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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 246 / 321
Phenaridine DB09178
small molecule | CAS: 42045-97-6

Phenaridine (2,5-Dimethylfentanyl) is a synthetic fentanyl derivative opioid. It was developed in 1972, and is used for surgical anasthesia in Russia. Phenaridine has similar effects to fentanyl. In rat studies, it was less potent than fentanyl. Side effects …

Kategori:
AminesAminopyridinesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenazepam DB19164
small molecule | CAS: 51753-57-2

Phenazepam is under investigation in clinical trial NCT03017430 (Pregabalin for Opiate Withdrawal Syndrome).

Kategori:
Adjuvants, ImmunologicAntiarrhythmic agentsAnticonvulsants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenazocine DB13606
small molecule | CAS: 58073-76-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsBenzomorphan Derivatives +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenazopyridine Approved DB01438
small molecule | CAS: 94-78-0

Phenazopyridine, also known as Pyridium, is a urinary tract analgesic used for the short-term management of urinary tract irritation and its associated unpleasant symptoms such as burning and pain during urination. In the USA, this drug was previously marked …

Kategori:
AminesAminopyridinesAntipruritics and Local Anesthetics +6
Target Protein:
Sodium channel protein type 1 subunit alphaGroup A nerve fibers
Waktu ParuhThe mean eliminatio…
Vol. DistribusiSmall, trace quanti…
KlirensThis drug is rapidl…
Genetik -
Phencyclidine DB03575
small molecule | CAS: 77-10-1

A hallucinogen formerly used as a veterinary anesthetic, and briefly as a general anesthetic for humans. Phencyclidine is similar to ketamine in structure and in many of its effects. Like ketamine, it can produce a dissociative state. It exerts its pharmacolo…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Inhibitors +11
Target Protein:
Glutamate receptor ionotropic, NMDA 3AGlutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 2A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phendimetrazine Approved DB01579
small molecule | CAS: 634-03-7

Phendimetrazine is a weight loss medication. Phendimetrazine is chemically related to amphetamines and is a Schedule III drug under the Convention on Psychotropic Substances and in the US since 1970.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Alpha-1A adrenergic receptorSodium-dependent noradrenaline transporterAlpha-1B adrenergic receptor
Waktu Paruh19-24 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenelzine Approved DB00780
small molecule | CAS: 51-71-8

Phenelzine, with the formula ?-phenylethylhydrazine, is a monoamine oxidase inhibiting antidepressant that is effective in the treatment of panic disorder and social anxiety disorder.[A15753] It was developed by Parke Davis and originally FDA approved on June…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +33
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] BAmine oxidase [copper-containing] 3 +4
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
small molecule | CAS: 2257-09-2

Phenethyl Isothiocyanate has been used in trials studying the prevention and treatment of Leukemia, Lung Cancer, Tobacco Use Disorder, and Lymphoproliferative Disorders.

Kategori:
Aldehyde Dehydrogenase, antagonists & inhibitorsAnticarcinogenic AgentsAntineoplastic Agents +8
Target Protein:
Actin, aortic smooth muscleActin, cytoplasmic 1ATP synthase subunit beta, mitochondrial +42
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenethylamine DB04325
small molecule | CAS: 64-04-0

Deskripsi belum tersedia.

Kategori:
AminesCentral Nervous System AgentsCentral Nervous System Depressants +2
Target Protein:
5-hydroxytryptamine receptor 2APrimary amine oxidaseSerine protease 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pheneticillin Approved DB13337
small molecule | CAS: 147-55-7

Pheneticillin (or phenethicillin) is a penicillin antibiotic which is approved for use internationally.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pheneturide DB13362
small molecule | CAS: 90-49-3

Deskripsi belum tersedia.

Kategori:
AmidesAnticonvulsantsCentral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenformin Approved DB00914
small molecule | CAS: 114-86-3

A biguanide hypoglycemic agent with actions and uses similar to those of metformin. Although it is generally considered to be associated with an unacceptably high incidence of lactic acidosis, often fatal, it is still available in some countries. (From Martin…

Kategori:
Alimentary Tract and MetabolismAmidinesBiguanides +9
Target Protein:
5'-AMP-activated protein kinase catalytic subunit alpha-15'-AMP-activated protein kinase subunit gamma-15'-AMP-activated protein kinase subunit beta-1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenglutarimide DB13413
small molecule | CAS: 1156-05-4

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenibut DB13455
small molecule | CAS: 1078-21-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenindamine Approved DB01619
small molecule | CAS: 82-88-2

Phenindamine is an antihistamine. Phenindamine blocks the effects of the naturally occurring chemical histamine in your body. Antihistamines such as phenindamine appear to compete with histamine for histamine H1- receptor sites on effector cells. The antihist…

Kategori:
Antihistamines for Systemic UseHistamine AgentsHistamine Antagonists +2
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenindione Approved DB00498
small molecule | CAS: 83-12-5

An indandione that has been used as an anticoagulant. Phenindione has actions similar to warfarin, but it is now rarely employed because of its higher incidence of severe adverse effects. (From Martindale, The Extra Pharmacopoeia, 30th ed, p234)

Kategori:
AnticoagulantsBlood and Blood Forming OrgansHematologic Agents +4
Target Protein:
Vitamin K epoxide reductase complex subunit 1
Waktu Paruh5-10 hours
Vol. Distribusi-
Klirens-
Genetik -
Pheniprazine DB09250
small molecule | CAS: 55-52-7

Pheniprazine is an irreversible and nonselective monoamine oxidase inhibitor (MAOI) of the hydrazine chemical class that was used as an antidepressant in the 1960s. In addition, it was used for the treatment of other conditions, such as angina pectoris and sc…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pheniramine Approved DB01620
small molecule | CAS: 86-21-5

Pheniramine is a first-generation antihistamine in the alkylamine class, similar to [brompheniramine] and [chlorpheniramine].[A181628] It is used in some over-the-counter allergy as well as cold & flu products in combination with other drugs. Pheniramine's …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseAntihistamines for Topical Use +10
Target Protein:
Histamine H4 receptorHistamine H1 receptorNuclear receptor subfamily 1 group I member 3
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
Klirens-
Genetik -
Phenmetrazine Approved DB00830
small molecule | CAS: 134-49-6

A sympathomimetic drug used primarily as an appetite depressant. Its actions and mechanisms are similar to dextroamphetamine.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnti-Obesity Agents +8
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Waktu Paruh16 to 31 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenobarbital Approved DB01174
small molecule | CAS: 50-06-6

A barbituric acid derivative that acts as a nonselective central nervous system depressant. It promotes binding to inhibitory gamma-aminobutyric acid subtype receptors, and modulates chloride currents through receptor channels. It also inhibits glutamate indu…

Kategori:
Anticholinergic AgentsAnticonvulsantsBarbiturates +57
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7 +4
Waktu Paruh53 to 118 hours (me…
Vol. Distribusi-
Klirens-
Genetik -
Phenol Approved DB03255
small molecule | CAS: 108-95-2

Phenol is an antiseptic and disinfectant. It is active against a wide range of micro-organisms including some fungi and viruses, but is only slowly effective against spores. Phenol has been used to disinfect skin and to relieve itching. Phenol is also used as…

Kategori:
AnestheticsAnesthetics, LocalAnti-Infective Agents +19
Target Protein:
Carbonic anhydrase 1Carbonic anhydrase 4Carbonic anhydrase 12 +5
Waktu Paruh-
Vol. DistribusiAt I5 min after exp…
KlirensIn rabbits, 72% is …
Genetik -
Phenolphthalein Approved DB04824
small molecule | CAS: 77-09-8

Phenolphthalein was withdrawn in Canada due to concerns with carcinogenicity in 1997.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesCompounds used in a research, industrial, or household setting +7
Target Protein:
UDP-glucuronosyltransferase 1A9Nuclear receptor subfamily 1 group I member 2Nuclear receptor subfamily 1 group I member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 98-67-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 143-74-8

Phenolsulfonphthalein or otherwise called phenol red is a pH indicator commonly used in cell biology laboratories. Phenolsulfonphthalein is being investigated for use clinically due to its weak estrogen mimicking actions [A174964].

Kategori:
Benzene DerivativesColoring AgentsCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenoperidine DB13605
small molecule | CAS: 562-26-5

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnestheticsAnesthetics, General +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenothiazine DB11447
small molecule | CAS: 92-84-2

Phenothiazine (PTZ) is an organic thiazine compound.

Kategori:
Agents that reduce seizure thresholdAnti-Infective AgentsAntiparasitic Agents +3
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenothrin DB13717
small molecule | CAS: 26002-80-2

Deskripsi belum tersedia.

Kategori:
AgrochemicalsAntiparasitic Products, Insecticides and RepellentsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenoxybenzamine Approved DB00925
small molecule | CAS: 59-96-1

An alpha-adrenergic antagonist with long duration of action. It has been used to treat hypertension and as a peripheral vasodilator.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +13
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorAlpha-2A adrenergic receptor +6
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenoxyethanol Approved DB11304
small molecule | CAS: 122-99-6

Phenoxyethanol is a colorless liquid with a pleasant odor. It is a glycol ether used as a perfume fixative, insect repellent, antiseptic, solvent, preservative, and also as an anesthetic in fish aquaculture. Phenoxyethanol is an ether alcohol with aromatic pr…

Kategori:
AlcoholsAnestheticsAnti-Infective Agents +5
Waktu Paruh-
Vol. DistribusiA pharmacokinetic s…
Klirens-
Genetik -
Phenoxymethylpenicillin Approved DB00417
small molecule | CAS: 87-08-1

Phenoxymethylpenicillin is a narrow spectrum antibiotic also commonly referred to as Penicillin V or Penicillin VK.[A178609] It is a phenoxymethyl analog of Penicillin G, or [benzylpenicillin]. An orally active naturally penicillin, phenoxymethylpenicillin is…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
MecA PBP2' (penicillin binding protein 2')Penicillin-binding protein 1AD-alanyl-D-alanine carboxypeptidase DacB +2
Waktu ParuhUpon oral administr…
Vol. DistribusiFollowing intraveno…
Klirens-
Genetik -
small molecule | CAS: 3818-37-9

Phenoxypropazine is a non-selective and irreversible monoamine oxidase enzyme inhibitor (MAOI), belonging to the _hydrazine_ chemical class. It was marketed as an antidepressant in 1961 but was later withdrawn in 1966 because of its hepatotoxic potential.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenprobamate DB13354
small molecule | CAS: 673-31-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCarbamic Acid EstersCentral Nervous System Depressants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenprocoumon Approved DB00946
small molecule | CAS: 435-97-2

Coumarin derivative that acts as a long-acting oral anticoagulant.

Kategori:
4-HydroxycoumarinsAnticoagulantsBenzopyrans +16
Target Protein:
Vitamin K epoxide reductase complex subunit 1
Gen Terkait:
CYP2C9 CYP2C9 VKORC1
Waktu Paruh5-6 days
Vol. Distribusi-
Klirens-
Genetik 3 Varian
Phenserine DB04892
small molecule | CAS: 101246-66-6

Phenserine is under development by Axonyx, a US biopharmaceutical company that focuses on treatments for dementia. Phenserine is a next generation acetylcholinesterase (AChE) inhibitor indicated for the treatment of AD. Unlike currently marketed AChE inhibito…

Kategori:
Acids, AcyclicAlkaloidsCarbamates +11
Target Protein:
AcetylcholinesteraseCholinesteraseAmyloid-beta precursor protein
Waktu Paruh8 to 10 hours
Vol. Distribusi-
Klirens-
Genetik -
Phensuximide Approved DB00832
small molecule | CAS: 86-34-0

Phensuximide is a member of the succinimide class with anticonvulsant properties. It suppresses the paroxysmal three cycle per second spike and wave EEG pattern associated with lapses of consciousness in petit mal seizures. The frequency of attacks is reduced…

Kategori:
AnticonvulsantsCentral Nervous System DepressantsImides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phentermine Approved DB00191
small molecule | CAS: 122-09-8

Phentermine is a sympathomimetic amine anorectic agent and it was introduced in 1959 as part of an anti-obesity combination drug.[A174361, A174364] It is chemically related to amphetamine and it is commonly referred to as an atypical amphetamine.[A174370] Phe…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +22
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Phentolamine Approved DB00692
small molecule | CAS: 50-60-2

Phentolamine is a reversible, non-selective alpha-adrenergic blocker that induces vasodilation. While initially introduced to the market for the treatment of hypertension, this clinical use was halted due to cardiovascular and gastrointestinal adverse effects…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +15
Target Protein:
Alpha-1 adrenergic receptorsD(2) dopamine receptorAlpha-2 adrenergic receptors +1
Waktu ParuhPhentolamine has a …
Vol. DistribusiWhile there is limi…
Klirens-
Genetik -
Phenyl aminosalicylate Approved DB06807
small molecule | CAS: 133-11-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 937-34-8

Deskripsi belum tersedia.

Kategori:
Sulfur AcidsSulfur CompoundsSulfuric Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenyl salicylate Approved DB11071
small molecule | CAS: 118-55-8

Phenyl salicylate is a 2-hydroxybenzoic acid phenyl ester. It is utilized in some manufacturing processes of polymers, lacquers, adhesives, waxes, as well as polishes. It is an active ingredient in some pharmaceutical products as a mild analgesic for pain rel…

Kategori:
Acids, CarbocyclicAnti-Infective Agents, LocalBenzene Derivatives +7
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhMean half-life of 1…
Vol. DistribusiSteady-state plasma…
KlirensPlease refer to [DB…
Genetik -
small molecule | CAS: 195868-36-1

Deskripsi belum tersedia.

Kategori:
Compounds used in a research, industrial, or household settingMacromolecular SubstancesOrganosilicon Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Hematopoietic prostaglandin D synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-glucose 4-epimerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 122-78-1

Deskripsi belum tersedia.

Kategori:
AldehydesOils, Volatile
Target Protein:
Primary amine oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenylacetic acid Approved DB09269
small molecule | CAS: 103-82-2

Phenylacetic acid is an organic compound containing a phenyl functional group and a carboxylic acid functional group. It is a white solid with a disagreeable odor. Because it is used in the illicit production of phenylacetone (used in the manufacture of subst…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmmonium Ion Binding Activity +5
Waktu Paruh-
Vol. Distribusi19.2 ± 3.3 L.
Klirens-
Genetik -
small molecule | CAS: 28047-15-6

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenylalanine Approved DB00120
small molecule | CAS: 63-91-2

Phenylalanine is an essential aromatic amino acid that is a precursor of melanin, [dopamine], [noradrenalin] (norepinephrine), and [thyroxine].

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +7
Target Protein:
Tyrosine 3-monooxygenaseTyrosine aminotransferaseLarge neutral amino acids transporter small subunit 2 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxypeptidase A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 5241-58-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Substance-P receptorGenome polyproteinGenome polyprotein +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 52735-71-4

Deskripsi belum tersedia.

Target Protein:
Chymotrypsinogen B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12251–12300 dari 16004
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