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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 249 / 272
Tetroxoprim DB15976
small molecule | CAS: 53808-87-0

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tetryzoline Approved DB06764
small molecule | CAS: 84-22-0

Tetryzoline, also known as tetrahydrozoline, is a derivative of imidazoline with central and peripheral alpha (?)-adrenergic properties.[A231769] Available since the 1950s, tetryzoline is a selective ?<sub>1</sub>-receptor agonist [A231774] that is used as a…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +20
Target Protein:
Alpha-1 adrenergic receptorsAlpha-2C adrenergic receptorAlpha-2 adrenergic receptors
Waktu ParuhFollowing ocular ad…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
small molecule

Betalutin has been used in trials studying the treatment of Non-Hodgkin Lymphoma and Relapsed, Diffuse Large B-cell Lymphoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tezacaftor Approved DB11712
small molecule | CAS: 1152311-62-0

Tezacaftor is a drug of the cystic fibrosis transmembrane conductance regulator (CFTR) potentiator class.[L1595] It was developed by Vertex Pharmaceuticals and FDA approved in combination with [ivacaftor] to manage cystic fibrosis.[L6814] This drug was approv…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesCytochrome P-450 CYP1A2 Inhibitors +33
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Tezacitabine DB06433
small molecule | CAS: 171176-43-5

A synthetic purine nucleoside analogue with potential antineoplastic activity.

Kategori:
Antineoplastic AgentsDeoxyribonucleosidesEnzyme Inhibitors +6
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tezampanel DB06354
small molecule | CAS: 154652-83-2

Tezampanel is an AMPA receptor antagonist.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, AMPA, antagonists & inhibitors
Target Protein:
Glutamate receptor ionotropic, kainate 1Gamma-aminobutyric acid type B receptor subunit 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tezepelumab Approved DB15090
biotech | CAS: 1572943-04-4

Asthma is a heterogeneous chronic obstructive respiratory disease with both "type 2" (T2) and T2-low endotypes characterized by reduced airflow, chronic inflammation, and airway remodelling.[A243764, A243769] Thymic stromal lymphopoietin (TSLP), an innate ple…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Thymic stromal lymphopoietin
Waktu ParuhTezepelumab has an …
Vol. DistribusiTezepelumab has a c…
KlirensTezepelumab has an …
Genetik -
Tezosentan DB06558
small molecule | CAS: 180384-57-0

Tezosentan is an intravenous endothelin receptor A/B antagonist. Tezosentan was initially developed for vasodilation in patients with acute heart failure but studies have shown that it does not assist in the treatment of dyspnea or prevent cardiovascular even…

Kategori:
Cardiovascular AgentsReceptors, EndothelinVasodilating Agents
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhA pronounced and ra…
Vol. Distribusi-
Klirens-
Genetik -
TG-100801 DB05075
small molecule | CAS: 867331-82-6

TG100801 is a topically applied kinase inhibitor in macular degeneration patients. It is administered noninvasively as an eye drop and is designed to suppress VEGF mediated leakage and additional kinase targets associated with inflammation, edema, and angioge…

Kategori:
Benzene Derivatives
Target Protein:
Vascular endothelial growth factor CVascular endothelial growth factor DVascular endothelial growth factor A, long form +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
TG-1042 DB18435
biotech

TG-1042 (formerly known as ASN-002) is a recombinant adenovirus carrying the cDNA coding sequence for the human interferon gamma gene.

Waktu Paruh-
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TG01 vaccine DB17123
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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TG100-115 DB05552
small molecule | CAS: 677297-51-7

An NSAID that inhibits PI-3K gamma and delta.

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG4010 DB06584
biotech | CAS: 350485-85-7

A bivalent cancer vaccine comprised of a modified vaccinia virus Ankara (MVA) strain encoding human mucin 1 (MUC1) and interleukin-2 (IL-2) with potential immunostimulating and antineoplastic activities. Originally developed for the eradication of smallpox, M…

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsCarbohydrates +6
Target Protein:
Mucin-1Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG4023 DB06108
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
TGAAC09 DB06363
biotech

tgAAC09 is an investigational vaccine that utilizes an AAV vector to deliver genes that encode HIV proteins. It was under investigation in clinical trials NCT00482027 and NCT00888446 for the treatment of HIV Infection.

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TGAAC94 DB06175
small molecule

tgAAC94 is a recombinant adeno-associated virus serotype 2 (AAV2) vector containing the cDNA for a human tumor necrosis factor receptor (TNFR)-immunoglobulin (IgG1) Fc fusion (TNFR:Fc) gene. It was under investigation in clinical trials to treat Inflammatory …

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 1373958-68-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingXanthenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TH0318 DB05145
biotech

TH0318 is a stabilized analogue of human GLP-1 (glucagon-like peptide-1) under investigation for the treatment of type 2 diabetes.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Thalagen DB17714
biotech

Thalagen is a branded product developed by San Rocco Therapeutics. It consists of autologous CD34-positive hematopoietic progenitor cells transduced with TNS9.3.55, a lentiviral vector encoding the normal human beta-globin gene. It is being investigated for t…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Thalidomide Approved DB01041
small molecule | CAS: 50-35-1

A piperidinyl isoindole originally introduced as a non-barbiturate hypnotic, thalidomide was withdrawn from the market due to teratogenic effects. It has been reintroduced and used for a number of inflammatory disorders and cancers. Thalidomide displays immun…

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +38
Target Protein:
Tumor necrosis factorProtein cereblonDNA +1
Waktu ParuhThe half-life of th…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Thallium Tl-201 DB15361
small molecule | CAS: 15064-65-0

Thallium Tl-201 is under investigation in clinical trial NCT02697760 (The CZT Dynamic Myocardial Perfusion Imaging).

Kategori:
IsotopesRadioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thallous chloride Approved DB09316
small molecule | CAS: 7791-12-0

Thallous chloride (also known as Thallium(I) chloride) is a colourless solid intermediate in the isolation of thallium from its ores. It is created from the treatment of thallium(I) sulfate with hydrochloric acid. This solid crystallizes in the caesium chlori…

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh91% of the blood ra…
Vol. Distribusi3–10 L/kg
KlirensApproximately 4-8% …
Genetik -
THE-630 DB16750
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Theanine DB12444
small molecule | CAS: 3081-61-6

Theanine, a precursor of ethylamine, is found in green tea. It is under investigation in clinical trial NCT00291070 (Effects of L-Theanine in Boys With ADHD).

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thebacon DB13458
small molecule | CAS: 466-90-0

Deskripsi belum tersedia.

Kategori:
Cough and Cold PreparationsOpium Alkaloids and Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thenalidine Approved DB04826
small molecule | CAS: 86-12-4

Withdrawn from the Canadian, US, and UK markets in 1963 due to concerns involving neutropenia.

Kategori:
Antihistamines for Systemic UseAntihistamines for Topical UseAntipruritics, Incl. Antihistamines, Anesthetics, Etc. +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 326-91-0

Thenoyltrifluoroacetone is a chelating agent and inhibitor of cellular respiration.

Kategori:
ButanonesChelating AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
Liver carboxylesterase 1Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theobromine DB01412
small molecule | CAS: 83-67-0

Theobromine (3,7-dimethylxanthine) is the principle alkaloid in Theobroma cacao (the cacao bean) and other plants. A xanthine alkaloid that is used as a bronchodilator and as a vasodilator. It has a weaker diuretic activity than theophylline and is also a les…

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +15
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theodrenaline DB12927
small molecule | CAS: 13460-98-5

Theodrenaline is under investigation in clinical trial NCT01311414 (Effect of Cafedrine/Theodrenaline and Urapidil on Cerebral Oxygenation).

Kategori:
Adrenergic and Dopaminergic AgentsAgents that produce hypertensionAlcohols +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theophylline Approved DB00277
small molecule | CAS: 58-55-9

A methylxanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant activities. Mechanistically, theophylline acts as a phosphodiesterase inhibitor, adenosine receptor blocker, and histo…

Kategori:
Agents that reduce seizure thresholdAlkaloidsAnti-Asthmatic Agents +32
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +12
Gen Terkait:
CYP1A2
Waktu Paruh8 hours
Vol. Distribusi* 0.3 to 0.7 L/kg
Klirens* 0.29 mL/kg/min [P…
Genetik 1 Varian
Theralizumab DB15717
biotech | CAS: 906068-56-2

Theralizumab is a humanized anti-CD28 monoclonal antibody designed for treating autoimmune diseases and cancer. After the first human trial, it was withdrawn due to severe toxicity (likely due to lymphopenia and human cytokine release).[A216527,A216532]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thermomyces lanuginosus Approved DB10973
biotech

Thermomyces lanuginosus allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiabendazole Approved DB00730
small molecule | CAS: 148-79-8

2-Substituted benzimidazole first introduced in 1962. It is active against a variety of nematodes and is the drug of choice for strongyloidiasis. It has CNS side effects and hepatototoxic potential. (From Smith and Reynard, Textbook of Pharmacology, 1992, p91…

Kategori:
AnthelminticsAnti-Infective AgentsAntifungals for Dermatological Use +18
Target Protein:
Fumarate reductase flavoprotein subunit
Waktu ParuhThe half-life for t…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 67-16-3

Deskripsi belum tersedia.

Kategori:
PyrimidinesSulfur CompoundsThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10023-48-0

Deskripsi belum tersedia.

Target Protein:
Thiamine-phosphate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamphenicol DB08621
small molecule | CAS: 15318-45-3

Deskripsi belum tersedia.

Kategori:
AlcoholsAmphenicolsAnti-Bacterial Agents +8
Target Protein:
Dr hemagglutinin structural subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamylal Approved DB01154
small molecule | CAS: 77-27-0

A barbiturate that is administered intravenously for the production of complete anesthesia of short duration, for the induction of general anesthesia, or for inducing a hypnotic state. (From Martindale, The Extra Pharmacopoeia, 30th ed, p919)

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +22
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3ATP-sensitive inward rectifier potassium channel 8ATP-sensitive inward rectifier potassium channel 11 +1
Waktu ParuhAlthough no studies…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Arsenate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiazinam DB13420
small molecule | CAS: 2338-21-8

Deskripsi belum tersedia.

Kategori:
AminesAntihistamines for Systemic UseAntipsychotic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activatorSerine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiethylperazine Approved DB00372
small molecule | CAS: 1420-55-9

A dopamine antagonist that is particularly useful in treating the nausea and vomiting associated with anesthesia, mildly emetic cancer chemotherapy agents, radiation therapy, and toxins. This piperazine phenothiazine does not prevent vertigo or motion sicknes…

Kategori:
AntiemeticsAntihistamines for Systemic UseAntipsychotic Agents +16
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyclomaltodextrin glucanotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiocellobiose DB03263
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiocitrulline DB03953
small molecule | CAS: 156719-37-8

Deskripsi belum tersedia.

Kategori:
AmidesAmino AcidsAmino Acids, Diamino +4
Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 602-41-5

Thiocolchicoside is a semi-synthetic derivative of the colchicine, a natural anti-inflammatory glycoside which originates from the flower seeds of _Superba gloriosa_. It is a muscle relaxant with anti-inflammatory and analgesic effects. It has potent convul…

Kategori:
AlkaloidsCentral Nervous System DepressantsMuscle Relaxants +2
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Glycine receptor subunit alpha-2 +6
Waktu ParuhApproximately 7.7h …
Vol. DistribusiThe apparent volume…
KlirensPrimarily extrarena…
Genetik -
Thioctamide DB15963
small molecule | CAS: 940-69-2

Deskripsi belum tersedia.

Kategori:
CoenzymesEnzymes and CoenzymesFatty Acids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 137314-40-0

A salt of alpha-lipoic acid and tromethamine; may be useful in treating vascular stress in patients with diabetes.

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Genetik -
small molecule | CAS: 51555-87-4

Thiodigalactoside is a solid. This compound belongs to the dihexoses. These are disaccharides containing two hexose carbohydrates. This medication is known to target galectin-1, heat-labile enterotoxin b chain, neurocan core protein, and lactose permease.

Kategori:
CarbohydratesGalactosidesGlycosides +2
Target Protein:
Heat-labile enterotoxin B chainLactose permeaseNeurocan core protein +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12401–12450 dari 13591
Sebelumnya Halaman 249 / 272 Berikutnya