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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (12560)

Halaman 241 / 252
small molecule

Deskripsi belum tersedia.

Kategori:
Vanadates
Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 58-98-0

A uracil nucleotide containing a pyrophosphate group esterified to C5 of the sugar moiety. [PubChem]

Target Protein:
UDP-N-acetylglucosamine 2-epimeraseHisto-blood group ABO system transferaseGalactose-1-phosphate uridylyltransferase +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Alpha,alpha-trehalose-phosphate synthase [UDP-forming]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycosyl transferaseLgtC
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-glucose 4-epimerase
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-glucose 4-epimerase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-N-acetylmuramoylalanine--D-glutamate ligaseUDP-N-acetylmuramate--L-alanine ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
UDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligaseUDP-N-acetylmuramoylalanine--D-glutamate ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urocortin-2 DB13033
biotech | CAS: 351999-18-3

Urocortin 2 has been investigated for the basic science of Heart Failure and Cardiovascular Disease.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +3
Target Protein:
Corticotropin-releasing factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urofollitropin Approved DB00094
biotech | CAS: 97048-13-0

Urofollitropin is a urinary-derived follicle-stimulating hormone (FSH) that is extracted and purified from human urine samples. It consists of two non-covalently linked, non-identical glycoproteins designated as the alpha- and beta- subunits. The alpha- and b…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesGonadotropins +9
Target Protein:
Follicle-stimulating hormone receptor
Waktu ParuhCirculation half li…
Vol. DistribusiTime to peak in pla…
Klirens-
Genetik -
Urokinase Approved DB00013
biotech | CAS: 9039-53-6

Urokinase is an endogenous peptide that is cleaved in the presence of plasmin between lysine 158 and isoleucine 159 to yield active urokinase.[A191943] Urokinase remains connected between these 2 chains by a sulfhydryl bond.[A191943] Urokinase was granted …

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +15
Target Protein:
PlasminogenUrokinase plasminogen activator surface receptorPlasminogen activator inhibitor 1 +5
Waktu ParuhUrokinase has a hal…
Vol. DistribusiThe volume of distr…
KlirensData regarding the …
Genetik -
Urolithin A DB15464
small molecule | CAS: 1143-70-0

Urolithin A is a metabolite of ellagic acid. It has been demonstrated to stimulate mitophagy and improve muscle health in old animals and in preclinical models of aging.[A179494]

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
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Ursadiol DB14555
small molecule | CAS: 37384-13-7

Deskripsi belum tersedia.

Waktu Paruh-
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Ursodeoxycholic acid Approved DB01586
small molecule | CAS: 128-13-2

Ursodeoxycholic acid (UDCA), also known as ursodiol, is a naturally-occurring bile acid that constitutes a minor fraction of the human bile acid pool.[A256272,A256277] UDCA has been used to treat liver disease for decades: its first use in traditional medicin…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +15
Target Protein:
Aldo-keto reductase family 1 member C2Biliverdin reductase ASolute carrier family 23 member 2 +1
Waktu ParuhThe estimated half-…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Ursolic acid DB15588
small molecule | CAS: 77-52-1

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +13
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Phospholipase A2DNA polymerase catalytic subunit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urtoxazumab DB17806
biotech | CAS: 502496-16-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
USL-311 DB15265
small molecule | CAS: 1373268-67-7

USL-311 is under investigation in clinical trial NCT02765165 (Phase 1/2 Study of USL311 Alone and in Combination With Lomustine in Subjects With Advanced Solid Tumors and Relapsed/Recurrent Glioblastoma Multiforme (GBM)).

Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Usnea barbata Approved DB14351
biotech

Usnea barbata is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Ustekinumab Approved DB05679
biotech | CAS: 815610-63-0

Ustekinumab is a human immunoglobulin (Ig) G1 kappa monoclonal antibody directed against interleukin(IL)-12 and IL-23, which are cytokines that are involved in immune and inflammatory responses.[A187349] It was generated via recombinant human IL-12 immunizati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Interleukin-23Interleukin-12 subunit beta
Waktu ParuhFollowing administr…
Vol. DistribusiThe total volume of…
KlirensThe median apparent…
Genetik -
Ustilago nuda hordei Approved DB10835
biotech

Ustilago nuda hordei is a fungus which can provoke allergic reactions. Ustilago nuda hordei extract is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Utidelone DB17575
small molecule

Utidelone (UTD1), a novel microtubule stabilizing agent, is an epothilone B analogue produced by genetic engineering.[A257544,A257549] It is under investigation in clinical trials for various cancers.

Waktu Paruh-
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Utomilumab DB15113
biotech | CAS: 1417318-27-4

Utomilumab is under investigation in clinical trial NCT03318900 (T Cell Immunotherapy for Advanced Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Utreloxastat DB18154
small molecule | CAS: 1213269-96-5

Deskripsi belum tersedia.

Waktu Paruh-
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Klirens-
Genetik -
Uttroside B DB18633
small molecule | CAS: 88048-09-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
UV1 DB18470
biotech

UV1 is a cancer vaccine consisting of p719-20, p728, and p725 synthetic peptides representing fragments of the hTERT subunit

Waktu Paruh-
Vol. Distribusi-
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Genetik -
UX053 DB18558
biotech

UX053 is an mRNA encoding the human glycogen debranching enzyme.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Uzansertib DB17571
small molecule | CAS: 2088852-47-3

Uzansertib is under investigation in clinical trial NCT02587598 (Study of INCB053914 in Subjects With Advanced Malignancies).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
V-SARS DB15812
biotech

[COVID-19 convalescent plasma] is currently being acquired from recovered COVID-19 patients and used as prophylaxis for the virus. This therapeutic concept was applied to the development of V-SARS, which heat inactivates the plasma, and packages it into a onc…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
V1003 DB05046
small molecule

V1003 is an intranasal formulation of buprenorphine, an opiate analgesic, for the management of post-operative pain in hospital and home settings. Buprenorphine is a well-known analgesic and the intranasal formulation has the potential to provide a convenient…

Target Protein:
Kappa-type opioid receptorMu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V116517 DB16060
small molecule | CAS: 1073616-61-1

V116517 is under investigation in clinical trial NCT01688947 (Analgesic Efficacy and Safety of V116517 in Subjects With Moderate to Severe Chronic Pain Due to Postherpetic Neuralgia (PHN)).

Kategori:
AminesPyridines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
V24343 DB05201
small molecule

The anti-obesity drug, V24343, acts by targeting the CB1 receptor in the brain and suppressing a person's appetite.

Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V590 DB16437
biotech

The V590 vaccine was developed on Merck’s recombinant vesicular stomatitis virus (rVSV) platform that was previously used to develop its Ebola Zaire virus vaccine, ERVEBO®[A226818, L30573, L30578]. By teaming up with IAVI, Merk developed a vaccine that does n…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
V591 DB16438
biotech

The V591 vaccine, part of Merck’s COVID-19 vaccine programming, was developed using a modified measles vaccine virus as a vector for COVID-19 antigen delivery[L30593]. Through Merck’s acquisition of Thermis in May 2020, they were able to leverage Thermis’ pla…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
VA-MENGOC-BC® DB15800
biotech

VA-MENGOC-BC is a meningococcal B and C vaccine and an outer membrane vesicle (OMV)-based vaccine. The OMVs contain over 100 proteins, and are derived from meningococcal group B and capsular polysaccharide of meningococcal group C. As there already exists a p…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vabicaserin DB12071
small molecule | CAS: 887258-95-9

Vabicaserin has been used in trials studying the health services research and treatment of Schizophrenia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vaborbactam Approved DB12107
small molecule | CAS: 1360457-46-0

Vaborbactam is a ?-lactamase inhibitor based on a cyclic boronic acid pharmacophore.[A32053] It has been used in trials investigating the treatment of bacterial infections in subjects with varying degrees of renal insufficiency. In August 2017, a combination …

Kategori:
AcidsAcids, NoncarboxylicAnti-Infective Agents +6
Target Protein:
Beta-lactamaseBeta-lactamaseCarbapenem-hydrolyzing beta-lactamase KPC +7
Waktu ParuhThe half life of va…
Vol. DistribusiThe steady-state vo…
KlirensThe mean renal clea…
Genetik -
VAC-52150 DB17781
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vactosertib DB15310
small molecule | CAS: 1352608-82-2

Vactosertib is under investigation in clinical trial NCT03724851 (Vactosertib in Combination With Pembrolizumab in Metastatic Colorectal or Gastric Cancer).

Kategori:
AminesEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
TGF-beta receptor type-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vadadustat Approved DB12255
small molecule | CAS: 1000025-07-9

One of the most common symptoms of advanced renal disease is anemia, caused primarily by the inability of the kidney to respond to anemic conditions with a corresponding increase in [erythropoietin] (EPO) production.[A244165] The treatment of anemia associate…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntianemic Preparations +20
Target Protein:
Egl nine homolog 1Prolyl hydroxylase EGLN2Prolyl hydroxylase EGLN3 +2
Waktu ParuhIn patients with di…
Vol. DistribusiThe apparent volume…
KlirensIn healthy subjects…
Genetik -
biotech | CAS: 1436390-64-5

Vadastuximab Talirine has been used in trials studying the treatment of Acute myeloid leukemia, Myelodysplastic Syndrome, Acute Myelogenous Leukemia, and Acute Promyelocytic Leukemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Myeloid cell surface antigen CD33
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vadimezan DB06235
small molecule | CAS: 117570-53-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +4
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vafidemstat DB16446
small molecule | CAS: 1357362-02-7

Vafidemstat is under investigation in clinical trial NCT03867253 (Testing the Safety and Preliminary Efficacy of the New Drug ORY-2001 in Mild to Moderate Alzheimer's Disease).

Kategori:
Oxazoles
Target Protein:
Lysine-specific histone demethylase 1AAmine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valaciclovir Approved DB00577
small molecule | CAS: 124832-26-4

Valaciclovir (valacyclovir), also known as _Valtrex_, is an antiviral drug that has been used to manage and treat various herpes infections for more than 2 decades. It was initially approved by the FDA in 1995 [FDA label] and marketed by GlaxoSmithKline [L56…

Kategori:
Acyclovir and prodrugAmino AcidsAmino Acids, Branched-Chain +19
Target Protein:
Thymidine kinaseDNA polymerase catalytic subunit
Waktu ParuhThe plasma eliminat…
Vol. DistribusiCerebrospinal fluid…
KlirensRenal clearance of …
Genetik -
Valanafusp alfa DB15336
biotech | CAS: 1815583-32-4

Valanafusp alfa is under investigation in clinical trial NCT03071341 (Extension Study Evaluating Long Term Safety and Activity of AGT-181 in Children With MPS I).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valbenazine Approved DB11915
small molecule | CAS: 1025504-45-3

Valbenazine is a modified metabolite of [tetrabenazine], and it is currently being approved for the treatment of various movement disorders, particularly tardive dyskinesia and chorea associated with Huntington's disease.[L47885,A261135] Tardive dyskinesia ha…

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +11
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhBoth Valbenazine an…
Vol. DistribusiThe mean steady-sta…
KlirensValbenazine has a m…
Genetik -
Valdecoxib Approved DB00580
small molecule | CAS: 181695-72-7

Valdecoxib was removed from the Canadian, U.S., and E.U. markets in 2005 due to concerns about a possible increased risk of heart attack and stroke.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +29
Target Protein:
Prostaglandin G/H synthase 2Carbonic anhydrase 2Carbonic anhydrase 3
Waktu Paruh8-11 hours
Vol. Distribusi* 86 L
Klirens* oral cl=6 L/h * …
Genetik -
Valerian Approved DB13196
biotech | CAS: 8057-49-6

Valerian is extracted from a herb that is a perennial flowering plant. Valerian root is reported to have sedative and anxiolytic effects however its mechanism of action is not completely understood. Valerian has been used in the treatment of conditions includ…

Kategori:
AngiospermsBiological ProductsCentral Nervous System Depressants +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valganciclovir Approved DB01610
small molecule | CAS: 175865-60-8

Valganciclovir hydrochloride (Valcyte, manufactured by Roche) is an antiviral medication used to treat cytomegalovirus infections. As the L-valyl ester of ganciclovir, it is actually a prodrug for ganciclovir. After oral administration, it is rapidly converte…

Kategori:
Agents that reduce seizure thresholdAnti-Infective AgentsAntiinfectives for Systemic Use +13
Target Protein:
DNA polymerase catalytic subunitDNA
Waktu ParuhApproximately 4.08 …
Vol. Distribusi* 0.703 ± 0.134 L/kg
Klirens* 3.07+/- 0.64 mL/m…
Genetik -
Menampilkan 12001–12050 dari 12560
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