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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 250 / 252
Zipalertinib DB18763
small molecule | CAS: 1661854-97-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Zipeprol DB13564
small molecule | CAS: 34758-83-3

Deskripsi belum tersedia.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +1
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Ziprasidone Approved DB00246
small molecule | CAS: 146939-27-7

Disorders such as schizophrenia and bipolar disorder can significantly impair mood, cognition, and behavior.[A190525] These mental illnesses can often be accompanied by comorbidities such as depression and substance abuse, and can significantly impact the qua…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +45
Target Protein:
D(2) dopamine receptorNeuronal acetylcholine receptor subunit alpha-75-hydroxytryptamine receptor 2A +24
Waktu ParuhThe half life of zi…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent s…
Genetik -
biotech | CAS: 2377668-38-5

Deskripsi belum tersedia.

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Zirconium chloride hydroxide Approved DB15479
small molecule | CAS: 10119-31-0

Deskripsi belum tersedia.

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small molecule | CAS: 1314-23-4

Deskripsi belum tersedia.

Kategori:
Compounds used in a research, industrial, or household settingDental AlloysDental Materials +4
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Genetik -
biotech

Zirconium panitumumab Zr-89 is under investigation in clinical trial NCT05423197 (Study Evaluating Zr-panitumumab for Assessment of Suspected Metastatic Lesions on 18F-FDG-PET/CT in Head and Neck Squamous Cell Carcinoma).

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Ziresovir DB15145
small molecule | CAS: 1422500-60-4

Ziresovir is under investigation in clinical trial NCT03699202 (Anti-RSV Study in Chinese Patients (ASCENT)).

Kategori:
Anti-Infective AgentsAntiviral AgentsAzepines +3
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Ziritaxestat DB15403
small molecule | CAS: 1628260-79-6

Ziritaxestat is under investigation in clinical trial NCT03798366 (A Clinical Study to Test How Effective and Safe GLPG1690 is for Patients With Systemic Sclerosis).

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ZK-805623 DB04432
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
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Zk-806450 DB02112
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
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ZK-93423 DB17063
small molecule | CAS: 83910-44-5

ZK-93423 is a beta-carboline with muscle relaxant activity with agonistic properties at the benzodiazepine receptor.[A253172]

Kategori:
Anti-Anxiety AgentsAnticonvulsantsCentral Nervous System Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2
Waktu Paruh-
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ZM-39923 DB17064
small molecule | CAS: 273727-89-2

ZM-39923 is a small molecule that inhibits Janus kinase and human tissue transglutaminase (TGM2).[A253177]

Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK3
Waktu Paruh-
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Zofenoprilat DB08766
small molecule | CAS: 75176-37-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +1
Target Protein:
Cytosol aminopeptidase
Waktu Paruh-
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Zofin DB16519
biotech

Zofin, previously known as Organicell Flow, is a nanoparticle-based therapeutic derived from perinatal sources which is manufactured in a way that retains the naturally occurring microRNAs without the addition of other substances[L31323].

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Zolazepam DB11555
small molecule | CAS: 31352-82-6

Zolazepam is a pyrazolodiazepinone derivative used as an anaesthetic in veterinary medicine. Zolazepam is typically used in combination with the NMDA antagonist tiletamine or the ?2 adrenoceptor agonist xylazine. It is around four times the potency of diazepa…

Kategori:
Anti-Anxiety AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
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Zolbetuximab Approved DB15118
biotech | CAS: 1496553-00-4

Zolbetuximab is under investigation in clinical trial NCT01630083 (Efficacy and Safety of IMAB362 in Combination With the EOX Regimen for CLDN18.2-positive Gastric Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Claudin-18
Waktu Paruh-
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Zoledronic acid Approved DB00399
small molecule | CAS: 118072-93-8

Zoledronic acid, or CGP 42'446,[A203120] is a third generation, nitrogen containing bisphosphonate similar to [ibandronic acid], [minodronic acid], and [risedronic acid].[A203111] Zoledronic acid is used to treat and prevent multiple forms of osteoporosis, hy…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +5
Target Protein:
Geranylgeranyl pyrophosphate synthaseHydroxylapatiteFarnesyl pyrophosphate synthase
Waktu ParuhZoledronic acid has…
Vol. Distribusi-
KlirensZoledronic acid has…
Genetik -
Zoliflodacin DB12817
small molecule | CAS: 1620458-09-4

Zoliflodacin has been used in trials studying the basic science and treatment of Gonorrhoea.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +5
Target Protein:
DNA gyrase subunit ADNA gyrase subunit B
Waktu Paruh-
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Zolimidine DB13593
small molecule | CAS: 1222-57-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord)
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Zolmitriptan Approved DB00315
small molecule | CAS: 139264-17-8

Zolmitriptan is a member of the triptan class of 5-hydroxytryptamine(5-HT)<sub>1B/1D/(1F)</sub> receptor agonists used to treat acute migraine.[A462, L12978] [Sumatriptan] was the first triptan to be developed, but had poor oral bioavailability and lipophilic…

Kategori:
Agents that produce hypertensionAminesAnalgesics +24
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1F +5
Gen Terkait:
GNB3
Waktu ParuhZolmitriptan has a …
Vol. DistribusiZolmitriptan has a …
KlirensZolmitriptan has a …
Genetik 1 Varian
Zolpidem Approved DB00425
small molecule | CAS: 82626-48-0

Zolpidem, also known as _Ambien_, is a hypnotic drug that was initially approved by the FDA in 1992 [FDA label]. Zolpidem improves sleep in patients with insomnia. It is aimed for use in patients with difficulties initiating sleep. This drug decreases the ti…

Kategori:
Benzodiazepine hypnotics and sedativesCentral Nervous System AgentsCentral Nervous System Depressants +21
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-2 +2
Waktu ParuhThe average zolpide…
Vol. Distribusi0.54 to 0.68 L/kg (…
KlirensIn a clinical trial…
Genetik -
Zomepirac DB04828
small molecule | CAS: 33369-31-2

Zomepirac, formerly marketed as Zomax tablets, was associated with fatal and near-fatal anaphylactoid reactions. The manufacturer voluntarily removed Zomax tablets from the Canadian, US, and UK markets in March 1983.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +15
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Prostaglandin D2 receptor 2
Waktu Paruh-
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Zonisamide Approved DB00909
small molecule | CAS: 68291-97-4

Zonisamide is a sulfonamide anticonvulsant used as an adjunctive therapy in adults with partial-onset seizures.[L42530,L42535] Zonisamide may act by blocking repetitive firing of voltage-gated sodium channels, leading to a reduction of T-type calcium channel…

Kategori:
Agents causing hyperkalemiaAmidesAnti-epileptic Agent +32
Target Protein:
Sodium channel protein type 1 subunit alphaSodium channel protein type 2 subunit alphaSodium channel protein type 3 subunit alpha +29
Waktu ParuhIn plasma, the elim…
Vol. DistribusiFollowing a 400 mg …
KlirensIn patients not tak…
Genetik -
Zopiclone Approved DB01198
small molecule | CAS: 43200-80-2

Zopiclone is a novel hypnotic agent used in the treatment of insomnia. Its mechanism of action is based on modulating benzodiazepine receptors. In addition to zopiclone's benzodiazepine pharmacological properties it also has some barbiturate-like properties.

Kategori:
Aza CompoundsBenzodiazepine hypnotics and sedativesCentral Nervous System Agents +16
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +2
Waktu ParuhElimination half li…
Vol. Distribusi-
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Genetik -
small molecule | CAS: 139570-93-7

Zoptarelin doxorubicin has been used in trials studying the treatment of Breast Cancer, Ovarian Cancer, Prostate Cancer, Endometrial Cancer, and Urothelial Carcinoma, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAnthracyclinesCarbohydrates +12
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh-
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Genetik -
Zorevunersen DB16912
biotech | CAS: 2415330-04-8

Deskripsi belum tersedia.

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Zorubicin DB11618
small molecule | CAS: 54083-22-6

Zorubicin is a drug of the anthracycline class - a class of medications that have historically demonstrated effective chemotherapy for a variety of cancer types.

Kategori:
AnthracyclinesAnthracyclines and Related SubstancesAntibiotics, Antineoplastic +6
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Zosuquidar DB06191
small molecule | CAS: 167354-41-8

Zosuquidar is a compound of antineoplastic drug candidates currently under development. It is now in "Phase 3" of clinical tests in the United States. Its action mechanism consists of the inhibition of P-glycoproteins; other drugs with this mechanism include …

Kategori:
BenzocycloheptenesDrug Resistance, MultipleHeterocyclic Compounds, Fused-Ring +1
Target Protein:
ATP-dependent translocase ABCB1Phosphatidylcholine translocator ABCB4
Waktu Paruh-
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Zotarolimus DB18761
small molecule | CAS: 221877-54-9

Zotarolimus is an immunosuppressant under investigation for use in drug-eluting stents.

Kategori:
Anti-Bacterial AgentsLactonesMacrolides
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
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Zotatifin DB16408
small molecule | CAS: 2098191-53-6

Zotatifin is under investigation in clinical trial NCT04092673 (Study of Eft226 in Subjects With Selected Advanced Solid Tumor Malignancies).

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Zotepine Approved DB09225
small molecule | CAS: 26615-21-4

Zotepine, with the formula (2-chloro-11-(2-dimethyl-amino-ethoxy)-dibenzo thiepin, is a neuroleptic drug. It was designed and synthesized by Fujisawa Pharmaceutical Co Ltd.[A31855] It has been used as an antipsychotic in Japan, India and some places in Europe…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +21
Target Protein:
D(1) dopamine receptorD(2) dopamine receptor5-hydroxytryptamine receptor 2A +4
Waktu ParuhThe half-life of zo…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Zotiraciclib DB16656
small molecule | CAS: 1204918-72-8

Zotiraciclib is under investigation in clinical trial NCT02942264 (Zotiraciclib (TG02) Plus Dose-dense or Metronomic Temozolomide Followed by Randomized Phase II Trial of Zotiraciclib (TG02) Plus Temozolomide Versus Temozolomide Alone in Adults With Recurrent…

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 9Tyrosine-protein kinase Fyn +1
Waktu Paruh-
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Zotizalkib DB19238
small molecule | CAS: 2648641-36-3

Deskripsi belum tersedia.

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Zoxazolamine DB19372
small molecule | CAS: 61-80-3

Deskripsi belum tersedia.

Kategori:
Antigout PreparationsAntirheumatic AgentsBenzoxazoles and derivatives +8
Target Protein:
Small conductance calcium-activated potassium channel protein 2
Waktu Paruh-
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ZSTK-474 DB12904
small molecule | CAS: 475110-96-4

ZSTK474 has been used in trials studying the treatment of Neoplasms.

Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
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ZUBERITAMAB DB19443
biotech | CAS: 2251143-19-6

Zuberitamab is under investigation in clinical trial NCT06642909 (A Phase II Study of Zuberitamab Injection in Patients With Primary Membranous Nephropathy).

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Zucapsaicin Approved DB09120
small molecule | CAS: 25775-90-0

Zucapsaicin, the cis-isomer of capsaicin, is a topical analgesic used to treat osteoarthritis of the knee and other neuropathic pain. It is a modulator of transient receptor potential cation channel subfamily V member 1 (TRPV-1), also known as the vanilloid o…

Kategori:
AlkaloidsAlkenesAlkynes +25
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhIn rats, the elimin…
Vol. Distribusi-
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Zuclopenthixol Approved DB01624
small molecule | CAS: 53772-83-1

Zuclopenthixol, also known as Zuclopentixol or Zuclopenthixolum, is an antipsychotic agent. Zuclopenthixol is a thioxanthene-based neuroleptic with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine rece…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +34
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +4
Waktu Paruh20 hours (range 12-…
Vol. Distribusi20 L/kg.
Klirensapproximately 0.9 L…
Genetik -
Zunsemetinib DB16502
small molecule | CAS: 1640282-42-3

ATI-450 was under investigation in clinical trials (NCT05279417 and NCT05216224) for treating patients with rheumatoid arthritis and hidradenitis suppurativa, respectively. Additionally, ATI-450 was studied in a terminated trial (NCT05511519) to treat patient…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
MAP kinase-activated protein kinase 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Zuranolone Approved DB15490
small molecule | CAS: 1632051-40-1

Zuranolone is a neuroactive steroid that acts as a positive allosteric modulator of the GABA<sub>A</sub> receptors. Unlike other more common GABA<sub>A</sub> positive allosteric modulators on the market like benzodiazepines, zuranolone can modulate both synap…

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +9
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3GABA(A) Receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe mean apparent c…
Genetik -
small molecule | CAS: 29584-22-3

Zuretinol acetate has been used in trials studying the treatment of Impaired Dark Adaptation, RP (Retinitis Pigmentosa), Retinitis Pigmentosa (RP), and LCA (Leber Congenital Amaurosis).

Kategori:
Adjuvants, ImmunologicAlkenesAnticarcinogenic Agents +14
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Genetik -
ZYCOV-D DB15892
biotech

The ZYCOV-D vaccine candidate was developed by Cadila Healthcare Ltd. based in India[A219758]. The vaccine was developed using a DNA vaccine platform with a non-replicating and non-integrating plasmid carrying the gene of interest[L16503]. Once the plasmid D…

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ZYIL-1 DB18184
small molecule | CAS: 2455519-86-3

Deskripsi belum tersedia.

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Zytron Approved DB11768
small molecule | CAS: 299-85-4

Zytron (DMPA) is under investigation for the treatment and health services research of HIV, Lactation, Contraception, Postpartum Depression, and Immune Cells (Mucosal and Systemic). DMPA has been investigated for the prevention, treatment, and basic science o…

Kategori:
AminesOrganophosphorus CompoundsSulfur Compounds
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Chymase
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Subtilisin Carlsberg
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small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase TEM
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small molecule

Deskripsi belum tersedia.

Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferase
Waktu Paruh-
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Genetik -
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