Hasil Filter

3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (3253)

Halaman 25 / 66
Fanapanel DB12393
small molecule | CAS: 161605-73-8

Fanapanel has been investigated for the treatment of Visual Acuity.

Kategori:
Heterocyclic Compounds, Fused-RingOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Farampator DB15012
small molecule | CAS: 211735-76-1

Farampator is under investigation in clinical trial NCT00113022 (Org 24448 to Treat Major Depression).

Kategori:
Oxazoles
Target Protein:
Glutamate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Faropenem DB12190
small molecule | CAS: 106560-14-9

Faropenem has been used in trials studying the treatment of Tuberculosis, Pulmonary Tuberculosis, and Community Acquired Pneumonia.

Kategori:
AmidesAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasiglifam DB12491
small molecule | CAS: 1000413-72-8

Fasiglifam has been used in trials studying the treatment of Chronic Kidney Disease, Type 2 Diabetes Mellitus, and Diabetes Mellitus, Type 2.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Free fatty acid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasinumab DB12157
biotech | CAS: 1190239-42-9

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic pain[A241045] and has demonstrated significantly greater pain relief and functional improvement as …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Beta-nerve growth factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Favipiravir Approved DB12466
small molecule | CAS: 259793-96-9

Discovered by Toyama Chemical Co., Ltd. in Japan, favipiravir is a modified pyrazine analog that was initially approved for therapeutic use in resistant cases of influenza.[A191688,A191721] The antiviral targets RNA-dependent RNA polymerase (RdRp) enzymes, wh…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +11
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'RNA-directed RNA polymerase catalytic subunit
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe recommended ora…
Genetik -
Fedratinib Approved DB12500
small molecule | CAS: 936091-26-8

Fedratinib, also known as SAR302503 and TG101348, is a tyrosine kinase inhibitor used to treat intermediate-2 and high risk primary and secondary myelofibrosis.[A183176,L8090] It is an anilinopyrimidine derivative.[A183188] Fedratinib was granted FDA appro…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase JAK1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of fe…
Genetik -
Feladilimab DB16415
biotech

Feladilimab is under investigation in clinical trial NCT04128696 (Study of GSK3359609 and Pembrolizumab in Programmed Death Receptor 1-ligand 1 Positive Recurrent or Metastatic Head and Neck Squamous Cell Carcinoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felcisetrag DB12725
small molecule | CAS: 916075-84-8

Felcisetrag (TD-8954) has been used in trials studying the treatment of Enteral Feeding Intolerance and Gastrointestinal Motility Disorder.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felzartamab DB16375
biotech | CAS: 2197112-39-1

Felzartamab is under investigation in clinical trial NCT04145440 (Trial to Assess Safety and Efficacy of MOR202 in Anti-pla2r + Membranous Nephropathy (Amn)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenamole DB12506
small molecule | CAS: 5467-78-7

Fenamole has been investigated for the supportive care of Side Effects and Dental Plaque.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fencamfamin DB01463
small molecule | CAS: 1209-98-9

Fencamfamin (Glucoenergan, Reactivan) is a stimulant which was developed in the 1960s as an appetite suppressant, but was later withdrawn for this application due to problems with dependence and abuse. It is around half the potency of [dexamphetamine], and is…

Kategori:
Bridged-Ring CompoundsCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Sodium-dependent dopamine transporterD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenfluramine Approved DB00574
small molecule | CAS: 458-24-2

Dravet syndrome is a pediatric encephalopathy that typically manifests within the first year of life following exposure to elevated temperatures. It is characterized by recurrent pharmacoresistant seizures, which increase in frequency and severity with diseas…

Kategori:
Alimentary Tract and MetabolismAminesAnticonvulsants +27
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2C +4
Waktu ParuhFenfluramine has an…
Vol. DistribusiFenfluramine has an…
KlirensFenfluramine has a …
Genetik -
Fenobam DB12931
small molecule | CAS: 57653-26-6

Fenobam is under investigation in clinical trial NCT00637221 (Open Label Study Investigating Safety and Efficacy of Fenobam anhydrous 50 mg - 150 mg on Prepulse Inhibition Tests and Continuous Performance Tasks, Adults With Fragile X Syndrome).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenofibric acid Approved DB13873
small molecule | CAS: 42017-89-0

Fenofibric acid is a lipid-lowering agent that is used in severe hypertriglyceridemia, primary hyperlipidemia, and mixed dyslipidemia. It works to decrease elevated low-density lipoprotein cholesterol, total cholesterol, triglycerides, apolipoprotein B, while…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnticholesteremic Agents +17
Target Protein:
Peroxisome proliferator-activated receptor alphaFatty acid-binding protein, liverMatrix metalloproteinase-25 +3
Waktu ParuhFollowing once dail…
Vol. DistribusiThe volume of distr…
KlirensIn five elderly vol…
Genetik -
Fenoterol Approved DB01288
small molecule | CAS: 13392-18-2

Fenoterol is an adrenergic beta-2 agonist that is used as a bronchodilator and tocolytic.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +28
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenpropidin Approved DB12728
small molecule | CAS: 67306-00-7

Fenpropidin has been investigated for the treatment of Hernia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingFungicides, Industrial +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenthion DB11412
small molecule | CAS: 55-38-9

Fenthion is an _organothiophosphate_ drug used as an insecticide, avicide, and acaricide. Its mode of action is explained by cholinesterase enzyme inhibition, which is similar to other organophosphates. Fenthion is listed as a restricted use compound by the U…

Kategori:
AgrochemicalsCholinergic AgentsCholinesterase Inhibitors +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferrous bisglycinate Approved DB11210
small molecule | CAS: 20150-34-9

Ferrous bisglycinate is a chelate that is used as a source of dietary iron. Forming a ring structure when reacting with glycine, ferrous bisglycinate acts as both a chelate and a nutritionally functional [A27250]. It is found in foods for food enrichment or i…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsIron Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fevipiprant DB12011
small molecule | CAS: 872365-14-5

Fevipiprant has been used in trials studying the treatment of Asthma, Atopic Dermatitis, and Allergic Rhinitis.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fexinidazole Approved DB12265
small molecule | CAS: 59729-37-2

Human African trypanosomiasis (HAT, also colloquially referred to as sleeping sickness), caused by _T. brucei gambiense_ and _T. brucei rhodesiense_, remains a moderate risk (>1/10,000 inhabitants per year in endemic areas) despite focussed control efforts. T…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAntiparasitic Products, Insecticides and RepellentsAntiprotozoals +43
Waktu ParuhFexinidazole, M1, a…
Vol. DistribusiFexinidazole has an…
KlirensFexinidazole has a …
Genetik -
Fezakinumab DB12344
biotech | CAS: 1007106-86-6

Fezakinumab has been used in trials studying the treatment of Atopic Dermatitis and Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fiacitabine DB12901
small molecule | CAS: 69123-90-6

Fiacitabine has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-Infective AgentsAntineoplastic AgentsAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fialuridine DB15427
small molecule | CAS: 69123-98-4

Fialuridine is under investigation in clinical trial NCT01337466 (Biodistribution and Dosimetry Evaluation of [124I]FIAU).

Kategori:
Anti-Infective AgentsAntiviral AgentsArabinonucleosides +7
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fianlimab DB18858
biotech | CAS: 2126132-98-5

Fianlimab is under investigation in clinical trial NCT06190951 (A Trial to Learn if Fianlimab and Cemiplimab Are Safe and Work Better Than Anti-pd1 Alone in Adult Participants With Resectable Stage 3 or 4 Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fibronectin DB15150
biotech

Fibronectin is under investigation in clinical trial NCT01812239 (Vaginal Progesterone in Twins With Short Cervix).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsCarbohydrates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fidanacogene elaparvovec Approved DB16783
biotech | CAS: 1954659-47-2

Fidanacogene elaparvovec is a liver-specific adeno-associated virus (AAV) vector containing a codon-optimized human coagulation FIX gene that was investigated as a potential treatment for hemophilia B.[L46691] Hemophilia B is a rare X-linked genetic disorder …

Kategori:
Adeno-associated Viral Vector TherapiesHepatotoxic Agents
Target Protein:
Coagulation factor IX (F9)
Waktu Paruh-
Vol. DistribusiIn a monkey biodist…
KlirensClearance of vector…
Genetik -
Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Figopitant DB12122
small molecule | CAS: 502422-74-4

Figopitant is under investigation in clinical trial NCT02209714 (Safety, Tolerability and Pharmacodynamics After Oral Administration of BIIF 1149 BS in Healthy Male Volunteers).

Kategori:
AcetamidesAmidesBenzene Derivatives
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filgotinib Approved DB14845
small molecule | CAS: 1206161-97-8

Rheumatoid arthritis (RA) is a chronic, autoimmune, systemic, and inflammatory disease that causes synovial joint symptoms and can limit range of motion in severe cases.[A221451,A221456] The disease is associated with extra-articular manifestations, progressi…

Kategori:
Antineoplastic and Immunomodulating AgentsArthritis, Rheumatoid, drug therapyImmunosuppressive Agents +5
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe half-life of fi…
Vol. Distribusi-
Klirens-
Genetik -
Filgrastim Approved DB00099
biotech | CAS: 121181-53-1

Filgrastim is a short-acting recombinant, non-pegylated human granulocyte colony-stimulating factor (G-CSF) analog produced by recombinant DNA technology. It has an amino acid sequence identical to endogenous G-CSF, but it is non-glycosylated unlike the endog…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBiological Factors +10
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhAfter intravenous a…
Vol. DistribusiAfter intravenous a…
KlirensClearance rates of …
Genetik -
Filociclovir DB12438
small molecule | CAS: 632325-71-4

Filociclovir is under investigation in clinical trial NCT01433835 (Safety and Pharmacokinetics of Single Oral Doses of Filociclovir in Healthy Volunteers).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filorexant DB12158
small molecule | CAS: 1088991-73-4

Filorexant has been used in trials studying the prevention and treatment of Migraine, Headache, Polysomnography, Diabetic Neuropathy, Painful, and Major Depressive Disorder, Recurrent.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fimaporfin DB17253
small molecule | CAS: 1443547-43-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finasteride Approved DB01216
small molecule | CAS: 98319-26-7

Finasteride is a synthetic 4-azasteroid compound [L10565] and specific inhibitor of steroid Type II 5?-reductase, which is an intracellular enzyme that converts the androgen testosterone into 5?-dihydrotestosterone (DHT). It works in a similar fashion as [dut…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +22
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 2Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +1
Waktu ParuhIn healthy young su…
Vol. DistribusiThe volume of distr…
KlirensIn healthy young su…
Genetik -
Fingolimod Approved DB08868
small molecule | CAS: 162359-55-9

Multiple sclerosis, or MS, is a devastating inflammatory disease that often progresses and causes severe neurological, physical, and cognitive effects.[A176474] Fingolimod is a sphingosine 1-phosphate receptor modulator for the treatment of relapsing-remittin…

Kategori:
AlcoholsAminesAmino Alcohols +16
Target Protein:
D(3) dopamine receptorSphingosine kinase 1Sphingosine 1-phosphate receptor 5 +4
Waktu ParuhThe half-life of fi…
Vol. DistribusiThe volume of distr…
KlirensFingolimod blood cl…
Genetik -
Fipaxalparant DB18124
small molecule | CAS: 1195941-38-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysophosphatidic acid receptor 1Lysophosphatidic acid receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Firategrast DB12732
small molecule | CAS: 402567-16-2

Firategrast has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FK-614 DB12557
small molecule | CAS: 193012-35-0

FK614 has been used in trials studying the treatment of Diabetes Mellitus.

Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fletikumab DB12356
biotech | CAS: 1357158-22-5

Fletikumab is under investigation in clinical trial NCT01038674 (Safety and Tolerability of Anti-IL-20 in Subjects With Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluasterone DB06250
small molecule | CAS: 112859-71-9

Has antiproliferative effects on HIV-1 and reduces HIV-1 replication.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fludeoxyglucose (18F) Approved DB09502
small molecule | CAS: 63503-12-8

Fludeoxyglucose F 18 Injection is a positron emitting radiopharmaceutical containing no-carrier added radioactive 2-deoxy-2-[18F]fluoro-D-g1ucose, which is used for diagnostic purposes in conjunction with Positron Emission Tomography (PET). It is administered…

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDeoxy Sugars +10
Waktu Paruh10-13 minutes
Vol. DistribusiFludeoxyglucose F 1…
KlirensFludeoxyglucose F 1…
Genetik -
Fludrocortisone Approved DB00687
small molecule | CAS: 127-31-1

Fludrocortisone is a synthetic mineralocorticoid used in conjunction with [hydrocortisone] to replace missing endogenous corticosteroids in patients with adrenal insufficiency.[A187169,A187187] It is functionally similar to [aldosterone], the body's primary e…

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +18
Target Protein:
Androgen receptorMineralocorticoid receptorGlucocorticoid receptor
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensPopulation pharmaco…
Genetik -
Fluindione Approved DB13136
small molecule | CAS: 957-56-2

Fluindione is under investigation for the treatment of Venous Thrombosis, Pulmonary Embolism, Permanent Atrial Fibrillation, and Anticoagulating Treatment on a Duration at Least 12-month-old Superior. Fluindione has been investigated for the treatment of Bloo…

Kategori:
AnticoagulantsBlood and Blood Forming OrgansCytochrome P-450 CYP2C9 Substrates +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flumazenil Approved DB01205
small molecule | CAS: 78755-81-4

Fumazenil is an imidazobenzodiazepine derivative and a potent benzodiazepine receptor antagonist that competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex, thereby reversing the effects of benz…

Kategori:
AntidotesBenzazepinesBenzodiazepine Antagonist +9
Target Protein:
Translocator proteinGamma-aminobutyric acid receptor subunit gamma-2Gamma-aminobutyric acid receptor subunit alpha-2 +5
Waktu ParuhInitial distributio…
Vol. Distribusi* 0.9 to 1.1 L/kg
Klirens* 1 L/hr/kg [health…
Genetik -
Fluocinolone DB12553
small molecule | CAS: 807-38-5

Fluocinolone has been used in trials studying the treatment and prevention of Candida Infection, Oral Lichen Planus, Macular Degeneration, and Choroidal Neovascularization.

Kategori:
Fused-Ring CompoundsPregnadienesPregnanes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluocinonide Approved DB01047
small molecule | CAS: 356-12-7

A topical glucocorticoid used in the treatment of eczema.

Kategori:
Adrenal Cortex HormonesAnti-Allergic AgentsAnti-Inflammatory Agents +24
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluocortin DB13223
small molecule | CAS: 33124-50-4

Fluocortin has been studied as a corticosteroid for treatment of dermatitis and eczema Spain [A174817].

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids, Dermatological Preparations +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluorescein Approved DB00693
small molecule | CAS: 2321-07-5

A phthalic indicator dye that appears yellow-green in normal tear film and bright green in a more alkaline medium, such as the aqueous humor, and is used therapeutically as a diagnostic aid in corneal injuries and corneal trauma. It has been approved by FDA f…

Kategori:
BSEP/ABCB11 SubstratesColoring AgentsColouring Agents +21
Target Protein:
Organic anion transporter 3Immunoglobulin kappa variable 2-30DNA
Waktu Paruh-
Vol. Distribusi* 0.5 L/kg
Klirens* renal cl=1.75 mL/…
Genetik -
small molecule | CAS: 140616-46-2

Fluorescein lisicol has been used in trials studying the diagnostic of Pharmacokinetics, Hepatic Cirrhosis, Hepatitis, Viral, Human, Nonalcoholic Steatohepatitis, and Non-Alcoholic Fatty Liver Disease.

Kategori:
Heterocyclic Compounds, Fused-RingSpiro CompoundsXanthenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1201–1250 dari 3253
Sebelumnya Halaman 25 / 66 Berikutnya