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6694

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6694 (100.0%)

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Halaman 25 / 134
biotech

Autologous peripheral blood-derived CD34+ cells, or CLBS119 (a proprietary version being developed by Caladrius Biosciences, Inc.), are hematopoietic stem cells.[L27741] It is also a cell therapy being investigated by Caladrius Biosciences in the clinical tri…

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AV-101 DB12878
small molecule | CAS: 153152-32-0

AV-101 has been used in trials studying the treatment of Neuropathic Pain.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsSweetening Agents
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AV-COVID-19 DB15802
biotech

AV-COVID-19 is a vaccine composed of autologous dendritic cells loaded with SARS-CoV-2 antigens and with or without Granulocyte-macrophage colony-stimulating factor (GM-CSF). The vaccine is created from the receiving patients’ isolated peripheral blood mon…

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AV608 DB05072
small molecule

AV608 is a NK-1 antagonist. It is developed for the treatment of Social anxiety disorder (SAD), irritable bowel syndrome (IBS) and overactive bladder (OAB).

Target Protein:
Substance-P receptor
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AVA-4746 DB18022
small molecule | CAS: 422268-99-3

Deskripsi belum tersedia.

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AVA-6000 DB17398
small molecule | CAS: 1841402-73-0

Deskripsi belum tersedia.

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Avacincaptad pegol Approved DB15165
biotech | CAS: 1613641-69-2

Avacincaptad pegol is an RNA aptamer covalently bound to a branched polyethylene glycol (PEG) molecule. It was developed to treat an advanced form of age-related macular degeneration (AMD) called geographic atrophy (GA).[L47696] AMD is the leading cause of vi…

Kategori:
Aptamers, NucleotideComplement Inactivating AgentsComplement Inactivator Proteins
Target Protein:
Complement C5
Waktu ParuhThe estimated appar…
Vol. DistribusiLimited information…
KlirensLimited information…
Genetik -
Avacopan Approved DB15011
small molecule | CAS: 1346623-17-3

Anti-neutrophil cytoplasmic (auto)antibody (ANCA)-associated vasculitis (AAV) is a rare (estimated incidence of 3 cases per 100,000 per year) form of "pauci-immune" systemic small-vessel vasculitis typified by the presence of ANCAs in the serum.[A240249, A240…

Kategori:
AminesAntineoplastic and Immunomodulating AgentsComplement 5a Receptor Antagonist +22
Target Protein:
C5a anaphylatoxin chemotactic receptor 1
Waktu ParuhA single 30 mg dose…
Vol. DistribusiAvacopan has an app…
KlirensAvacopan has an est…
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Avagacestat DB11893
small molecule | CAS: 1146699-66-2

Avagacestat has been investigated for the basic science and treatment of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors +4
Target Protein:
Gamma-secretase subunit APH-1ANicastrinGamma-secretase subunit APH-1B +2
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Avalglucosidase alfa Approved DB16099
biotech | CAS: 1802558-87-7

Avalglucosidase alfa, or NeoGAA, is a drug for enzyme replacement therapy specifically designed for Pompe disease, a rare inherited neuromuscular disorder caused by the deficiency of the alpha-glucosidase (GAA) enzyme. GAA is an essential enzyme that hydrolyz…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean avalglucos…
Vol. DistribusiThe volume of distr…
KlirensThe mean avalglucos…
Genetik -
biotech | CAS: 2227000-30-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Avanafil Approved DB06237
small molecule | CAS: 330784-47-9

Avanafil is a phosphodiesterase-5 (PDE5) inhibitor used in the treatment of erectile dysfunction. In comparison with other drugs of the same class, it shows greater selectivity for PDE5 over PDE6 than both [sildenafil] and [vardenafil] but less selectivity th…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A Substrates +9
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu ParuhStudies have demons…
Vol. DistribusiThe apparent volume…
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Avasopasem DB18481
small molecule

Deskripsi belum tersedia.

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Avelumab Approved DB11945
biotech | CAS: 1537032-82-8

Avelumab is a human IgG1 lambda monoclonal antibody that binds programmed cell death ligand-1 (PD-L1) to block its interaction with its receptors found on T cells and antigen-presenting cells.[A261496] Avelumab was first approved by the FDA on March 23, 2017.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe geometric mean …
KlirensThe total systemic …
Genetik -
Avenciguat DB18882
small molecule | CAS: 1579514-06-9

Avenciguat is under investigation in clinical trial NCT05282121 (A Study to Test Whether BI 685509 Alone or in Combination With Empagliflozin Helps People With Liver Cirrhosis Caused by Viral Hepatitis or Non-alcoholic Steatohepatitis (NASH) Who Have High Blo…

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AVI-4557 DB05447
small molecule

AVI-4557 is an oral antisense compound that selectively inhibits the metabolic enzyme cytochrome P450 3A4 (CYP), a liver enzyme responsible for the metabolism or breakdown of approximately half of currently marketed drugs. Studies indicate that AVI-4557 can s…

Target Protein:
Hepatocyte nuclear factor 4-alpha
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AVI-5126 DB05726
small molecule

AVI-526 is an improved formulation of [AVI-4557], developed for use on Vein Grafts before use in Heart by-Pass Graft Surgery. AVI-526 works by silencing a gene known as c-myc, a key regulatory gene involved in cardiovascular restenosis. The drug was under inv…

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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Avicin D DB17240
small molecule | CAS: 197787-20-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosides
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Avilamycin DB11375
small molecule | CAS: 11051-71-1

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +2
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Aviptadil DB06260
small molecule | CAS: 40077-57-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsErectile DysfunctionGastrointestinal Hormones +9
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Avizakimab DB18842
biotech | CAS: 2229685-51-0

Avizakimab is under investigation in clinical trial NCT03371251 (Study of BOS161721 in Systemic Lupus Erythematosus (SLE) Patients on a Background of Limited Standard of Care).

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AVN-944 DB05500
biotech

AVN944 is a biotech drug that demonstrated a statistically meaningful impact on IMPDH and other proteins that are critical to activities in cancer cells, including nucleotide biosynthesis, energy and metabolism, DNA replication, apoptosis and cell cycle contr…

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
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Avobenzone Approved DB09495
small molecule | CAS: 70356-09-1

Avobenzone is dibenzoyl methane derivative. It is oil soluble ingredient. Avobenzone has the ability to absorb ultraviolet light over wider range of wavelengths. It is included in many commercially available sunscreens which are used as wide spectrum sunscree…

Kategori:
Compounds used in a research, industrial, or household settingCosmeticsDermatologicals +4
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Avoralstat DB12120
small molecule | CAS: 918407-35-9

Avoralstat has been used in trials studying the prevention of HAE and Hereditary Angioedema.

Kategori:
Acids, CarbocyclicAlkenesAmides +6
Target Protein:
Kallikrein-2Kininogen-1
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Avotaciclib DB16652
small molecule | CAS: 1983983-41-0

Avotaciclib is under investigation in clinical trial NCT03579836 (Evaluation of Safety and Efficacy in BEY1107 in Monotherapy Gemcitabine Combination in Patient With Pancreatic Cancer).

Target Protein:
Cyclin-dependent kinase 1
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Avotermin DB11955
biotech | CAS: 182212-66-4

Juvista has been investigated for the treatment, prevention, and basic science of Scars, Keloid, and Cicatrix.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
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AVR-RD-01 DB17651
biotech

AVR-RD-01 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ cells that transduced with Lentiviral Vector/alpha-galactosidase A (AGA) encoding for the human AGA complementary deoxyribonucleic acid…

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AVR-RD-02 DB17650
biotech

AVR-RD-02 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ enriched hematopoietic stem cells (HSCs) that have been genetically modified _ex vivo_ with a lentiviral vector (LV) to contain a ribon…

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AVR118 DB04979
biotech

AVR118 represents a new type of biopolymer chemistry that also possesses novel immunomodulator activity. This non-toxic peptide-nucleic acid, which to date has shown no indication of human toxicity, appears to stimulate the proinflammatory responses required …

Kategori:
HIVNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
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AVXS-301 DB17943
biotech

AVXS-301 consists of an adeno-associated virus serotype 9 (AAV9) designed to express the superoxide dismutase 1 (SOD1) gene. It is being investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).[L47077]

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AX200 DB05093
small molecule

AX200, which has been developed for the treatment of stroke, is the most advanced drug candidate and is halfway through the process of gaining clinical approval. The expression of the endogenous AX200 protein in the brain is increased after brain damage. Thus…

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Axatilimab Approved DB16388
biotech | CAS: 2155851-88-8

Axatilimab is a humanized IgG4 monoclonal antibody produced in Chinese hamster ovary cells.[L51194] It is targeted against macrophage colony-stimulating factor 1 receptor (CSF-1R), causing a reduction in circulating levels of monocytes and macrophages respons…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Macrophage colony-stimulating factor 1 receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
Axicabtagene ciloleucel Approved DB13915
biotech

Axicabtagene ciloleucel is an anti-CD19 chimeric antigen receptor (CAR) T-cell therapy. The drug has a unique mechanism of action, as it utilizes the patient's own T cells, which play a central role in immune response to cancer.[A216163] Once T-cells are coll…

Kategori:
AntigensAntigens, CDAntigens, Differentiation +16
Target Protein:
B-lymphocyte antigen CD19
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AZ-3102 DB18502
small molecule

AZ-3102 is a Biphenyl-substituted L-ido configured deoxynojirimycin derivative

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Azacitidine Approved DB00928
small molecule | CAS: 320-67-2

Azacitidine is a pyrimidine nucleoside analogue with anti-neoplastic activity. It differs from cytosine by the presence of nitrogen in the C5-position, key in its hypomethylating activity.[A1406,A1413,A1415] Two main mechanisms of action have been proposed fo…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
DNA (cytosine-5)-methyltransferase 1RNADNA
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients given a…
KlirensAzacitidine has an …
Genetik -
Azadirachtin DB19419
small molecule | CAS: 11141-17-6

Azadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).

Kategori:
AgrochemicalsAzadirachtaCompounds used in a research, industrial, or household setting +5
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Azafenidin DB19031
small molecule | CAS: 68049-83-2

Azafenidin is under investigation in clinical trial NCT01726582 (Pancreas Cancer: Molecular Profiling as a Guide to Therapy Before and After Surgery ("Personalized Medicine")).

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Azaperone DB11376
small molecule | CAS: 1649-18-9

Azaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs and elephants. At the same time, th…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Butyrophenones +11
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
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AZD-0328 DB12145
small molecule | CAS: 220099-91-2

AZD0328 has been used in trials studying the treatment and basic science of Schizophrenia and Alzheimer's Disease.

Kategori:
Receptors, Nicotinic
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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AZD-1236 DB11961
small molecule | CAS: 459814-89-2

AZD1236 has been used in trials studying the basic science and treatment of Cystic Fibrosis and Chronic Obstructive Pulmonary Disease.

Kategori:
AmidesImidazolesImidazolidines +2
Target Protein:
Macrophage metalloelastase
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AZD-1305 DB11766
small molecule | CAS: 872045-91-5

AZD1305 has been used in trials studying the treatment and basic science of Atrial Flutter, Atrial Fibrillation, and Left Ventricle Function.

Kategori:
Acids, AcyclicAza Compounds
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AZD-1480 DB12588
small molecule | CAS: 935666-88-9

AZD1480 has been used in trials studying the treatment of Solid Malignancies, Post-Polycythaemia Vera, Primary Myelofibrosis (PMF), and Essential Thrombocythaemia Myelofibrosis.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
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AZD-1981 DB11946
small molecule | CAS: 802904-66-1

AZD1981 has been used in trials studying the treatment and basic science of Asthma, Postmenopausal, Pharmakokinetic, Asthma Patients, and Drug Interaction, among others.

Target Protein:
Prostaglandin D2 receptor 2
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AZD-2066 DB12644
small molecule | CAS: 934282-55-0

AZD2066 has been used in trials studying the treatment and basic science of Pain, Chronic Pain, Reflux Episodes, Neuropathic Pain, and Diabetic Neuropathy, among others.

Target Protein:
Metabotropic glutamate receptor 5
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AZD-3043 DB12576
small molecule | CAS: 579494-66-9

AZD3043 has been used in trials studying the treatment and basic science of Safety, Sedation, Tolerability, and Pharmacokinetics.

Kategori:
Acids, CarbocyclicCentral Nervous System DepressantsHypnotics and Sedatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
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AZD-3839 DB12368
small molecule | CAS: 1227163-84-9

AZD3839 has been used in trials studying the basic science of Safety, Tolerability, Alzheimer's Disease, and Blood Concentration.

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-4547 DB12247
small molecule | CAS: 1035270-39-3

AZD4547 has been used in trials studying the treatment of Cancer, LYMPHOMA, Gastric Cancer, Adenocarcinoma, and Solid Neoplasm, among others.

Target Protein:
Fibroblast growth factor receptor 1
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AZD-5423 DB12280
small molecule | CAS: 1034148-04-3

AZD5423 has been used in trials studying the basic science and treatment of Asthma, Bioavailability and AUC, and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AcetatesAcids, AcyclicAmides +4
Target Protein:
Glucocorticoid receptor
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AZD-5672 DB11804
small molecule | CAS: 780750-65-4

Azd5672 has been used in trials studying the basic science and treatment of Pharmacokinetics, Renal Impairment, and Rheumatoid Arthritis.

Kategori:
AcetamidesAmidesAnti-HIV Agents +5
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AZD-5991 DB14792
small molecule | CAS: 2143010-83-5

AZD-5991 is under investigation in clinical trial NCT03218683 (Study of AZD5991 in Relapsed or Refractory Haematologic Malignancies.).

Kategori:
Antineoplastic Agents
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