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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 245 / 252
small molecule | CAS: 21411-53-0

Pristinamycin IIA is a macrolide antibiotic, a member of the streptogramin A group of antibiotics, and one component of pristinamycin. It is produced by Streptomyces graminofaciens and other bacteria.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
Streptogramin A acetyltransferase
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small molecule | CAS: 23152-29-6

One of the components of virginiamycin, a cyclic polypeptide antibiotic complex from streptomyces virginiae, s. Loidensis, s. Mitakaensis, s. Pristina-spiralis, s. Ostreogriseus, and others. It is used to treat infections with gram-positive organisms and as a…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic +1
Target Protein:
Large ribosomal subunit protein eL37
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Virulizin DB17098
biotech | CAS: 216586-46-8

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicBodily SecretionsComplex Mixtures +1
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biotech

Virus Specific T-Cells (VSTs) are a target therapy that are generated for specific viral antigens. These products are generated from virus-naive or virus-experienced autologous or allogenic sources. Antigens identified as an immune target are presented by ant…

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VIS-410 DB19067
biotech | CAS: 2043950-09-8

VIS-410 is under investigation in clinical trial NCT03040141 (Study of Efficacy and Safety of IV VIS410 Plus Oseltamivir Versus Oseltamivir in Hospitalized Adults With Influenza A).

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Visilizumab DB12053
biotech | CAS: 219716-33-3

Visilizumab has been investigated for the treatment of Ulcerative Colitis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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Vismodegib Approved DB08828
small molecule | CAS: 879085-55-9

Vismodegib is an orally active small molecule that inhibits the hedgehog signaling pathway by binding to and inhibiting the transmembrane protein smoothened homologue (SMO).[A258613,A258618,L45803] It was discovered by high-throughput screening of a library o…

Kategori:
AmidesAminesAniline Compounds +18
Target Protein:
Protein smoothened
Waktu ParuhThe half-life of vi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Visnadine DB13355
small molecule | CAS: 477-32-7

Deskripsi belum tersedia.

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingPeripheral Vasodilators +1
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small molecule | CAS: 934960-96-0

Deskripsi belum tersedia.

Kategori:
AminesBenzoquinonesBenzylammonium Compounds +8
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Vistusertib DB11925
small molecule | CAS: 1009298-59-2

Vistusertib is under investigation for the treatment of Advanced Gastric Adenocarcinoma.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTOR
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Visugromab DB18894
biotech | CAS: 2556646-63-8

Visugromab is under investigation in clinical trial NCT06059547 (Neoadjuvant Immunotherapy in Combination With the Anti-gdf-15 Antibody Visugromab (CTL-002) for Treatment of Muscle Invasive Bladder Cancer).

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VIT-100 DB05865
small molecule

VIT-100 was developed by ItherX Pharmaceuticals of San Diego. In preclinical studies, companyl has shown that VIT-100 inhibits the growth of cells taken from multiple keloid biopsies as compared to the same keloidal cells treated with a control. It is believe…

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small molecule | CAS: 15713-12-9

Deskripsi belum tersedia.

Target Protein:
5-methyltetrahydrofolate--homocysteine S-methyltransferase
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Vitamin E Approved DB00163
small molecule | CAS: 59-02-9

In 1922, vitamin E was demonstrated to be an essential nutrient[A32448]. Vitamin E is a term used to describe 8 different fat soluble tocopherols and tocotrienols, alpha-tocopherol being the most biologically active[A176104]. Vitamin E acts as an antioxidant,…

Kategori:
AntioxidantsBasic Ointments and ProtectantsBenzopyrans +23
Target Protein:
SEC14-like protein 4SEC14-like protein 3SEC14-like protein 2 +7
Waktu Paruh44 hours in prematu…
Vol. Distribusi0.41L/kg in prematu…
Klirens6.5mL/hr/kg in prem…
Genetik -
Vitamin K7 DB15664
small molecule | CAS: 83-69-2

Deskripsi belum tersedia.

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Vitespen DB06400
biotech | CAS: 492448-75-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +3
Waktu Paruh-
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Vixarelimab DB16350
biotech | CAS: 2243320-83-2

Vixarelimab is under investigation in clinical trial NCT03816891 (A Study to Assess the Efficacy, Safety, and Tolerability of KPL-716 in Reducing Pruritus in Prurigo Nodularis).

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Vixtimotamab DB17393
biotech | CAS: 2243775-32-6

Deskripsi belum tersedia.

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VK-0214 DB17670
small molecule | CAS: 852949-30-5

Deskripsi belum tersedia.

Target Protein:
Thyroid hormone receptor beta
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VK-2809 DB15137
small molecule | CAS: 852948-13-1

VK-2809 is under investigation in clinical trial NCT02927184 (Safety and Tolerability of VK2809 in Patients With Primary Hypercholesterolemia and Non-Alcoholic Fatty Liver Disease).

Kategori:
Organophosphorus Compounds
Target Protein:
Thyroid hormone receptor beta
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VL-2397 DB17796
small molecule | CAS: 1186200-57-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +1
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VLTS-589 DB05430
small molecule

VLTS-589 consists of plasmid encoding the angiomatrix protein Del-1 in conjunction with poloxamer 188 for the treatment of peripheral vascular disease.

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VLTS-934 DB05597
small molecule

VLTS-934 was developed by Valentis inc. for the treatment of Peripheral Arterial Disease (PAD). It was under investigation in clinical trial NCT00113009 (Trial of VLTS-934 in Subjects With Intermittent Claudication Secondary to Peripheral Arterial Disease).

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VLX-1005 DB18307
small molecule | CAS: 1532593-30-8

Deskripsi belum tersedia.

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Arachidonate 12-lipoxygenase, 12R-type
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VLX-1570 DB16030
small molecule | CAS: 1956378-23-6

VLX-1570 is under investigation in clinical trial NCT02372240 (A Study of VLX1570 and Dexamethasone in Myeloma Patients).

Kategori:
Benzene Derivatives
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VM4-037 DB15319
small molecule | CAS: 1071470-72-8

VM4-037 is under investigation in clinical trial NCT00884520 (An Exploratory, Open Label, Multi-Center, Non-Randomized Study of [F-18]VM4-037).

Kategori:
AmidesAmino Acids, Peptides, and ProteinsFluorine Radioisotopes +4
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VMD-928 DB18052
small molecule | CAS: 1802770-18-8

Deskripsi belum tersedia.

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VO659 DB18160
biotech | CAS: 1479142-52-3

VO659 is an antisense oligonucleotide being investigated for the treatment of Huntington's disease.

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Voacamine DB04877
small molecule | CAS: 3371-85-5

Voacamine is an alkaloid isolated from the bark of the _Pescheria fuchsiae folia_ tree. It is an antimalarial drug approved for use in several African countries. Voacamine is also under investigation for use in modulating multidrug-resistance in tumor cells.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +5
Target Protein:
ATP-dependent translocase ABCB1
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biotech | CAS: 2490556-51-7

Vobramitamab duocarmazine is under investigation in clinical trial NCT05551117 (A Study of Vobramitamab Duocarmazine in Participants With Metastatic Castration Resistant Prostate Cancer and Other Solid Tumors).

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biotech | CAS: 1300724-82-6

Vocimagene amiretrorepvec is under investigation in clinical trial NCT02576665 (A Study of Toca 511, a Retroviral Replicating Vector, Combined With Toca FC in Patients With Solid Tumors or Lymphoma (Toca 6)).

Kategori:
Amino Acids, Peptides, and ProteinsAminohydrolasesEnzymes +4
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Voclosporin Approved DB11693
small molecule | CAS: 515814-01-4

Lupus nephritis (LN) is a type of glomerulonephritis occurring in patients with systemic lupus erythematosus (SLE). LN is a significant cause of renal failure, morbidity, and death in patients with SLE. Within 10 years of being diagnosed with SLE, 5-20% of …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsCalcineurin Inhibitor Immunosuppressant +16
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 1 +1
Waktu ParuhThe average termina…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent s…
Genetik -
Vodudeutentan DB17410
small molecule | CAS: 2364365-83-1

Deskripsi belum tersedia.

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Vofatamab DB14781
biotech | CAS: 1312305-12-6

Vofatamab is under investigation in clinical trial NCT02401542 (Dose Escalation, Expansion Study of Vofatamab (B-701) in Treatment of Locally Advanced or Metastatic Urothelial Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Volagidemab DB16421
biotech | CAS: 1233956-13-2

Volagidemab is under investigation in clinical trial NCT03117998 (Multiple Dose Study to Evaluate the Efficacy, Safety and Pharmacodynamics of REMD-477 in Subjects With Type 1 Diabetes Mellitus).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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Volanesorsen Approved DB15067
biotech | CAS: 915430-78-3

Volanesorsen is an antisense oligonucleotide that binds to apoC-III mRNA to prevent its translation.[L16621] It is indicated to treat familial chylomicronemia, a genetic condition that prevents breakdown of triglycerides and chylomicrons.[L16621] This drug is…

Kategori:
CarbohydratesGlycosidesLipid Modifying Agents +4
Target Protein:
Apolipoprotein C-III
Waktu ParuhVolanesorsen has a …
Vol. DistribusiThe volume of distr…
KlirensThe exact rate of c…
Genetik -
Volasertib DB12062
small molecule | CAS: 755038-65-4

Volasertib has been used in trials studying the treatment of Leukemia, Neoplasms, Leukemia, Myeloid, Acute, Myelodysplastic Syndromes, and Leukemia, Monocytic, Acute, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase PLK1
Waktu Paruh-
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Volinanserin DB16351
small molecule | CAS: 139290-65-6

Volinanserin is under investigation in clinical trial NCT00464243 (Efficacy and Safety of Volinanserin on Sleep Maintenance Insomnia - Polysomnographic Study).

Kategori:
Antidepressive AgentsBenzene DerivativesCentral Nervous System Depressants +7
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH25-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A
Waktu Paruh-
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Volixibat DB13914
small molecule | CAS: 1025216-57-2

Volixibat, also known as SHP626 or LUM002, is an investigational drug that will potentially be used for the treatment of Non-Alcoholic Steatohepatitis (NASH). If approved for use, it will be the first available agent for the treatment of NASH. Volixibat is…

Kategori:
CarbohydratesHeterocyclic Compounds, Fused-RingLipid Regulating Agents +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
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Volociximab DB06647
biotech | CAS: 558480-40-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +10
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Klirens-
Genetik -
biotech | CAS: 2092457-20-8

Volrubigene ralaparvovec is under investigation in clinical trial NCT03223194 (Gene Transfer Clinical Study in Crigler-najjar Syndrome).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Volrustomig DB18893
biotech | CAS: 2407760-40-9

Volrustomig is under investigation in clinical trial NCT06097728 (MEDI5752 in Combination With Carboplatin Plus Pemetrexed in Unresectable Pleural Mesothelioma).

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Von Willebrand factor human Approved DB13133
biotech | CAS: 109319-16-6

The human von Willebrand factor (vWF) is a human plasma-derived vWF, an endogenous large multimeric plasma glycoprotein involved in hemostasis. It serves a dual role in hemostasis by mediating platelet adhesion and aggregation at the site of blood vessel inju…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chainAsialoglycoprotein receptor 1 +1
Waktu ParuhIn patients with Ty…
Vol. DistribusiThe volume of distr…
KlirensIn patients with Ty…
Genetik -
Vonafexor DB18782
small molecule | CAS: 1192171-69-9

Deskripsi belum tersedia.

Target Protein:
Bile acid receptor
Waktu Paruh-
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Vonicog alfa Approved DB12872
biotech

Vonicog alfa is a recombinant human von Willebrand factor (rVWF) produced from Chinese hamster ovary cells.[A264444] Used to treat von Willebrand Disease (vWD), it mimics the biological actions of endogenous VWF,[L51274] which is a critical plasma glycoprotei…

Kategori:
von Willebrand Factor
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chain
Waktu ParuhIn Study 071001, th…
Vol. Distribusi-
KlirensIn Study 071001, th…
Genetik -
Vonlerolizumab DB16352
biotech | CAS: 1638935-72-4

Vonlerolizumab is under investigation in clinical trial NCT03029832 (A Study of MOXR0916 in Combination With Atezolizumab Versus Atezolizumab Alone in Participants With Untreated Locally Advanced or Metastatic Urothelial Carcinoma Who Are Ineligible for Cispl…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
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Genetik -
Vonoprazan Approved DB11739
small molecule | CAS: 881681-00-1

Vonoprazan is a potassium-competitive acid blocker (PCAB) that inhibits H<sup>+</sup>, K<sup>+</sup>-ATPase-mediated gastric acid secretion. PCABs represent an alternative to proton-pump inhibitors for the treatment of acid-related disorders. Unlike proton-pu…

Kategori:
Alimentary Tract and MetabolismAmidesCytochrome P-450 CYP2B6 Substrates +17
Target Protein:
Hydrogen potassium ATPase
Waktu ParuhVonoprazan has an e…
Vol. DistribusiVonoprazan has an a…
KlirensVonoprazan has an a…
Genetik -
Vopratelimab DB15378
biotech | CAS: 2039148-04-2

Vopratelimab is under investigation in clinical trial NCT02904226 (JTX-2011 Alone and in Combination With Anti-PD-1 or Anti-CTLA-4 in Subjects With Advanced and/or Refractory Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vorapaxar Approved DB09030
small molecule | CAS: 618385-01-6

Vorapaxar is a tricyclic himbacine-derived selective inhibitor of protease activated receptor (PAR-1) indicated for reducing the incidence of thrombotic cardiovascular events in patients with a history of myocardial infarction (MI) or with peripheral arterial…

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +11
Target Protein:
Proteinase-activated receptor 1
Waktu ParuhVorapaxar has an ef…
Vol. Distribusi424 L
Klirens-
Genetik -
Vorasidenib Approved DB17097
small molecule | CAS: 1644545-52-7

Vorasidenib is a first-in-class dual isocitrate dehydrogenase-1 (IDH1) and isocitrate dehydrogenase-2 (IDH2) inhibitor.[A264209] It works by suppressing the levels of D-2-hydroxyglutarate (2-HG), an oncometabolite produced by mutant IDH1 and IDH2 isoforms.[L5…

Kategori:
AminesBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Substrates +26
Target Protein:
Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrialIsocitrate dehydrogenase [NAD] subunit beta, mitochondrialIsocitrate dehydrogenase [NAD] subunit gamma, mitochondrial +2
Waktu ParuhThe mean (CV%) stea…
Vol. DistribusiThe mean (CV%) volu…
KlirensThe mean (CV%) stea…
Genetik -
Menampilkan 12201–12250 dari 12560
Sebelumnya Halaman 245 / 252 Berikutnya