Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 24 / 134
Asparagine Approved DB00174
small molecule | CAS: 70-47-3

A non-essential amino acid that is involved in the metabolic control of cell functions in nerve and brain tissue. It is biosynthesized from aspartic acid and ammonia by asparagine synthetase. (From Concise Encyclopedia Biochemistry and Molecular Biology, 3rd …

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Target Protein:
Sodium-coupled neutral amino acid transportersNeutral amino acid transporter B(0)Asparagine synthetase [glutamine-hydrolyzing] +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspartame DB00168
small molecule | CAS: 22839-47-0

Flavoring agent sweeter than sugar, metabolized as phenylalanine and aspartic acid.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +13
Target Protein:
Taste receptor type 1 member 3Taste receptor type 1 member 2Transient receptor potential cation channel subfamily V member 1
Waktu ParuhAt room temperature…
Vol. Distribusi-
Klirens-
Genetik -
Aspartic acid Approved DB00128
small molecule | CAS: 56-84-8

One of the non-essential amino acids commonly occurring in the L-form. It is found in animals and plants, especially in sugar cane and sugar beets. It may be a neurotransmitter.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2AGlutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 1 +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
(S)-2-haloacid dehalogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspoxicillin DB13816
small molecule | CAS: 63358-49-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astemizole Approved DB00637
small molecule | CAS: 68844-77-9

Astemizole is a long-acting, non-sedating second generation antihistamine used in the treatment of allergy symptoms. It was withdrawn from market by the manufacturer in 1999 due to the potential to cause arrhythmias at high doses, especially when when taken …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzimidazoles +27
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated delayed rectifier potassium channel KCNH1 +1
Waktu Paruh1 day
Vol. Distribusi-
Klirens-
Genetik -
Astodrimer DB11854
biotech | CAS: 1379746-42-5

Astodrimer has been used in trials studying the treatment and prevention of Bacterial Vaginosis. It is a lysine-based dendrimer with naphthalene disulfonic acid surface groups.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
Envelope glycoprotein gp160
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AstraZeneca COVID-19 Vaccine Approved DB15656
biotech | CAS: 2420395-83-9

The AstraZeneca COVID-19 Vaccine (previously known as ChAdOx1 nCoV-19 or AZD1222) is one of several vaccines developed in 2020 for the prevention of COVID-19 caused by SARS-CoV-2.[L12669,L32649] The ChAdOx1 viral vector was developed at the University of Oxfo…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asunaprevir Approved DB11586
small molecule | CAS: 630420-16-5

Asunaprevir, also named BMS-650032, is a potent hepatitis C virus (HCV) NS3 protease inhibitor. It has been shown to have a very high efficacy in dual-combination regimens with daclatasvir in patients chronically infected with HCV genotype 1b.[A32528] It was …

Kategori:
AmidesAntiinfectives for Systemic UseAntiviral Agents +35
Target Protein:
Gag-Pol polyproteinGenome polyprotein
Waktu ParuhClinical pharmacoki…
Vol. DistribusiThe registered volu…
KlirensClinical pharmacoki…
Genetik -
Asundexian DB19088
small molecule | CAS: 2064121-65-7

Asundexian is under investigation in clinical trial NCT05686070 (A Study to Test Asundexian for Preventing a Stroke Caused by a Clot in Participants After an Acute Ischemic Stroke or After a High-risk Transient Ischemic Attack, a So-called Mini Stroke).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Coagulation factor XI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-301 DB16507
biotech

AT-301 was under investigation in clinical trial NCT01675284 to evaluate the safety, reactogenicity, and humoral immune responses to an inactivated H5N1 influenza vaccine

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-7519 DB08142
small molecule | CAS: 844442-38-2

AT7519 is a selective inhibitor of certain Cyclin Dependent Kinases (CDKs) leading to tumour regression. It is developed by Astex for the treatment of solid tumours and haematological malignancies.

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitors
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT1022 DB04995
small molecule

AT1022 is a hydromorphone skin patch designed to provide rapid and sustained delivery of a potent opiate for the management of severe pain. AT1022 incorporates PassPort(TM) system, developed to deliver protein and peptide drugs, small-molecule drugs, genes a…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT2220 DB05200
small molecule

AT2220 is an experimental, oral therapy for the treatment of Pompe disease and belongs to a class of molecules known as pharmacological chaperones. It is a small molecule designed to act as a pharmacological chaperone that specifically binds, stabilizes, and …

Target Protein:
Lysosomal alpha-glucosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT3022 DB05172
small molecule

AT3022, the Altea Therapeutics’s fentanyl citrate transdermal patch designed to provide safe and rapid management of moderate to severe chronic pain.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATA-100 DB18329
biotech

ATA-100 is an adeno-associated virus serotype 9 carrying the human Fukutin-Related protein gene and target sequence of the miR-208a

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atacicept DB06399
biotech | CAS: 845264-92-8

Atacicept is a recombinant fusion protein combined with the extracellular ligand binding portion of TACI.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ataciguat DB12805
small molecule | CAS: 254877-67-3

Ataciguat has been investigated for the basic science of Aortic Valve Stenosis.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +5
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ataluren Approved DB05016
small molecule | CAS: 775304-57-9

Ataluren is a novel, orally administered drug that targets nonsense mutations. Ataluren is approved for use by the European Medicines Agency to treat Duchenne Muscular Dystrophy in patients aged 5 years and older who are able to walk. More specifically, atalu…

Kategori:
Musculo-Skeletal SystemOAT1/SLC22A6 inhibitorsOAT3/SLC22A8 Inhibitors +3
Target Protein:
Dystrophin
Waktu ParuhAtaluren plasma hal…
Vol. Distribusi-
Klirens-
Genetik -
Atazanavir Approved DB01072
small molecule | CAS: 198904-31-3

Atazanavir (formerly known as BMS-232632) is an antiretroviral drug of the protease inhibitor (PI) class. Like other antiretrovirals, it is used to treat infection of human immunodeficiency virus (HIV). Atazanavir is distinguished from other PIs in that it ca…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +45
Target Protein:
Pol polyproteinGag-Pol polyprotein
Gen Terkait:
UGT1A1 UGT1A1 UGT1A1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn patients with HI…
KlirensIn patients with HI…
Genetik 3 Varian
small molecule | CAS: 433937-93-0

Atecegatran metoxil has been used in trials studying the basic science and prevention of Nonvalvular Atrial Fibrillation, Persistent or Permanent Nonvalvular Atrial Fibrillation, and Persistent or Permanent Non-valvular Atrial Fibrillation.

Kategori:
Azetines
Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atexakin alfa DB19234
biotech | CAS: 143631-61-2

Atexakin alfa is under investigation in clinical trial NCT05435742 (SON-080 in Patients With Persistent Chemotherapy-induced Peripheral Neuropathy (CIPN)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atezolizumab Approved DB11595
biotech | CAS: 1380723-44-3

Atezolizumab is a humanized monoclonal antibody used to prevent the interaction of PD-L1 and PD-1, removing inhibition of immune responses seen in some cancers.[A18493,L7489] This medication is reserved for patients whose tumors express PD-L1, cannot receive …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhThe half life of at…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of at…
Genetik -
ATG-101 DB17162
biotech

ATG-101 is a novel PD-L1/4-1BB bispecific antibody that was designed to block the binding of immunosuppressive PD-1/PD-L1 and conditionally induce 4-1BB stimulation, thus activating anti-tumor immune effectors, while delivering enhanced anti-tumor activity, w…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATI-1013 DB18185
biotech

ATI-1013 is a fully human nicotine-specific monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aticaprant DB12341
small molecule | CAS: 1174130-61-0

Aticaprant has been used in trials studying the health services research and basic science of Anxiety Disorders and Alcohol Dependence.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +5
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atidarsagene autotemcel Approved DB17538
biotech

Atidarsagene autotemcel, sold under the brand name Libmeldy, is a gene therapy comprising genetically modified autologous CD34+ enriched hematopoietic stem and progenitor cells transduced _ex vivo_ using a lentiviral vector encoding the human arylsulfatase A …

Kategori:
Alimentary Tract and MetabolismAutologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene Therapy +2
Target Protein:
Human Arylsulfatase A mRNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atilotrelvir DB19439
small molecule | CAS: 2850365-55-6

Atilotrelvir is under investigation in clinical trial NCT05041907 (Finding Treatments for COVID-19: A Trial of Antiviral Pharmacodynamics in Early Symptomatic COVID-19 (PLATCOV)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atisnolerbart DB19418
biotech | CAS: 2456308-79-3

Atisnolerbart is under investigation in clinical trial NCT06602739 (A Study to Demonstrate the Effect of REGN5713-5715 on Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Birch Pollen Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atlantic mackerel Approved DB15542
biotech

Atlantic mackerel allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atogepant Approved DB16098
small molecule | CAS: 1374248-81-3

Atogepant is an oral antagonist of calcitonin gene-related peptide (CGRP) receptors indicated for the prevention of episodic migraine headaches. It was developed by AbbVie and received FDA approval under the brand name Qulipta in September 2021.[L38814] While…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Atoltivimab Approved DB15898
biotech | CAS: 2135632-29-8

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhAtoltivimab adminis…
Vol. DistribusiAtoltivimab adminis…
KlirensAtoltivimab adminis…
Genetik -
Atomoxetine Approved DB00289
small molecule | CAS: 83015-26-3

Atomoxetine is a selective norepinephrine (NE) reuptake inhibitor used for the treatment of attention deficit hyperactivity disorder (ADHD). Also known as the marketed product Strattera, atomoxetine is used with other treatment modalities (psychological, educ…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterNMDA receptor +2
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +3
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe clearance rate …
Genetik 6 Varian
Atorvastatin Approved DB01076
small molecule | CAS: 134523-00-5

Atorvastatin (Lipitor®), is a lipid-lowering drug included in the statin class of medications. By inhibiting the endogenous production of cholesterol in the liver, statins lower abnormal cholesterol and lipid levels, and ultimately reduce the risk of cardiova…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +37
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseDipeptidyl peptidase 4Aryl hydrocarbon receptor +2
Gen Terkait:
KIF6 HMGCR CYP3A4
Waktu ParuhThe half-life of at…
Vol. DistribusiThe reported volume…
KlirensThe registered tota…
Genetik 3 Varian
Atosiban Approved DB09059
small molecule | CAS: 90779-69-4

Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used intravenously to halt premature labor. Although initial studies suggested it could be used as a nasal spray and hence would not require hospital admission, it is not used in that fo…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormone Antagonists +8
Target Protein:
Oxytocin receptorVasopressin V1a receptorVasopressin V1b receptor +1
Waktu ParuhAtosiban does not c…
Vol. DistribusiAtosiban has a mean…
KlirensAtosiban has a mean…
Genetik -
ATP DB00171
small molecule | CAS: 56-65-5

An adenine nucleotide containing three phosphate groups esterified to the sugar moiety. In addition to its crucial roles in metabolism adenosine triphosphate is a neurotransmitter.

Kategori:
Adenine NucleotidesAdenosine TriphosphateDietary Supplements +7
Target Protein:
Tyrosine-protein kinase ABL1ATP-binding cassette sub-family C member 6ATP-binding cassette sub-family C member 4 +39
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Atractylodes japonica root oil is obtained from the roots of Atractylodes japonica, which is a herb native to eastern Asia. It is present in some cosmetic products such as whitening creams as an active ingredient and lubricant for skin irritation. Atractylode…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atrazine DB07392
small molecule | CAS: 1912-24-9

Atrazine is a selective triazine herbicide. Inhalation hazard is low and there are no apparent skin manifestations or other toxicity in humans. Acutely poisoned sheep and cattle may show muscular spasms, fasciculations, stiff gait, increased respiratory rates…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingHerbicides +3
Target Protein:
Photosynthetic reaction center cytochrome c subunitReaction center protein H chainReaction center protein L chain +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atropine Approved DB00572
small molecule | CAS: 51-55-8

Atropine is an alkaloid originally synthesized from Atropa belladonna. It is a racemic mixture of d-and l-hyoscyamine, of which only l-hyoscyamine is pharmacologically active.[A251670,L42835] Atropine is generally available as a sulfate salt and can be admini…

Kategori:
Adjuvants, AnesthesiaAgents producing tachycardiaAgents that produce hypertension +32
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhFollowing intraveno…
Vol. DistribusiAtropine is distrib…
KlirensFollowing intraveno…
Genetik -
ATSN-101 DB18327
biotech

ATSN-101 is a adeno-associated virus serotype 5 encoding human retinal guanylate cyclase 1 gene (AAV5-GUCY2D)

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Attapulgite Approved DB01574
small molecule | CAS: 12174-11-7

Attapulgite is a magnesium aluminium phyllosilicate which occurs in a type of clay soil common to the Southeastern United States. When used in medicine, it physically binds to acids and toxic substances in the stomach and digestive tract. For that reason, it …

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsAntidotes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATX-101 DB05780
small molecule

ATX-101 (medical), sodium deoxycholate for subcutaneous injection, is being evaluated as a treatment for the reduction of localized fat deposits. This includes treatment of superficial lipomas (benign tumors of soft tissue composed of mature fat cells), fat d…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATX-201 DB05765
small molecule

ATX-201 is one of a family of novel compounds that inhibits microtubule polymerization. It is developed by Kythera Biopharmaceuticals, Inc. for the treatment of actinic keratosis. The company announced the decision to discontinue its ATX-201 clinical program…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Auranofin Approved DB00995
small molecule | CAS: 34031-32-8

Auranofin is a gold salt that is capable of eliciting pharmacologic actions that suppress inflammation and stimulate cell-mediated immunity. It has subsequently been listed by the World Health Organization as a member of the antirheumatic agent category. Aura…

Kategori:
Antiinflammatory and Antirheumatic ProductsAntirheumatic AgentsDrugs that are Mainly Renally Excreted +6
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aurodox DB04124
small molecule | CAS: 12704-90-4

Aurodox is an antibiotic obtained from a streptomyces variant considered as possibly effective against streptococcus pyogenes infections. It may promote growth in poultry.

Kategori:
AlkenesAnti-Bacterial AgentsAnti-Infective Agents +2
Target Protein:
Elongation factor Tu-B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aurothioglycanide Approved DB19361
small molecule | CAS: 16925-51-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AUTO3 DB17364
biotech

AUTO3 is bicistronic chimeric antigen receptor T-cell therapy investigated for acute lymphoblastic leukemia (ALL). It is an investigational chimeric antigen receptor (CAR) T cell treatment targeting CD19 and CD22.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2365453-34-3

Autogene cevumeran is an mRNA-based cancer vaccine targeting an unspecified amount of tumour-associated antigens. It is being investigated for cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Autologous DNP-conjugated tumour vaccine, or melanoma vaccine, is an investigational autologous cell vaccine technology for melanoma.[A254806]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Autologous pancreatic islet therapy involves isolating the patient's own insulin-producing cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1151–1200 dari 6694
Sebelumnya Halaman 24 / 134 Berikutnya