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12560

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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 247 / 252
WT-1 427 long DB17354
biotech | CAS: 935395-33-8

Deskripsi belum tersedia.

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WT-1 A1 DB17352
small molecule | CAS: 852243-39-1

Deskripsi belum tersedia.

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WU-NK-101 DB18350
biotech

WU-NK-101 is an allogeneic CD3-depleted, CD56-enriched activated natural killer-cell product

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WVE-N531 DB17848
biotech

Deskripsi belum tersedia.

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WX-UK1 DB05476
small molecule | CAS: 255374-84-6

WX-UK1 is a 3-amidinophenylalanine-based non-cytotoxic small molecule that belongs to a new class of drugs. In animal models, WX-UK1 blocks tumor cell invasion, metastasis and primary tumor growth by inhibiting serine proteases and the urokinase Plasminogen A…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Urokinase plasminogen activator surface receptor
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X-165 DB18053
small molecule | CAS: 1815589-34-4

Deskripsi belum tersedia.

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X-396 DB13104
small molecule | CAS: 1365267-27-1

X-396 has been used in trials studying the treatment of Advanced Solid Tumors and Non-small Cell Lung Cancer.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
ALK tyrosine kinase receptor
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Xaliproden DB06393
small molecule | CAS: 135354-02-8

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNervous System +5
Target Protein:
5-hydroxytryptamine receptor 1A
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Xanomeline Approved DB15357
small molecule | CAS: 131986-45-3

Schizophrenia is a complex disease involving a number of different neurotransmitters, including serotonin, dopamine, and acetylcholine.[A264509] Positive symptoms (e.g. hallucinations, delusions) have traditionally been attributed to increased dopaminergic ac…

Kategori:
Autonomic AgentsCentral Nervous System AgentsCholinergic Agents +18
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe half-life of xa…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
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Xanthan gum Approved DB11253
small molecule | CAS: 11138-66-2

Xanthan gum is a polysaccharide gum derived from* Xanthomonas campestris* by a pure-culture fermentation process and purified by recovery with isopropyl alcohol. The major constituents include D-glucose, D-mannose, and D-glucuronic acid. Xanthan gum is a dire…

Kategori:
AntigensAntigens, BacterialBiological Factors +9
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Xanthinol Approved DB09092
small molecule | CAS: 2530-97-4

Xanthinol is a very potent water-soluble derivative of niacin that can be found in diet supplements. It is also known as xanthinol nicotinate. [L1079] Xaninthol is known to be a potent vasodilator that can easily pass through the cell membrane and once inside…

Kategori:
Cardiovascular AgentsHeterocyclic Compounds, Fused-RingNicotinic Acids +6
Target Protein:
NAD(P) transhydrogenase, mitochondrialGlyceraldehyde-3-phosphate dehydrogenaseIsocitrate dehydrogenase [NAD] subunit alpha, mitochondrial +3
Waktu ParuhThe reported elimin…
Vol. DistribusiThe volume of distr…
KlirensThe total body clea…
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Xanthium strumarium pollen Approved DB10356
biotech

Xanthium strumarium pollen is the pollen of the Xanthium strumarium plant. Xanthium strumarium pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Xanthohumol DB15359
small molecule | CAS: 6754-58-1

Xanthohumol is under investigation in clinical trial NCT01367431 (Xanthohumol and Metabolic Syndrome).

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +7
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XAV-19 DB15895
biotech

XAV-19 is an intravenous antibody-based treatment targeted towards SARS-CoV-2 and other coronaviruses[L16553,L16558]. The therapy concept is based on [COVID-19 convalescent plasma]. However, rather than using human plasma, XAV-19 is a heterologous swine glyco…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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XC221 DB16503
small molecule

XC221 was investigated in clinical trials to treat patients with respiratory infections, including influenza, COVID-19, and other acute viral upper respiratory infections.

Kategori:
Experimental Unapproved Treatments for COVID-19
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Xeligekimab DB18869
biotech | CAS: 2382921-73-3

Xeligekimab is under investigation in clinical trial NCT06028490 (A Study of Il4r? Monoclonal Antibody in Patients With Uncontrolled Seasonal Allergic Rhinitis.).

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XEN-2174 DB05012
small molecule | CAS: 701909-57-1

XEN-2174 is a synthetic drug modeled on a peptide from the venom of a cone shell found on Australia's Great Barrier Reef. XEN-2174 represents a new class of molecules, called the chi conopeptides that selectively inhibit the Norepinephrine Transporter (NET). …

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Sodium-dependent noradrenaline transporter
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XEN-D0101 DB06020
small molecule

XEN-D0101 is an investigational drug developed by Xention Inc. for the treatment of Atrial Fibrillation. XEN-D0101 works by being a selective antagonist of the voltage-gated potassium channel Kv1.5.

Kategori:
Kv1.5 Potassium Channel, antagonists & inhibitorsSulfur Compounds
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XEN-D0501 DB18673
small molecule

XEN-D0501 is a tetrahydronaphthyl urea-based selective TRPV1 antagonist being investigated for the treatment of erythromelalgia.

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Xenon DB13453
small molecule | CAS: 7440-63-3

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +7
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Xenon Xe-129 Approved DB17386
small molecule | CAS: 13965-99-6

Hyperpolarized Xenon-129 (Xe-129) is a contrast agent used in the lung's clinical magnetic resonance imaging (MRI). Lung MRIs are challenging due to the low proton density of this tissue, as well as the presence of artifacts due to respiration and cardiovascu…

Kategori:
Contrast MediaDiagnostic Uses of ChemicalsHyperpolarized Contrast Agent +3
Waktu ParuhXenon-129 in a 75% …
Vol. DistribusiXenon is readily di…
KlirensNot available.
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Xenon-133 Approved DB09315
small molecule | CAS: 14932-42-4

Xenon-133 is an inhaled radionuclide used for lung imaging, imaging blood flow in the brain, and to assess pulmonary function.

Kategori:
Diagnostic RadiopharmaceuticalsElementsGases +6
Waktu ParuhHalf Life 5.245 days
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Xentuzumab DB14871
biotech | CAS: 1417158-65-6

Xentuzumab is under investigation in clinical trial NCT02191891 (Xentuzumab (BI 836845) Plus Afatinib in Patients With Epidermal Growth Factor Receptor (EGFR) Mutant Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Xenysalate DB13815
small molecule | CAS: 3572-52-9

Deskripsi belum tersedia.

Kategori:
DermatologicalsMedicated Shampoos
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Xevinapant DB16305
small molecule | CAS: 1071992-99-8

Deskripsi belum tersedia.

Kategori:
Benzene Derivatives
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
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small molecule | CAS: 157435-10-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 2-beta
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XL-888 DB12981
small molecule | CAS: 1149705-71-4

XL888 has been used in trials studying the treatment of Cancer and Melanoma.

Kategori:
Acids, CarbocyclicAza CompoundsHSP90 Heat-Shock Proteins, antagonists & inhibitors
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XL019 DB05243
small molecule

XL019 is a selective inhibitor of the cytoplasmic tyrosine kinase JAK2. An IND for XL019 was filed by Exelixis in May 2007.

Target Protein:
Tyrosine-protein kinase JAK2
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XL228 DB05184
small molecule

XL228 is a novel anticancer compound designed to inhibit the insulin-like growth factor type-1 receptor (IGF1R), Src and Abl tyrosine kinases – targets that play crucial roles in cancer cell proliferation, survival and metastasis.

Target Protein:
Insulin-like growth factor 1 receptorProto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase ABL1 +1
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XL281 DB05190
small molecule

XL281 is a novel anticancer compound designed to potently inhibit the RAS/RAF/MEK/ERK signaling pathway. Mutational activation of RAS occurs in about 30 percent of all human tumors, including non-small cell lung, pancreatic, and colon cancer. XL281 is a speci…

Target Protein:
Serine/threonine-protein kinase B-rafRAF proto-oncogene serine/threonine-protein kinase
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XL418 DB05204
small molecule

XL418 is a novel anticancer compound.

Target Protein:
Tyrosine-protein kinase BTK
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XL765 DB05241
small molecule

XL765 is an orally available small molecule that has been shown in preclinical studies to selectively inhibit the activity of phosphoinositide-3 kinase (PI3K) and mammalian target of rapamycin (mTOR). It is being developed by Exelixis, Inc.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform +2
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XL820 DB05146
small molecule | CAS: 1123889-88-2

XL820 is investigated for use/treatment in solid tumors. XL820 is a solid. The proteins that XL820 inhibit include platelet-derived growth factor receptor beta (PDGFR), mast/stem cell growth factor receptor KIT, vascular endothelial growth factor receptor 2, …

Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor KitPlatelet-derived growth factor receptor alpha +1
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XL844 DB05149
small molecule

XL844 is investigated for the use and treatment solid tumors. XL844 is a solid. XL844 is a potent inhibitor of the checkpoint kinases CHK1 and CHK2, which induce cell cycle arrest in response to a variety of DNA damaging agents. Known drug targets of XL844 in…

Target Protein:
Serine/threonine-protein kinase Chk2Serine/threonine-protein kinase Chk1
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XL999 DB05014
small molecule | CAS: 921206-68-0

XL999 has the potential to provide benefit to patients with lung cancer and acute myelogenous leukemia. XL999 is a new chemical entity that inhibits a spectrum of receptor tyrosine kinases (RTKs) with growth promoting and angiogenic properties, including FGFR…

Target Protein:
Fibroblast growth factor receptor 3Fibroblast growth factor receptor 1Vascular endothelial growth factor receptor 2 +3
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XmAb 2513 DB06324
biotech

XmAb 2513 is a humanized monoclonal antibody that targets the antigen CD30, a molecule expressed on the surface of a number of tumor cell types. It has been investigated for the treatment of hodgkin’s lymphoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Tumor necrosis factor receptor superfamily member 8
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XmAb24306 DB17526
biotech

XmAb24306 is an investigational cancer immunotherapy. It is a heterodimeric interleukin (IL)-15/IL-15-receptor alpha (IL-15Ra) complex fused to a bispecific Fc domain.

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biotech

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XMT-2056 DB18230
biotech

XMT-2056 is a HER2-targeted antibody-drug conjugate (ADC) consisting of a HER2-targeted antibody conjugated with a stimulator of interferon genes (STING) agonist payload.

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XPro1595 DB16454
biotech | CAS: 2489785-77-3

XPro1595 is an investigational dominant-negative protein that neutralizes soluble TNF.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +10
Target Protein:
Tumor necrosis factor
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XR5944 DB06364
small molecule | CAS: 343247-32-5

XR5944 is a DNA bis-intercalating anticancer drug. It has both intercalating and antineoplastic activities.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
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XTL-001 DB05405
biotech | CAS: 339991-45-6

XTL001 is an investigational monoclonal antibody (MAb) product developed by XTL Biopharmaceuticals to evaluate the safety profile and antiviral activity of the compound in patients chronically infected with hepatitis B virus (HBV).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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XTL-6865 DB06058
small molecule

XTL-6865 is a combination of two fully human monoclonal antibodies (Ab68 and Ab65) against the hepatitis C virus E2 envelope protein. It is being developed to prevent HCV re-infection following a liver transplant and for the treatment of chronic HCV disease.

Target Protein:
Genome polyprotein
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XV638 DB02702
small molecule | CAS: 183854-11-7

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
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Xylazine DB11477
small molecule | CAS: 7361-61-7

Xylazine is a clonidine analog used as a non-opioid tranquilizer in veterinary medicine and as an emetic, especially in cats.[A9095,L42675,A251420] It acts as an agonist at ?2 adrenoceptors; however, its affinity is lower than the one reported for other ?2 ad…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +15
Target Protein:
Alpha-2B adrenergic receptorAlpha-2C adrenergic receptorAlpha-2 adrenergic receptors
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Xylitol DB11195
small molecule | CAS: 87-99-0

Xylitol is a naturally occurring five-carbon sugar alcohol found in most plant material, including many fruits and vegetables. Xylitol-rich plant materials include birch and beechwood [A22081]. It is widely used as a sugar substitute and in "sugar-free" food …

Kategori:
AlcoholsCarbohydratesCompounds used in a research, industrial, or household setting +8
Target Protein:
Xylose isomeraseXylose isomeraseXylose isomerase +2
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Xylometazoline Approved DB06694
small molecule | CAS: 526-36-3

Xylometazoline is an imidazoline derivative [A228523] with sympathomimetic and nasal decongestant activity. Xylometazoline works by binding to alpha (?)-adrenergic receptors to cause vasoconstriction of nasal blood vessels.[A228508] Xylometazoline is avail…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +17
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-1A adrenergic receptor +3
Waktu ParuhNo information is a…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Xylose Approved DB09419
small molecule | CAS: 58-86-6

Xylose is a monosaccharide of the aldopentose type consisted of five carbon atoms and an aldehyde functional group. Xylose is a sugar isolated from wood. D-Xylose is a sugar widely used as a diabetic sweetener in food and beverage. Xylose has also been used a…

Kategori:
CarbohydratesMonosaccharidesPentoses
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
Y-27632 DB08756
small molecule | CAS: 146986-50-7

Y-27632 is an inhibitor of Rho-associated protein kinase. It inhibits calcium sensitization to affect smooth muscle relaxation.

Kategori:
Antihypertensive AgentsCardiovascular AgentsCentral Nervous System Agents +6
Target Protein:
ProthrombincAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alpha +2
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YA-101 DB18121
small molecule | CAS: 151602-49-2

Deskripsi belum tersedia.

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