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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Halaman 243 / 252
VCA-894A DB18609
biotech

VCA-894A is a synthetic 2'-O-methoxyethyl phosphorothioate oligoribonucleotide sodium salt consisting of 19 nucleotide residues with the sequence 5'-MeCMeUGMeUGGAAGMeUGAGGGMeCMeCAG-3'

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Vebicorvir DB18784
small molecule | CAS: 2090064-66-5

Deskripsi belum tersedia.

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Vebreltinib DB16823
small molecule | CAS: 1440964-89-5

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
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Vecabrutinib DB16657
small molecule | CAS: 1510829-06-7

Vecabrutinib is under investigation in clinical trial NCT03037645 (Safety, PK, PD, and Antitumor Activity of Vecabrutinib (SNS-062) in B Lymphoid Cancers).

Kategori:
Amines
Target Protein:
Tyrosine-protein kinase BTK
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Vedolizumab Approved DB09033
biotech | CAS: 943609-66-3

Vedolizumab is a recombinant humanized IgG1 monoclonal antibody directed against the human lymphocyte ?4?7 integrin, a key mediator of gastrointestinal inflammation implicated in diseases like ulcerative colitis or Crohn's disease.[L48216] ?4?7 integrin facil…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-4Integrin beta-7
Waktu ParuhVedolizumab has a l…
Vol. DistribusiSerum apparent volu…
KlirensVedolizumab clearan…
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Vedroprevir DB12037
small molecule | CAS: 1098189-15-1

Vedroprevir has been investigated for the treatment of Hepatitis C, Chronic.

Kategori:
Antiviral AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
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small molecule | CAS: 15966-93-5

Deskripsi belum tersedia.

Target Protein:
Vascular endothelial growth factor receptor 2
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VEGFR2-169 DB16152
small molecule | CAS: 673478-49-4

VEGFR2-169 is under investigation in clinical trial NCT00655785 (Antiangiogenic Peptide Vaccine Therapy With Gemcitabine in Treating Patient With Pancreatic Cancer (Phase1/2)).

Kategori:
Amino Acids, Peptides, and ProteinsCancer VaccinesEnzymes +15
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Veglin DB05890
small molecule | CAS: 1220118-27-3

VEGF-AS (Veglin) is an anti-angiogenesis non-chemotherapy drug (angiogenesis inhibitor) that was developed by VasGene Therapeutics, Inc. for the treatment of a variety of malignancies including mesothelioma. Veglin is one of several newly developed non-chemot…

Target Protein:
Vascular endothelial growth factor A, long form
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Velafermin DB06493
small molecule | CAS: 697766-75-9

Velafermin was a novel investigational protein therapeutic, also known as fibroblast growth factor-20 (FGF-20), which promotes both epithelial and mesenchymal cell proliferation in vitro and has demonstrated activity in multiple animal models. Velafermin was …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
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Velaglucerase alfa Approved DB06720
biotech | CAS: 884604-91-5

Velaglucerase alfa is a gene-activated human recombinant glucocerebrosidase used for the treatment of Type 1 Gaucher disease, caused by a deficiency of the lysosomal enzyme glucocerebrosidase. Additionally, Velaglucerase alfa has also been investigated for us…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +1
Target Protein:
Lysosomal acid glucosylceramidase
Waktu Paruh11-12 minutes.
Vol. DistribusiThe mean volume of …
KlirensMean clearance rang…
Genetik -
Veldoreotide DB12777
biotech | CAS: 252845-37-7

Somatoprim is under investigation for the treatment of Acromegaly.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
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Veliflapon DB16346
small molecule | CAS: 128253-31-6

Veliflapon is under investigation in clinical trial NCT00353067 (Veliflapon (Dg-031)to Prevent Heart Attacks or Stroke in Patients With a History of Heart Attack or Unstable Angina).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +7
Target Protein:
Arachidonate 5-lipoxygenase-activating protein
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Veligrotug DB18976
biotech | CAS: 2728655-31-8

Veligrotug is under investigation in clinical trial NCT00791544 (Dose Finding Study of AVE1642 in Patients With Advanced or Metastatic Liver Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Velmanase alfa Approved DB12374
biotech | CAS: 1492823-75-2

Velmanase alfa is a recombinant human lysosomal alpha-mannosidase developed for enzyme replacement therapy to treat alpha-mannosidosis. Alpha-mannosidosis is a rare autosomal recessive lysosomal storage disorder. Patients with alpha-mannosidosis have a geneti…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Waktu ParuhAt the end of intra…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
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Velmupressin DB18783
small molecule | CAS: 1647119-61-6

Deskripsi belum tersedia.

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Velneperit DB12889
small molecule | CAS: 342577-38-2

Velneperit has been used in trials studying the treatment of Obesity.

Target Protein:
Neuropeptide Y receptor type 5
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Velpatasvir Approved DB11613
small molecule | CAS: 1377049-84-7

Velpatasvir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiinfectives for Systemic Use +22
Target Protein:
Nonstructural protein 5A
Waktu Paruh15h [FDA Label].
Vol. Distribusi1.4-1.6 L/kg [A191…
KlirensEstimated 0.12 L/h/…
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Velsecorat DB16347
small molecule | CAS: 1196509-60-0

Velsecorat is under investigation in clinical trial NCT02479412 (A Multiple Dosing (14 Days) Study to Assess Efficacy and Safety of Three Dose Levels of AZD7594, Given Once Daily by Inhalation, in Patients With Mild to Moderate Asthma).

Kategori:
Dioxins and Dioxin-like CompoundsHeterocyclic Compounds, Fused-RingPyrazoles
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Veltuzumab DB05656
biotech | CAS: 728917-18-8

Veltuzumab is a monoclonal antibody which, as of October 2009, is undergoing Phase I/II clinical trials for the treatment of non-Hodgkin's lymphoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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Vemircopan DB18012
small molecule | CAS: 2086178-00-7

Deskripsi belum tersedia.

Target Protein:
Complement factor D
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Vemurafenib Approved DB08881
small molecule | CAS: 918504-65-1

Vemurafenib is a competitive kinase inhibitor with activity against BRAF kinase with mutations like V600E.[A31269] It exerts its function by binding to the ATP-binding domain of the mutant BRAF.[A31270] Vemurafenib was co-developed by Roche and Plexxikon and …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimation of t…
KlirensThe total body clea…
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Venadaparib DB17105
small molecule | CAS: 1681017-83-3

Deskripsi belum tersedia.

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Venanprubart DB18891
biotech | CAS: 2635407-50-8

Venanprubart is under investigation in clinical trial NCT05781451 (Anti-btla Agonist Therapy in Subjects With Primary Sjogren's Syndrome).

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Venetoclax Approved DB11581
small molecule | CAS: 1257044-40-8

Venetoclax is a BCL-2 inhibitor that was initially approved by the FDA in April 2016 [FDA label]. Proteins in the B cell CLL/lymphoma 2 (BCL-2) family are important regulators of the apoptotic (programmed cell death) process [A18565], [A18566]. Venetoclax is…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe half-life of ve…
Vol. DistribusiThe population esti…
KlirensMainly hepatic [FDA…
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Venglustat DB14966
small molecule | CAS: 1401090-53-6

Venglustat is under investigation in clinical trial NCT01674036 (Safety, Tolerability and Pharmacokinetics of Genz-682452 in Healthy Men).

Kategori:
Acids, AcyclicEnzyme Inhibitors
Target Protein:
Ceramide glucosyltransferase
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Venlafaxine Approved DB00285
small molecule | CAS: 93413-69-5

Venlafaxine is an antidepressant and a serotonin and norepinephrine reuptake inhibitor (SNRI). Its active metabolite, [desvenlafaxine], works by blocking the reuptake of serotonin and norepinephrine, which are key neurotransmitters in mood regulation. Venlafa…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAmines +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +2
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe apparent volume…
KlirensMean ± SD plasma ap…
Genetik 5 Varian
biotech | CAS: 2724922-85-2

Deskripsi belum tersedia.

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Vepafestinib DB18779
small molecule | CAS: 2129515-96-2

Deskripsi belum tersedia.

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Vepdegestrant DB19006
small molecule | CAS: 2229711-68-4

Vepdegestrant is under investigation in clinical trial NCT05909397 (A Study of ARV-471 (PF-07850327) Plus Palbociclib Versus Letrozole Plus Palbociclib in Participants With Estrogen Receptor Positive, Human Epidermal Growth Factor Negative Advanced Breast Can…

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Vepsitamab DB18211
biotech | CAS: 2413453-53-7

Deskripsi belum tersedia.

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Veralipride DB13523
small molecule | CAS: 66644-81-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntipsychotic Agents +12
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Verapamil Approved DB00661
small molecule | CAS: 52-53-9

Verapamil is a phenylalkylamine calcium channel blocker used in the treatment of high blood pressure, heart arrhythmias, and angina,[L8791] and was the first calcium channel antagonist to be introduced into therapy in the early 1960s.[A188514] It is a member …

Kategori:
ACE Inhibitors and Calcium Channel BlockersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +50
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent P/Q-type calcium channel subunit alpha-1A +10
Gen Terkait:
ADRB1
Waktu ParuhSingle-dose studies…
Vol. DistribusiVerapamil has a ste…
KlirensSystemic clearance …
Genetik 1 Varian
Verbenone DB15977
small molecule | CAS: 80-57-9

Deskripsi belum tersedia.

Kategori:
Bridged-Ring CompoundsMonoterpenesTerpenes
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biotech | CAS: 2364604-87-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Vercirnon DB15250
small molecule | CAS: 698394-73-9

Vercirnon is a novel, orally active anti-inflammatory agent that targets a chemokine receptor protein implicated in both Crohn's disease and ulcerative colitis, the two principal forms of IBD. It is under investigation in clinical trial NCT01611805 (Japanese …

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
C-C chemokine receptor type 9
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Verdinexor DB12207
small molecule | CAS: 1392136-43-4

Kpt 335 is under investigation in clinical trial NCT02431364 (Trial of Safety and Tolerability of Oral Verdinexor (Verdinexor) in Healthy Adults).

Kategori:
Acids, AcyclicAcrylatesAmides
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Verdiperstat DB12440
small molecule | CAS: 890655-80-8

Verdiperstat has been used in trials studying the basic science and treatment of Multiple System Atrophy (MSA).

Kategori:
Pyrimidines
Target Protein:
Myeloperoxidase
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Verekitug DB19096
biotech | CAS: 2768386-15-6

Verekitug is under investigation in clinical trial NCT06164704 (A Study to Investigate the Efficacy and Safety of Verekitug (UPB-101) in Participants With Chronic Rhinosinusitis With Nasal Polyps).

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Vericiguat Approved DB15456
small molecule | CAS: 1350653-20-1

Vericiguat is a direct stimulator of soluble guanylate cyclase (sGC) used in the management of systolic heart failure to reduce mortality and hospitalizations.[L31153] A key component of the NO-sGC-cGMP signaling pathway that helps to regulate the cardiovascu…

Kategori:
BCRP/ABCG2 SubstratesCardiac TherapyGuanylate Cyclase Stimulators +8
Target Protein:
Retinal guanylyl cyclase 1Guanylate cyclase soluble subunit beta-1
Waktu ParuhIn patients with he…
Vol. DistribusiIn healthy subjects…
KlirensVericiguat is a low…
Genetik -
Verinurad DB11873
small molecule | CAS: 1352792-74-5

Verinurad has been used in trials studying the basic science and treatment of Gout, Gout and Hyperuricemia, and Gout and Asymptomatic Hyperuricemia.

Kategori:
Acids, AcyclicAntigout PreparationsAntirheumatic Agents +3
Target Protein:
Solute carrier family 22 member 12
Waktu Paruh-
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biotech | CAS: 295371-00-5

Verpasep caltespen is a recombinant chimeric protein composed of the heat shock protein 65 (Hsp65) from _Mycobacterium bovis_, and the human papilloma viral (HPV) protein E7. Hsp65, similar to other members of its family of proteins, elicits a strong immune r…

Target Protein:
Keratin, type II cytoskeletal 7E3 ubiquitin-protein ligase UBR4
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Verteporfin Approved DB00460
small molecule | CAS: 129497-78-5

Verteporfin, marketed as Visudyne, is a benzoporphyrin derivative comprising a 50:50 mixture of two isomers: [CL-315555] and [CL-315585]. It is used as a photosensitizer in photodynamic therapy to eliminate abnormal blood vessels in wet form macular degenerat…

Kategori:
Antineovascularisation AgentsDermatologicalsEENT Drugs, Miscellaneous +10
Waktu ParuhFollowing intraveno…
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Verticillium albo-atrum Approved DB10850
biotech

Verticillium albo-atrum is a fungus which can provoke allergic reactions. Verticillium albo-atrum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Veru-111 DB16462
small molecule | CAS: 1332881-26-1

VERU-111, an investigational drug intended for various therapeutic uses, was under investigation in clinical trials NCT04842747, NCT03752099, NCT04388826, NCT04844749, NCT05008510, and NCT05079360. These trials aimed to evaluate its efficacy, safety, and tole…

Kategori:
Experimental Unapproved Treatments for COVID-19Heterocyclic Compounds, Fused-Ring
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Verubecestat DB12285
small molecule | CAS: 1286770-55-5

Verubecestat is under investigation for the treatment of Alzheimer's Disease, Prodromal Alzheimer's disease, and Amnestic Mild Cognitive Impairment. Verubecestat is Merck’s investigational oral ?-site amyloid precursor protein cleaving enzyme (BACE1 or ? …

Kategori:
Sulfur CompoundsThiazines
Target Protein:
Beta-secretase 1
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Verubulin DB05585
small molecule | CAS: 827031-83-4

Antineoplastic; a small-molecule inhibitor of microtubule formation that is not a substrate for multidrug resistance pumps.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Verucerfont DB12512
small molecule | CAS: 885220-61-1

Verucerfont has been used in trials studying the treatment of Congenital Adrenal Hyperplasia.

Kategori:
Aza CompoundsOxazolesReceptors, Corticotropin-Releasing Hormone, antagonists & inhibitors
Target Protein:
Corticotropin-releasing factor receptor 1
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Verzistobart DB18895
biotech | CAS: 2649466-18-0

Verzistobart is under investigation in clinical trial NCT06056895 (Triple Immune Checkpoint Inhibition for Advanced or Metastatic PD-(L)1 Refractory Merkel Cell Carcinoma).

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Vesatolimod DB12687
small molecule | CAS: 1228585-88-3

Vesatolimod has been used in trials studying the treatment of Hepatitis B and Chronic Hepatitis B.

Kategori:
Anti-Infective AgentsAntiviral AgentsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Toll-like receptor 7
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