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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 242 / 282
Setiptiline DB09304
small molecule | CAS: 57262-94-9

Setiptiline is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). In Japan, the company Mochida started its commercialization for the treatment of depression started in 1989.

Kategori:
Antidepressive Agents, TetracyclicDibenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Alpha-2 adrenergic receptorsSerotonin Receptors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setmelanotide Approved DB11700
small molecule | CAS: 920014-72-8

Setmelanotide is the first available treatment for patients with pro-opiomelanocortin, proprotein subilisin/kexin type 1, or leptin deficiencies.[L24474] It is an agonist of the melanocortin 4 receptor.[A224449] Earlier attempts at agonizing MC4R (such as LY2…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Obesity Agents +19
Target Protein:
Melanocortin receptor 4
Waktu ParuhThe elimination had…
Vol. DistribusiThe apparent volume…
KlirensA 3mg subcutaneous …
Genetik -
Setogepram DB15447
small molecule | CAS: 1002101-19-0

Setogepram is under investigation in clinical trial NCT03184584 (Open-Label Rollover Study of PBI 4050 in Subjects With Alström Syndrome).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
G-protein coupled receptor 84Free fatty acid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setrobuvir DB12051
small molecule | CAS: 1071517-39-9

Setrobuvir has been used in trials studying the treatment of Hepatitis C, Chronic.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolinesSulfonamides +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevasemten DB18983
small molecule | CAS: 2417395-15-2

Sevasemten is under investigation in clinical trial NCT05291091 (Phase 2 Study of EDG-5506 in Becker Muscular Dystrophy (GRAND CANYON)).

Waktu Paruh-
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Sevelamer Approved DB00658
small molecule | CAS: 52757-95-6

Sevelamer is a phosphate binding drug used to prevent hyperphosphataemia in patients with chronic renal failure. It is marketed by Genzyme under the trade name Renagel.

Kategori:
AminesBile Acid SequestrantsChelating Agents +9
Target Protein:
Phosphate
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seviprotimut-L DB16328
biotech

Seviprotimut-L is under investigation in clinical trial NCT01546571 (Study of a Melanoma Vaccine in Stage Iib, Iic, and III Melanoma Patients).

Waktu Paruh-
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Sevirumab DB17771
biotech | CAS: 138660-96-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seviteronel DB12275
small molecule | CAS: 1610537-15-9

Seviteronel has been used in trials studying the treatment of CRPC, Prostate Cancer, and Castration-resistant Prostate Cancer.

Kategori:
Antineoplastic AgentsCytochrome P-450 Enzyme InhibitorsEnzyme Inhibitors
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevoflurane Approved DB01236
small molecule | CAS: 28523-86-6

Sevoflurane is an ether inhalation anesthetic agent used to induce and maintain general anesthesia.[L42340] It is a volatile, non-flammable compound with a low solubility profile and blood/gas partition coefficient.[L42340] Sevoflurane was patented in 1972, w…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +17
Target Protein:
GABA(A) ReceptorGlycine receptor subunit alpha-1Glutamate receptor 1 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiPatients given low-…
KlirensIn patients given l…
Genetik -
Sevuparin DB15007
small molecule

Sevuparin is under investigation in clinical trial NCT03853421 (Placebo-controlled Study to Determine the Safety and Tolerability of Subcutaneous Doses of Sevuparin).

Kategori:
CarbohydratesGlycosaminoglycansPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SF1126 DB05210
small molecule

SF1126 is an integrin-targeted PI3 kinase inhibitor.

Kategori:
Amino Acids, Peptides, and ProteinsBenzopyransHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Phosphatidylinositol 3-kinase regulatory subunit alphaPhosphatidylinositol 3-kinase regulatory subunit betaPhosphatidylinositol 3-kinase regulatory subunit gamma +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGI-1776 DB12494
small molecule | CAS: 1025065-69-3

SGI-1776 has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias.

Waktu Paruh-
Vol. Distribusi-
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SGN-30 DB05471
biotech

SGN-30 is an engineered monoclonal antibody (mAb) that reacts with significant affinity to the CD30 antigen, which is highly expressed on a variety of hematologic malignancies as compared to on normal cells. SGN-30 has been shown to induce direct anti-cancer…

Target Protein:
Nuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGN-B6A DB18377
biotech | CAS: 2764774-91-4

Sigvotatug vedotin (SGN-B6A) is a humanized immunoglobulin G1 anti-integrin beta-6 monoclonal antibody conjugated to monomethyl auristatin E.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
SGS-742 DB05010
small molecule | CAS: 123690-78-8

SGS-742 has been used in trials studying the treatment of Seizures and Metabolic Disease.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingGABA Agents +4
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
SGS518 DB05042
small molecule

SGS518, a novel antagonist for the 5HT6 subtype of the serotonin receptor, is being developed as a treatment for Cognitive Impairment Associated with Schizophrenia (CIAS).

Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SGX-523 DB06314
small molecule | CAS: 1022150-57-7

A MET receptor tyrosine kinase inhibitor.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Shark liver oil DB11088
biotech | CAS: 68990-63-6

Shark oil is extracted from the livers of sharks, which can account for up to 25% of their total body weight. The 3 main targeted species are the deep sea shark (Centrophorus squamosus), the dogfish (Sqaulus acanthias), and the basking shark (Cetorhinus maxim…

Waktu Paruh-
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Genetik -
Shea butter DB14311
biotech | CAS: 194043-92-0

Shea butter is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanecarboxylic AcidsCyclohexanes +3
Target Protein:
3-phosphoshikimate 1-carboxyvinyltransferase3-phosphoshikimate 1-carboxyvinyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SHR-A1904 DB18702
biotech

SHR-A1904 is under investigation in clinical trial NCT04877717 (A Study of SHR-A1904 in Patients With Advanced Solid Cancer).

Waktu Paruh-
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Genetik -
Siagoside DB12351
small molecule | CAS: 100345-64-0

Siagoside (Sygen, AGF 2) has been investigated for the treatment of Parkinson Disease. It is a naturally occurring substance in the nerve cell’s membrane that is thought to play a role in cell growth, development, and repair. Siagoside completed phase 2 trial…

Kategori:
Acidic GlycosphingolipidsCarbohydratesGangliosides +7
Waktu Paruh-
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Klirens-
Genetik -
Sibeprenlimab DB18919
biotech | CAS: 2382896-07-1

Sibeprenlimab is under investigation in clinical trial NCT05248659 (Phase 2/3 Open-label Trial of Sibeprenlimab in the Treatment of Immunoglobulin a Nephropathy).

Waktu Paruh-
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Sibutramine Approved DB01105
small molecule | CAS: 106650-56-0

Sibutramine (trade name Meridia in the USA, Reductil in Europe and other countries), usually as sibutramide hydrochloride monohydrate, is an orally administered agent for the treatment of obesity. It is a centrally acting stimulant chemically related to amphe…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +23
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Gen Terkait:
GNB3
Waktu Paruh1.1 hours
Vol. Distribusi-
Klirens* Oral cl=1750 L/h …
Genetik 1 Varian
Sifalimumab DB12773
biotech | CAS: 1006877-41-3

Sifalimumab is a fully human monoclonal antibody targeting interferon-alpha. The levels of interferon-alpha are elevated in many patients with active systemic lupus erythematosus (SLE, or lupus) and other autoimmune disorders, and may be associated with disea…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Interferon alpha-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIG-001 DB17826
biotech

SIG-001 is a cultured human retinal pigment epithelial cell line (ARPE-19) genetically modified with a non-viral vector to express B domain deleted human factor VIII protein, encapsulated within two-layer modified alginate spheres.

Waktu Paruh-
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Genetik -
SIG-205 DB18548
biotech

SIG-205 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express human native alpha-L-iduronidase enzyme (hIDUA), encapsulated within two-layer modified alginate spheres

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SIG-207 DB18547
biotech

SIG-207 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express Human alpha-galactosidase A (alpha-Gal A), encapsulated within two-layer modified alginate spheres

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
siG12D LODER DB16329
biotech

siG12D LODER is under investigation in clinical trial NCT01676259 (A Phase 2 Study of Sig12d LODER in Combination With Chemotherapy in Patients With Locally Advanced Pancreatic Cancer).

Waktu Paruh-
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Genetik -
Silatecan DB12384
small molecule | CAS: 220913-32-6

Silatecan has been used in trials studying the treatment of GBM, Tumors, Gliosarcoma, Solid Malignancies, and Glioblastoma Multiforme, among others.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sildenafil Approved DB00203
small molecule | CAS: 139755-83-2

In eliciting its mechanism of action, sildenafil ultimately prevents or minimizes the breakdown of cyclic guanosine monophosphate (cGMP) by inhibiting cGMP specific phosphodiesterase type 5 (PDE5) [F3850, F3853, F3856, F3859, F3883, F3886, L5611, L5614]. The …

Kategori:
Agents Causing Muscle ToxicityAmidesCardiovascular Agents +33
Target Protein:
Plasma protease C1 inhibitorcGMP-specific 3',5'-cyclic phosphodiesteraseRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma +3
Gen Terkait:
ACE GNB3
Waktu ParuhThe terminal phase …
Vol. DistribusiThe mean steady-sta…
KlirensThe total body clea…
Genetik 2 Varian
Silibinin DB09298
small molecule | CAS: 22888-70-6

Silibinin is the major active constituent of silymarin, a standardized extract of the milk thistle seeds, containing a mixture of flavonolignans consisting of silibinin, isosilibinin, silicristin, silidianin and others. Silibinin is presented as a mixture of …

Kategori:
Alimentary Tract and MetabolismAntineoplastic AgentsAntineoplastic Agents, Phytogenic +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silicic acid DB14138
small molecule | CAS: 1343-98-2

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicSilicon Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silicon Approved DB12982
small molecule | CAS: 7440-21-3

Silicon is under investigation in clinical trial NCT00103246 (Photodynamic Therapy Using Silicon Phthalocyanine 4 in Treating Patients With Actinic Keratosis, Bowen's Disease, Skin Cancer, or Stage I or Stage II Mycosis Fungoides).

Kategori:
Diet, Food, and NutritionElementsFood +5
Waktu Paruh-
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Klirens-
Genetik -
Silicon dioxide Approved DB11132
small molecule | CAS: 7631-86-9

Silicon dioxide, or silica, is an oxide of silicon with the chemical formula SiO2. It is found in nature as agate, amethyst, chalcedony, cristobalite, flint, sand, QUARTZ, and tridymite as transparent and tasteless crystals. Inhalation of fine crystals is tox…

Kategori:
ColloidsComplex MixturesCompounds used in a research, industrial, or household setting +6
Target Protein:
Macrophage receptor MARCO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silmitasertib DB15408
small molecule | CAS: 1009820-21-6

Silmitasertib is under investigation in clinical trial NCT03904862 (Testing the Safety and Tolerability of CX-4945 in Patients With Recurrent Medulloblastoma Who May or May Not Have Surgery).

Kategori:
Casein Kinase II, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Casein kinase II subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silodosin Approved DB06207
small molecule | CAS: 160970-54-7

Silodosin is a selective antagonist of alpha(?)-1 adrenergic receptors that binds to the ?<sub>1A</sub> subtype with the highest affinity. ?1-adrenergic receptors regulate smooth muscle tone in the bladder neck, prostate, and prostatic urethra: the ?<sub>1A</…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +15
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu ParuhThe elimination hal…
Vol. DistribusiSilodosin has an ap…
KlirensAfter intravenous a…
Genetik -
Silodrate Approved DB14116
small molecule | CAS: 12408-47-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siltuximab Approved DB09036
biotech | CAS: 541502-14-1

Siltuximab is a chimeric (human-mouse) monoclonal immunoglobulin G1-kappa antibody produced in a Chinese hamster ovary (CHO) cell line by recombinant DNA technology. Siltuximab prevents the binding of IL-6 to soluble and membrane-bound IL-6 receptors by formi…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Interleukin-6
Waktu ParuhThe mean terminal h…
Vol. DistribusiBased on population…
KlirensBody weight was ide…
Genetik -
Silver Approved DB12965
small molecule | CAS: 7440-22-4

Silver (Ag) is a chemical element that belongs in the family of transition metals in the periodic table. It has a high electrical conductivity, thermal conductivity, and reflectivity. Silver exists as a pure elemental form, alloy with other metals, and minera…

Kategori:
Antiseptics and DisinfectantsDermatologicalsElements +4
Target Protein:
MetallothioneinCeruloplasminAlbumin +1
Waktu ParuhThe biological half…
Vol. DistribusiFollowing exposure …
Klirens-
Genetik -
Silver cation DB14521
small molecule | CAS: 14701-21-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver citrate DB11233
small molecule | CAS: 126-45-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver oxide DB15668
small molecule | CAS: 20667-12-3

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Infective AgentsElectrolytes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 9015-51-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Infective Agents, Local +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Silver sulfadiazine Approved DB05245
small molecule | CAS: 22199-08-2

Silver sulfadiazine is a sulfa derivative topical antibacterial used primarily on second- and third-degree burns.

Kategori:
AmidesAminesAniline Compounds +14
Target Protein:
DNADihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simendan DB12286
small molecule | CAS: 131741-08-7

Simendan is under investigation in clinical trial NCT00527059 (Renal Effects of Levosimendan in Patients Admitted With Acute Decompensated Heart Failure).

Kategori:
Antiarrhythmic agentsCardiotonic AgentsCardiovascular Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 910562-13-9

Simenepag isopropyl has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simeprevir Approved DB06290
small molecule | CAS: 923604-59-5

Simeprevir is a hepatitis C virus (HCV) NS3/4A protease inhibitor indicated in patient's with HCV genotype 1 for the treatment of chronic hepatitis C virus (HCV) infection. HCV is a single-stranded RNA virus that is categorized into nine distinct genotypes, w…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +37
Target Protein:
Genome polyproteinNS3 proteaseGenome polyprotein
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of si…
Genetik -
Simethicone Approved DB09512
small molecule | CAS: 8050-81-5

Simethicone is a silicon based surfactant that decreases the surface tension of gastrointestinal gas bubbles to facilitate their elimination.[A228308] It has a favourable safety profile as it is not systemically absorbed.[A228308] Simethicone has been in u…

Kategori:
Antifoaming AgentsCompounds used in a research, industrial, or household settingDermatologicals +9
Waktu ParuhSimethicone is not …
Vol. DistribusiSimethicone is not …
KlirensSimethicone is not …
Genetik -
Menampilkan 12051–12100 dari 14063
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