12741 DB12057
small molecule | CAS: 610782-82-6

ORM-12741 has been used in trials studying the basic science and treatment of Alzheimer's Disease.

Kategori:
Adrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +2
Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORM-13070 C-11 DB15324
small molecule | CAS: 1227170-74-2

ORM-13070 C-11 is under investigation in clinical trial NCT00735774 (Suitability of 11C-ORM-13070 as a PET Tracer).

Kategori:
Carbon Radioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ormeloxifene DB13310
small molecule | CAS: 31477-60-8

Ormeloxifene is a third-generation selective estrogen receptor (ER) modulator. In India, ormeloxifene has been marketed since the 1990s as a non-hormonal, non-steroidal oral contraceptive taken once a week,[A251450] and it was later introduced for the treatme…

Kategori:
Adrenal Cortex HormonesBenzopyransChromans +13
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu ParuhIn healthy, non-lac…
Vol. DistribusiIn healthy women, t…
KlirensIn healthy, non-lac…
Genetik -
Ornidazole DB13026
small molecule | CAS: 16773-42-5

Ornidazole has been used in trials studying the prevention of Elective Colorectal Surgery.

Kategori:
AmebicidesAnti-Infective AgentsAntibacterials for Systemic Use +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ornipressin DB13464
biotech | CAS: 3397-23-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsCoagulants +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ornithine Approved DB00129
small molecule | CAS: 70-26-8

Produced during the urea cycle, ornithine is an amino acid produced from the splitting off of urea from arginine. L-Ornithine allows for the disposal of excess nitrogen and acts as a precursor of citrulline and arginine.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +9
Target Protein:
Ornithine aminotransferase, mitochondrialOrnithine transcarbamylase, mitochondrialArginase-1 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orotic acid DB02262
small molecule | CAS: 65-86-1

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialOrotate phosphoribosyltransferaseDihydroorotate dehydrogenase (quinone), mitochondrial +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orotidylic acid DB02957
small molecule | CAS: 2149-82-8

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORP-101 DB16072
small molecule | CAS: 1820753-68-1

ORP-101 is under investigation in clinical trial NCT04129619 (A Comparison of the Effects of ORP-101 Versus Placebo in Adult Patients With Irritable Bowel Syndrome With Diarrhea (IBS-D)).

Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orphenadrine Approved DB01173
small molecule | CAS: 83-98-7

A muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.

Kategori:
Agents producing tachycardiaAminesAnti-Dyskinesia Agents +41
Target Protein:
Glutamate receptor ionotropic, NMDA 2DGlutamate receptor ionotropic, NMDA 1Glutamate receptor ionotropic, NMDA 3B +4
Waktu Paruh13-20 hours
Vol. Distribusi-
Klirens-
Genetik -
Orris Approved DB10413
biotech

Orris allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ortataxel DB11669
small molecule | CAS: 186348-23-2

Ortataxel has been used in trials studying the treatment of Lymphoma, Lung Cancer, Glioblastoma, and Kidney Cancer.

Kategori:
Antineoplastic AgentsCyclodecanesCycloparaffins +3
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orteronel DB12066
small molecule | CAS: 566939-85-3

Orteronel has been investigated for the treatment of Prostate Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lactose operon repressor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orthosiphon aristatus leaf Approved DB15838
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orticumab DB16653
biotech | CAS: 1314241-10-5

Orticumab is under investigation in clinical trial NCT04776629 (A Proof-of-activity Study With Orticumab in Subjects With Psoriasis and Cardiometabolic Risk Factors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Orvepitant DB12427
small molecule | CAS: 579475-18-6

Orvepitant has been used in trials studying the treatment of Depressive Disorder, Depressive Disorder, Major, Post-Traumatic Stress Disorder, and Posttraumatic Stress Disorder (PTSD).

Kategori:
Antidepressive AgentsCentral Nervous System Depressants
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORY-1001 DB16848
small molecule | CAS: 1401966-39-9

Deskripsi belum tersedia.

Kategori:
AminesCycloparaffinsPolyamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oryctolagus cuniculus hair Approved DB10898
biotech

European rabbit hair is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12551–12600 dari 17430
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