Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 241 / 282
Selpercatinib Approved DB15685
small molecule | CAS: 2152628-33-4

Selpercatinib is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A202052, L13604] Enhanced RET (Rearranged during transfection) oncogene expression is a hallmark of many cancers. Although …

Kategori:
Agents that produce hypertensionAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3 +3
Waktu ParuhSelpercatinib has a…
Vol. DistribusiSelpercatinib has a…
KlirensSelpercatinib has a…
Genetik -
Seltorexant DB14961
small molecule | CAS: 1452539-75-1

Seltorexant is under investigation in clinical trial NCT03494907 (A Study to Evaluate the Effects of Single-dose Seltorexant on Electrocardiogram Intervals in Healthy Adult Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selumetinib Approved DB11689
small molecule | CAS: 606143-52-6

Activation of the Raf-MEK-ERK signalling pathway is known to be implemented in several types of malignancies; thus, mitogen-activated protein kinase kinase (MEK) inhibitors such as selumetinib are important tools that can target the problematic overactivity o…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +18
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1Dual specificity mitogen-activated protein kinase kinase 2
Waktu ParuhSelumetinib is char…
Vol. DistribusiThe mean apparent v…
KlirensThe clearance of se…
Genetik -
Selurampanel DB12367
small molecule | CAS: 912574-69-7

Selurampanel has been investigated in Adrenocortical Adenoma and Sarcoma, Endometrial Stromal.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semagacestat DB12463
small molecule | CAS: 425386-60-3

Semagacestat has been used in trials studying the treatment of Alzheimer Disease.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmyloid Precursor Protein Secretases, antagonists & inhibitors +2
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semaglutide Approved DB13928
small molecule | CAS: 910463-68-2

Semaglutide is a glucagon-like peptide 1 (GLP-1) analog used to manage type 2 diabetes along with lifestyle changes, such as dietary restrictions and increased physical activity.[A31421,L8681] Other members of this drug class include [Exenatide] and [Liraglut…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhOne of the major pr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Semapimod DB12094
small molecule | CAS: 352513-83-8

Semapimod has been used in trials studying the treatment of Crohn Disease.

Kategori:
AmidesAmidinesAmines +9
Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semorinemab DB15234
biotech | CAS: 2159141-27-0

Semorinemab is under investigation in clinical trial NCT03289143 (A Study to Evaluate the Efficacy and Safety of RO7105705 in Patients With Prodromal to Mild Alzheimer's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semuloparin DB06294
small molecule

Deskripsi belum tersedia.

Kategori:
AnticoagulantsCarbohydratesCardiovascular Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semzuvolimab DB18920
biotech | CAS: 2409099-32-5

Semzuvolimab is under investigation in clinical trial NCT03149211 (To Investigate the Efficacy and Safety of UB-421 Monotherapy in HIV-1 Infected Adults).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Retroviral Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senaparib DB17163
small molecule | CAS: 1401682-78-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senicapoc DB06280
small molecule | CAS: 289656-45-7

Senicapoc (ICA-17043) is a novel Gardos channel blocker.[A259068] It is being investigated for the treatment of sickle cell disease.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Intermediate conductance calcium-activated potassium channel protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senlizumab DB17894
biotech | CAS: 336128-48-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sennosides DB11365
small molecule | CAS: 517-43-1

Sennosides (also known as senna glycoside or senna) is a medication used to treat constipation[FDA Label][L771] and empty the large intestine before surgery. The medication is taken by mouth or via the rectum[FDA Label]. It typically begins working in minutes…

Kategori:
Alimentary Tract and MetabolismAnthracenesAnthraquinones +13
Target Protein:
Aquaporin-3Reverse transcriptase/RNaseH
Waktu ParuhThe half life of ra…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ra…
Genetik -
Senrebotase DB12626
biotech | CAS: 1290102-81-6

Senrebotase has been used in trials studying the treatment of Neuralgia, Postherpetic and Urinary Bladder, Overactive.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seocalcitol DB04258
small molecule | CAS: 134404-52-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsCholestanesCholestenes +11
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEP-363856 DB15665
small molecule | CAS: 1310426-33-5

SEP-363856 is a novel psychotropic drug being investigated for the treatment of schizophrenia. Unlike other drugs used for this condition, SEP-363856 does not bind to the dopamine D2 receptors, but exerts actions on the trace amine–associated receptor 1 (TAA…

Target Protein:
5-hydroxytryptamine receptor 1ATrace amine-associated receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepantronium DB17062
small molecule | CAS: 753440-91-4

Sepantronium is a compound that suppresses survivin expression in a dose and time-dependent manner, and causes broad-range apoptosis.[A253167]

Kategori:
NaphthalenesQuinones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepetaprost DB12043
small molecule | CAS: 1262873-06-2

Sepetaprost has been used in trials studying the treatment of Open Angle-glaucoma, Ocular Hypertension, and Mild Open Angle-glaucoma (OAG).

Kategori:
EthersEthers, Cyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEphB4-HSA DB14797
biotech

SEphB4-HSA is under investigation in clinical trial NCT02495896 (Recombinant EphB4-HSA Fusion Protein With Standard Chemotherapy Regimens in Treating Patients With Advanced or Metastatic Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepiapterin DB16326
small molecule | CAS: 17094-01-8

Sepiapterin is under investigation in clinical trial NCT03519711 (A Study of CNSA-001 in Primary Tetrahydrobiopterin (BH4) Deficient Participants With Hyperphenylalaninemia).

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepofarsen DB16327
biotech | CAS: 2227173-68-2

Sepofarsen is under investigation in clinical trial NCT03913143 (A Study to Evaluate Efficacy, Safety, Tolerability and Exposure After a Repeat-dose of Sepofarsen (QR-110) in LCA10 (ILLUMINATE)).

Kategori:
OphthalmologicalsSensory Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepranolone DB12972
small molecule | CAS: 516-55-2

Sepranolone has been investigated for the treatment of Premenstrual Dysphoric Disorder.

Kategori:
AnestheticsCentral Nervous System AgentsCentral Nervous System Depressants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seproxetine DB06731
small molecule | CAS: 126924-38-7

Seproxetine is also known as (S)-norfluoxetine. It is a selective serotonin reuptake inhibitor (SSRI). It is an active metabolite of fluoxetine. Seproxetine was being investigated by Eli Lilly as an antidepressant but development was never completed and the d…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2C19 Inhibitors +14
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu Paruh4-16 days
Vol. Distribusi-
Klirens-
Genetik -
SER-100 DB16013
small molecule | CAS: 383123-18-0

SER-100 is under investigation in clinical trial NCT01987284 (SER100 in Isolated Systolic Hypertension).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Nociceptin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SER-287 DB18204
biotech

SER-287 comprises healthy microbiome-derived Gram positive bacterial spores.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serabelisib DB14935
small molecule | CAS: 1268454-23-4

Serabelisib is under investigation in clinical trial NCT02625259 (A Study to Evaluate the Relative Bioavailability, Effect of Food, and Gastric Potential Hydrogen (pH) Modification on the Pharmacokinetics of TAK-117 (MLN1117) in Healthy Participants).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingOxazines
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seractide acetate Approved DB09334
biotech | CAS: 39295-97-1

Seractide acetate is the acetate salt of full length human corticotropin.

Target Protein:
Adrenocorticotropic hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seralutinib DB18072
small molecule | CAS: 1619931-27-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seratrodast DB06739
small molecule | CAS: 112665-43-7

Seratrodast (INN) is a thromboxane receptor antagonist used primarily in the treatment of asthma.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Asthmatic Agents +27
Target Protein:
Thromboxane A2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serdemetan DB12027
small molecule | CAS: 881202-45-5

Serdemetan has been used in trials studying the treatment of Neoplasms.

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Target Protein:
E3 ubiquitin-protein ligase Mdm2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serdexmethylphenidate Approved DB16629
small molecule | CAS: 1996626-29-9

Attention Deficit Hyperactivity Disorder (ADHD) is an early-onset neurodevelopmental disorder that often extends into adulthood and is characterized by developmentally inappropriate and impaired attention, impulsivity, and motor hyperactivity.[A230698, A23070…

Kategori:
Agents that produce hypertensionCentral Nervous System AgentsCentral Nervous System Stimulants +12
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 1A
Waktu ParuhFollowing a single …
Vol. DistribusiSerdexmethylphenida…
KlirensSerdexmethylphenida…
Genetik -
Serelaxin DB05794
biotech | CAS: 99489-94-8

Recombinant human relaxin is a hormone produced during pregnancy that facilitates the birth process by causing a softening and lengthening of the cervix and the pubic symphysis (the place where the pubic bones come together).It is a heterodimer protein secret…

Kategori:
Cardiac TherapyVasodilators Used in Cardiac Diseases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seribantumab DB11857
biotech | CAS: 1334296-12-6

Seribantumab has been used in trials studying the treatment of NSCLC, Heregulin, Adenocarcinoma, Colorectal Cancer, and Solid Tumor Cancers, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serine DB00133
small molecule | CAS: 56-45-1

A non-essential amino acid occurring in natural form as the L-isomer. It is synthesized from glycine or threonine. It is involved in the biosynthesis of purines; pyrimidines; and other amino acids.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +3
Target Protein:
Cystathionine beta-synthaseL-serine dehydratase/L-threonine deaminaseSerine racemase +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Threonine--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serlopitant DB12973
small molecule | CAS: 860642-69-9

Serlopitant has been investigated for the treatment of Prurigo Nodularis.

Kategori:
Heterocyclic Compounds, Fused-RingNeurokinin-1 Receptor AntagonistsNeurotransmitter Agents
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sermorelin Approved DB00010
biotech | CAS: 86168-78-7

Sermorelin acetate is the acetate salt of an amidated synthetic 29-amino acid peptide (GRF 1-29 NH 2 ) that corresponds to the amino-terminal segment of the naturally occurring human growth hormone-releasing hormone (GHRH or GRF) consisting of 44 amino acid r…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesDiagnostic Agents +13
Target Protein:
Growth hormone-releasing hormone receptor
Waktu Paruh11-12 min
Vol. Distribusi-
Klirens-
Genetik -
Serotonin DB08839
small molecule | CAS: 50-67-9

For temporary relief of nervousness, anxiety, mood swings, joint pains, weakness, drowsiness, itching and lethargy. Not evaluated by the FDA, homeopathic product.

Kategori:
AminesAntidepressive AgentsAutacoids +19
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 75-hydroxytryptamine receptor 2B +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SerpinPC DB17698
biotech

SerpinPC is a mutated alpha-1-antitrypsin (?1AT) and serine protease inhibitor being investigated for the treatment of hemophilia.[A258993]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serplulimab DB17451
biotech | CAS: 2231029-82-4

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Serrapeptase DB13131
biotech | CAS: 95077-02-4

Serrapeptase is a proteolytic enzyme preparation used concomitantly with an antibiotic in osteoarticular infections. Serratiopeptidase is under investigation in clinical trial NCT02493179 (Efficacy Evaluation of the (Serodase 5 mg Tablet) in the Treatment of …

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sertaconazole Approved DB01153
small molecule | CAS: 99592-32-2

Sertaconazole nitrate is an antifungal medication of the imidazole class. It is available in topical formulations for the treatment of skin infections such as athlete's foot.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +8
Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sertindole Approved DB06144
small molecule | CAS: 106516-24-9

Sertindole, a neuroleptic, is one of the newer antipsychotic medications available. Serdolect is developed by the Danish pharmaceutical company H. Lundbeck. It is a phenylindole derivative used in the treatment of schizophrenia. It was first marketed in 1996 …

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +22
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C +5
Waktu Paruh3 days
Vol. Distribusi-
Klirens-
Genetik -
Sertraline Approved DB01104
small molecule | CAS: 79617-96-2

Sertraline is a popular antidepressant medication commonly known as a selective serotonin reuptake inhibitor (SSRI), and is similar to drugs such as [Citalopram] and [Fluoxetine]. Despite marked structural differences between compounds in this drug class, SSR…

Kategori:
Agents that reduce seizure thresholdAminesAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent dopamine transporterSigma receptor +2
Gen Terkait:
CYP2C19 CYP2C19
Waktu ParuhThe elimination hal…
Vol. DistribusiSertraline is widel…
KlirensIn pharmacokinetic …
Genetik 2 Varian
Sesame oil DB11172
biotech | CAS: 8008-74-0

Sesame oil is a commonly used vegetable oil in Asia and flavoring enhancer in various culinary practices. It is extracted from sesame seeds and contains linoleic acid, oleic acid, palmitic acid, stearic acid and other fatty acids. Sesame oil is reported to po…

Kategori:
Biological ProductsComplex MixturesDiet, Food, and Nutrition +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2379806-98-9

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setanaxib DB16869
small molecule | CAS: 1218942-37-0

Deskripsi belum tersedia.

Kategori:
PyrazolesPyridines
Target Protein:
NADPH oxidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Setipiprant DB12562
small molecule | CAS: 866460-33-5

Setipiprant has been investigated for the treatment of Seasonal Allergic Rhinitis, asthma and scalp hair loss (Androgenetic Alopecia).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prostaglandin D2 receptorProstaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 12001–12050 dari 14063
Sebelumnya Halaman 241 / 282 Berikutnya