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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 244 / 272
Talotrexin DB06178
small molecule | CAS: 113857-87-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Talquetamab Approved DB16678
biotech | CAS: 2226212-40-2

Talquetamab is a IgG4-PAA bispecific G protein-coupled receptor class C group 5 member D (GPRC5D)-directed CD3 T-cell engager. It consists of two arms - anti-GPRC5D and anti-CD3 arms - linked by two interchain disulfide bonds, each arm comprising a heavy and …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +7
Target Protein:
T-cell surface glycoprotein CD3G-protein coupled receptor family C group 5 member D
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensTalquetamab clearan…
Genetik -
Talsaclidine DB12287
small molecule | CAS: 147025-53-4

Talsaclidine has been used in trials studying the treatment of Alzheimer Disease.

Waktu Paruh-
Vol. Distribusi-
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Talsupram DB09191
small molecule | CAS: 21489-20-3

Talsupram is a selective norepinephrine reuptake inhibitor (NRI). It was under research for the treatment of depression in 1960 and 1970 but it was never marketed. Talsupram presents a similar structure to [citalopram].

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Talviraline DB07885
small molecule | CAS: 163451-80-7

Talviraline has been used in trials studying the treatment of HIV Infections.

Kategori:
Acquired Immunodeficiency SyndromeHeterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamatinib DB07159
small molecule | CAS: 841290-80-0

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase SYKProto-oncogene tyrosine-protein kinase receptor Ret
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taminadenant DB18811
small molecule | CAS: 1337962-47-6

Deskripsi belum tersedia.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamnorzatinib DB19201
small molecule | CAS: 1646839-59-9

Tamnorzatinib is under investigation in clinical trial NCT03176277 (A Study of ONO-7475 in Patients With Acute Leukemias).

Target Protein:
Tyrosine-protein kinase MerTyrosine-protein kinase receptor UFO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamoxifen Approved DB00675
small molecule | CAS: 10540-29-1

Tamoxifen is a non-steroidal antiestrogen used to treat estrogen receptor positive breast cancers as well as prevent the incidence of breast cancer in high risk populations.[A1025,L7799,L7802] Tamoxifen is used alone or as an adjuvant in these treatments.[L77…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +64
Target Protein:
Estrogen receptorEstrogen receptor betaProtein kinase C +7
Gen Terkait:
CYP2D6 F5
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ta…
Genetik 2 Varian
biotech | CAS: 2148334-68-1

Tamrintamab pamozirine is an antibody-drug conjugate targeted against DPEP3.

Kategori:
Antibody-drug Conjugates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamsulosin Approved DB00706
small molecule | CAS: 106133-20-4

Tamsulosin is a selective alpha-1A and alpha-1B adrenoceptor antagonist that exerts its greatest effect in the prostate and bladder, where these receptors are most common.[Label] It is indicated for the treatment of signs and symptoms of benign prostatic hype…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu ParuhThe half life in fa…
Vol. Distribusi16L after intraveno…
Klirens2.88L/h.[Label]
Genetik -
Tanaproget DB04787
small molecule | CAS: 304853-42-7

Tanaproget (NSP-989) is an investigational non-steroidal progestin. It is a high affinity, high efficacy agonist of the progesterone receptor (PR) with a much more selective binding profile relative to most conventional progestins. Because of this tanaproget …

Kategori:
Heterocyclic Compounds, Fused-RingOxazinesReceptors, Progesterone, agonists +1
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandospirone DB12833
small molecule | CAS: 87760-53-0

Tandospirone has been used in trials studying the treatment of Schizophrenia.

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Agents +8
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tandutinib DB05465
small molecule | CAS: 387867-13-2

MLN518 is a novel, oral, small molecule designed to inhibit type III receptor tyrosine kinases, including FLT3, (platelet-derived growth-factor receptor) PDGFR and c-KIT. Tyrosine kinases are enzymes involved in several cellular processes and are known to be …

Kategori:
Heterocyclic Compounds, Fused-RingPotential QTc-Prolonging AgentsQTc Prolonging Agents +1
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Platelet-derived growth factor D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanespimycin DB05134
small molecule | CAS: 75747-14-7

Tanespimycin, manufactured by Conforma Therapeutics is under development as a small molecule inhibitor of heat shock protein 90 (HSP90). It is developed for the treatment of several types of cancer, solid tumors or chronic myelogenous leukemia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tanezumab DB12335
biotech | CAS: 880266-57-9

Tanezumab has been investigated for the treatment of Osteoarthritis, Knee and Neuralgia, Postherpetic.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanfanercept DB19142
biotech | CAS: 2119738-70-2

Tanfanercept is under investigation in clinical trial NCT06400589 (A Study to Evaluate the Efficacy and Safety of Tanfanercept (HL036) in Dry Eye Disease).

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Tangerine Approved DB10637
biotech

Tangerine allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Vol. Distribusi-
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Genetik -
Tangerine peel DB14316
biotech

Tangerine peel is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
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Genetik -
Taniborbactam DB16338
small molecule | CAS: 1613267-49-4

Taniborbactam is under investigation in clinical trial NCT03840148 (Safety and Efficacy Study of Cefepime/vnrx-5133 in Patients With Complicated Urinary Tract Infections).

Kategori:
AcidsAcids, NoncarboxylicBoron Compounds
Waktu Paruh-
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Genetik -
Taniraleucel DB18311
biotech

Deskripsi belum tersedia.

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Tannic acid Approved DB09372
small molecule | CAS: 1401-55-4

Tannic acid is a polyphenolic compound. It is a type of the commercially available tannins. It acts as a weak acid. Tannic acid is found in the nutgalls formed by insects on twigs of certain oak trees (Quercus infectoria and other Quercus species). It is remo…

Kategori:
Benzene DerivativesBiopolymersCompounds used in a research, industrial, or household setting +4
Target Protein:
Anoctamin-1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tanshinone I DB16886
small molecule | CAS: 568-73-0

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanzisertib DB11798
small molecule | CAS: 899805-25-5

Tanzisertib has been used in trials studying the treatment of Fibrosis, Discoid Lupus, Pulmonary Fibrosis, Interstitial Lung Disease, and Lung Diseases, Interstitial, among others.

Kategori:
AlcoholsCarbon RadioisotopesCyclohexanes +6
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tapencarium DB17821
small molecule

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Waktu Paruh-
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Genetik -
Tapentadol Approved DB06204
small molecule | CAS: 175591-23-8

Tapentadol is a centrally-acting synthetic analgesic with a dual mechanism of action. It is a mu-opioid receptor agonist that also inhibits norepinephrine reuptake.[A260721, A36596] Tapentadol was first approved by the FDA on November 20, 2008. The extende…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAnalgesics +25
Target Protein:
Mu-type opioid receptorSodium-dependent noradrenaline transporterKappa-type opioid receptor +2
Waktu ParuhThe terminal half-l…
Vol. DistribusiTapentadol is widel…
KlirensThe total clearance…
Genetik -
Tapinarof Approved DB06083
small molecule | CAS: 79338-84-4

Tapinarof is a novel, first-in-class, small-molecule AhR agonist that is indicated for the treatment of adult psoriasis. It is available as a topical cream to be applied to the affected area once daily.[L41845, A248790] Tapiranof was first discovered as a met…

Kategori:
AntipsoriaticsAntipsoriatics for Topical UseAryl Hydrocarbon Receptor Agonist +11
Target Protein:
Aryl hydrocarbon receptor
Waktu ParuhDue to the insuffic…
Vol. DistribusiThe Vss of tapinaro…
Klirens-
Genetik -
Tapotoclax DB17166
small molecule | CAS: 1883727-34-1

Deskripsi belum tersedia.

Target Protein:
Induced myeloid leukemia cell differentiation protein Mcl-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taprenepag DB12623
small molecule | CAS: 752187-80-7

Taprenepag has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.

Kategori:
Acids, AcyclicAmidesFatty Acids +5
Target Protein:
Prostaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarafenacin DB18810
small molecule | CAS: 385367-47-5

Deskripsi belum tersedia.

Target Protein:
Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Taraxacum officinale leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Tarazepide DB06435
small molecule | CAS: 141374-81-4

Deskripsi belum tersedia.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2411896-53-0

Tarcocimab tedromer is under investigation in clinical trial NCT06270836 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer Compared With Sham Treatment in Participants With Moderately Severe to Severe Non-proliferative Diabetic Retinopathy (…

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Vol. Distribusi-
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Genetik -
Tarenflurbil DB05289
small molecule | CAS: 51543-40-9

Tarenflurbil is an investigational drug that was studied in patients with mild Alzheimer's disease. It is a selective amyloid lowering agent (SALA) that reduces levels of the toxic peptide amyloid beta 42 (A?42) in cultured human cells and in animal models. A…

Kategori:
Acids, AcyclicAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarextumab DB12104
biotech | CAS: 1359940-55-8

Tarextumab has been used in trials studying the treatment of Solid Tumors, Stage IV Pancreatic Cancer, and Stage IV Small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tariquidar DB06240
small molecule | CAS: 206873-63-4

Deskripsi belum tersedia.

Kategori:
Drug Resistance, MultipleHeterocyclic Compounds, Fused-RingP-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarlatamab Approved DB17256
biotech | CAS: 2307488-83-9

Tarlatamab is a first-in-class T-cell engager used to treat extensive-stage small cell lung cancer.[L50748] It is a bispecific monoclonal antibody that targets CD3 expressed on the surface of T-cells and delta-like ligand 3 (DLL3), an inhibitory ligand that s…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific Monoclonal Antibodies +5
Target Protein:
Delta-like protein 3T-cell surface glycoprotein CD3
Waktu ParuhThe median terminal…
Vol. DistribusiAt steady-state, th…
KlirensThe systemic cleara…
Genetik -
Tarloxotinib DB14944
small molecule | CAS: 1636938-13-0

Tarloxotinib is under investigation in clinical trial NCT03743350 (NSCLC Exon 20 or HER2-activating Mutations).

Target Protein:
Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tartronate DB03680
small molecule

Deskripsi belum tersedia.

Target Protein:
NAD-dependent malic enzyme, mitochondrialNADP-dependent malic enzyme, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-102 DB08937
small molecule | CAS: 733030-01-8

TAS-102 (Taiho Pharma USA, Inc.) is an anti-cancer drug under development and in stage 3 clinical trials for the treatment of colorectal cancer. It is composed of the thymidine phosphorylase inhibitor (TPI) tipiracil and the cytotoxin trifluridine. Trifluridi…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +4
Waktu Paruh-
Vol. Distribusi-
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TAS-106 DB06656
small molecule | CAS: 180300-43-0

TAS-106 is a new nucleoside antimetabolite. TAS-106 has demonstrated strong antitumor activity without serious toxicity in nude rat models bearing human tumours [A31693].

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
Waktu Paruh-
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Genetik -
TAS-108 DB05966
small molecule | CAS: 229634-97-3

Deskripsi belum tersedia.

Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
TAS-116 DB14876
small molecule | CAS: 1260533-36-5

TAS-116 is under investigation in clinical trial NCT02965885 (A Study of TAS-116 in Patients With Solid Tumors).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Heat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-117 DB15054
small molecule | CAS: 1402602-94-1

TAS-117 is under investigation in clinical trial NCT03017521 (K-BASKET, TAS-117, PI3K/AKT Gene Aberration).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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Genetik -
TAS-303 DB18808
small molecule | CAS: 1449371-87-2

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasimelteon Approved DB09071
small molecule | CAS: 609799-22-6

Tasimelteon is a selective dual melatonin receptor agonist indicated for the treatment of Non-24-Hour Sleep-Wake Disorder (N24HSWD). Occurring commonly in blind individuals without light perception, this condition is often characterized by periods of night-ti…

Kategori:
Central Nervous System DepressantsCycloparaffinsCytochrome P-450 CYP1A2 Substrates +11
Target Protein:
Melatonin receptor type 1AMelatonin receptor type 1B
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent oral v…
Klirens-
Genetik -
Tasisulam DB11941
small molecule | CAS: 519055-62-0

Tasisulam has been used in trials studying the treatment and basic science of Melanoma, Lymphoma, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TASO-001 DB17463
biotech

TASO-001 is a transforming growth factor (TGF)-beta 2 specific antisense oligodeoxynucleotide.

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Genetik -
Tasosartan DB01349
small molecule | CAS: 145733-36-4

Tasosartan is a long-acting angiotensin II (AngII) receptor blocker. Its long duration of action has been attributed to its active metabolite enoltasosartan. It is used to treat patients with essential hypertension.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin II receptor blockers (ARBs), plain +4
Target Protein:
Type-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taspoglutide DB14027
small molecule | CAS: 275371-94-3

Taspoglutide is a pharmaceutical drug, a glucagon-like peptide-1 agonist (GLP-1 agonist), under investigation for treatment of type 2 diabetes being codeveloped by Ipsen and Roche. In September 2010 Roche halted Phase III clinical trials due to incidences of …

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Hormones +5
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12151–12200 dari 13591
Sebelumnya Halaman 244 / 272 Berikutnya