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2279

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Halaman 24 / 46
Isatuximab Approved DB14811
biotech | CAS: 1461640-62-9

Isatuximab (formerly SAR650984) is a humanized, IgG1-derived monoclonal antibody (mAb) produced from a Chinese hamster ovary (CHO) cell line.[L12099,A191799] Structurally, isatuximab is comprised of two identical immunoglobulin kappa light chains and two iden…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. DistribusiThe predicted volum…
KlirensTotal clearance dec…
Genetik -
Islatravir DB15653
small molecule | CAS: 865363-93-5

Islatravir is under investigation in clinical trial NCT04233216 (Doravirine/islatravir (DOR/ISL) in Heavily Treatment-experienced (HTE) Participants for Human Immunodeficiency Virus Type 1 (HIV-1) Infection (MK-8591A-019)).

Kategori:
AlcoholsAnti-Infective AgentsAnti-Retroviral Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isoeugenol Approved DB14188
small molecule | CAS: 97-54-1

Isoeugenol is a commonly used fragrance added to many commercially available products, and occurs naturally in the essential oils of plants such as ylang-ylang. It is also a significant dermatologic sensitizer and allergen, and as a result has been restricted…

Kategori:
Acids, CarbocyclicAlkenesAllyl Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isoflavone DB12007
small molecule | CAS: 574-12-9

Isoflavone is a soy phytoestrogen and a biologically active component of several agriculturally important legumes such as soy, peanut, green peas, chick peas and alfalfa [A33103]. Soybean is an exceptionally rich source of dietary isoflavones, where the avera…

Kategori:
BenzopyransChromonesDrugs that are Mainly Renally Excreted +4
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gamma
Waktu ParuhThe half-life of is…
Vol. DistribusiIsoflavones are rea…
KlirensIn a human study, t…
Genetik -
Isoleucine DB00167
small molecule | CAS: 73-32-5

An essential branched-chain aliphatic amino acid found in many proteins. It is an isomer of leucine. It is important in hemoglobin synthesis and regulation of blood sugar and energy levels.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Short/branched chain specific acyl-CoA dehydrogenase, mitochondrialBranched-chain-amino-acid aminotransferase, cytosolicBranched-chain-amino-acid aminotransferase, mitochondrial +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 961-29-5

Isoliquiritigenin is a precursor to several flavonones in many plants.

Kategori:
BenzopyransChromonesEnzyme Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isopropyl alcohol Approved DB02325
small molecule | CAS: 67-63-0

An isomer of 1-propanol. It is a colorless liquid having disinfectant properties. It is used in the manufacture of acetone and its derivatives and as a solvent. Topically, it is used as an antiseptic.

Kategori:
AlcoholsAntiseptics and DisinfectantsCompounds used in a research, industrial, or household setting +5
Target Protein:
Nitric oxide synthase 3Oxysterols receptor LXR-betaHeme oxygenase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isosorbide mononitrate Approved DB01020
small molecule | CAS: 16051-77-7

Isosorbide mononitrate is an organic nitrate with vasodilating properties. It is an anti-anginal agent that works by relaxing the smooth muscles of both arteries and veins, but but predominantly veins to reduce cardiac preload.[L11698, L11743] Isosorbide mono…

Kategori:
AlcoholsAntianginal AgentsCarbohydrates +14
Target Protein:
Guanylate cyclase soluble subunit alpha-2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe total body clea…
Genetik -
biotech | CAS: 2413386-21-5

Ispectamab debotansine is an antibody drug conjugate comprised of an anti-B cell maturation (BCMA) IgG1 humanized antibody conjugated covalently to the dibenzocyclooctyne (DBCO) noncleavable linker maytansinoid warhead.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Itepekimab DB16206
biotech | CAS: 2226742-52-3

Itepekimab is under investigation in clinical trial NCT03546907 (Proof-of-concept Study to Assess the Efficacy, Safety and Tolerability of SAR440340 (Anti-il-33 Mab) in Patients With Moderate-to-severe Chronic Obstructive Pulmonary Disease (COPD)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ivabradine Approved DB09083
small molecule | CAS: 155974-00-8

Ivabradine is a novel heart rate lowering medicine for the symptomatic management of stable angina pectoralis and symptomatic chronic heart failure. Ivabradine, brand name Corlanor, was approved by the FDA in April 2015 for the treatment of chronic heart fai…

Kategori:
BenzazepinesBradycardia-Causing AgentsCardiac Therapy +10
Target Protein:
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2
Waktu Paruh2 hours.
Vol. Distribusi~100 L.
KlirensTotal clearance is …
Genetik -
Ivacaftor Approved DB08820
small molecule | CAS: 873054-44-5

Ivacaftor (also known as Kalydeco or VX-770) is a drug used for the management of Cystic Fibrosis (CF). It is manufactured and distributed by Vertex Pharmaceuticals. It was approved by the Food and Drug Administration on January 31, 2012[L768], and by Health …

Kategori:
AminesAniline CompoundsBenzene Derivatives +20
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Gen Terkait:
CFTR
Waktu ParuhIn a clinical study…
Vol. DistribusiAfter oral administ…
KlirensThe CL/F (SD) for t…
Genetik 1 Varian
Ivermectin Approved DB00602
small molecule | CAS: 70288-86-7

Ivermectin is a semi-synthetic antiparasitic medication derived from avermectins, a class of highly-active broad-spectrum antiparasitic agents isolated from the fermentation products of _Streptomyces avermitilis_.[L31453] Ivermectin itself is a mixture of two…

Kategori:
Agents Causing Muscle ToxicityAgrochemicalsAnthelmintics +25
Target Protein:
Glutamate-gated chloride channel subunit betaGlutamate-gated chloride channel alpha
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Ivonescimab DB18931
biotech | CAS: 2428381-53-5

Ivonescimab is under investigation in clinical trial NCT05184712 (Phase 3 Clinical Study of AK112 for NSCLC Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ivosidenib Approved DB14568
small molecule | CAS: 1448347-49-6

Ivosidenib is a first-in-class isocitrate dehydrogenase-1 (IDH1) inhibitor. IDH1 is an enzyme that is often mutated and overexpressed in some cancers, leading to aberrant cell growth and proliferation.[A248750] Ivosidenib inhibits mutated IDH1, blocking the e…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +26
Target Protein:
Isocitrate dehydrogenase [NADP] cytoplasmic
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
IVT-8086 DB18381
biotech

IVT-8086 is a humanized secreted frizzled-related protein-2 monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ixekizumab Approved DB11569
biotech | CAS: 1143503-69-8

Ixekizumab is a humanized immunoglobulin G subclass 4 (IgG4) monoclonal antibody (mAb) against interleukin-17A (IL-17A) and prevents it from interacting with the IL-17A receptor. As IL-17A is a pro-inflammatory cytokine involved in inflammation and immune res…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Interleukin-17A
Waktu Paruh13 days
Vol. DistribusiThe mean (geometric…
Klirens0.39 L/day
Genetik -
Izokibep DB19081
biotech | CAS: 2226130-02-3

Izokibep is under investigation in clinical trial NCT05623345 (Psoriatic Arthritis Study of Izokibep).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Izuralimab DB18933
biotech | CAS: 2329669-80-7

Izuralimab is under investigation in clinical trial NCT05879185 (A Study of Xmab23104 in People With Sarcoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
J147 DB13957
small molecule | CAS: 1146963-51-0

J147 is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging. [A31606,A31607,A31608] It is a curcumin derivative and a potent neurogenic and neuroprotective drug candidate initially develo…

Kategori:
AlkanesBenzene DerivativesCatechols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Janssen COVID-19 Vaccine Approved DB15857
biotech

The Janssen COVID-19 vaccine (Ad26.COV2.S) is a recombinant vaccine that contains an adenovirus serotype 26 (Ad26) vector expressing a stabilized SARS-CoV-2 spike protein. The vaccine was created in collaboration with Johnson and Johnson (J&J), Janssen Pharma…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JB991 DB05081
small molecule

JB991 is a cyclopentenone prostaglandin analogue intended for treatment of psoriasis. The drug exerts marked antiproliferative and pro-apoptotic effect in human keratinocytes and fibroblasts in vitro. In addition a closely related cyclopentenone prostaglandin…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
jCell DB17906
biotech

jCell is an human retinal progenitor cell therapy for retinitis pigmentosa.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-27390467 DB06962
small molecule | CAS: 1025795-11-2

JNJ-27390467 is a potent, nonpeptide inhibitor of human mast cell tryptase.

Target Protein:
Tryptase beta-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KAb201 DB17210
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB001 DB05222
biotech

KB001 is a Humaneered™ PEGylated monoclonal antibody fragment for the treatment of life-threatening Pseudomonas aeruginosa infections, a common problem of cystic fibrosis and mechanically ventilated patients.

Target Protein:
Low calcium response locus protein V
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB002 DB05194
small molecule

KB002 is an engineered human IgG1k antibody engineered human. It is developed for the treatment of autoimmune diseases, initially rheumatoid arthritis.

Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaGranulocyte-macrophage colony-stimulating factorGM-CSF receptor alpha subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ketorolac Approved DB00465
small molecule | CAS: 74103-06-3

Ketorolac is a Non-steroidal anti-inflammatory drug (NSAID) and is commercially available as an oral tablet, injectable, nasal spray and as an ophthalmic solution.[L6358][L6508][L11055][L3674][L11070] It's analgesic properties make it a useful pain manage…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +26
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhKetorolac trometham…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Kinetin Approved DB11336
small molecule | CAS: 525-79-1

Kinetin is a cytokinin which are plant hormones promotes cell division and plant growth. It was shown to naturally exist in DNA of organisms including humans and various plants. While kinetin is used in tissue cultures to produce new plants, it is also found …

Kategori:
CytokininsGrowth SubstancesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kisspeptin-10 DB16210
biotech | CAS: 374675-21-5

Kisspeptin-10 is under investigation in clinical trial NCT03771326 (KP-10 and Insulin Secretion in Men).

Kategori:
Amino Acids, Peptides, and ProteinsGenes, Tumor SuppressorIntercellular Signaling Peptides and Proteins +5
Target Protein:
KiSS-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KITE-585 DB17409
biotech

KITE-585 is an autologous, fully-human anti-B cell maturation antigen (BCMA) chimeric antigen receptor (CAR) T cell therapy. It is being investigated in the treatment of multiple myeloma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Konjac mannan DB14963
small molecule | CAS: 37220-17-0

Konjac mannan is under investigation in clinical trial NCT01709955 (The Effects of Glucomannan on Weight Loss).

Kategori:
CarbohydratesGastrointestinal AgentsLaxatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KRN-330 DB19075
biotech

Anti-a33 fully-human monoclonal antibody is under investigation in clinical trial NCT00838578 (Phase I/II Study of KRN330 Plus Irinotecan in Patients With Metastatic Colorectal Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KRN-5500 DB15215
small molecule | CAS: 151276-95-8

KRN-5500 is under investigation in clinical trial NCT00002923 (KRN5500 in Treating Patients With Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-3972-T DB17441
biotech | CAS: 2170699-22-4

L-3972-T is one of the components of the human papilloma virus (HPV) type 16 E6/E7 synthetic long peptide (SLP) vaccine ISA101b.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Acetylleucine Approved DB16956
small molecule | CAS: 1188-21-2

Levacetylleucine (L-acetylleucine) is a modified acetylated derivative of the amino acid [leucine]. The racemic (i.e. DL-) form has been available in France since 1957 for the treatment of vertigo.[A264439] Observational studies in patients with Niemann-Pi…

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +7
Waktu ParuhThe half-life of le…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
L-cysteic acid DB03661
small molecule | CAS: 498-40-8

L-cysteic acid is a beta-sulfoalanine. It is an amino acid with a C-terminal sulfonic acid group which has been isolated from human hair oxidized with permanganate. It occurs normally in the outer part of the sheep's fleece, where the wool is exposed to light…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +1
Target Protein:
M-phase inducer phosphatase 2Peptide deformylaseTyrosine-protein phosphatase non-receptor type 1 +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Glutamine Approved DB00130
small molecule | CAS: 56-85-9

A non-essential amino acid present abundantly throughout the body and is involved in many metabolic processes. It is synthesized from glutamic acid and ammonia. It is the principal carrier of nitrogen in the body and is an important energy source for many cel…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids and Derivatives +8
Target Protein:
CTP synthase 1AmidophosphoribosyltransferaseGlutamine synthetase
Waktu ParuhThe half life of el…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesMonosaccharides
Target Protein:
Ferrichrome-iron receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Rhamnitol DB02399
small molecule | CAS: 488-28-8

Deskripsi belum tersedia.

Target Protein:
L-rhamnose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-tartaric acid DB09459
small molecule | CAS: 87-69-4

Tartaric acid is a white crystalline organic acid that occurs naturally in many plants, most notably in grapes.Tartaric is an alpha-hydroxy-carboxylic acid, is diprotic and aldaric in acid characteristics, and is a dihydroxyl derivative of succinic acid.

Kategori:
Acids, AcyclicCarbohydratesChelating Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Labetuzumab DB05097
biotech | CAS: 219649-07-7

Labetuzumab is a humanized monoclonal antibody to carcinoembryonic antigen that inhibits tumor growth. It is used in radioimmunotherapy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Cell adhesion molecule CEACAM5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lactic acid Approved DB04398
small molecule | CAS: 50-21-5

A normal intermediate in the fermentation (oxidation, metabolism) of sugar. The concentrated form is used internally to prevent gastrointestinal fermentation. (From Stedman, 26th ed) Sodium lactate is the sodium salt of lactic acid, and has a mild saline tast…

Kategori:
Basic Ointments and ProtectantsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +6
Target Protein:
Bifunctional protein PutANimA-related protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lactitol Approved DB12942
small molecule | CAS: 585-86-4

Lactitol, also known as 4-?-D-galactopyranosyl-D-glucitol, is a sugar alcohol synthesized from [lactose].[A190918] It is used in food manufacturing as a nutritive sweetener and is approximately 35% as sweet as table sugar (i.e. [sucrose]).[A190912] Clinically…

Kategori:
AlcoholsAlimentary Tract and MetabolismCarbohydrates +15
Waktu ParuhThe average half-li…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Lactose Approved DB04465
small molecule | CAS: 63-42-3

A disaccharide of glucose and galactose in human and cow milk. It is used in pharmacy for tablets, in medicine as a nutrient, and in industry.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +9
Target Protein:
Galectin-3SialidaseBeta-galactosidase +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lactulose Approved DB00581
small molecule | CAS: 4618-18-2

Lactulose is a synthetic disaccharide derivative of lactose that is most commonly used as a laxative agent despite also being formally indicated to serve as an adjunct therapy in treating portal-systemic encephalopathy (PSE).[FDA Label,L6199,L6202] Despite be…

Kategori:
Acidifying ActivityAlimentary Tract and MetabolismAmmonia Detoxicants +8
Target Protein:
Evolved beta-galactosidase subunit alpha
Waktu ParuhThe data regarding …
Vol. DistribusiNegligible amounts …
KlirensNegligible amounts …
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Camphor 5-monooxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lamivudine Approved DB00709
small molecule | CAS: 134678-17-4

A reverse transcriptase inhibitor and zalcitabine analog in which a sulfur atom replaces the 3' carbon of the pentose ring. It is used to treat Human Immunodeficiency Virus Type 1 (HIV-1) and hepatitis B (HBV).

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +26
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHDNA +1
Waktu Paruh5 to 7 hours (healt…
Vol. DistribusiApparent volume of …
Klirens* Renal clearance =…
Genetik -
Lanadelumab Approved DB14597
biotech | CAS: 1426055-14-2

Lanadelumab, also known as DX-2930, is a human IgG1 monoclonal antibody designed for subcutaneous self-injection.[L4538] It is a fully human immunoglobulin, k-light-chain made in recombinant Chinese Hamster Ovary cells.[L4537] It has been granted priority rev…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Plasma kallikrein
Waktu ParuhLanadelumab has a h…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Lanimostim DB06559
small molecule | CAS: 117276-75-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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