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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 237 / 252
Trichlormethiazide Approved DB01021
small molecule | CAS: 133-67-5

A thiazide diuretic with properties similar to those of hydrochlorothiazide. (From Martindale, The Extra Pharmacopoeia, 30th ed, p830)

Kategori:
Antihypertensive AgentsBenzothiadiazinesCardiovascular Agents +13
Target Protein:
Solute carrier family 12 member 3Solute carrier family 12 member 1Sodium/potassium-transporting ATPase subunit alpha-1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75-87-6

Deskripsi belum tersedia.

Kategori:
AlcoholsEthylene GlycolsGlycols
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichloroacetate Approved DB11152
small molecule | CAS: 76-03-9

Trichloroacetate, or trichloroacetic acid, is a strong acid prepared by the reaction of chlorine with acetic acid in the presence of a suitable catalyst. In clinical chemistry and biochemistry, it is used as a precipitant of macromolecules including proteins,…

Kategori:
AcetatesAcids, AcyclicCaustics +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichophyton rubrum Approved DB10915
biotech

Trichophyton rubrum is a fungus which can provoke allergic reactions. Trichophyton rubrum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichophyton verrucosum Approved DB11295
small molecule

Trichophyton verrucosum is a fungus which can provoke allergic reactions. Trichophyton verrucosum extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichostatin A DB04297
small molecule | CAS: 58880-19-6

Deskripsi belum tersedia.

Kategori:
AminesAnti-Infective AgentsAntifungal Agents +9
Target Protein:
Histone deacetylase 7Histone deacetylase 8Acetoin utilization protein +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triciribine DB12405
small molecule | CAS: 35943-35-2

Triciribine has been used in trials studying the treatment of Leukemia, Ovarian Cancer, HER2/Neu Negative, Breast Adenocarcinoma, and Stage IV Breast Cancer, among others.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61966-08-3

Deskripsi belum tersedia.

Kategori:
NaphthalenesNucleic Acids, Nucleotides, and NucleosidesNucleotides
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triclabendazole Approved DB12245
small molecule | CAS: 68786-66-3

Triclabendazole, manufactured by Novartis pharmaceuticals, is an antihelminthic drug that was approved by the FDA in February 2019 for the treatment of fascioliasis in humans.[FDA label, L5452] Fascioliasis is a parasitic infection often caused by the helmi…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +34
Target Protein:
CruzipainExcretory Secretory (ES) proteins
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Triclocarban Approved DB11155
small molecule | CAS: 101-20-2

Triclocarban, with the chemical formula C13H9Cl3N2O [L2675] is an antibacterial agent that is particularly effective against Gram-positive bacteria such as *Staphylococcus aureus*. It is a bacteriostatic compound that has been found in antibacterial soaps and…

Kategori:
AmidesAminesAnilides +10
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADPH] FabI
Waktu Paruh10 hours [L2680]
Vol. Distribusi-
KlirensAfter a pharmacokin…
Genetik -
Triclofos Approved DB06753
small molecule | CAS: 306-52-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triclosan Approved DB08604
small molecule | CAS: 3380-34-5

An aromatic ether that is phenol which is substituted at C-5 by a chloro group and at C-2 by a 2,4-dichlorophenoxy group. It is widely used as a preservative and antimicrobial agent in personal care products such as soaps, skin creams, toothpaste and deodoran…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +11
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH] FabIEnoyl-[acyl-carrier-protein] reductase [NADH]Enoyl-[acyl-carrier-protein] reductase [NADH] FabI +7
Waktu ParuhThe terminal plasma…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2433-96-7

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Target Protein:
Lipase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tricyclazole DB02891
small molecule | CAS: 41814-78-2

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tridecactide DB15687
small molecule | CAS: 22006-64-0

Tridecactide, also known as alpha-corticotropin 1-13, is a deacetylated and deaminated alpha-melanocyte stimulating hormone, which may have antipyretic, anti-inflammatory, and antimicrobial effects.[A203210] Tridecactide, along with [metenkefalin], are under …

Kategori:
Experimental Unapproved Treatments for COVID-19Melanocyte-Stimulating Hormones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tridihexethyl DB00505
small molecule | CAS: 60-49-1

Tridihexethyl is a synthetic anticholinergic agent which has been shown in experimental and clinical studies to have a pronounced antispasmodic and antisecretory effect on the gastrointestinal tract. Tridihexethyl is an antimuscarinic, anticholinergic drug. T…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +7
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2943-75-1

Deskripsi belum tersedia.

Kategori:
NaphthalenesQuinonesSilicon Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triethylenetetramine Approved DB06824
small molecule | CAS: 112-24-3

Triethylenetatramine (TETA), also known as trientine, is a potent and selective copper (II)-selective chelator. It is a structural analog of linear polyamine compounds, [spermidine] and [spermine]. TETA was first developed in Germany in 1861 and its chelating…

Kategori:
Alimentary Tract and MetabolismAminesChelating Agents +11
Target Protein:
Carbonic anhydrase 14
Waktu ParuhThe mean terminal h…
Vol. DistribusiTETA is widely dist…
KlirensIn healthy adult vo…
Genetik -
small molecule | CAS: 7360-38-5

Triethylhexanoin is an ingredient of cosmetic products as a fragrant solvent.

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingExcipients +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trifarotene Approved DB12808
small molecule | CAS: 895542-09-3

Trifarotene is a topical retinoid cream used in the treatment of acne vulgaris that was first approved for use in the United States in October 2019.[L9013] Retinoids are a class of medications structurally and functionally analogous to [vitamin A], though lat…

Kategori:
AlkenesAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +11
Target Protein:
Retinoic acid receptor gammaRetinoic acid receptor betaRetinoic acid receptor alpha
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
Klirens-
Genetik -
Trifluoperazine Approved DB00831
small molecule | CAS: 117-89-5

A phenothiazine with actions similar to chlorpromazine. It is used as an antipsychotic and an antiemetic.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptorCalmodulin-1Calmodulin-3 +6
Waktu Paruh10-20 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thiamine-phosphate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75-89-8

A non-aqueous co-solvent that serves as tool to study protein folding. It is also used in various pharmaceutical, chemical and engineering applications.

Kategori:
Alcohols
Target Protein:
Alcohol dehydrogenase 1CGTPase HRasAlcohol dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 406-95-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trifluperidol DB13552
small molecule | CAS: 749-13-3

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesButyrophenones +11
Target Protein:
Chymase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triflupromazine Approved DB00508
small molecule | CAS: 146-54-3

A phenothiazine used as an antipsychotic agent and as an antiemetic.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntidepressive Agents +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2B +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trifluridine Approved DB00432
small molecule | CAS: 70-00-8

Trifluridine is a fluorinated pyrimidine nucleoside that is structurally related to [idoxuridine] [A35271]. It is an active antiviral agent in ophthalmic solutions used mainly in the treatment of primary keratoconjunctivitis and recurrent epithelial keratitis…

Kategori:
Anti-Infective AgentsAntimetabolitesAntineoplastic Agents +20
Target Protein:
Thymidylate synthaseDNAThymidylate synthase
Waktu ParuhAfter administratio…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Triflusal Approved DB08814
small molecule | CAS: 322-79-2

Triflusal is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a derivative. The benefits of this agent are the lack of action over the arachidonic acid pathway, the driven production of nitric oxide and the in…

Kategori:
Acids, CarbocyclicAnticoagulantsAntiplatelet agents +8
Target Protein:
Prostaglandin G/H synthase 1Nuclear factor NF-kappa-B p105 subunitNitric oxide synthase, inducible +1
Waktu ParuhIn the healthy huma…
Vol. DistribusiThe reported volume…
KlirensRenal clearance is …
Genetik -
Trifolium pratense pollen Approved DB15530
biotech

Trifolium pratense pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Folic Acid and DerivativesVitamin B ComplexVitamins
Target Protein:
Serine hydroxymethyltransferase, cytosolic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trilaciclib Approved DB15442
small molecule | CAS: 1374743-00-6

Trilaciclib, or G1T28, is a CDK4 and CDK6 inhibitor, indicated to reduce the incidence of chemotherapy induced myelosuppression in patients before topotecan-containing or platinum and etoposide-containing chemotherapy for extensive stage small cell lung cance…

Kategori:
BCRP/ABCG2 SubstratesCyclin-dependent Kinase 4 InhibitorsCyclin-dependent Kinase 6 Inhibitors +16
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6Cyclin-dependent kinase 9 +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Trilostane Approved DB01108
small molecule | CAS: 13647-35-3

Trilostane is an inhibitor of 3 beta-hydroxysteroid dehydrogenase used in the treatment of Cushing's syndrome. It was withdrawn from the United States market in April 1994.

Kategori:
Abortifacient AgentsAbortifacient Agents, SteroidalAdrenal Cortex Hormones +20
Target Protein:
3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 13 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2Estrogen receptor +1
Waktu Paruh8 hours.
Vol. Distribusi-
Klirens-
Genetik -
Trimazosin DB09206
small molecule | CAS: 35795-16-5

Trimazosin is a sympatholytic alpha blocker.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +7
Target Protein:
Alpha-1D adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimebutine Approved DB09089
small molecule | CAS: 39133-31-8

Trimebutine is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu opioid agonist effects. It is marketed for the treatment of irritable bowel syndrome (IBS) and lower gastrointestinal…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents producing tachycardia +27
Target Protein:
Mu-type opioid receptorVoltage-dependent L-type calcium channelCalcium-activated potassium channel +5
Waktu ParuhThe elimination hal…
Vol. DistribusiTrimebutine is most…
Klirens-
Genetik -
Trimegestone DB13129
small molecule | CAS: 74513-62-5

Trimegestone has been used in trials studying the treatment of Postmenopause.

Kategori:
Fused-Ring CompoundsGenito Urinary System and Sex HormonesNorpregnadienes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimesic acid DB08632
small molecule | CAS: 554-95-0

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetazidine Approved DB09069
small molecule | CAS: 5011-34-7

Trimetazidine is a piperazine derivative indicated for the symptomatic treatment of stable angina pectoris in patients inadequately controlled or intolerant to first line therapies.[L33015] Trimetazidine has been studied as a treatment for angina pectoris sin…

Kategori:
Cardiac TherapyCardiovascular AgentsPiperazines +1
Target Protein:
3-ketoacyl-CoA thiolase, mitochondrial
Waktu ParuhIn young, healthy s…
Vol. DistribusiThe volume of distr…
KlirensTrimetazidine clear…
Genetik -
Trimethobenzamide Approved DB00662
small molecule | CAS: 138-56-7

Trimethobenzamide is a novel antiemetic which prevents nausea and vomiting in humans. Its actions are unclear but most likely involves the chemoreceptor trigger zone (CTZ). In dogs pretreated with trimethobenzamide HCl, the emetic response to apomorphine is i…

Kategori:
Acids, CarbocyclicAmidesAminoalkyl Ethers +10
Target Protein:
D(2) dopamine receptor
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Trimethoprim Approved DB00440
small molecule | CAS: 738-70-5

Trimethoprim is an antifolate antibacterial agent that inhibits bacterial dihydrofolate reductase (DHFR), a critical enzyme that catalyzes the formation of tetrahydrofolic acid (THF) - in doing so, it prevents the synthesis of bacterial DNA and ultimately con…

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAnti-Infective Agents +32
Target Protein:
Dihydrofolate reductaseDihydrofolate reductase
Waktu ParuhTrimethoprim half-l…
Vol. DistribusiTrimethoprim is ext…
KlirensFollowing oral admi…
Genetik -
small molecule | CAS: 13957-55-6

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2453-03-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethyllysine DB03977
small molecule | CAS: 19253-88-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Calmodulin-2Calmodulin-1Calmodulin-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetrexate Approved DB01157
small molecule | CAS: 52128-35-5

A nonclassical folic acid inhibitor through its inhibition of the enzyme dihydrofolate reductase. It is being tested for efficacy as an antineoplastic agent and as an antiparasitic agent against pneumocystis pneumonia in AIDS patients. Myelosuppression is its…

Kategori:
Acids, AcyclicAcids, AldehydicAnti-Infective Agents +18
Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh11 to 20 hours
Vol. Distribusi* 20 ± 8 L/m2 * 36…
Klirens* 38 +/- 15 mL/min/…
Genetik -
Trimipramine Approved DB00726
small molecule | CAS: 739-71-9

Tricyclic antidepressant similar to imipramine, but with more antihistaminic and sedative properties.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +44
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +15
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +5
Waktu Paruh11-18 hrs
Vol. Distribusi-
Klirens-
Genetik 8 Varian
Trioxsalen Approved DB04571
small molecule | CAS: 3902-71-4

Trioxsalen (trimethylpsoralen, trioxysalen or trisoralen) is a furanocoumarin and a psoralen derivative obtained from several plants, mainly Psoralea corylifolia. Like other psoralens it causes photosensitization of the skin. It is administered either topical…

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +11
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tripamide DB15959
small molecule | CAS: 73803-48-2

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingMembrane Transport Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triphendiol DB06588
small molecule | CAS: 1213777-80-0

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triptolide DB12025
small molecule | CAS: 38748-32-2

Triptolide has been used in trials studying the treatment of HIV, Crohn's Disease, Intestinal Diseases, Gastrointestinal Diseases, and Digestive System Diseases, among others.

Kategori:
Adrenal Cortex HormonesAlkylating DrugsAntineoplastic Agents +10
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triptorelin Approved DB06825
small molecule | CAS: 57773-63-4

Triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH). Possessing greater potency than endogenous LHRH, triptorelin reversibly represses gonadotropin secretion. After chronic, continuous administration, this age…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +23
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiAfter a single IV d…
KlirensIn healthy male vol…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
AzurinThiazole tautomerasePantothenate synthetase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11801–11850 dari 12560
Sebelumnya Halaman 237 / 252 Berikutnya