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13591

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Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 251 / 272
Tibolone Approved DB09070
small molecule | CAS: 5630-53-5

Tibolone is a synthetic steroid hormone drug, which is mainly non-selective in its binding profile, acting as an agonist primarily at estrogen receptors (ER), with a preference for ER alpha [L1874]. Tibolone (Livial, Org OD 14), produced by Organon (West O…

Kategori:
Anabolic AgentsAntineoplastic Agents, HormonalCardiovascular Agents +12
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. Distribusi-
KlirensElimination of tibo…
Genetik -
Tibulizumab DB14848
biotech | CAS: 1849636-24-3

Tibulizumab is under investigation in clinical trial NCT03736772 (A Study of LY3090106 in Japanese and Caucasian Healthy Participants).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ticagrelor Approved DB08816
small molecule | CAS: 274693-27-5

Ticagrelor, or AZD6140, was first described in the literature in 2003.[A204170,A2903] Ticagrelor is an ADP derivative developed for its P2Y<sub>12</sub> receptor antagonism.[A2903] Unlike [clopidogrel], ticagrelor is not a prodrug.[A2903] It is marketed by As…

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +37
Target Protein:
P2Y purinoceptor 12
Waktu ParuhTicagrelor has a pl…
Vol. DistribusiThe steady state vo…
KlirensThe renal clearance…
Genetik -
Ticarcillin Approved DB01607
small molecule | CAS: 34787-01-4

An antibiotic derived from penicillin similar to carbenicillin in action.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Penicillin binding protein 2a
Waktu Paruh1.1 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech

Tick-borne encephalitis (TBE) is a disease caused by the TBE virus (TBEV), transmitted by ticks from the genus _Ixodes_. The disease course is variable. Some patients will be asymptomatic or experience a mild febrile illness, while others will experience the …

Kategori:
VaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ticlatone DB13613
small molecule | CAS: 70-10-0

Deskripsi belum tersedia.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ticlopidine Approved DB00208
small molecule | CAS: 55142-85-3

Ticlopidine is an effective inhibitor of platelet aggregation. It is a prodrug that is metabolised to an active form, which blocks the ADP receptor that is involved in GPIIb/IIIa receptor activation leading to platelet aggregation. Ticlopidine is marketed und…

Kategori:
Antiplatelet agentsBlood and Blood Forming OrgansCardiovascular Agents +36
Target Protein:
Platelet-activating factor receptorP2Y purinoceptor 12
Waktu ParuhHalf-life following…
Vol. DistribusiThe volume of distr…
KlirensTiclopidine clearan…
Genetik -
Tideglusib DB12129
small molecule | CAS: 865854-05-3

Tideglusib is under the investigation for the development of treatments for Alzheimer's disease and for progressive supranuclear palsy. It is reported to be a potent anti-inflammatory and neuroprotective that is a non-ATP competitive inhibitor of glycogen syn…

Kategori:
Glycogen Synthase Kinase 3, antagonists & inhibitorsSulfur CompoundsThiazoles
Target Protein:
Glycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 30986-62-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyLiver Therapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tidutamab DB18839
biotech | CAS: 2148354-90-7

Tidutamab is under investigation in clinical trial NCT04590781 (Safety and Efficacy of Xmab18087 ± Pembrolizumab in Advanced Merkel Cell Carcinoma or Extensive-stage Small Cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 144-12-7

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tienilic acid DB04831
small molecule | CAS: 40180-04-9

Tienilic acid, or ticrynafen, is a diuretic drug with uric acid-lowering action which was marketed for the treatment of hypertension. It was withdrawn in 1982 after case reports in the United States suggested a link between ticrynafen and hepatitis. (Manier e…

Kategori:
AcetatesAcids, AcyclicAntigout Preparations +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tifacogin DB06437
small molecule | CAS: 148883-56-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tifcemalimab DB18914
biotech | CAS: 2236068-83-8

Tifcemalimab is under investigation in clinical trial NCT06095583 (Phase 3 Study of Toripalimab Alone or in Combination With Tifcemalimab as Consolidation Therapy in Patients With Limited-stage Small Cell Lung Cancer (LS-SCLC)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tifuvirtide DB05413
biotech | CAS: 251562-00-2

Tifuvirtide is the first members of a new class of anti-HIV drugs which is also called fusion inhibitors. It has received fast-track designation from the FDA and is in Phase I/II clinical testing.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Viral +14
Target Protein:
Plasma serine protease inhibitor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigapotide DB04985
biotech | CAS: 848084-83-3

Tigapotide is a synthetic 15-mer peptide that is derived from the natural sequence of amino acids of the prostate secretory protein (PSP94), one of three predominant proteins found in human seminal fluid.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesProteins +2
Target Protein:
Small ribosomal subunit protein uS2
Waktu Paruh0.35 hours to 1.45 …
Vol. Distribusi-
Klirens-
Genetik -
Tigatuzumab DB15101
biotech | CAS: 918127-53-4

Tigatuzumab is under investigation in clinical trial NCT00991796 (CS-1008 With Carboplatin/Paclitaxel in Chemotherapy naïve Subjects With Metastatic or Unresectable Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigecycline Approved DB00560
small molecule | CAS: 220620-09-7

Tigecycline is a glycylcycline antibiotic developed and marketed by Wyeth under the brand name Tygacil. It was developed in response to the growing prevalence of antibiotic resistance in bacteria such as Staphylococcus aureus. It was granted fast-track approv…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
16S ribosomal RNA30S ribosomal protein S930S ribosomal protein S12 +3
Waktu Paruh27-43 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 943001-56-7

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigozertinib DB19239
small molecule | CAS: 2660250-10-0

Tigozertinib (BLU-945) is currently under investigation in clinical trial NCT04862780 (Phase 1/?2 Study Targeting EGFR Resistance Mechanisms in NSCLC) for the treatment of NSCLC.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tigulixostat DB18799
small molecule | CAS: 1287766-55-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TIK-301 DB16909
small molecule | CAS: 118702-11-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Melatonin receptor type 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilactase Approved DB13761
biotech | CAS: 9031-11-2

Tilactase is a beta-D-galactosidase obtained from _Aspergillus oryzae_. It is produced as a chewable tablet that has to be taken before the consumption of a lactose-containing meal.[A27172] The beta-D-galactosidase us a large monomeric multi-domain enzyme of …

Kategori:
Alimentary Tract and MetabolismAntifoaming Agentsbeta-Galactosidase +8
Target Protein:
Lactose
Waktu ParuhTilactase half-life…
Vol. DistribusiTilactase is not ab…
KlirensTilactase is not ab…
Genetik -
Tilarginine Approved DB11815
small molecule | CAS: 17035-90-4

Tilarginine has been investigated for the basic science, treatment, and diagnostic of Obesity, Type 2 Diabetes, Ocular Physiology, and Regional Blood Flow.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +4
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilavonemab DB17014
biotech | CAS: 2096513-89-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilbroquinol Approved DB13222
small molecule | CAS: 7175-09-9

Tilbroquinol was approved in France, Morocco, and Saudi Arabia but it has been withdrawn in France and Saudi Arabia markets mainly due to its hepatotoxicity risk outweighing the drug benefit [L5467]. In Morocco, the drug has been limited to use in the treatme…

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tildacerfont DB18545
small molecule | CAS: 1014983-00-6

Tildacerfont is a corticotropin-releasing factor receptor-1 antagonist containing an unfused thiazole ring

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tildipirosin DB11470
small molecule | CAS: 328898-40-4

Tildipirosin is a veterinary antibiotic.

Kategori:
Anti-Bacterial AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tildrakizumab Approved DB14004
biotech | CAS: 1326244-10-3

Tildrakizumab is a high-affinity, humanized, IgG1 ? antibody targeting interleukin 23 p19 that shows promise in the evolution of treatment strategy in chronic plaque psoriasis [A32255]. The Food and Drug Administration (FDA) approved ILUMYA (tildrakizumab-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-23
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe geometric mean …
KlirensThe mean (CV%) syst…
Genetik -
Tilia americana pollen Approved DB10732
biotech

Tilia americana pollen is the pollen of the Tilia americana plant. Tilia americana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilidine DB13787
small molecule | CAS: 51931-66-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAnalgesicsCentral Nervous System Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilmanocept Approved DB15373
small molecule | CAS: 1185986-76-8

Tilmanocept is under investigation in clinical trial NCT03241446 (Pharmacokinetics and Dosimetry of Tc 99m Tilmanocept Following a Single Intravenous Dose Administration in Male and Female Subjects Diagnosed With Rheumatoid Arthritis (RA)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilpisertib DB18798
small molecule | CAS: 2065153-41-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilsotolimod DB16341
biotech | CAS: 1948266-37-2

Tilsotolimod is under investigation in clinical trial NCT03865082 (Study of Tilsotolimod in Combination With Nivolumab and Ipilimumab for the Treatment of Solid Tumors (ILLUMINATE-206)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Toll-like receptor 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TILT-123 DB17519
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiludronic acid Approved DB01133
small molecule | CAS: 89987-06-4

Tiludronate, or (4-chlorophenyl)thio-methylene-1,1-bisphosphonate, is a first generation bisphosphonate similar to [etidronic acid] and [clodronic acid].[A1923,A203111] These drugs were developed to mimic the action of pyrophosphate, a regulator of calcificat…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +6
Target Protein:
HydroxylapatiteAdenosine triphosphate (ATP)Tyrosine-protein phosphatase non-receptor type 12 +3
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe volume of distr…
KlirensTiludronic acid has…
Genetik -
Timbetasin DB19119
biotech | CAS: 77591-33-4

Timbetasin is under investigation in clinical trial NCT05555589 (Assessment of the Safety and Efficacy of 0.1% RGN-259 Ophthalmic Solution for the Treatment of NK: SEER-2).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timcodar DB12761
small molecule | CAS: 179033-51-3

Timcodar has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timepidium DB13850
small molecule | CAS: 97094-64-9

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timolol Approved DB00373
small molecule | CAS: 26839-75-8

Timolol is a nonselective beta-adrenergic antagonist given in an eye drop solution to reduce intraocular pressure, or pressure in the eyes.[L6724] It is also used in tablet form as a drug to treat hypertension.[L6727] Timolol was first approved by the FDA in …

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +28
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorEndolysin
Waktu ParuhTimolol half-life w…
Vol. Distribusi1.3 - 1.7 L/kg [L6]…
KlirensOne pharmacokinetic…
Genetik -
Timolumab DB18597
biotech | CAS: 1073538-99-4

Timolumab is a recombinant, fully-human, IgG4 immunoglobulin with antigen-binding specificity for human vascular adhesion protein-1 (VAP-1).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14325-05-4

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinengotinib DB17384
small molecule | CAS: 2230490-29-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinidazole Approved DB00911
small molecule | CAS: 19387-91-8

A nitroimidazole antitrichomonal agent effective against _Trichomonas vaginalis_, _Entamoeba histolytica_, and _Giardia lamblia_ infections.

Kategori:
Alimentary Tract and MetabolismAlkylating DrugsAnti-Bacterial Agents +24
Target Protein:
DNA
Waktu ParuhThe elimination hal…
Vol. Distribusi* 50 L
Klirens-
Genetik -
Tinlarebant DB17832
small molecule | CAS: 1821327-95-0

Deskripsi belum tersedia.

Target Protein:
Retinol-binding protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinlorafenib DB17082
small molecule | CAS: 2573781-75-4

Tinlorafenib (PF-07284890) is a potent, selective, highly brain-penetrant, small-molecule inhibitor of BRAF V600 mutations.[A253992]

Kategori:
Heterocyclic Compounds, Fused-RingSulfonamides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinodasertib DB18796
small molecule | CAS: 1464151-33-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinoridine DB13001
small molecule | CAS: 24237-54-5

Tinoridine is under investigation in clinical trial NCT01224756 (Efficacy of Tinoridine in Treating Pain and Inflammation in Adults).

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinostamustine DB15147
small molecule | CAS: 1236199-60-2

Tinostamustine is under investigation in clinical trial NCT03452930 (Tinostamustine With or Without Radiation Therapy in Treating Patients With Newly Diagnosed MGMT-Unmethylated Glioblastoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiocarlide DB13608
small molecule | CAS: 910-86-1

Deskripsi belum tersedia.

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsDrugs for Treatment of Tuberculosis +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12501–12550 dari 13591
Sebelumnya Halaman 251 / 272 Berikutnya