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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 240 / 321
Parathiazine DB15978
small molecule | CAS: 84-08-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parathyroid hormone Approved DB05829
biotech | CAS: 9002-64-6

Parathyroid hormone (PTH) is a single-chain polypeptide composed of 84 amino acids. Available as Preotact, it is an identical form of human recombinant hormome which produced as a fusion protein undergoeing post-translational processing involving the cleava…

Kategori:
Amino Acids, Peptides, and ProteinsCalcium HomeostasisCalcium-Regulating Hormones and Agents +7
Target Protein:
Parathyroid hormone 2 receptorParathyroid hormone/parathyroid hormone-related peptide receptor
Waktu Paruh1.5 hours.
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
biotech | CAS: 172867-62-8

Parathyroid Hormone-Related Protein 1-36 is under investigation in clinical trial NCT00853723 (Comparison Study of Pthrp and PTH to Treat Osteoporosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pardoprunox DB12061
small molecule | CAS: 269718-84-5

Pardoprunox has been used in trials studying the treatment of Early Stage Parkinson's Disease and Advanced Stage Parkinson's Disease. Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parecoxib Approved DB08439
small molecule | CAS: 198470-84-7

Parecoxib is a water-soluble and injectable prodrug of valdecoxib. It is marketed as Dynastat in the European Union. Parecoxib is a COX2 selective inhibitor in the same category as celecoxib (Celebrex) and rofecoxib (Vioxx). As it is injectable, it can be use…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Target Protein:
Prostaglandin G/H synthase 2Lactotransferrin
Waktu Paruh22 minutes (parecox…
Vol. Distribusi-
Klirens-
Genetik -
Parethoxycaine DB19380
small molecule | CAS: 94-23-5

Parethoxycaine is a local anesthetic that was previously approved in the US.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pargeverine DB15783
small molecule | CAS: 13479-13-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pargyline Approved DB01626
small molecule | CAS: 555-57-7

Pargyline is a monoamine oxidase inhibitor with antihypertensive properties.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +12
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paricalcitol Approved DB00910
small molecule | CAS: 131918-61-1

Paricalcitol is a synthetic vitamin D analog. Paricalcitol has been used to reduce parathyroid hormone levels. Paricalcitol is indicated for the prevention and treatment of secondary hyperparathyroidism associated with chronic renal failure.

Kategori:
Anti-Parathyroid AgentsBone Density Conservation AgentsCalcium Homeostasis +16
Target Protein:
Vitamin D3 receptor
Waktu Paruh4 to 6 hours
Vol. Distribusi* 30.8 ± 7.5 L [CKD…
Klirens* 1.49 +/- 0.60 L/h…
Genetik -
biotech | CAS: 2259927-72-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paritaprevir Approved DB09297
small molecule | CAS: 1216941-48-8

Paritaprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into ni…

Kategori:
AmidesAmino AcidsAmino Acids, Cyclic +27
Target Protein:
Genome polyproteinGag-Pol polyprotein
Waktu Paruh5.5 hr [FDA Label]
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
Parnaparin Approved DB09260
small molecule | CAS: 9005-49-6

Parnaparin is an heparin of low molecular weight with antithrombotic effects.

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paromomycin Approved DB01421
small molecule | CAS: 7542-37-2

An oligosaccharide antibiotic produced by various streptomyces. [PubChem]

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmebicides +10
Target Protein:
30S ribosomal protein S1016S ribosomal RNASmall ribosomal subunit protein uS2 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paroxetine Approved DB00715
small molecule | CAS: 61869-08-7

Paroxetine is a selective serotonin reuptake inhibitor (SSRI) drug commonly known as Paxil. It has a variety of uses, including the treatment of anxiety disorders, major depression, posttraumatic stress disorder, and symptoms of menopause, among others.[T653]…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 2A +9
Gen Terkait:
ABCB1 CYP2D6 CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiParoxetine has a la…
KlirensThe apparent oral c…
Genetik 7 Varian
PARPI F-18 DB18657
small molecule | CAS: 1883580-48-0

PARPI F-18 is a diagnostic agent under investigation for use in the management of glioblastoma multiforme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parsaclisib DB14867
small molecule | CAS: 1426698-88-5

Parsaclisib is under investigation in clinical trial NCT03126019 (An Open-Label Study of Parsaclisib in Relapsed or Refractory Follicular Lymphoma (CITADEL-203)).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsPhosphatidylinositol-3-kinase (Pi3K) inhibitors +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parsatuzumab DB14897
biotech | CAS: 1312797-14-0

Parsatuzumab is under investigation in clinical trial NCT01366131 (Study Evaluating the Safety and Efficacy of MEGF0444A in Combination With Carboplatin, Paclitaxel and Bevacizumab in Patients With Advanced or Recurrent Non-Squamous Non-Small Cell Lung Cancer…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parthenolide Approved DB13063
small molecule | CAS: 20554-84-1

Parthenolide has been used in trials studying the diagnostic of Allergic Contact Dermatitis.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +8
Target Protein:
Proto-oncogene c-RelTranscription factor RelBInhibitor of nuclear factor kappa-B kinase subunit beta +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PAS-004 DB18611
small molecule

PAS-004 is an allosteric MEK 1/2 inhibitor being developed by Pasithea Therapeutics. It is being investigated for the treatment of neurofibromatosis 1 and Noonan syndrome.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pascolizumab DB06560
biotech | CAS: 331243-22-2

Pascolizumab (SB 240683) is a humanized anti-interleukin-4 antibody with therapeutic potential in asthma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Target Protein:
Interleukin-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pasireotide Approved DB06663
small molecule | CAS: 396091-73-9

Pasireotide is a synthetic long-acting cyclic hexapeptide with somatostatin-like activity. It is marketed as a diaspartate salt called Signifor, which is used in the treatment of Cushing's disease.

Kategori:
Amino Acids, Peptides, and ProteinsBradycardia-Causing AgentsCytochrome P-450 CYP3A Inhibitors +22
Target Protein:
Somatostatin receptor type 3Somatostatin receptor type 1Somatostatin receptor type 2 +1
Waktu ParuhThe half-life is 12…
Vol. DistribusiPasireotide is wide…
KlirensThe clearance in he…
Genetik -
PAT-1251 DB16735
small molecule | CAS: 2098884-52-5

PAT-1251 is under investigation in clinical trial NCT04054245 (PAT-1251 in Treating Patients With Primary Myelofibrosis, Post-polycythemia Vera Myelofibrosis, or Post-essential Thrombocytosis Myelofibrosis).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PAT-SM6 DB17406
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pateclizumab DB14997
biotech | CAS: 1202526-59-7

Pateclizumab is under investigation in clinical trial NCT01225393 (A Study to Evaluate the Efficacy and Safety of MLTA3698A in Combination With a Disease-Modifying Anti-Rheumatic Drug (DMARD) Compared With Adalimumab in Combination With a DMARD in Patients Wi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patent Blue Approved DB13967
small molecule | CAS: 25305-77-5

Patent blue is aniline dye and it is one of the most common dyes used.[A32573] It is a sodium or calcium salt of diethylammonium hydroxide inner salt.[A32574] It has the chemical designation of (4-(alpha-(p-(diethylamino)phenyl)-2,4-disulfobenzylidene)-2,5-cy…

Kategori:
AminesAniline CompoundsColoring Agents +4
Target Protein:
Albumin
Waktu ParuhThe elimination hal…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Patidegib DB12655
small molecule | CAS: 1037210-93-7

Patidegib has been investigated for the treatment of Conventional Chondrosarcoma.

Kategori:
Alkaloids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2376210-48-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patiromer Approved DB09263
small molecule | CAS: 1260643-52-4

Patiromer is a powder for suspension in water for oral administration, approved in the U.S. as Veltassa in October, 2015. Patiromer is supplied as patiromer sorbitex calcium which consists of the active moiety, patiromer, a non-absorbed potassium-binding poly…

Kategori:
Cation Exchange ResinsCompounds used in a research, industrial, or household settingMacromolecular Substances +3
Target Protein:
Potassium
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patisiran Approved DB14582
biotech | CAS: 1420706-45-1

Patisiran is a first in class short interfering RNA for the treatment of patients with polyneuropathy caused by hereditary transthyretin-mediated amyloidosis [L4220]. It is marketed as Onpattro which is formulated as patisiran within a liposome envelope for b…

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingDecreased RNA Integrity +12
Target Protein:
Transthyretin mRNA
Waktu ParuhPatisiran has a ter…
Vol. DistribusiThe steady state vo…
KlirensThe total body clea…
Genetik -
Patritumab DB12090
biotech | CAS: 1262787-83-6

Patritumab has been used in trials studying the treatment of LUNG CANCER, Solid Tumors, Neoplasms by Site, Head and Neck Neoplasms, and Non-small Cell Lung Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patulin DB15586
small molecule | CAS: 149-29-1

Deskripsi belum tersedia.

Kategori:
Biological FactorsCompounds used in a research, industrial, or household settingMutagens +6
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patupilone DB03010
small molecule | CAS: 152044-54-7

Epothilone B is a 16-membered macrolide that mimics the biological effects of taxol.

Kategori:
Anti-Bacterial AgentsAntimitotic AgentsAntineoplastic Agents +9
Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-4B chain +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pavinetant DB11692
small molecule | CAS: 941690-55-7

Pavinetant has been used in trials studying the basic science and treatment of Safety and Schizophrenia.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingQuinolines +3
Target Protein:
Neuromedin-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paxalisib DB15186
small molecule | CAS: 1382979-44-3

GDC-0084 is under investigation in clinical trial NCT03696355 (Study of GDC-0084 in Pediatric Patients With Newly Diagnosed Diffuse Intrinsic Pontine Glioma or Diffuse Midline Gliomas).

Kategori:
Enzyme Inhibitors
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pazopanib Approved DB06589
small molecule | CAS: 444731-52-6

Pazopanib is a small molecule inhibitor of multiple protein tyrosine kinases with potential antineoplastic activity. It is developed by GlaxoSmithKline and was FDA approved on October 19, 2009.

Kategori:
AmidesAngiogenesis InhibitorsAntineoplastic Agents +36
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +7
Gen Terkait:
UGT1A1 HCP5
Waktu Paruh35 hours. Oral abso…
Vol. DistribusiVd steady state, IV…
KlirensCL, cancer patient,…
Genetik 2 Varian
Pazufloxacin DB11774
small molecule | CAS: 127045-41-4

Pazufloxacin is under investigation in clinical trial NCT02592096 (Pazufloxacin Mesilate Ear Drops Clinical Trial Protocol).

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PB-722 DB18447
biotech

PB-722 is a long-acting glucagon receptor agonist.[L48260]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBCAR20A DB17189
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBCAR269A DB17188
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBFT02 DB18580
biotech

PBFT02 is a non-replicating recombinant adeno-associated virus serotype 1 vector delivering human GRN gene encoding the protein progranulin.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBGM01 DB18581
biotech

PBGM01 is a non-replicating recombinant adeno-associated virus serotype hu68 vector, which contains human GLB1 transgene encoding the galactosidase beta 1 enzyme.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBI-1402 DB05480
small molecule

PBI-1402 is a small molecule synthetic compound with oral Bioavailability. The compound activates neutrophils, enhancing their survival and activation with comparable efficacy to GM-CSF, G-CSF and EPO, which are currently used to treat anemia. However, it ha…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBKR03 DB18138
biotech

PBKR03 is a non-replicating recombinant adeno-associated virus serotype hu68 vector, containing a transgene encoding the human galactosylceramidase (GALC) enzyme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBR-06 F-18 DB17020
small molecule | CAS: 1003581-94-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBT-1033 DB05565
small molecule | CAS: 747408-78-2

Deskripsi belum tersedia.

Target Protein:
Microtubule-associated protein tau
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBT-434 Approved DB16965
small molecule | CAS: 1232840-87-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCI-27483 DB13000
small molecule | CAS: 871266-63-6

PCI-27483 has been used in trials studying the treatment of Pancreatic Cancer, Ductal Adrenocarcinoma, and Exocrine Pancreatic Cancer.

Kategori:
AmidesAmidinesAmino Acids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCLX-001 DB15567
small molecule | CAS: 1215011-08-7

PCLX-001 is a first-in-kind N-Myristoyltransferase (NMT) inhibitor being developed by [Pacylex Pharmaceuticals](https://pacylex.com). Current studies have shown that PCLX-001 works differently than other known cancer drugs and has high activity and positive r…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCO-371 DB14946
small molecule | CAS: 1613373-33-3

PCO-371 is under investigation in clinical trial NCT02475616 (A Single Ascending Dose Study of PCO371 in Healthy Volunteers).

Kategori:
Imidazoles
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCS-499 DB15122
small molecule | CAS: 1268605-91-9

PCS-499 is under investigation in clinical trial NCT01487109 (A Phase 2 Study to Evaluate the Safety and Efficacy of CTP-499 in Type 2 Diabetic Nephropathy Patients).

Kategori:
DeuteriumHeterocyclic Compounds, Fused-RingPurines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11951–12000 dari 16004
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