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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 238 / 252
Tritoqualine Approved DB13711
small molecule | CAS: 14504-73-5

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UseCholagogues and CholereticsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRK-001 DB18577
biotech

TRK-001 is an autologous regulatory T-cell therapy. It is being investigated for the prevention of graft rejection following solid organ transplantation.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRK-250 DB18500
biotech

TRK-250 is a small interfering RNA agent that targets human transforming growth factor-beta 1 (TGF-?1) messenger RNA.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troclosene DB15960
small molecule | CAS: 2782-57-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiviral Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trofinetide Approved DB06045
small molecule | CAS: 853400-76-7

Trofinetide is a novel synthetic analog of [glypromate], also known as glycine–proline–glutamate (GPE), a naturally occurring protein in the brain and the N-terminal tripeptide of insulin-like growth factor 1 (IGF-1).[A258438] Trofinetide was approved by the …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +11
Waktu ParuhThe effective elimi…
Vol. DistribusiFollowing oral admi…
KlirensNo information is a…
Genetik -
Trolamine salicylate Approved DB11079
small molecule | CAS: 2174-16-5

Trolamine salicylate is an organic compound or a salt formed between triethanolamine and salicylic acid. Triethanolamine neutralizes the acidity of the salicylic acid. It is a topical analgesic used for temporary relief of minor pain associated with arthritis…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnti-Inflammatory Agents +11
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. DistribusiTopical administrat…
Klirens-
Genetik -
Troleandomycin Approved DB13179
small molecule | CAS: 2751-09-9

A macrolide antibiotic that is similar to erythromycin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +18
Target Protein:
50S ribosomal protein L3250S ribosomal protein L4Nuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tromantadine Approved DB13288
small molecule | CAS: 53783-83-8

Tromantadine is marketed as Viru-Merz in the Czech Republic [L5740]. It is an antiviral used in the treatment of herpes zoster and simplex.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tromethamine Approved DB03754
small molecule | CAS: 77-86-1

An organic amine proton acceptor. It is used in the synthesis of surface-active agents and pharmaceuticals; as an emulsifying agent for cosmetic creams and lotions, mineral oil and paraffin wax emulsions, as a biological buffer, and used as an alkalizer. (Fro…

Kategori:
AlcoholsBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +12
Target Protein:
S-adenosylmethionine decarboxylase proenzymeAmyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropatepine DB13252
small molecule | CAS: 27574-24-9

Tropatepine has been used in France for its antiparkinsons activities [A175024].

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropicamide Approved DB00809
small molecule | CAS: 1508-75-4

Tropicamide is an alkaloid atropine?derived anticholinergic drug and a non?selective antagonist of muscarinic acetylcholine (mACh) receptors.[A230103] Usually available in ophthalmic formulations, tropicamide is used to cause mydriasis and cycloplegia for eye…

Kategori:
Anticholinergic AgentsAutonomic AgentsCholinergic Agents +8
Target Protein:
Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhTropicamide has a p…
Vol. DistribusiNo information can …
KlirensNo information can …
Genetik -
Tropifexor DB16343
small molecule | CAS: 1383816-29-2

Tropifexor is under investigation in clinical trial NCT02516605 (A Multi-part, Double Blind Study to Assess Safety, Tolerability and Efficacy of Tropifexor (LJN452) in PBC Patients).

Kategori:
Heterocyclic Compounds, Fused-RingThiazoles
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropinone DB01874
small molecule | CAS: 532-24-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tropisetron Approved DB11699
small molecule | CAS: 89565-68-4

Tropisetron is an indole derivative with antiemetic activity. As a selective serotonin receptor antagonist, tropisetron competitively blocks the action of serotonin at 5HT3 receptors, resulting in suppression of chemotherapy- and radiotherapy-induced nausea a…

Kategori:
Alimentary Tract and MetabolismAntiarrhythmic agentsAntidepressive Agents +14
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh5.7 h.
Vol. Distribusi400-600 L.
Klirens1800 ml/min.
Genetik -
biotech | CAS: 931101-84-7

Troplasminogen alfa is under investigation in clinical trial NCT00144014 (Safety and Efficacy Study in Acute Ischaemic Stroke).

Kategori:
Amino Acids, Peptides, and ProteinsBeta-GlobulinsBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troriluzole DB15079
small molecule | CAS: 1926203-09-9

Troriluzole is under investigation in clinical trial NCT03701399 (Troriluzole in Adult Subjects With Spinocerebellar Ataxia).

Kategori:
Nervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trotabresib DB17421
small molecule | CAS: 1706738-98-8

Trotabresib is an oral, potent, and reversible inhibitor of the epigenetic target bromodomain and extra-terminal (BET) proteins.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trovafloxacin Approved DB00685
small molecule | CAS: 147059-72-1

Trovafloxacin is a broad spectrum antibiotic that has been commonly marketed under the brand name Trovan by Pfizer. It exerts its antibacterial activity by inhibiting the uncoiling of supercoiled DNA in various bacteria by blocking the activity of DNA gyrase …

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhFollowing oral admi…
Vol. Distribusi-
Klirens-
Genetik -
Troxacitabine DB04961
small molecule | CAS: 145918-75-8

Troxacitabine is a nucleoside analog with antineoplastic activity. There has been growing interest in its development for the treatment of patients with refractory lymphoproliferative conditions.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAntineoplastic Agents +3
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troxerutin DB13124
small molecule | CAS: 7085-55-4

Troxerutin has been used in trials studying the treatment of Chronic Venous Insufficiency.

Kategori:
AnticoagulantsBenzopyransCapillary Stabilizing Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troxipide DB13419
small molecule | CAS: 30751-05-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRU-015 DB05580
small molecule | CAS: 1169717-01-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRV-120027 DB12199
small molecule | CAS: 1234510-46-3

TRV120027 has been used in trials studying the treatment of Heart Failure and Kidney Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-518 DB17534
biotech | CAS: 1427683-53-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-E-002-1 DB17264
small molecule | CAS: 1803036-93-2

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX1 DB05863
biotech

TRX1 is a humanized antibody that binds to the CD4 receptor found on a subset of T cells. TRX1 is being developed for the potential treatment of autoimmune diseases in collaboration with Genentech, Inc. TolerRx is currently conducting a Phase I clinical study…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypan blue free acid Approved DB09158
small molecule | CAS: 2538-83-2

Trypan blue is a diazo dye used in ophthalmic cataract surgery to stain the anterior capsule in the presence of a mature cataract. This is done to aid in visualization before creating the continuous curvilinear capsulorhexis.

Kategori:
ArylsulfonatesArylsulfonic AcidsAzo Compounds +12
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trypsin Approved DB11237
small molecule | CAS: 9002-07-7

Trypsin is a serine protease that plays an essential role in protein hydrolysis and absorption in mammals. When converted from its zymogen trypsinogen, trypsin is available as an active peptide hydrolase (EC 3.4.21.4) form to cleave peptide chains, mainly at …

Kategori:
Blood and Blood Forming OrgansDermatologicalsEndopeptidases +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tryptamine DB08653
small molecule | CAS: 61-54-1

Deskripsi belum tersedia.

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Target Protein:
Amine oxidase [flavin-containing] B5-hydroxytryptamine receptor 2AAmine oxidase [flavin-containing] A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tryptophan Approved DB00150
small molecule | CAS: 73-22-3

An essential amino acid that is necessary for normal growth in infants and for nitrogen balance in adults. It is a precursor of indole alkaloids in plants. It is a precursor of serotonin (hence its use as an antidepressant and sleep aid). It can be a precurso…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +14
Target Protein:
Indoleamine 2,3-dioxygenase 1Tryptophan--tRNA ligase, cytoplasmicTryptophan--tRNA ligase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tryptophanamide DB04537
small molecule | CAS: 20696-57-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Tryptophan--tRNA ligase, cytoplasmicTryptophan--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Tryptophan--tRNA ligase, cytoplasmicTryptophan--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSHA-102 DB18599
biotech

TSHA-102 is a recombinant serotype 9 adeno-associated virus encoding a codon-optimized human MECP2 gene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSHA-104 DB18225
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSHA-105 DB18328
biotech

TSHA-105 is an adeno-associated virus serotype 9 (AAV9) vector with an engineered transgene encoding the human SLC13A5 protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSHA-120 DB16985
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TSN-084 DB18306
small molecule | CAS: 2412309-60-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TST10088 DB05151
small molecule

TST10088 is a recombinant variant of a plant toxin belonging to the family of class II ribosome inactivating proteins. These molecules efficiently kill cells by activating preprogrammed death pathways known as apoptosis. TST10088 has been designed and enginee…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TT-232 DB12088
small molecule | CAS: 147159-51-1

Tln 232 is under investigation in clinical trial NCT00422786 (Phase II Study of CAP-232 in Patients With Refractory Metastatic Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Target Protein:
Pyruvate kinase PKM
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TTI-101 DB17578
small molecule | CAS: 432001-19-9

Deskripsi belum tersedia.

Kategori:
AmidesBenzene DerivativesNaphthalenes +3
Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TTP889 DB05131
small molecule

TTP889, an orally bioavailable selective inhibitor of the intrinsic coagulation pathway, is being developed as an anticoagulant for the treatment of thromboembolic disorders. TTP889 is the only known selective small molecule inhibitor of Factor IX, a key enzy…

Target Protein:
Coagulation factor IX
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
TTX-MC138 DB18628
biotech

TTX-MC138 is an antisense oligonucleotide targeting miR-10b.[L48335] It is under investigation for the treatment of various metastatic cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TTX-siPDL1 DB18550
biotech

TTX-siPDL1 is an siRNA-based modulator of programmed death-ligand 1.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TU-514 DB01991
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycoconjugatesLipids
Target Protein:
UDP-3-O-[3-hydroxymyristoyl] N-acetylglucosamine deacetylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tubimod DB17745
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tubocurarine Approved DB01199
small molecule | CAS: 57-95-4

Tubocurarine is a non-depolarizing neuromuscular blocking agent and the first identified curare alkaloid.[A216008] Curare is one of the names used to describe plant-derived poisons used by indigenous South Americans to coat the tips of hunting arrows and dart…

Kategori:
AlkaloidsAminesAnticholinergic Agents +23
Target Protein:
Neuronal acetylcholine receptor subunit alpha-25-hydroxytryptamine receptor 3AAcetylcholinesterase +1
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Tucatinib Approved DB11652
small molecule | CAS: 937263-43-9

Tucatinib is a kinase inhibitor drug used with [trastuzumab] and [capecitabine] in the treatment of unresectable or metastatic HER-2 positive breast cancer. It was developed by Seattle Genetics and approved by the FDA on April 17, 2020.[L12951] Tucatinib is a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +18
Target Protein:
Receptor tyrosine-protein kinase erbB-2Receptor tyrosine-protein kinase erbB-3
Waktu ParuhA pharmacokinetic s…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
biotech | CAS: 339986-90-2

Tucotuzumab celmoleukin is under investigation in clinical trial NCT00016237 (Interleukin-2 Combined With Monoclonal Antibody Therapy in Treating Patients With Kidney, Bladder, or Lung Cancer That Has Not Responded to Previous Treatment).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulathromycin A DB11474
small molecule | CAS: 217500-96-4

Tulathromycin is a macrolide antibiotic used to treat bovine respiratory disease in cattle and swine respiratory disease in pigs. It is marketed by Pfizer Inc. under the tradename Draxxin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulisokibart DB18719
biotech | CAS: 2648504-55-4

PRA023 is a humanized monoclonal antibody directed to vascular endothelial growth inhibitor, also known as tumour necrosis factor (TNF)-like ligand 1A (TL1A) and TNF superfamily member 15. It is being investigated for ulcerative colitis.

Target Protein:
Tumor necrosis factor ligand superfamily member 15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11851–11900 dari 12560
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