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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 238 / 282
Sacubitril Approved DB09292
small molecule | CAS: 149709-62-6

Sacubitril is a prodrug neprilysin inhibitor used in combination with valsartan to reduce the risk of cardiovascular events in patients with chronic heart failure (NYHA Class II-IV) and reduced ejection fraction. It was approved by the FDA after being given t…

Kategori:
Acids, AcyclicAgents causing angioedemaAmino Acids +13
Target Protein:
Neprilysin
Waktu ParuhThe half life of sa…
Vol. Distribusi103 L
Klirens-
Genetik -
Sacubitrilat DB14127
small molecule | CAS: 149709-44-4

A metabolite of LCZ696 with neprilysin inhibitory activity.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +4
Target Protein:
Neprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Safflower oil Approved DB09446
biotech | CAS: 8001-23-8

Safflower (_Carthamus tinctorius_ L) is a herbaceous plant in the Asteraceae family. Extracted from the seeds of safflowers, safflower oil is a rich source of various saturated fatty acids, monounsaturated fatty acid (oleic acid) or essential n-6 polyunsatura…

Kategori:
Biological ProductsComplex MixturesDiet, Food, and Nutrition +10
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Safinamide Approved DB06654
small molecule | CAS: 133865-89-1

Safinamide is for the treatment of parkinson's disease. It was approved in Europe in February 2015, and in the United States on March 21, 2017.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +27
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh22 h
Vol. Distribusi1.8 litres/kg
Klirenstotal oral clearanc…
Genetik -
Safingol DB11924
small molecule | CAS: 15639-50-6

Safingol has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
AlcoholsAminesAmino Alcohols +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Safrazine DB09253
small molecule | CAS: 33419-68-0

Safrazine is a member of the hydrazine family with non-selective and irreversible inhibitor effects against monoamine oxidases. In 1960, it was used as an antidepressant but it is now discontinued.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Safusidenib DB18745
small molecule | CAS: 1898206-17-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sage Approved DB10982
biotech

Sage allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sage oil DB11199
biotech | CAS: 8022-56-8

Sage oil is extracted from sage or *Salvia officinalis*, the herb commonly used for culinary purposes. *Salvia officinalis* is a common sage and a member of the genus *Salvia*, that includes aromatic and perennial plants with flowers. Essential oil has been t…

Kategori:
Agents that reduce seizure thresholdNon-Standardized Food Allergenic ExtractNon-Standardized Plant Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sagopilone DB12391
small molecule | CAS: 305841-29-6

Sagopilone has been used in trials studying the treatment of Melanoma, Neoplasms, CNS Disease, Breast Cancer, and Breast Neoplasms, among others. It is a so-called fully synthetic epothilone and is the first such compound to be in clinical development to comb…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sakuranetin DB08517
small molecule | CAS: 2957-21-3

Deskripsi belum tersedia.

Kategori:
BenzopyransBiological FactorsChromones +3
Target Protein:
Adenosine receptor A2bAdenosine receptor A1Adenosine receptor A3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salicin DB19357
small molecule | CAS: 138-52-3

Deskripsi belum tersedia.

Kategori:
AlcoholsAnalgesicsAnalgesics, Non-Narcotic +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salicylamide Approved DB08797
small molecule | CAS: 65-45-2

Salicylamide is the common name for the substance o-hydroxybenzamide, or amide of salicyl. Salicylamide is a non-prescription drug with analgesic and antipyretic properties. It has similar medicinal uses to aspirin. Salicylamide is used in combination with bo…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25395-22-6

Deskripsi belum tersedia.

Kategori:
Amides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salicylanilide Approved DB19376
small molecule | CAS: 87-17-2

Deskripsi belum tersedia.

Kategori:
AmidesAminesAnilides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salicylic acid Approved DB00936
small molecule | CAS: 69-72-7

A compound obtained from the bark of the white willow and wintergreen leaves, and also prepared synthetically. It has bacteriostatic, fungicidal, and keratolytic actions. Its salts, the salicylates, are used as analgesics.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +35
Target Protein:
Carbonic anhydrase 6Carbonic anhydrase 12Carbonic anhydrase 2 +5
Waktu Paruh-
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Salirasib DB12681
small molecule | CAS: 162520-00-5

Salirasib has been used in trials studying the diagnostic of Carcinoma, Non-Small-Cell Lung.

Kategori:
Acids, CarbocyclicAlcoholsAntineoplastic Agents +11
Target Protein:
Serine/threonine-protein kinase mTORGTPase NRas
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salix alba bark Approved DB14274
biotech

Salix alba bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Herbs and Natural Products
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salix lasiolepis pollen Approved DB10752
biotech

Salix lasiolepis pollen is the pollen of the Salix lasiolepis plant. Salix lasiolepis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salmeterol Approved DB00938
small molecule | CAS: 89365-50-4

Salmeterol is a long-acting beta-2 adrenergic receptor agonist drug that is currently prescribed for the treatment of asthma and chronic obstructive pulmonary disease COPD.[L11545,L11548,L11551,L11554,L11557] It has a longer duration of action than the short-…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +35
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe half life of sa…
Vol. DistribusiIn asthmatic patien…
KlirensThe average clearan…
Genetik -
Salmon calcitonin Approved DB00017
biotech | CAS: 47931-85-1

Synthetic peptide, 32 residues long formulated as a nasal spray.

Kategori:
Amino Acids, Peptides, and ProteinsBone Density Conservation AgentsBone Density, drug effects +15
Target Protein:
Calcitonin receptor
Waktu ParuhHalf-life eliminati…
Vol. Distribusi0.15 to 0.3 L/kg
Klirens-
Genetik -
Salsalate Approved DB01399
small molecule | CAS: 552-94-3

Salsalate is a nonsteroidal anti-inflammatory agent for oral administration. Salsalate's mode of action as an anti-inflammatory and antirheumatic agent may be due to inhibition of synthesis and release of prostaglandins. The usefulness of salicylic acid, the …

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +17
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe parent compound…
Vol. Distribusi-
Klirens-
Genetik -
Saltikva DB18462
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 96574-01-5

Salvianolic acid A is under investigation in clinical trial NCT03908242 (Phase I Study of Continuous Administration of Salvianolic Acid A Tablet).

Kategori:
Acids, CarbocyclicAntineoplastic AgentsCinnamates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 121521-90-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde ReductaseAldehyde Reductase, antagonists & inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salvinorin A DB12327
small molecule | CAS: 83729-01-5

Salvinorin A has been investigated for the basic science of Pharmaceutical Preparations.

Kategori:
AlkaloidsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samalizumab DB12636
biotech | CAS: 1073059-33-2

Samalizumab has been used in trials studying the treatment of Multiple Myeloma and B-cell Chronic Lymphocytic Leukemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samarium DB12403
small molecule | CAS: 7440-19-9

Samarium has been used in trials studying the treatment and prevention of Pain, Cancer, Metastasis, Prostate Cancer, and Metastatic Osteosarcoma, among others.

Kategori:
ElementsLanthanoid Series ElementsMetals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samarium (153Sm) lexidronam Approved DB05273
small molecule | CAS: 122575-21-7

Samarium Sm 153 lexidronam is a radioactive medication used to treat pain caused by cancer that has spread to the bone. It is a radiopharmaceutical. Radiopharmaceuticals are radioactive agents that may be used to diagnose some diseases by studying the functio…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticCentral Nervous System Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samarium Sm-153 DB12905
small molecule | CAS: 15766-00-4

Samarium 153 has been used in trials studying the supportive care of Pain, Lung Cancer, Breast Cancer, Prostate Cancer, and Metastatic Cancer.

Kategori:
ElementsIsotopesLanthanoid Series Elements +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samatasvir DB12660
small molecule | CAS: 1312547-19-5

Samatasvir has been used in trials studying the treatment of Hepatitis C, Chronic, Chronic Hepatitis C Virus, and Chronic Hepatitis C Infection.

Kategori:
Acids, AcyclicHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samidorphan Approved DB12543
small molecule | CAS: 852626-89-2

[Olanzapine] is an effective atypical antipsychotic that, like other antipsychotics, is associated with weight gain, metabolic dysfunction, and increased risk of type II diabetes.[A235638, A235643] Samidorphan is a novel opioid antagonist structurally related…

Kategori:
AlkaloidsAntipsychotic AgentsCentral Nervous System Agents +17
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu ParuhSamidorphan has a m…
Vol. DistribusiSamidorphan followi…
KlirensSamidorphan has a m…
Genetik -
small molecule | CAS: 141646-08-4

Sanfetrinem cilexetil is under investigation in clinical trial NCT05388448 (EBA, Safety and Tolerability of Sanfetrinem Cilexetil).

Kategori:
Amides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapablursen DB18608
biotech | CAS: 2273007-95-5

Sapablursen is a synthetic 2'-O-(2-methoxyethyl)-modified antisense oligonucleotide linked to a tri-antennary cluster of N-acetyl galactosamine (GalNAc3) sugars targeting transmembrane protease, serine 6 messenger ribonucleic acid

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapacitabine DB06365
small molecule | CAS: 151823-14-2

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapanisertib DB11836
small molecule | CAS: 1224844-38-5

Sapanisertib has been used in trials studying the treatment of HCC, Solid Tumor, Gliosarcoma, Liver Cancer, and Glioblastoma, among others.

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapitinib DB12183
small molecule | CAS: 848942-61-0

Sapitinib has been used in trials studying the treatment and basic science of Neoplasms, Breast Cancer, Breast Neoplasms, Metastatic Cancer, and Metastatic Breast Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saprisartan DB01347
small molecule | CAS: 146623-69-0

Saprisartan is an AT1 receptor antagonist. It is based on medications of losartan's prototypical chemical structure. The mode of (functional) AT1 receptor antagonism has been characterized as insurmountable/noncompetitive for saprisartan. It is very likely t…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +6
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapropterin Approved DB00360
small molecule | CAS: 62989-33-7

Sapropterin (tetrahydrobiopterin or BH4) is a cofactor in the synthesis of nitric oxide. It is also essential in the conversion of phenylalanine to tyrosine by the enzyme phenylalanine-4-hydroxylase; the conversion of tyrosine to L-dopa by the enzyme tyrosine…

Kategori:
Alimentary Tract and MetabolismAminesBCRP/ABCG2 Inhibitors +15
Target Protein:
Phenylalanine-4-hydroxylaseNitric oxide synthase 3Tyrosine 3-monooxygenase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saquinavir Approved DB01232
small molecule | CAS: 127779-20-8

Saquinavir is an HIV-1 protease inhibitor used in combination with [ritonavir] and other antiretrovirals for the treatment of human immunodeficiency virus-1 (HIV-1) infection. In 1995 it became the first protease inhibitor approved by the FDA, followed shortl…

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +44
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh-
Vol. DistribusiThe steady-state vo…
KlirensThe systemic cleara…
Genetik -
SAR-125844 DB15382
small molecule | CAS: 1116743-46-4

SAR-125844 is under investigation in clinical trial NCT01391533 (Study of SAR125844 Single Agent Administered as Slow Intravenous Infusion in Adult Patients With Advanced Malignant Solid Tumors).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfur Compounds +1
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR-405838 DB12541
small molecule | CAS: 1303607-60-4

SAR405838 has been used in trials studying the treatment of Neoplasm Malignant.

Kategori:
Heterocyclic Compounds, Fused-RingP-glycoprotein substrates
Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR-439459 DB17864
biotech | CAS: 2114339-57-8

SAR-439459 is a pan-transforming Growth Factor-beta (TGF?) neutralizing antibody.[A259862] Developed by Sanofi, it is being investigated for the treatment of cancers and Osteogenesis Imperfecta.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR421869 DB17909
biotech

SAR421869 is a Lentiviral Vector Containing The Human My07A Gene currently being investigated for the treatment of retinitis pigmentosa associated with Usher syndrome 1B gene defect.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR422459 DB17908
biotech

SAR422459 is a Lentiviral Vector Containing The Human Abca4 Gene that is currently being investigated to treat Stargardt disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR443122 DB16492
small molecule | CAS: 2125450-76-0

SAR443122, was investigated in several clinical trials to evaluate its safety and efficacy. NCT04469621 was studied in severe COVID-19 patients, while NCT05588843 is currently recruiting participants with ulcerative colitis. Additionally, NCT04781816, which w…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR445136 DB17708
biotech

SAR445136 is an investigational zinc finger nuclease gene-edited cell therapy. It consists of autologous CD34+ hematopoietic stem precursor cells (HSPC) modified ex vivo by zinc finger nucleases (ZFN) that target the BCL11A gene erythroid-specific enhancer (E…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 110880-55-2

Sar9, Met (O2)11-Substance P is a neurokinin-1 receptor agonist. It is an analog of the naturally occurring human neuropeptide Substance P, which can be found throughout the body, including in the airways of humans and many other species.

Kategori:
Amino Acids, Peptides, and ProteinsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saracatinib DB11805
small molecule | CAS: 379231-04-6

Saracatinib has been investigated for the treatment of Cancer, Osteosarcoma, Ovarian Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cancer.

Kategori:
Antineoplastic AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +6
Target Protein:
Proto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase ABL1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11851–11900 dari 14063
Sebelumnya Halaman 238 / 282 Berikutnya