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12560

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9109 (72.5%)
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12560 (100.0%)

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Halaman 244 / 252
Vesencumab DB15428
biotech | CAS: 1205533-60-3

Vesencumab is under investigation in clinical trial NCT00747734 (A Study of MNRP1685A in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
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Vesnarinone DB12082
small molecule | CAS: 81840-15-5

Vesnarinone has been used in trials studying the treatment of HIV Infections and Sarcoma, Kaposi.

Kategori:
Adjuvants, ImmunologicAnti-Infective AgentsAntineoplastic Agents +8
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3AVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu Paruh-
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biotech

Vespula maculifrons venom protein is an extract of Vespula maculifrons venom. Vespula maculifrons venom protein is used in allergenic testing.

Kategori:
Bee and Wasp VenomCell-mediated ImmunityIncreased Histamine Release +2
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VG161 DB18469
biotech

VG161 is an oncolytic virus therapy under investigation for the treatment of cholangiocarcinoma.

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VGA039 DB18385
biotech

VGA039 is an IgG4 monoclonal antibody directed against protein S.

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VGB-R04 DB18615
biotech

VGB-R04 is an adeno-associated viral vector delivering human FIX Padua gene.

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VGM-R02b DB18256
biotech

Deskripsi belum tersedia.

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VGV-1 DB05328
small molecule

VGV-1 is a potential salvage therapy for treatment of HIV infected people who have failed anti-retroviral therapy.

Target Protein:
Gag-Pol polyprotein
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Vibecotamab DB18872
biotech | CAS: 2138442-13-2

Vibecotamab is under investigation in clinical trial NCT05285813 (A Phase II Study of Vibecotamab (Xmab14045) for MRD- Positive AML and MDS After Hypomethylating Agent Failure).

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Vibegron Approved DB14895
small molecule | CAS: 1190389-15-1

Vibegron is a potent, selective beta-3 adrenergic receptor (?3) agonist that relaxes the detrusor smooth muscle of the bladder, thereby increasing bladder capacity.[L28305] Vibegron was first approved in Japan in September 2018 for the treatment of overactive…

Kategori:
Adrenergic AgonistsAdrenergic beta-3 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-3 adrenergic receptor
Waktu ParuhThe terminal plasma…
Vol. DistribusiThe mean apparent v…
KlirensThere is limited in…
Genetik -
Vibostolimab DB16420
biotech | CAS: 2231305-30-7

Vibostolimab is under investigation in clinical trial NCT04303169 (Substudy 02C: Safety and Efficacy of Pembrolizumab in Combination With Investigational Agents or Pembrolizumab Alone in Participants With Stage III Melanoma Who Are Candidates for Neoadjuvant …

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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Vibriolysin DB05135
small molecule | CAS: 69598-88-5

Vibriolysin is a proteolytic enzyme secreted by the marine microorganism Vibrio proteolyticus. It is a new agent for enzymatic debridement, shown to rapidly and thoroughly hydrolyze burn wound eschar within full-thickness wounds.

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Vicagrel DB16349
small molecule | CAS: 1314081-53-2

Vicagrel is under investigation in clinical trial NCT03599284 (The Efficacy, Safety and Pharmacokinetic of Antiplatelet Therapy for Vicagrel).

Kategori:
Acids, CarbocyclicAntiplatelet agentsCytochrome P-450 CYP2C19 Substrates +2
Target Protein:
P2Y purinoceptor 12
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Vicriviroc DB06652
small molecule | CAS: 306296-47-9

Vicriviroc, also known as SCH 417690 and SCH-D, is currently in clinical trials for the management of HIV-1. This pyrimidine based drug inhibits the interaction of HIV-1 with CCR5, preventing viral entry into cells. This drug was developed by Schering-Plough.

Kategori:
Cytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +2
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
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Vidarabine Approved DB00194
small molecule | CAS: 24356-66-9

A nucleoside antibiotic isolated from Streptomyces antibioticus. It has some antineoplastic properties and has broad spectrum activity against DNA viruses in cell cultures and significant antiviral activity against infections caused by a variety of viruses su…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +17
Target Protein:
Adenosine receptor A2bDNA polymerase catalytic subunitThymidine kinase +1
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Vidofludimus DB15446
small molecule | CAS: 717824-30-1

Vidofludimus is under investigation in clinical trial NCT03722576 (Vidofludimus Calcium for Primary Sclerosing Cholangitis).

Kategori:
Acids, AcyclicBenzene Derivatives
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
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VidPrevtyn Beta Approved DB16427
biotech

VidPrevtyn Beta is an adjuvanted, recombinant COVID-19 vaccine developed collaboratively by GlaxoSmithKline (GSK) and Sanofi Pasteur.[L49691] It comprises a recombinant SARS-CoV-2 spike protein (B.1.351 strain) - produced by recombinant DNA technology using a…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
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Vidutolimod DB17500
biotech | CAS: 147063-80-7

Vidutolimod is a Toll-like receptor 9 (TLR9) agonist. It is an investigational cancer vaccine.

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Vigabatrin Approved DB01080
small molecule | CAS: 68506-86-5

Vigabatrin is an analog of gamma-aminobutyric acid ([GABA]), the main inhibitory neurotransmitter in the central nervous system, used in the treatment of refractory seizures and infantile spasms.[L13616] It irreversibly inhibits the enzyme responsible for GAB…

Kategori:
Acids, AcyclicAminobutyratesAnti-epileptic Agent +15
Target Protein:
4-aminobutyrate aminotransferase, mitochondrial
Waktu ParuhThe terminal half-l…
Vol. DistribusiVigabatrin is widel…
KlirensThe oral clearance …
Genetik -
Vilamakitug DB18978
biotech | CAS: 2458202-06-5

Vilamakitug is under investigation in clinical trial NCT05201352 (Evaluation of Efficacy of Trifluridine/tipiracil Plus an Anti-il-1? True Human Antibody Versus Trifluridine/tipiracil Plus Placebo in Metastatic Colorectal Cancer Patients After Failure of Oxal…

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Vilanterol Approved DB09082
small molecule | CAS: 503068-34-6

Vilanterol is a selective long-acting ?2-adrenergic agonist (LABA) with inherent 24-hour activity for the once-daily treatment of COPD and asthma.[A7737] This is in response to the need for longer-acting ?2-adrenergic agonists to overcome poor patient complia…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +19
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhThe effective half-…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
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Vilastobart DB19327
biotech | CAS: 2760549-50-4

Vilastobart is under investigation in clinical trial NCT04896697 (Vilastobart (XTX101) Monotherapy and Vilastobart and Atezolizumab Combination Therapy in Advanced Solid Tumors).

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Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Vildagliptin Approved DB04876
small molecule | CAS: 274901-16-5

Vildagliptin (LAF237) is an orally active antihyperglycemic agent that selectively inhibits the dipeptidyl peptidase-4 (DPP-4) enzyme. It is used to manage type II diabetes mellitus, where GLP-1 secretion and insulinotropic effects are impaired.[A232488] By i…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +11
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensAfter intravenous a…
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Vilobelimab DB16416
biotech | CAS: 2250440-41-4

Vilobelimab is a chimeric monoclonal immunoglobulin G4 (IgG4) antibody that binds to the soluble form of human C5a with high affinity. It consists of mouse anti-human complement factor 5a (C5a) monoclonal binding sites (variable regions of heavy and light cha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Complement C5
Waktu ParuhThe elimination hal…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Viloxazine Approved DB09185
small molecule | CAS: 46817-91-8

Viloxazine is a selective norepinephrine reuptake inhibitor.[L41685] For decades, an immediate-release formulation of viloxazine has been used in Europe as an antidepressant. It was first approved in the UK in 1974; however, the immediate-release formulation …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +46
Target Protein:
Sodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C +10
Waktu ParuhThe mean (± SD) hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Viltolarsen Approved DB15005
biotech | CAS: 2055732-84-6

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albeit a less seve…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD gene (exon 53 viltolarsen target site)
Waktu ParuhViltolarsen has a r…
Vol. DistribusiViltolarsen has a s…
KlirensViltolarsen has a r…
Genetik -
Viminol DB13353
small molecule | CAS: 21363-18-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
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Vimseltinib DB17520
small molecule | CAS: 1628606-05-2

Deskripsi belum tersedia.

Target Protein:
Macrophage colony-stimulating factor 1 receptor
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Vinbarbital DB13377
small molecule | CAS: 125-42-8

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +2
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Vinblastine Approved DB00570
small molecule | CAS: 865-21-4

Antitumor alkaloid isolated from Vinca rosea. (Merck, 11th ed.)

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +37
Target Protein:
Tubulin beta-2A chainTubulin alpha-1A chainTubulin beta chain +4
Waktu ParuhTriphasic: 35 min, …
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Vincristine Approved DB00541
small molecule | CAS: 57-22-7

Vincristine is an antitumor vinca alkaloid isolated from Vinca Rosea. It is marketed under several brand names, many of which have different formulations such as Marqibo (liposomal injection) and Vincasar. Vincristine is indicated for the treatment of acute l…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntimitotic Agents +33
Target Protein:
Tubulin beta chainTubulin alpha-4A chain
Waktu ParuhWhen intravenously …
Vol. DistribusiWithin 15 to 30 min…
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Vindesine Approved DB00309
small molecule | CAS: 53643-48-4

Vinblastine derivative with antineoplastic activity against cancer. Major side effects are myelosuppression and neurotoxicity. Vindesine is used extensively in chemotherapy protocols (antineoplastic combined chemotherapy protocols).

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +19
Target Protein:
Tubulin beta-1 chain
Waktu Paruh24 hours.
Vol. Distribusi-
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Vinflunine Approved DB11641
small molecule | CAS: 162652-95-1

Vinflunine is a third-generation member of the vinca alkaloid family with anti-tumour actions. It was first described in 1998 at the Pierre Fabre research center in France. Like other vinca agents, vinflunine is an anti-mitotic agent that induces a cell cycle…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Tubulin beta chain
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe terminal volume…
KlirensThe total blood cle…
Genetik -
Vinorelbine Approved DB00361
small molecule | CAS: 71486-22-1

Vinorelbine is an anti-mitotic chemotherapy drug that is used in the treatment of several types of malignancies, including breast cancer and non-small cell lung cancer (NSCLC) [L1998]. It was initially approved in the USA in 1990's for the treatment of NSCLC…

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +23
Target Protein:
Tubulin beta chain
Waktu ParuhThe terminal phase …
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Vinpocetine DB12131
small molecule | CAS: 42971-09-5

Vinpocetine has been investigated for the treatment of Epilepsy.

Kategori:
Agents causing hyperkalemiaAlkaloidsAntiarrhythmic agents +25
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Vintafolide DB05168
small molecule | CAS: 742092-03-1

Vintafolide is a folate-targeted chemotherapeutic conjugate (folate vitamin + vinca alkaloid) in clinical stage development as a treatment for folate-receptor positive cancers.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
Folate receptor alphaFolate receptor betaFolate receptor gamma
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Vinylglycine DB03214
small molecule | CAS: 70982-53-5

Vinylglycine is an irreversible inhibitor of aspartate aminotransferase.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
L-amino-acid oxidase1-aminocyclopropane-1-carboxylate synthase-like protein 1
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small molecule | CAS: 1184-84-5

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAlkenes +4
Target Protein:
Phosphonoacetaldehyde hydrolase
Waktu Paruh-
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Viomycin Approved DB06827
small molecule | CAS: 32988-50-4

Viomycin is a tuberactinomycin antibiotic that was used to treat Mycobacterium tuberculosis until it was replaced by the less toxic capreomycin. These drugs bind RNA in bacterial ribosomes and inhibit protein synthesis. Viomycin was derived from the actinomyc…

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAnti-Bacterial Agents +8
Target Protein:
16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyA
Waktu Paruh-
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Vipadenant DB06625
small molecule | CAS: 442908-10-3

Deskripsi belum tersedia.

Kategori:
Adenosine A2 Receptor AntagonistsNeurotransmitter AgentsPurinergic Agents +2
Target Protein:
Adenosine receptor A2a
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Viper antivenom Approved DB14114
biotech

Viper antivenom consists of antibodies derived from horses immunized and subsequently developed antibodies against snake venoms. ANAVIP, an equine-derived antivenom made with venom from _Bothrops asper_ and _Crotalus durissus_, was first approved by the FDA o…

Kategori:
Antivenins
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Vipoglanstat DB18126
small molecule | CAS: 1360622-01-0

Deskripsi belum tersedia.

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VIR201 DB05110
biotech

is an experimental therapeutic vaccine currently in clinical trial. The aim of therapeutic vaccines is to augment the body's immune response to HIV and to delay or prevent progression to AIDS.

Target Protein:
Interferon gamma
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biotech

Viral macrophage inflammatory protein-II (vMIP) is a highly basic protein and human chemokine analog encoded by human herpesvirus-8. The structure of vMIP consists of 71 residues and is a monomer under most conditions. It helps its virus evade the host immune…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +10
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Viralym-C DB17975
biotech

Viralym-C is an investigational T-cell immunotherapy developed by ViraCyte. It consists of Human Leukocyte Antigen (HLA)-matched cytomegalovirus (CMV)-specific T lymphocytes. It was granted FDA orphan designation in January 2017 and investigated for the treat…

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Menampilkan 12151–12200 dari 12560
Sebelumnya Halaman 244 / 252 Berikutnya