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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 238 / 272
Spebrutinib DB11764
small molecule | CAS: 1202757-89-8

Spebrutinib has been used in trials studying the treatment of Rheumatoid Arthritis, Lymphoma, Large B-Cell, Diffuse, and Leukemia Lymphocytic Chronic B-Cell.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spermaceti DB16556
biotech | CAS: 8002-23-1

Deskripsi belum tersedia.

Kategori:
AlcoholsCetaceaLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spermidine DB03566
small molecule | CAS: 124-20-9

Spermidine is a polyamine formed from putrescine. It is found in almost all tissues in association with nucleic acids. It is found as a cation at all pH values, and is thought to help stabilize some membranes and nucleic acid structures. It is a precursor of …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +2
Target Protein:
Thioredoxin reductase 1, cytoplasmicBeta-1 adrenergic receptorBeta-2 adrenergic receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spermine DB00127
small molecule | CAS: 71-44-3

Spermine is a spermidine-derived biogenic polyamine found as a polycation at all pH values. Found in various tissues and organisms, it often acts as an essential growth factor in some bacterial species. Spermine is associated with nucleic acids, particularly …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +4
Target Protein:
Spermine synthaseCarbonic anhydrase 4Glutamate receptor ionotropic, NMDA 1 +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Spesolimab Approved DB15626
biotech | CAS: 2097104-58-8

Spesolimab is an interleukin-36 (IL-36) receptor antagonist. It is a humanized monoclonal immunoglobulin G1 antibody that was produced in Chinese hamster ovary (CHO) cells by recombinant DNA technology. The biosimilar of the drug, spesolimab-sbzo, was first a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-1 receptor-like 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiBased on the popula…
KlirensIn the linear dose …
Genetik -
SPG302 DB18103
small molecule | CAS: 2274723-90-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SPG601 DB18742
small molecule

SPG601 is being investigated for the treatment of fragile X syndrome.

Waktu Paruh-
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SPH-3127 DB19108
small molecule | CAS: 1399849-02-5

SPH-3127 is under investigation in clinical trial NCT05359068 (Study to Evaluate the Efficacy and Safety of SPH3127 in Patients With Mild-moderate Essential Hypertension).

Kategori:
Oxazines
Waktu Paruh-
Vol. Distribusi-
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Sphingosine DB03203
small molecule | CAS: 123-78-4

An amino alcohol with a long unsaturated hydrocarbon chain. Sphingosine and its derivative sphinganine are the major bases of the sphingolipids in mammals. (Dorland, 28th ed)

Kategori:
AlcoholsAminesAmino Alcohols +2
Target Protein:
Choline-phosphate cytidylyltransferase BGenome polyproteinGenome polyprotein +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sphinxolide B DB04783
small molecule

Deskripsi belum tersedia.

Target Protein:
Actin, alpha skeletal muscle
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spinosad Approved DB08823
small molecule | CAS: 168316-95-8

Spinosad is a pediculicide mixture of spinosyn A and spinosyn D (in an approximately 5:1 ratio, respectively) used in the topical treatment of head lice in children (four years old and older) and in adults. Spinosad is an insecticide based on a compound found…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +6
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. DistribusiNo distribution if …
Klirens-
Genetik -
Spiperone DB17056
small molecule | CAS: 749-02-0

Spiperone is a dopamine antagonist that binds dopamine and serotonin receptors.[A253142]

Kategori:
Antipsychotic AgentsButyrophenonesCentral Nervous System Agents +9
Target Protein:
Alpha-1A adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spirapril Approved DB01348
small molecule | CAS: 83647-97-6

Spirapril is an ACE inhibitor antihypertensive drug used to treat hypertension. Spirapril is converted to the active spiraprilat after administration. ACE inhibitors are used primarily in treatment of hypertension and congestive heart failure.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +9
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh30 to 35 hours
Vol. Distribusi-
Klirens-
Genetik -
Spironolactone Approved DB00421
small molecule | CAS: 52-01-7

Spironolactone is a potassium-sparing diuretic. It binds to mineralocorticoid receptors and functions as aldosterone antagonists.[A178192] It promotes sodium and water excretion and potassium retention.[A11837] Spironolactone was originally developed purely f…

Kategori:
Agents causing hyperkalemiaAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +19
Target Protein:
Mineralocorticoid receptorGlucocorticoid receptorAndrogen receptor +4
Waktu ParuhThe mean half-life …
Vol. Distribusi-
Klirens-
Genetik -
SPK-1001 DB17973
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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SPL23-2 DB17866
biotech

SPL23-2 is an antisense oligonucleotide (ASO) targeting the W1282X nonsense mutation associated with a severe form of cystic fibrosis.[L46767]

Waktu Paruh-
Vol. Distribusi-
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SPL84-23-1 DB18575
biotech

SPL84-23-1 is a sodium salt of 19-bp single-stranded RNA uniformly modified 2'-O-(2-methoxyethyl) phosphorothioate Antisense Oligonucleotide (ASO) consisting of 19 nucleotide residues with the sequence 5'-5MeC-5MeU-G-5MeC-A-A-5MeC-A-G-A-5MeU-G-G-A-A-G-A-5MeC-…

Waktu Paruh-
Vol. Distribusi-
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Sporisorium cruentum Approved DB10873
biotech

Sporisorium cruentum is a fungus which can provoke allergic reactions. Sporisorium cruentum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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SPP 301 DB05290
small molecule

SPP301 (Avosentan) is a potent and highly selective ET[A] receptor blocker and is clinically investigated in diabetic nephropathy. This study was designed to evaluate whether avosentan influences the pharmacokinetics of steroid oral contraceptives.

Target Protein:
Endothelin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SPP1148 DB05203
small molecule

SPP1148, the most promising compound from a new series of renin inhibitors for the treatment of hypertension and related end-organ disease.

Target Protein:
ReninAngiotensin-converting enzyme 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sprifermin DB12616
biotech | CAS: 890058-52-3

Sprifermin has been used in trials studying the treatment of Osteoarthritis, Knee and Cartilage Injury of Knee.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Squalane DB11420
small molecule | CAS: 111-01-3

Deskripsi belum tersedia.

Kategori:
AlkenesHydrocarbons, AcyclicPolyenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Squalene Approved DB11460
small molecule | CAS: 111-02-4

Squalene is originally obtained from shark liver oil. It is a natural 30-carbon isoprenoid compound and intermediate metabolite in the synthesis of cholesterol. It is not susceptible to lipid peroxidation and provides skin protection. It is ubiquitously distr…

Kategori:
AlkenesHydrocarbons, AcyclicPolyenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2892-62-8

Squaric acid dibutyl ester is under investigation in clinical trial NCT01971385 (Safety and Efficacy of Squaric Acid Dibutyl Ester for the Treatment of Herpes Labialis).

Kategori:
Adjuvants, ImmunologicAllergensAntigens +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SR 121463 DB05455
small molecule

SR 121463 is a nonpeptide aquaretic compound with potent selective antagonism of the vasopressin V2 (V1b) receptor subtype. It is a candidate for control of hyponatremia and in the treatment of syndrome of inappropriate secretion of anti-diuretic hormone (SIA…

Target Protein:
Vasopressin V1b receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SR 140333 DB05790
small molecule

SR 140333 is tachykinin antagonist which has potential to treat diarrhoea due to food allergy or inflammatory bowel disease.

Kategori:
Stereoisomerism
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SR-123781A DB05361
biotech | CAS: 232602-93-6

SR-123781A is a synthetic hexadecasaccharide Factor IIa and Xa antagonist. It is under investigation by Sanofi-Aventis and Organon for the treatment of thrombosis and acute coronary syndromes (ACS).

Kategori:
AnticoagulantsCarbohydratesHeparin and similars
Target Protein:
Coagulation factor XProthrombinAntithrombin-III +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SR-9009 DB14013
small molecule | CAS: 1379686-30-2

SR-9009 is a REV-ERB agonist. SR-9011 has been demonstrated that it is specifically lethal to cancer cells and oncogene-induced senescent cells, including melanocytic naevi, and has no effect on the viability of normal cells or tissues [A32628].

Kategori:
Sulfur Compounds
Target Protein:
Nuclear receptor subfamily 1 group D member 1Nuclear receptor subfamily 1 group D member 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SR-9011 DB14014
small molecule | CAS: 1379686-29-9

SR-9011 is a REV-ERB agonist. SR-9011 has been demonstrated that it is specifically lethal to cancer cells and oncogene-induced senescent cells, including melanocytic naevi, and has no effect on the viability of normal cells or tissues [A32628].

Kategori:
Sulfur Compounds
Target Protein:
Nuclear receptor subfamily 1 group D member 2Nuclear receptor subfamily 1 group D member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SR12813 DB04466
small molecule | CAS: 126411-39-0

Deskripsi belum tersedia.

Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRA-737 DB16876
small molecule | CAS: 1489389-18-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sri-9439 DB03351
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sri-9662 DB03060
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRT-1720 DB17057
small molecule | CAS: 925434-55-5

SRT-1720 is an activator of NAD(+)-dependent histone deacetylase SIRT1.[A253147]

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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SRT-2104 DB12186
small molecule | CAS: 1093403-33-8

SRT2104 has been investigated for the basic science and treatment of Sepsis, PSORIASIS, Atrophy, Muscular, and Diabetes Mellitus, Type 2.

Kategori:
Enzyme ActivatorsHeterocyclic Compounds, Fused-Ring
Target Protein:
NAD-dependent protein deacetylase sirtuin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRX-246 DB16968
small molecule | CAS: 512784-93-9

Deskripsi belum tersedia.

Kategori:
Antidiuretic Hormone Receptor AntagonistsAzetinesNatriuretic Agents
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SS1(dsFv)-PE38 DB17579
biotech

SS1(dsFv)-PE38 is a recombinant anti-mesothelin immunotoxin. SS1(dsFv)-PE38 is under investigation in clinical trial NCT01051934 (A Phase I Trial of SS1 (Dsfv) PE38 With Paclitaxel, Carboplatin, and Bevacizumab in Subjects With Unresectable Non-small Cell Lun…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ssCART-19 cells DB18653
biotech

ssCART-19 cells consist of autologous anti-CD19 Chimeric Antigen Receptors (CAR)-T cells expressing a short hairpin RNA (shRNA) against interleukin-6 (IL-6).

Waktu Paruh-
Vol. Distribusi-
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SSR-126517E DB05362
small molecule

SSR-126517E is a second generation synthetic pentasaccharide that binds antithrombin with such high affinity that it assumes a plasma half-life of 80 hours.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST-003 DB18197
biotech | CAS: 143896-17-7

ST-003 is a novel galanin receptor inhibitor being investigated for the treatment of primary sclerosing cholangitis.

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsNeuropeptides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST-101 DB12621
biotech | CAS: 887603-94-3

ST-101 is a small peptide antagonist of C/EBP? and T-type calcium channel activator. ST101 has been used in trials studying the treatment of Essential Tremor and Alzheimer's Disease.[A260411]

Kategori:
Indenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST-36 DB17275
biotech

ST-36 is a cell-penetrating dominant-negative form of activating transcription factor 5. In 2017, it received orphan drug designation by the FDA for the treatment of glioma.[L47341]

Waktu Paruh-
Vol. Distribusi-
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St. John's Wort Approved DB01323
biotech | CAS: 84082-80-4

Deskripsi belum tersedia.

Kategori:
AngiospermsAntidepressive AgentsAntidepressive Agents Indicated for Depression +33
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stachyose DB19276
small molecule | CAS: 470-55-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stannous chloride Approved DB11056
small molecule | CAS: 7772-99-8

Stannous chloride is used as a source of tin in radiopharmaceutical kits. Tin reduces technetium-99m, the active radiological agent, allowing it to form a complex with phosphate-containing moeities [A32700]. These complexes localize primarily in bone (40-50%)…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Stannous fluoride Approved DB11092
small molecule | CAS: 7783-47-3

Stannous Fluoride, or Tn(II) Fluoride, is a compound commonly used in toothpastes for the prevention of gingivitis, dental infections, cavities, and to relieve dental hypersensitivity. Although similar in function and activity to Sodium Fluoride (NaF), the co…

Kategori:
Alimentary Tract and MetabolismCaries Prophylactic AgentsCariostatic Agents +6
Waktu ParuhThe half-life for t…
Vol. DistribusiStannous fluoride i…
KlirensStimulated and nons…
Genetik -
Stannsoporfin DB04912
small molecule | CAS: 106344-20-1

Stannsoporfin is a competitive heme oxygenase (HO) inhibitor being developed by InfaCare, a subsidiary of WellSpring Pharmaceuticals, for the prevention of hyperbilirubinemia in infants at risk of developing jaundice.

Kategori:
Biological FactorsCoordination ComplexesEnzyme Inhibitors +4
Target Protein:
Heme oxygenase 1Heme oxygenase 2
Waktu Paruh3.8 hours following…
Vol. Distribusi-
Klirens-
Genetik -
Stanolone DB02901
small molecule | CAS: 521-18-6

A potent androgenic metabolite of testosterone. Dihydrotestosterone (DHT) is generated by a 5-alpha reduction of testosterone. Unlike testosterone, DHT cannot be aromatized to estradiol therefore DHT is considered a pure androgenic steroid.

Kategori:
5-Androstanon (3) DerivativesAlimentary Tract and MetabolismAnabolic Agents for Systemic Use +17
Target Protein:
Androgen receptorEstrogen receptorMineralocorticoid receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1164-91-6

Stanolone acetate is a synthetic androgen and anabolic steroid and a dihydrotestosterone ester that was never marketed.

Kategori:
P-glycoprotein substratesTestosterone and derivatives
Target Protein:
Androgen receptor17-beta-hydroxysteroid dehydrogenase type 1Estrogen receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stanozolol Approved DB06718
small molecule | CAS: 10418-03-8

Stanozolol is a synthetic anabolic steroid with therapeutic uses in treating hereditary angioedema. Stanozolol is derived from testosterone, and has been abused by several high profile professional athletes.

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +10
Target Protein:
Androgen receptorGlucocorticoid binding proteins
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11851–11900 dari 13591
Sebelumnya Halaman 238 / 272 Berikutnya