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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 239 / 282
Saralasin DB06763
small molecule | CAS: 34273-10-4

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAgents that produce hypertension +8
Target Protein:
Type-2 angiotensin II receptorType-1 angiotensin II receptor
Waktu Paruh-
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Genetik -
Sarcosine DB12519
small molecule | CAS: 107-97-1

Sarcosine has been investigated for the treatment of Schizophrenia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsN-substituted Glycines
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Genetik -
Sarecycline Approved DB12035
small molecule | CAS: 1035654-66-0

Sarecycline is a semi-synthetic derivative of tetracycline that was initially discovered by Paratek Pharmaceuticals from Boston, MA but then licensed to Warner Chilcott of Rockaway, NJ in July of 2007 [A40005]. After completing various phase-II and phase-III …

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Systemic UseAnti-Bacterial Agents +7
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Saredutant DB06660
small molecule | CAS: 142001-63-6

Saredutant (SR 48968) is a neurokinin-2 antagonist drug being developed as an antidepressant and anxiolytic by Sanofi-Aventis.

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +4
Target Protein:
Substance-K receptor
Waktu Paruh-
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Sargramostim Approved DB00020
biotech | CAS: 123774-72-1

Sargramostim is a human recombinant granulocyte macrophage colony-stimulating factor (GM-CSF) expressed in yeast. It is a glycoprotein that is 127 residues. Substitution of Leu23 leads to a difference from native protein.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaInterleukin-3 receptor subunit alphaCytokine receptor common subunit beta +2
Waktu Paruh-
Vol. Distribusi-
Klirens* 420 mL/min/m2 [No…
Genetik -
Sarilumab Approved DB11767
biotech | CAS: 1189541-98-7

Sarilumab is a fully human anti-interleukin 6 (IL-6) receptor monoclonal IgG1 antibody that binds to both membrane-bound and soluble IL-6 receptor forms, thus blocking the cis- and trans-inflammatory signalling cascades of IL-6.[A27262] Sarilumab was develope…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
Interleukin-6 receptor subunit alphaHigh affinity immunoglobulin gamma Fc receptor ILow affinity immunoglobulin gamma Fc region receptor II-a +3
Waktu ParuhThe half-life will …
Vol. DistribusiIn patients with rh…
KlirensSarilumab is not el…
Genetik -
Sarizotan DB06454
small molecule | CAS: 351862-32-3

Deskripsi belum tersedia.

Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptorD(3) dopamine receptor
Waktu Paruh-
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Saroglitazar DB13115
small molecule | CAS: 495399-09-2

Saroglitazar has been investigated for the treatment of Fatty Liver.

Kategori:
Acids, Carbocyclic
Waktu Paruh-
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Sarpogrelate DB12163
small molecule | CAS: 125926-17-2

Sarpogrelate has been investigated for the treatment of Diabetes Mellitus, Diabetic Nephropathy, Coronary Artery Disease, and Renal Insufficiency, Chronic.

Kategori:
Acids, AcyclicAntidepressive AgentsAntiplatelet agents +8
Target Protein:
5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sarracenia Purpurea Approved DB13965
biotech

_Sarracenia purpurea_, commonly known as the purple pitcher plant, northern pitcher plant, turtle socks, or side-saddle flower, is a perennial carnivorous plant in the family _Sarraceniaceae_. _Sarracenia purpurea_ attract and trap insects within their pitche…

Kategori:
Miscellaneous Analgesics and Antipyretics
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
biotech

SARS-CoV-2 mRNA vaccine (ARCoV) is a novel mRNA coronavirus vaccine that consists of a lipid nanoparticle-encapsulated mRNA encoding the receptor binding domain of SARS-CoV-2[A220048]. It is the first COVID-19 mRNA vaccine to be approved for clinical trials …

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biotech

The University of Queensland (UQ), in partnership with The Coalition for Epidemic Preparedeness Inovations (CEPI) and CSL has developed a COVID-19 candidate, SARS-CoV-2 Sclamp. The vaccine was developed using UQ’s rapid response ‘molecular clamp’ vaccine plat…

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biotech

Bimervax is an adjuvanted non-mRNA COVID-19 vaccine utilizing a SARS-CoV-2 recombinant spike (S) protein receptor binding domain (RBD) fusion heterodimer.[L48902] It is intended to elicit protection against Omicron XBB.1.5, one of the dominant circulating SAR…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
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Sarsagenin DB16928
small molecule | CAS: 126-19-2

Deskripsi belum tersedia.

Kategori:
CholestanesDrugs, Chinese HerbalFused-Ring Compounds +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Saruparib DB18982
small molecule | CAS: 2589531-76-8

Saruparib is under investigation in clinical trial NCT06380751 (Saruparib (AZD5305) Plus Camizestrant Compared With CDK4/6 Inhibitor Plus Endocrine Therapy or Plus Camizestrant in Hr-positive, Her2-negative (IHC 0, 1+, 2+/ ISH Non-amplified), BRCA1, BRCA2, or…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Sasanlimab DB18849
biotech | CAS: 2206792-50-7

Sasanlimab is under investigation in clinical trial NCT06218069 (Immuno-pet Imaging Responses Administered Immune Checkpoint Inhibitor).

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Satavaptan DB14923
small molecule | CAS: 185913-78-4

Satavaptan is under investigation in clinical trial NCT00359437 (Satavaptan in the Prevention of Ascites Recurrence in Patients With Ascites Due to Cirrhosis of the Liver).

Kategori:
Antidiuretic Hormone Receptor AntagonistsNatriuretic AgentsOxazines
Target Protein:
Vasopressin V2 receptor
Waktu Paruh-
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Genetik -
small molecule | CAS: 1039726-31-2

Deskripsi belum tersedia.

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Satralizumab Approved DB15762
biotech | CAS: 1535963-91-7

Satralizumab is a recombinant humanized monoclonal antibody targeted against human interleukin-6 (IL-6) receptors, similar to [tocilizumab], which is produced in Chinese hamster ovary cells and based on an IgG2 framework.[L15536] Satralizumab is used in the t…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe terminal half-l…
Vol. DistribusiSatralizumab is sub…
KlirensThe total clearance…
Genetik -
Satraplatin DB04996
small molecule | CAS: 129580-63-8

Satraplatin is a platinum compound that is currently under investigation as one treatment of patients with advanced prostate cancer who have failed previous chemotherapy. As an investigation drug, it has not yet received U.S. Food and Drug Administration (FDA…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsOrganometallic Compounds +1
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Savolitinib DB12048
small molecule | CAS: 1313725-88-0

Savolitinib has been used in trials studying the treatment and health services research of Tumor, Food Effect, Gastric Cancer, Health Subjects, and Colorectal Cancer, among others.

Kategori:
Tyrosine Kinase Inhibitors
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saxagliptin Approved DB06335
small molecule | CAS: 361442-04-8

Saxagliptin (rINN) is an orally active hypoglycemic (anti-diabetic drug) of the new dipeptidyl peptidase-4 (DPP-4) inhibitor class of drugs. FDA approved on July 31, 2009.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +20
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhSaxagliptin = 2.5 h…
Vol. Distribusi151 L
KlirensRenal clearance, si…
Genetik -
SB 11285 DB17511
small molecule

SB 11285 is a second-generation Stimulator of Interferon Genes (STING) agonist.[L45123] SB 11285 is under investigation in clinical trial NCT04096638 (Evaluating Safety and Efficacy of SB 11285 Alone and in Combination With Atezolizumab in Patients With Advan…

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Vol. Distribusi-
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Genetik -
SB 224289 DB17052
small molecule | CAS: 180083-23-2

SB-224289 is a small molecule with a high affinity for human 5-HT1B receptors.[A253122]

Kategori:
Piperidines
Target Protein:
5-hydroxytryptamine receptor 1B
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SB-1578 DB15294
small molecule | CAS: 937273-04-6

SB-1578 is under investigation in clinical trial NCT01235871 (A Single and Multiple-Dose Study of SB1578).

Kategori:
fms-Like Tyrosine Kinase 3, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingJanus Kinase 2, antagonists & inhibitors +1
Target Protein:
Tyrosine-protein kinase JAK2
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Klirens-
Genetik -
SB-218078 DB17051
small molecule | CAS: 135897-06-2

SB-218078 is a specific inhibitor of CHK1.[A253117]

Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-249553 DB05285
small molecule

SB-249553 is a vaccine that has MAGE-3 cancer antigen and the Adjuvant SBAS-2. It is also under by GlaxoSmithKline to treat melanoma and lung cancer.

Waktu Paruh-
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Genetik -
SB-269970 DB13988
small molecule | CAS: 201038-74-6

SB-269970 is an experimental drug developed by GlaxoSmithKline. In the studies performed with this agent, it has been suggested that SB-269970 acts either as a selective antagonist or inverse agonist of the serotonin receptor 7 (5-HT7).[A31816,A31817]

Kategori:
AmidesBenzene DerivativesSulfones +1
Target Protein:
5-hydroxytryptamine receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-649868 DB14822
small molecule | CAS: 380899-24-1

SB-649868 is under investigation in clinical trial NCT01030939 (Study to Investigate Safety, Tolerability, Pharmacokinetics and Cardiac Function After Repeat Doses of SB-649868 in Healthy-volunteers).

Kategori:
Carbon RadioisotopesHeterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Orexin/Hypocretin receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-705498 DB11883
small molecule | CAS: 501951-42-4

SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.

Kategori:
AmidesTRPV Cation Channels, antagonists & inhibitors
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-743921 DB05546
small molecule | CAS: 618430-39-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-773812 DB16042
small molecule | CAS: 630407-66-8

SB-773812 is under investigation in clinical trial NCT00259870 (SB-773812 Administered in Adults With Schizophrenia).

Waktu Paruh-
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Genetik -
SB220025 DB04338
small molecule

Deskripsi belum tersedia.

Kategori:
Calcium-Calmodulin-Dependent Protein Kinases, antagonists & inhibitors
Target Protein:
Mitogen-activated protein kinase 14Mitogen-activated protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB719125 DB16753
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
SBT-100 DB17215
biotech

SBT-100 is an anti-signal transducer and activator of transcription 3 (STAT3) B VHH13 single-domain antibody (sdAb). It was granted orphan drug designation by the FDA for the treatment of pancreatic cancer and osteosarcoma.[L44131,L44136]

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Genetik -
SBT-272 DB18037
small molecule | CAS: 2356106-71-1

Deskripsi belum tersedia.

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Genetik -
SC 41930 DB17101
small molecule | CAS: 120072-59-5

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +9
Target Protein:
Leukotriene B4 receptor 1Leukotriene B4 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SC-236 DB14059
small molecule | CAS: 170569-86-5

SC-236 is a potent, selective, orally active inhibitor of cyclooxygenase-2 (COX-2) [L2964] that has been studied in cancer therapy [A33375], lower back pain [A33376], and inflammation [A33373], [A33374],[L2962], [A33377].

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Cyclooxygenase 2Prostaglandin G/H synthase 2Nuclear factor NF-kappa-B complex
Waktu ParuhLong plasma half-li…
Vol. Distribusi-
Klirens-
Genetik -
SC-74020 DB01630
small molecule

Deskripsi belum tersedia.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
72 kDa type IV collagenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SC12267 DB05125
small molecule

SC12267 is a novel, small molecule agent from the class of DMARDs (disease modifying anti-rheumatic drug) for the therapy of autoimmune diseases such as rheumatoid arthritis or multiple sclerosis. Through highly selective inhibition of pyrimidine biosynthesis…

Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
scAAV9.U7.ACCA DB18582
biotech

scAAV9.U7.ACCA is a non-replicating recombinant adeno-associated virus vector containing 4 antisense sequences designed to target exon 2 in the human DMD gene under the control of U7 small nuclear non-coding RNA. Developed by Nationwide Children’s Hospital, i…

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Scallop Approved DB10623
biotech

Scallop allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Klirens-
Genetik -
Scarlet red Approved DB19136
small molecule | CAS: 85-83-6

Scarlet red is under investigation in clinical trial NCT00591916 (New Treatment for Donor Sites).

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household setting
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SCB-2019 DB15805
biotech

SCB-2019 is a recombinant trimeric S protein subunit vaccine candidate being investigated against COVID-19. This vaccine candidate resembles the native trimeric viral spike and is produced through mammalian cell-culture. The vaccine was developed and test…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
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Genetik -
SCH-486757 DB12782
small molecule | CAS: 524019-25-8

Sch 486757 has been used in trials studying the treatment of Cough.

Kategori:
Aza Compounds
Waktu Paruh-
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Genetik -
SCH-900271 DB12433
small molecule | CAS: 915210-50-3

Sch 900271 has been used in trials studying the treatment of Mixed Hyperlipidemia and Primary Hypercholesterolemia.

Target Protein:
Hydroxycarboxylic acid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Schisandra chinensis fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Scopolamine Approved DB00747
small molecule | CAS: 51-34-3

Scopolamine is a tropane alkaloid isolated from members of the _Solanaceae_ family of plants, similar to [atropine] and [hyoscyamine], all of which structurally mimic the natural neurotransmitter [acetylcholine].[A228423, A228763] Scopolamine was first synthe…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhThe half-life of sc…
Vol. DistribusiThe volume of distr…
KlirensIV infusion of 0.5 …
Genetik -
biotech

Centruroides (scorpion) Immune F(ab')2 (equine) is a purified preparation of immune globulin F(ab’)2 fragments that are derived from plasma of the horses immunized with venom of *C. noxius*, *C. l. limpidus*, *C. l. tecomanus*, and *C. s. suffusus*. It is int…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh159 ± 57 h [FDA lab…
Vol. DistribusiSteady state: 13.6 …
Klirens83.5 ± 38.4 ml/Hr […
Genetik -
Scriptaid DB17053
small molecule | CAS: 287383-59-9

Scriptaid is a histone deacetylase (HDAC) inhibitor researched for its anti-tumor properties.[A253127]

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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